Compile Data Set for Download or QSAR
Report error Found 200 Enz. Inhib. hit(s) with Target = 'Neuropeptide S receptor'
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477899(CHEMBL438162)
Affinity DataEC50:  0.646nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  0.676nMAssay Description:Agonist activity at human NPSR Ile107 expressed in HEK293 cells assessed as induction of calcium mobilization after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477901(CHEMBL437201)
Affinity DataEC50:  0.676nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477898(CHEMBL441576)
Affinity DataEC50:  0.708nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  0.851nMAssay Description:Agonist activity at human NPSR Asn107 expressed in HEK293 cells assessed as induction of calcium mobilization after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443390(CHEMBL1474387)
Affinity DataIC50: 0.960nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50418333(CHEMBL1765705)
Affinity DataEC50:  1.07nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as induction of calcium mobilization after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477880(CHEMBL430024)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322839(rac-N-(3-methyl-1-morpholinopentan-3-yl)-N-((1-met...)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as cAMP level after 30 mins by phosphate-buffered sal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443390(CHEMBL1474387)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced ERK activation after 20 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322839(rac-N-(3-methyl-1-morpholinopentan-3-yl)-N-((1-met...)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]Tyr10-NPS from neuropeptide S receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477895(CHEMBL409981)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477884(CHEMBL267034)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477893(CHEMBL398524)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477894(CHEMBL398483)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50417462(CHEMBL469696)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human recombinant GPR154 receptor expressed in HEK293 cells assessed as inhibition of neuropeptide S-induced increase of intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477883(CHEMBL400369)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443406(CHEMBL3086823)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477889([2Nal2]hNPS)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412701(CHEMBL525809)
Affinity DataEC50:  2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  2.24nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477900(CHEMBL437199)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477887(CHEMBL437389)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443409(CHEMBL3086836)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477885(CHEMBL252537)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443408(CHEMBL3086837)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443400(CHEMBL3086821)
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443390(CHEMBL1474387)
Affinity DataIC50: 3.5nMAssay Description:Displacement of [125I]Tyr10-NPS from human neuropeptide S receptor expressed in CHO cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477892(CHEMBL411392)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477882(CHEMBL413849)
Affinity DataEC50:  4.20nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443405(CHEMBL3086824)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50412707(CHEMBL230333)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443391(CHEMBL469695)
Affinity DataIC50: 5.30nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as cAMP level after 30 mins by phosphate-buffered sal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443404(CHEMBL3086825)
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443392(CHEMBL1472563)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced ERK activation after 20 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322839(rac-N-(3-methyl-1-morpholinopentan-3-yl)-N-((1-met...)
Affinity DataIC50: 6.70nMAssay Description:Displacement of [125I]Tyr10-NPS from human neuropeptide S receptor expressed in CHO cells after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322836(rac-N-(3-methyl-1-(piperidin-1-yl)pentan-3-yl)-N-(...)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477897(CHEMBL427638)
Affinity DataEC50:  8.10nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477896(CHEMBL268436)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443399(CHEMBL3086822)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443398(CHEMBL1514777)
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced ERK activation after 20 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50443407(CHEMBL3086838)
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced calcium mobilization aft...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50331943(5-phenyl-2-(2-(piperidine-1-carbonyl)phenyl)-2,3-d...)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant GPR154 receptor expressed in HEK293 cells assessed as inhibition of neuropeptide S-induced increase of intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322839(rac-N-(3-methyl-1-morpholinopentan-3-yl)-N-((1-met...)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) assessed as intracellular calcium level by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50331943(5-phenyl-2-(2-(piperidine-1-carbonyl)phenyl)-2,3-d...)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) assessed as intracellular calcium level by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322839(rac-N-(3-methyl-1-morpholinopentan-3-yl)-N-((1-met...)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant NPS receptor expressed in CHOK1 cells assessed as inhibition of NPS-induced calcium mobilization by FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50477881(CHEMBL2372117)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse recombinant NPS receptor expressed in HEK293 cells assessed as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Human)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50322839(rac-N-(3-methyl-1-morpholinopentan-3-yl)-N-((1-met...)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at neuropeptide S receptor (unknown origin) expressed in CHO cells assessed as inhibition of NPS-induced ERK activation after 20 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetNeuropeptide S receptor(Mouse)
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50479763(CHEMBL524693)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse NPSR expressed in HEK293 cells assessed as increase in intracellular calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
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