Compile Data Set for Download or QSAR
Report error Found 126 of affinity data for UniProtKB/TrEMBL: Q60613
TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474329BDBM474329(US10858365, Compound 116 | 7-(3-fluoro-1H-pyrazol-...)
Affinity DataIC50: 0.200nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474284BDBM474284(US10858365, Compound 69 | 7-(4-fluorophenyl)-2-((3...)
Affinity DataIC50: 0.300nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474287BDBM474287(US10858365, Compound 73 | 2-((3-(difluoromethoxy)p...)
Affinity DataIC50: 0.400nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474328BDBM474328(US10858365, Compound 114 | 7-(4-fluorophenyl)-2-(2...)
Affinity DataIC50: 0.400nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474223BDBM474223(2-(2,6-difluorobenzyl)-8-(2-(dimethylamino) pyridi...)
Affinity DataIC50: 0.400nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474330BDBM474330(US10858365, Compound 117 | 7-(4-fluoro-1H-pyrazol-...)
Affinity DataIC50: 0.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474281BDBM474281(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50: 0.600nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474222BDBM474222(5-(5-amino-2-(2,6-difluorobenzyl)-7-(4- fluorophen...)
Affinity DataIC50: 0.800nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474233BDBM474233(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50: 0.800nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474309BDBM474309(US10858365, Compound 99 | 2-((3-fluoropyridin-2-yl...)
Affinity DataIC50: 0.800nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474292BDBM474292(US10858365, Compound 79 | 5-(5-am i no-2-(2,6-difl...)
Affinity DataIC50: 0.900nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474315BDBM474315(US10858365, Compound 105-1 | 7-(4-fluorophenyl)-8-...)
Affinity DataIC50: 1nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474316BDBM474316(US10858365, Compound 105-2 | 7-(4-fluorophenyl)-8-...)
Affinity DataIC50: 1nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474288BDBM474288(US10858365, Compound 74 | 2-((3-(difluoromethoxy)p...)
Affinity DataIC50: 1.20nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474300BDBM474300(US10858365, Compound 89 | 7-(4-fluorophenyl)-2-((3...)
Affinity DataIC50: 1.30nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474245BDBM474245(2-(2,6-difluorobenzyl)-7-(4-fluorophenyl)-8-(2- me...)
Affinity DataIC50: 1.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474335BDBM474335(US10858365, Compound 122 | (S)-7-(4-fluorophenyl)-...)
Affinity DataIC50: 2.60nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474299BDBM474299(US10858365, Compound 88 | 8-(benzo[d]thiazol-6-yl)...)
Affinity DataIC50: 2.60nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474258BDBM474258(5-[5-amino-7-(4-fluorophenyl)-2-[(3-fluoropyrid in...)
Affinity DataIC50: 2.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474334BDBM474334(US10858365, Compound 121 | 2-(2,6-difluorobenzyl)-...)
Affinity DataIC50: 2.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474230BDBM474230(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 3.40nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474310BDBM474310(US10858365, Compound 100 | 2-((3*fluoropyridin-2-y...)
Affinity DataIC50: 3.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474301BDBM474301(US10858365, Compound 90 | 2-((3-fluoropyridin-2-yl...)
Affinity DataIC50: 3.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474337BDBM474337(US10858365, Compound 124 | 7-(azetidin-l-yl)-2-(2,...)
Affinity DataIC50: 3.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474224BDBM474224(5-(5-amino-2-[[3-(difluoromethoxy)pyridin-2-yl] me...)
Affinity DataIC50: 4.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474293BDBM474293(US10858365, Compound 80 | 5-(5-amino-2-((3-fluorop...)
Affinity DataIC50: 4.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474302BDBM474302(US10858365, Compound 91 | 2-(2,6-difluorobenzyl)-8...)
Affinity DataIC50: 5.10nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474263BDBM474263(5-(5-amino-7-(4-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 5.10nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474229BDBM474229(7-(4-fluorophenyl)-2-((3-fluoropyridin-2-yl) methy...)
Affinity DataIC50: 5.40nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474314BDBM474314(US10858365, Compound 104 | (R)-7-(4-fluorophenyl)-...)
Affinity DataIC50: 5.70nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474273BDBM474273(5-(5-amino-2-(2,6-difluorobenzyl)-7-(thiazol-2- yl...)
Affinity DataIC50: 5.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474285BDBM474285(US10858365, Compound 71 | 5-(5-amino-2-[[3-(difluo...)
Affinity DataIC50: 6.40nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474231BDBM474231(6-[[5-amino-7-(4-fluorophenyl)-8-[imidazo[1,2-a] p...)
Affinity DataIC50: 7.30nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474305BDBM474305(US10858365, Compound 95 | 5-(5-amino-7-(4-fluoroph...)
Affinity DataIC50: 8.90nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474333BDBM474333(US10858365, Compound 120 | 2-(2-(dimethylamino)eth...)
Affinity DataIC50: 9.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474256BDBM474256(8-(2-chloro-6-methylpyridin-4-yl)-7-(4- fluorophen...)
Affinity DataIC50: 9.60nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474221BDBM474221(8-(2,6-dimethylpyridin-4-yl)-7-(4-fluoropheny1)- 2...)
Affinity DataIC50: 10nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474239BDBM474239(2-(2,6-difluorobenzyl)-8-(2-(difluoromethoxy) pyri...)
Affinity DataIC50: 11nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474303BDBM474303(US10858365, Compound 92 | 5-[5-amino-2-[(2,6-diflu...)
Affinity DataIC50: 11nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474312BDBM474312(US10858365, Compound 102 | 2-((3-fluoropyridin-2-y...)
Affinity DataIC50: 11.2nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474283BDBM474283(US10858365, Compound 68 | 7-(4-fluorophenyl)-8-[im...)
Affinity DataIC50: 12nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474226BDBM474226(5-(5-amino-2-(2,6-difluorobenzyl)-7-(oxazol-2- y1)...)
Affinity DataIC50: 12nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474271BDBM474271(5-[5-amino-7-(4-nuorophenyl)-2-[(1,3-thiazol-2- yl...)
Affinity DataIC50: 13nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474237BDBM474237(5-(5-amino-7-(3-chlorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 13nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474270BDBM474270(5-(5-amino-7-(3-fluorophenyl)-2-((3-fluoropyrid in...)
Affinity DataIC50: 15nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474278BDBM474278(5-(5-amino-2-(2,6-difluorobenzyl)-7-(4-fluoroph en...)
Affinity DataIC50: 16nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474336BDBM474336(US10858365, Compound 123 | 2-(2,6-difluorobenzyl)-...)
Affinity DataIC50: 16.5nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474238BDBM474238(5-(5-amino-2-((3-fluoropyridin-2-yl)methyl)-7- (3-...)
Affinity DataIC50: 17nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474289BDBM474289(US10858365, Compound 75 | 8-(1H-benzo[d]imidazol-6...)
Affinity DataIC50: 17nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetAdenosine receptor A2a(Mouse)
TBA

US Patent
LigandChemical structure of BindingDB Monomer ID 474252BDBM474252(8-(2,6-dimethyIpyridin-4-yl)-7-(4-fluorophenyl)- 2...)
Affinity DataIC50: 18nMAssay Description:hADORA1/CHO (hA1 expressing) cells (Genscript) were plated at 1×104 cells/well into 384-well polystyrene plates one day before starting the experimen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

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