Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 5973
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103315(US8552199, 1-31)
Affinity DataIC50:  111nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103319(US8552199, 1-38)
Affinity DataIC50:  115nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103314(US8552199, 1-27)
Affinity DataIC50:  117nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103317(US8552199, 1-34)
Affinity DataIC50:  121nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103312(US8552199, 1-15)
Affinity DataIC50:  123nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103311(US8552199, 1-09)
Affinity DataIC50:  139nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103313(US8552199, 1-23)
Affinity DataIC50:  144nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103322(US8552199, 1-46)
Affinity DataIC50:  144nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103316(US8552199, 1-32)
Affinity DataIC50:  147nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103329(US8552199, 1-72)
Affinity DataIC50:  147nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103327(US8552199, 1-62)
Affinity DataIC50:  173nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103330(US8552199, 1-81)
Affinity DataIC50:  179nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103328(US8552199, 1-66)
Affinity DataIC50:  194nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103318(US8552199, 1-36)
Affinity DataIC50:  198nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103320(US8552199, 1-40)
Affinity DataIC50:  208nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103321(US8552199, 1-42)
Affinity DataIC50:  222nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103323(US8552199, 1-47)
Affinity DataIC50:  229nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103332(US8552199, 2)
Affinity DataIC50:  255nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103310(US8552199, 1-05)
Affinity DataIC50:  294nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103324(US8552199, 1-50)
Affinity DataIC50:  766nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103331(US8552199, 1-90)
Affinity DataIC50:  777nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103325(US8552199, 1-55)
Affinity DataIC50:  848nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103326(US8552199, 1-58)
Affinity DataIC50:  1.04E+3nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM103333(US8552199, 3-1)
Affinity DataIC50:  1.14E+3nMAssay Description:Calcium mobilization assay using MCHR1.More data for this Ligand-Target Pair
In DepthDetails US Patent