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Report error Found 287 of affinity data for UniProtKB/TrEMBL: P05413
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448435(CHEMBL3122088)
Affinity DataKd:  0.200nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) in DMPC liposomes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448436(CHEMBL3122087)
Affinity DataKd:  2.80nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) in DMPC liposomes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448440(CHEMBL1235508)
Affinity DataKd:  3.60nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) at 60 uM by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50212876(2,3-bis[(2,4-dichlorobenzyl)oxy]benzoic acid | CHE...)
Affinity DataKi:  4nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50639276(CHEMBL5543014)
Affinity DataKi:  24nMAssay Description:Binding affinity to FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50002838(5-[2-(4,5-Diphenyl-oxazol-2-yl)-phenoxy]-pentanoic...)
Affinity DataKi:  32nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50247996(5-(2-(trifluoromethyl)benzyl)-5,6,7,8,9,10-hexahyd...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human H-FABP by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM451164(US10709688, Example 4)
Affinity DataIC50: 52nMAssay Description:A Nunc black plate was used as a 96-well plate for the purpose of measurement, and to each well was added 40 μL of sodium phosphate buffer and a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448438(CHEMBL3122153)
Affinity DataKd:  74nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) at 10 uM in DMPC liposomes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM451161(US10709688, Ligand 1 | 4-(2-(1-(2-Methoxyphenyl)-5...)
Affinity DataIC50: 77nMAssay Description:A Nunc black plate was used as a 96-well plate for the purpose of measurement, and to each well was added 40 μL of sodium phosphate buffer and a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM489733(US10968163, Compound 4e)
Affinity DataKi:  80nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50197091(CHEMBL1738980)
Affinity DataKi:  90nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50197091(CHEMBL1738980)
Affinity DataKi:  93nMAssay Description:Displacement of Bodipy-labeled fatty acid from human FABP3 after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2018
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM489700(US10968163, Compound 3-B)
Affinity DataKi:  100nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468452(CHEMBL4283759 | US10968163, Compound 3e)
Affinity DataKi:  100nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50197087(CHEMBL3950316)
Affinity DataKi:  100nMAssay Description:Displacement of Bodipy-labeled fatty acid from human FABP3 after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2018
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50212875(2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3-...)
Affinity DataKi:  110nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50613583(CHEMBL5287034)
Affinity DataKi:  150nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448437(CHEMBL3122151 | Oleate)
Affinity DataKd:  159nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) at 10 uM in DMPC liposomes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468463(CHEMBL4290535 | US10968163, Compound 3i)
Affinity DataKi:  160nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468443(CHEMBL4287414 | US10968163, Compound 4b | US202303...)
Affinity DataKi:  170nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468456(CHEMBL4278244 | US10968163, Compound 3o)
Affinity DataKi:  180nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468442(CHEMBL4276759 | US10968163, Compound 4a)
Affinity DataKi:  190nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50212886([2'-(3-ethyl-4,5-diphenyl-furan-2-yl)-biphenyl-3-y...)
Affinity DataKi:  220nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50063855(CHEMBL3400905)
Affinity DataIC50: 230nMAssay Description:Inhibition of FABP4 (unknown origin) relative to linoleic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50212873(((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPH...)
Affinity DataKi:  250nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM451163(US10709688, Ligand 3 | US10709688, Example 3)
Affinity DataIC50: 280nMAssay Description:A Nunc black plate was used as a 96-well plate for the purpose of measurement, and to each well was added 40 μL of sodium phosphate buffer and a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468439(CHEMBL4293382 | US10968163, Compound 3p)
Affinity DataKi:  310nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50538236(CHEMBL4644782)
Affinity DataKi:  350nMAssay Description:Displacement of 1,8-ANS from recombinant human 6His-tagged FABP3 expressed in Escherichia coli BL21 DE3 incubated for 15 mins followed by 1,8-ANS add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50212882([2'-(5-ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3...)
Affinity DataKi:  360nMAssay Description:Displacement of 1,8-ANS from mFABP by fluorescence based-assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM489714(US10968163, Compound 3l)
Affinity DataKi:  370nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50197092(CHEMBL3947458)
Affinity DataKi:  380nMAssay Description:Inhibition of FABP3 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM451161(US10709688, Ligand 1 | 4-(2-(1-(2-Methoxyphenyl)-5...)
Affinity DataKd:  386nMAssay Description:A Nunc black plate was used as a 96-well plate for the purpose of measurement, and to each well was added 40 μL of sodium phosphate buffer and a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50197092(CHEMBL3947458)
Affinity DataKi:  390nMAssay Description:Displacement of Bodipy-labeled fatty acid from human FABP3 after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2018
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468477(CHEMBL4284051)
Affinity DataKi:  400nMAssay Description:Displacement of DAUDA from recombinant human N-terminal His-tagged FABP3 expressed in Escherichia coli BL21(DE3) after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50197086(CHEMBL3971182)
Affinity DataKi:  400nMAssay Description:Displacement of Bodipy-labeled fatty acid from human FABP3 after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2018
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448439(CHEMBL3122152)
Affinity DataKd:  401nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) at 10 uM in DMPC liposomes by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2014
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM451177(US10709688, Ligand 7)
Affinity DataKd:  414nMAssay Description:A Nunc black plate was used as a 96-well plate for the purpose of measurement, and to each well was added 40 μL of sodium phosphate buffer and a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM489698(US10968163, Compound 3-A | US10968163, Compound 3)
Affinity DataKi:  420nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468462(CHEMBL4287117 | US10968163, Compound 3g | US202303...)
Affinity DataKi:  420nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50063854(CHEMBL3400157)
Affinity DataIC50: 450nMAssay Description:Inhibition of FABP4 (unknown origin) relative to linoleic acidMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2016
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM451169(US10709688, Example 9)
Affinity DataIC50: 510nMAssay Description:A Nunc black plate was used as a 96-well plate for the purpose of measurement, and to each well was added 40 μL of sodium phosphate buffer and a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50525617(CHEMBL4560388)
Affinity DataKd:  520nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli assessed as degree of fluorescent shift by temperature-dependent fluorescence thermal s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468475(CHEMBL4279887 | US10968163, Compound 3j)
Affinity DataKi:  530nMAssay Description:FABP5 was purified and delipidated as described previously (Kaczocha, M. et al. 2012). FABP5 (30 μg), NBD-stearate (1 μM), and a competitor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2021
Entry Details
US Patent

TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50615302(CHEMBL5282728)
Affinity DataKd:  560nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli assessed as degree of fluorescent shift by temperature-dependent fluorescence thermal s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50152851(4-Carbazol-9-yl-butyric acid | 4-(9H-CARBAZOL-9-YL...)
Affinity DataIC50: 600nMAssay Description:Inhibition of FABP3 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468465(CHEMBL4288603 | US10968163, Compound 3l-A)
Affinity DataKi:  640nMAssay Description:Displacement of DAUDA from recombinant human N-terminal His-tagged FABP3 expressed in Escherichia coli BL21(DE3) after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50248238(9-(2-methylbenzyl)-8-(prop-1-en-2-yl)-2,3,4,9-tetr...)
Affinity DataIC50: 680nMAssay Description:Inhibition of human H-FABP by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50468443(CHEMBL4287414 | US10968163, Compound 4b | US202303...)
Affinity DataKi:  690nMAssay Description:Displacement of DAUDA from recombinant human N-terminal His-tagged FABP3 expressed in Escherichia coli BL21(DE3) after 20 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetFatty acid-binding protein, heart(Human)
Osaka University

Curated by ChEMBL
LigandPNGBDBM50429939(CHEMBL2334261 | US10709688, Example 6)
Affinity DataIC50: 695nMAssay Description:Inhibition of human FABP3 by 8-anilino-1-naphthalenesulfonic acid based fluorescence displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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