Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50012024
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553299BDBM50553299(CHEMBL4790404)
Affinity DataIC50: 20nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553304BDBM50553304(CHEMBL4748743)
Affinity DataIC50: 25nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553297BDBM50553297(CHEMBL4747234)
Affinity DataIC50: 25nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553300BDBM50553300(CHEMBL4796729)
Affinity DataIC50: 32nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50316771BDBM50316771((Z,Z)-5-(3-Chloro-4-hydroxy-benzylidene)-2-propyli...)
Affinity DataIC50: 40nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553289BDBM50553289(CHEMBL4763318)
Affinity DataIC50: 40nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553294BDBM50553294(CHEMBL4759157)
Affinity DataIC50: 50nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553287BDBM50553287(CHEMBL4745979)
Affinity DataIC50: 63nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553303BDBM50553303(CHEMBL4748038)
Affinity DataIC50: 79nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553302BDBM50553302(CHEMBL4751870)
Affinity DataIC50: 100nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553288BDBM50553288(CHEMBL4755800)
Affinity DataIC50: 158nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553295BDBM50553295(CHEMBL4758919)
Affinity DataIC50: 200nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553290BDBM50553290(CHEMBL4740803)
Affinity DataIC50: 200nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553293BDBM50553293(CHEMBL4757599)
Affinity DataIC50: 251nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553296BDBM50553296(CHEMBL4789340)
Affinity DataIC50: 501nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553292BDBM50553292(CHEMBL4760357)
Affinity DataIC50: 631nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553304BDBM50553304(CHEMBL4748743)
Affinity DataIC50: 794nMAssay Description:Immunomodulatory activity in human S1PR3 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553301BDBM50553301(CHEMBL4757038)
Affinity DataIC50: 1.00E+3nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553298BDBM50553298(CHEMBL4793543)
Affinity DataIC50: 1.00E+3nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 3(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553306BDBM50553306(CHEMBL4764124)
Affinity DataIC50: 1.00E+3nMAssay Description:Immunomodulatory activity in human S1PR3 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553291BDBM50553291(CHEMBL4743676)
Affinity DataIC50: 1.00E+3nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 1(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553305BDBM50553305(CHEMBL4744825)
Affinity DataIC50: 1.00E+3nMAssay Description:Immunomodulatory activity at human S1PR1 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553306BDBM50553306(CHEMBL4764124)
Affinity DataIC50: 1.00E+4nMAssay Description:Immunomodulatory activity in human S1PR4 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 4(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553304BDBM50553304(CHEMBL4748743)
Affinity DataIC50: 1.00E+4nMAssay Description:Immunomodulatory activity in human S1PR4 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553306BDBM50553306(CHEMBL4764124)
Affinity DataIC50: 1.00E+4nMAssay Description:Immunomodulatory activity at human S1PR2 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSphingosine 1-phosphate receptor 2(Human)
University of Dundee

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50553304BDBM50553304(CHEMBL4748743)
Affinity DataIC50: 1.00E+4nMAssay Description:Immunomodulatory activity at human S1PR2 expressed in CHO-K1 EDG1 beta-arrestin cells assessed as stimulation of beta-arrestin recruitment incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed