Compile Data Set for Download or QSAR
Report error Found 61 of affinity data for UniProtKB/TrEMBL: Q8VHL0
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394962BDBM50394962(CHEMBL1394231)
Affinity DataIC50: 11nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394962BDBM50394962(CHEMBL1394231)
Affinity DataIC50: 11nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394961BDBM50394961(CHEMBL2165788)
Affinity DataIC50: 14nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394961BDBM50394961(CHEMBL2165788)
Affinity DataIC50: 14nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394961BDBM50394961(CHEMBL2165788)
Affinity DataIC50: 23nMAssay Description:Inhibition of UT-B-mediated urea transport in wild type CD1 mouse erythrocytes incubated for 10 mins prior to urea addition by Stopped-flow light sca...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394962BDBM50394962(CHEMBL1394231)
Affinity DataIC50: 25.1nMAssay Description:Reversible inhibition of mouse UT-B-mediated urea transportMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394964BDBM50394964(CHEMBL1590659)
Affinity DataIC50: 32nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435308BDBM50435308(CHEMBL2391344)
Affinity DataIC50: 38nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435309BDBM50435309(CHEMBL2391345)
Affinity DataIC50: 43nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394967BDBM50394967(CHEMBL2165784)
Affinity DataIC50: 104nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394972BDBM50394972(CHEMBL1372659)
Affinity DataIC50: 153nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580922BDBM50580922(CHEMBL5087071)
Affinity DataIC50: 160nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394966BDBM50394966(CHEMBL2165785)
Affinity DataIC50: 196nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50322183BDBM50322183(CHEMBL1173569 | UT-A1 inhibitor D4 | 3-(4-ethylphe...)
Affinity DataIC50: 212nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580906BDBM50580906(CHEMBL5074722)
Affinity DataIC50: 240nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435310BDBM50435310(CHEMBL2391346)
Affinity DataIC50: 353nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394965BDBM50394965(CHEMBL2165786)
Affinity DataIC50: 468nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580917BDBM50580917(CHEMBL5077469)
Affinity DataIC50: 480nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394970BDBM50394970(CHEMBL2165781)
Affinity DataIC50: 537nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607929BDBM50607929(CHEMBL5279934)
Affinity DataIC50: 690nMAssay Description:Inhibition of UT-B in mouse erythrocyte incubated for 10 mins by stopped-flow light scattering assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580912BDBM50580912(CHEMBL5091945)
Affinity DataIC50: 690nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435306BDBM50435306(CHEMBL2391348)
Affinity DataIC50: 800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435305BDBM50435305(CHEMBL2391347)
Affinity DataIC50: 800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435307BDBM50435307(CHEMBL2391349)
Affinity DataIC50: 800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580905BDBM50580905(CHEMBL5082942)
Affinity DataIC50: 840nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50134204BDBM50134204(CHEMBL3740772)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of UT-B in mouse erythrocyte incubated for 15 mins by erythrocyte osmotic lysis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580911BDBM50580911(CHEMBL5075260)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580910BDBM50580910(CHEMBL5069410)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394969BDBM50394969(CHEMBL2165782)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580909BDBM50580909(CHEMBL5084723)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580908BDBM50580908(CHEMBL5083627)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580913BDBM50580913(CHEMBL5085745)
Affinity DataIC50: 1.49E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580900BDBM50580900(CHEMBL5081628)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580916BDBM50580916(CHEMBL5085556)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607929BDBM50607929(CHEMBL5279934)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of UT-B in mouse erythrocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580907BDBM50580907(CHEMBL5094101)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580903BDBM50580903(CHEMBL5080875)
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580914BDBM50580914(CHEMBL5072845)
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580899BDBM50580899(CHEMBL5081622)
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394963BDBM50394963(CHEMBL2165787)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580915BDBM50580915(CHEMBL5077837)
Affinity DataIC50: 3.47E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607934BDBM50607934(CHEMBL1374572)
Affinity DataIC50: 4.15E+3nMAssay Description:Inhibition of UT-B in mouse erythrocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580904BDBM50580904(CHEMBL5089501)
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394968BDBM50394968(CHEMBL2165783)
Affinity DataIC50: 5.29E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50394974BDBM50394974(CHEMBL1725922)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of UT-B in wild type CD1 mouse erythrocyte assessed as hemolysis after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580898BDBM50580898(CHEMBL5083889)
Affinity DataIC50: 5.82E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580918BDBM50580918(CHEMBL5070486)
Affinity DataIC50: 9.85E+3nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580901BDBM50580901(CHEMBL5085679)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50607931BDBM50607931(CHEMBL5289033)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of UT-B in C57BL/6J mouse erythrocyte incubated for 6 min by erythrocyte osmotic lysis based high-throughput screening assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetUrea transporter 1(Mouse)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50580902BDBM50580902(CHEMBL5082057)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse UT-B expressed in MDCK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
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