Compile Data Set for Download or QSAR
Report error Found 116 Enz. Inhib. hit(s) with all data for entry = 50046108
TargetVesicular acetylcholine transporter(Pacific electric ray)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039623BDBM50039623((2R,3R)-5-Amino-3-(4-phenyl-piperidin-1-yl)-1,2,3,...)
Affinity DataKi:  0.0130nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Pacific electric ray)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039613BDBM50039613(trans-3-(4-phenylpiperidin-1-yl)-1,2,3,4-tetrahydr...)
Affinity DataKi:  0.0550nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Pacific electric ray)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095010BDBM50095010(CHEMBL264437)
Affinity DataKi:  0.340nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Pacific electric ray)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018094BDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  1nMAssay Description:Binding affinity to VAChT Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039613BDBM50039613(trans-3-(4-phenylpiperidin-1-yl)-1,2,3,4-tetrahydr...)
Affinity DataKi:  1.30nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Pacific electric ray)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292907BDBM50292907((+/-)-trans-2-Hydroxy-3-(4-(4-fluorobenzoyl)piperi...)
Affinity DataKi:  2.70nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Torpedo californica electric organ synaptic vesiclesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095010BDBM50095010(CHEMBL264437)
Affinity DataKi:  5.80nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095015BDBM50095015(CHEMBL3589727)
Affinity DataKi:  7.30nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095011BDBM50095011(CHEMBL3589731)
Affinity DataKi:  8.90nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095024BDBM50095024(CHEMBL3589719)
Affinity DataKi:  9.20nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095080BDBM50095080(CHEMBL3590030)
Affinity DataKi:  9.70nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095068BDBM50095068(CHEMBL3589872)
Affinity DataKi:  11nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095014BDBM50095014(CHEMBL3589728)
Affinity DataKi:  12nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095057BDBM50095057(CHEMBL3589714)
Affinity DataKi:  16nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095071BDBM50095071(CHEMBL3589869)
Affinity DataKi:  17nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095059BDBM50095059(CHEMBL3589712)
Affinity DataKi:  17nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095010BDBM50095010(CHEMBL264437)
Affinity DataKi:  18nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095011BDBM50095011(CHEMBL3589731)
Affinity DataKi:  19nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095056BDBM50095056(CHEMBL3589715)
Affinity DataKi:  20nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018094BDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  20nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50329773BDBM50329773((-)-(2R,3R)-5-(2-fluoroethoxy)-3-(4-phenylpiperidi...)
Affinity DataKi:  20nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095075BDBM50095075(CHEMBL3589865)
Affinity DataKi:  20nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095013BDBM50095013(CHEMBL3589729)
Affinity DataKi:  23nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039613BDBM50039613(trans-3-(4-phenylpiperidin-1-yl)-1,2,3,4-tetrahydr...)
Affinity DataKi:  23nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Sprague-Dawley rat brain membranes incubated for 2 hrs by liquid scintillation counting based competi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095023BDBM50095023(CHEMBL3589720)
Affinity DataKi:  23nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095077BDBM50095077(CHEMBL3589863)
Affinity DataKi:  23nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50292907BDBM50292907((+/-)-trans-2-Hydroxy-3-(4-(4-fluorobenzoyl)piperi...)
Affinity DataKi:  24nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095015BDBM50095015(CHEMBL3589727)
Affinity DataKi:  24nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095071BDBM50095071(CHEMBL3589869)
Affinity DataKi:  25nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039623BDBM50039623((2R,3R)-5-Amino-3-(4-phenyl-piperidin-1-yl)-1,2,3,...)
Affinity DataKi:  25nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095064BDBM50095064(CHEMBL3589876)
Affinity DataKi:  25nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039613BDBM50039613(trans-3-(4-phenylpiperidin-1-yl)-1,2,3,4-tetrahydr...)
Affinity DataKi:  26nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095019BDBM50095019(CHEMBL3589724)
Affinity DataKi:  26nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095060BDBM50095060(CHEMBL3589711)
Affinity DataKi:  26nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095069BDBM50095069(CHEMBL3589871)
Affinity DataKi:  30nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095052BDBM50095052(CHEMBL3589716)
Affinity DataKi:  31nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095020BDBM50095020(CHEMBL3589723)
Affinity DataKi:  41nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095076BDBM50095076(CHEMBL3589864)
Affinity DataKi:  43nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095067BDBM50095067(CHEMBL3589873)
Affinity DataKi:  47nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018094BDBM50018094((1R,2R)-2-(4-Phenyl-piperidin-1-yl)-cyclohexanol |...)
Affinity DataKi:  47nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095019BDBM50095019(CHEMBL3589724)
Affinity DataKi:  48nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095074BDBM50095074(CHEMBL3589866)
Affinity DataKi:  54nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095017BDBM50095017(CHEMBL3589732)
Affinity DataKi:  55nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095016BDBM50095016(CHEMBL3589726)
Affinity DataKi:  56nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095063BDBM50095063(CHEMBL3589877)
Affinity DataKi:  59nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095061BDBM50095061(CHEMBL3589879)
Affinity DataKi:  59nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetVesicular acetylcholine transporter(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095018BDBM50095018(CHEMBL3589725)
Affinity DataKi:  60nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in PC12 cell membranes incubated for 2 hrs by liquid scintillation counting based competit...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378717BDBM50378717(CHEMBL1204031)
Affinity DataKi:  61nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095066BDBM50095066(CHEMBL3589874)
Affinity DataKi:  63nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
Institute of Radiopharmaceutical Cancer Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095013BDBM50095013(CHEMBL3589729)
Affinity DataKi:  65nMAssay Description:Displacement of (-)-[3H]pentazocine from sigma1 receptor in Sprague-Dawley rat cortical membranes incubated for 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2016
Entry Details Article
PubMed
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