Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50046610
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.960nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]spiperone from human dopamine D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121336(CHEMBL3622098)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121339(CHEMBL3622095)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121336(CHEMBL3622098)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121338(CHEMBL3622096)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121340(CHEMBL3622094)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121339(CHEMBL3622095)
Affinity DataKi:  600nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121338(CHEMBL3622096)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121343(CHEMBL3622103)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121341(CHEMBL3622093)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121343(CHEMBL3622103)
Affinity DataKi:  930nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121335(CHEMBL3622099)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121340(CHEMBL3622094)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121332(CHEMBL3622101)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121341(CHEMBL3622093)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121337(CHEMBL3622097)
Affinity DataKi:  3.60E+3nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121333(CHEMBL3622100)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121330(CHEMBL3622102)
Affinity DataKi:  4.10E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121333(CHEMBL3622100)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121330(CHEMBL3622102)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121332(CHEMBL3622101)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121342(CHEMBL3622092)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Universit Degli Studi Di Milano

Curated by ChEMBL
LigandPNGBDBM50121342(CHEMBL3622092)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed