TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.00400nMAssay Description:Inhibition of aromatase (unknown origin) transfected in human MCF7 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0150nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0150nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0180nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0300nMAssay Description:Aromatase inhibitor potency as iron-binding-related type II difference spectrumMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione as substrate after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of aromatase in human placental microsomeMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human placental microsome aromatase using [1beta,2beta3H]androstenedione as substrate by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.120nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.180nMpH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of aromatase in human JEG3 cells using [1beta-3H] androstenedione as substrate assessed as tritiated H2O release after 1 hr by scintillati...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione as substrate after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.210nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.220nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.260nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.330nMpH: 7.5 T: 2°CAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.350nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.390nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human placental microsome aromatase using [1beta,2beta3H]androstenedione as substrate by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Ligand Info
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:The extent of in vitro inhibition of aromatase activities was assessed using intact monolayers of JEG-3 cells. Aromatase activity was measured using ...More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.420nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Inhibition of aromatase (unknown origin) expressed in JEG-3 cellsMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.460nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of aromatase in human JEG-3 cells using [1beta-3H]androstenedione after 1 hr by scintillation spectrometryMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of aromatase in human JEG-3 cells using Androst-4-ene-3,17-dione as substrate incubated for 1 hr and measured by BCA assayMore data for this Ligand-Target Pair
TargetAromatase(Homo sapiens (Human))
State University Of New York Upstate Medical University
Curated by ChEMBL
State University Of New York Upstate Medical University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of aromatse in human JEG3 cells by scintillation spectrometryMore data for this Ligand-Target Pair