Compile Data Set for Download or QSAR
maximum 50k data
Found 599 of affinity data for UniProtKB/TrEMBL: Q79MP6
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336509(CHEMBL116455 | Mercapto-acetic acid | Mercaptoacet...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336510(7,8-dihydroxy-1-methoxy-3-methyl-10-oxo-1,10-dihyd...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50121953(2-mercaptoethanecarboxylic acid | 3-mercaptopropan...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336511((4R,5S,6S)-3-(benzo[b]thiophen-2-ylthio)-6-((R)-1-...)
Affinity DataKi:  180nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50336508(CHEMBL1673299 | sodium 2,3-diethylmaleate)
Affinity DataKi:  410nMAssay Description:Inhibition of Pseudomonas aeruginosa beta-lactamase IMP-1 assessed as hydrolysis of nitrocefin by UV spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa MBL IMP-1 using nitrocefin as substrate preincubated for 20 mins by UV-spectrophotometric analysisMore data for this Ligand-Target Pair
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50421220(CHEMBL2087628)
Affinity DataKi:  3.30E+3nMAssay Description:Inhibition of recombinant Pseudomonas aeruginosa MBL IMP-1 using nitrocefin as substrate preincubated for 20 mins by UV-spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530895((R)-4-(4-(2-(1H-pyrazol- 1-yl)ethyl)piperidin-1- y...)
Affinity DataIC50:  0.0500nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530978(4-[4-(pyridin-2- yloxy)piperidin-1-yl]-N1- [(3R)-p...)
Affinity DataIC50:  0.100nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530914((R)-N1-(1- aminopropan-2- yl)-4-(4- (hydroxymethyl...)
Affinity DataIC50:  0.120nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530974(4-[4-(pyridin-2- ylmethyl)piperidin-1-yl]-N1- [(3R...)
Affinity DataIC50:  0.120nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530956(4-[4-(2- hydroxyethoxy)piperidin-1- yl]-N1-[(3R)-p...)
Affinity DataIC50:  0.130nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530966(4-[4-(2- hydroxyethyl)piperidin-1- yl]-N1-[(3R)-py...)
Affinity DataIC50:  0.130nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530969(4-[4- (hydroxymethyl)piperidin- 1-yl]-N1-[(3R)-pyr...)
Affinity DataIC50:  0.160nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531045(N1-((R)-3-amino-2- hydroxypropyl)-4-(4-(2- oxooxaz...)
Affinity DataIC50:  0.190nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531034((R)-4-(4-(1H-imidazol-4-yl)piperidin-1-yl)-N1-(pyr...)
Affinity DataIC50:  0.220nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531036((S)-4-(4-(1H-imidazol-4-yl)piperidin-1-yl)-N1-(2,3...)
Affinity DataIC50:  0.240nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530955(4-[4-(2- fluoroethyl)piperidin-1-yl]- N1-[(3R)-pyr...)
Affinity DataIC50:  0.240nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531055((S)-N1-(1-amino-3- hydroxypropan-2-yl)-4-(4-(2- am...)
Affinity DataIC50:  0.240nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531035((R)-4-(4-(N-(2-aminoethyl)sulfamoyl)piperidin-1-yl...)
Affinity DataIC50:  0.25nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531037((R)-4-(4-(1H-imidazol-4-yl)piperidin-1-yl)-N1-(3-a...)
Affinity DataIC50:  0.260nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530960(1-{4-[(3R)-pyrrolidin-3- ylsulfamoyl]-3-sulfamoyl-...)
Affinity DataIC50:  0.310nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531042((R)-4-(4-(1H-imidazol-1- yl)piperidin-1-yl)-N1-(3-...)
Affinity DataIC50:  0.360nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530887((R)-N1-(1-aminopropan- 2-yl)-4-(4- (hydroxymethyl)...)
Affinity DataIC50:  0.370nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530893((R)-2-(1-(4-(N-(3-amino- 2- hydroxypropyl)sulfamoy...)
Affinity DataIC50:  0.390nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530948(N1-[(3R)-pyrrolidin-3-yl]-4- (4-sulfamoylpiperidin...)
Affinity DataIC50:  0.430nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530924(6-(azetidin-3-ylsulfonyl)-3-[4- (2-hydroxyethyl)pi...)
Affinity DataIC50:  0.450nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530910((R)-N1-(3-amino- 2-hydroxypropyl)- 4-(4- (hydroxym...)
Affinity DataIC50:  0.470nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530931(4-(4-hydroxypiperidin-1- yl)-N1-[(3R)-pyrrolidin-3...)
Affinity DataIC50:  0.470nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530962(1-{4-[(3R)-pyrrolidin-3- ylsulfamoyl]-3-sulfamoyl-...)
Affinity DataIC50:  0.5nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530938(4-[(3R)-3- (hydroxymethyl)pyrrolidin- 1-yl]-N1-[(3...)
Affinity DataIC50:  0.510nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530913(N1-(1,3- diaminopropan-2- yl)-4-(4- (hydroxymethyl...)
Affinity DataIC50:  0.520nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531032(Methyl 1-(4-(N-((R)- pyrrolidin-3-yl)sulfamoyl)-3-...)
Affinity DataIC50:  0.540nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530985((R)-N1-(3-amino-2-hydroxypropyl)-4-(4-(2-(methylsu...)
Affinity DataIC50:  0.550nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530889((R)-N1-(3-amino-2- hydroxypropyl)-4-(4- (hydroxyme...)
Affinity DataIC50:  0.560nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530912((S)-N1-(2,3- diaminopropyl)-4- (4- (hydroxymethyl)...)
Affinity DataIC50:  0.560nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531070((S)-N1-(1-amino-3-hydroxypropan-2-yl)-4-(4-(N-(2-a...)
Affinity DataIC50:  0.580nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530911(N1-(2- aminoethyl)-4-(4- (hydroxymethyl) piperidin...)
Affinity DataIC50:  0.580nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531053((R)-4-(4-(2-aminoethyl)piperidin-1-yl)-N1-(1-amino...)
Affinity DataIC50:  0.600nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530999((R)-N1-(3-amino-2- hydroxypropyl)-4-(4-(N-(2- amin...)
Affinity DataIC50:  0.610nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530957(4-[4- (fluoromethyl)piperidin-1- yl]-N1-[(3R)-pyrr...)
Affinity DataIC50:  0.610nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530949(4-[3-(2- hydroxyethyl)pyrrolidin-1- yl]-N1-[(3R)-p...)
Affinity DataIC50:  0.620nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531061((R)-N1-(3-amino-2-hydroxypropyl)- 4-(4-(3-aminopro...)
Affinity DataIC50:  0.670nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530890((R)-N1-(3-amino-2- hydroxypropyl)-4-(4- fluoro-4- ...)
Affinity DataIC50:  0.700nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530939(4-(4-hydroxy-4- methylpiperidin-1-yl)-N1- [(3R)-py...)
Affinity DataIC50:  0.700nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530988((R)-N1-(3-amino-2- hydroxypropyl)-4-(4- hydroxypip...)
Affinity DataIC50:  0.760nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530958(4-[4- (difluoromethyl)piperidin-1- yl]-N1-[(3R)-py...)
Affinity DataIC50:  0.770nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531057((S)-N1-(1-amino-3- hydroxypropan-2-yl)-4-(4- (amin...)
Affinity DataIC50:  0.770nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM531069((R)-4-(4-(1H-imidazol-2-yl)piperidin-1-yl)-N1-(3-a...)
Affinity DataIC50:  0.770nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Toho University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM530926(6-(azetidin-3-ylsulfonyl)-3-[4- (hydroxymethyl)pip...)
Affinity DataIC50:  0.850nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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