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Found 69 with Last Name = 'armour' and Initial = 'd'
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470670(CHEMBL149557)
Affinity DataKi:  0.0316nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50410193(CHEMBL356062 | GR-203040)
Affinity DataKi:  0.0501nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470675(CHEMBL344536)
Affinity DataKi:  0.0501nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470678(CHEMBL146885)
Affinity DataKi:  0.0501nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470683(CHEMBL356786)
Affinity DataKi:  0.0631nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470669(CHEMBL359188)
Affinity DataKi:  0.0631nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470672(CHEMBL434884)
Affinity DataKi:  0.0794nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470667(CHEMBL424301)
Affinity DataKi:  0.126nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470677(CHEMBL147776)
Affinity DataKi:  0.158nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470671(CHEMBL358575)
Affinity DataKi:  0.158nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470676(CHEMBL359255)
Affinity DataKi:  0.158nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibitory activity against human NK1 receptor was determinedMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470681(CHEMBL357029)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataKi:  0.251nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470674(CHEMBL342966)
Affinity DataKi:  0.501nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470680(CHEMBL343404)
Affinity DataKi:  0.501nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470673(CHEMBL144793)
Affinity DataKi:  0.794nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470668(CHEMBL147619)
Affinity DataKi:  0.794nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataKi:  0.794nMAssay Description:Binding affinity measured by displacement of tritiated radiolabeled substance P from cloned human NK1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470679(CHEMBL146210)
Affinity DataKi:  2nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50470682(CHEMBL343219)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50346332(2-Oxo-5-phenyl-1,2,3,5-tetrahydro-benzo[e][1,4]dia...)
Affinity DataKi:  10nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214736(CHEMBL304638)
Affinity DataKi:  32nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50213785(CHEMBL91475)
Affinity DataKi:  40nMAssay Description:Binding affinity measured by displacement of tritiated radiolabeled substance P from cloned human NK1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214732(CHEMBL64839)
Affinity DataKi:  40nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400788(CHEMBL2203612)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]dofetilide from human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214733(CHEMBL62597)
Affinity DataKi:  316nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214734(CHEMBL302163)
Affinity DataKi:  631nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214641(CHEMBL291650)
Affinity DataKi:  794nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214735(CHEMBL64698)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50214640(CHEMBL64862)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
Gsk

Curated by ChEMBL
LigandPNGBDBM50213784(CHEMBL91840)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity measured by displacement of tritiated radiolabeled substance P from cloned human NK1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.320nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor stably expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.630nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type A receptor stably expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50189399((S)-N-(3-(4-(2-(4-fluorophenyl)acetamido)piperidin...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of [125I]MIP-1beta binding to CCR5 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400791(CHEMBL2203619)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50189401(CHEMBL214818 | N-((S)-3-(3-(2-methyl-1H-benzo[d]im...)
Affinity DataIC50:  2nMAssay Description:Inhibition of [125I]MIP-1beta binding to CCR5 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400795(CHEMBL2203615)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50189394((S)-N-(3-(4-(3-benzyl-1H-1,2,4-triazol-1-yl)piperi...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [125I]MIP-1beta binding to CCR5 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50189400(CHEMBL213914 | N-[(1S)-3-[2'-(2-methyl-1H-1,3-benz...)
Affinity DataIC50:  6nMAssay Description:Inhibition of [125I]MIP-1beta binding to CCR5 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400794(CHEMBL2203616)
Affinity DataIC50:  6nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400787(CHEMBL2203613)
Affinity DataIC50:  8nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400788(CHEMBL2203612)
Affinity DataIC50:  9nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM50422155(CHEMBL443825)
Affinity DataIC50:  16nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400792(CHEMBL2203618)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50189397((S)-N-(3-(4-(5-benzyl-1,2,4-oxadiazol-3-yl)piperid...)
Affinity DataIC50:  20nMAssay Description:Inhibition of [125I]MIP-1beta binding to CCR5 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400796(CHEMBL2203614)
Affinity DataIC50:  20nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50400790(CHEMBL2203620)
Affinity DataIC50:  21.5nMAssay Description:Displacement of [125I]MIP-1beta from CCR5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM50072427(1-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-2,4-d...)
Affinity DataIC50:  25nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Glaxo Wellcome

Curated by ChEMBL
LigandPNGBDBM50422157(CHEMBL345786)
Affinity DataIC50:  32nMAssay Description:Concentration required to displace [125I]Bolton-Hunter CCK-8 from human Cholecystokinin type B receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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