Affinity DataKi: 0.5nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita Degli Studi Di Milano
Universita Degli Studi Di Milano
Affinity DataKi: 25nM ΔG°: -43.1kJ/mole IC50: 460nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of Cy3B conjugated serotonin analogue binding to human recombinant 5-HT2C receptor expressed in Swiss mouse 3T3 cell membranes after 60 mi...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita Degli Studi Di Milano
Universita Degli Studi Di Milano
Affinity DataKi: 61nM ΔG°: -40.9kJ/mole IC50: 530nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibition of COX2 in mouse J774 cells assessed as inhibition of LPS-induced PGE2 production by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.98nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 4.17nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant HDAC6 using AMC-K(Ac)GL as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 5.01nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 7.08nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 7.08nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of COX2-dependent PGE2 production in LPS-stimulated mouse J774 cells by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 7.59nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 9.5nMAssay Description:Inhibition of COX2 in mouse J774 cells assessed as inhibition of LPS-induced PGE2 production by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant HDAC6 using AMC-K(Ac)GL as substrate by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 11.0nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 12.9nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of COX2 in mouse J774 cells assessed as inhibition of LPS-induced PGE2 production by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of COX2-dependent PGE2 production in LPS-stimulated mouse J774 cells by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 17.0nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 18.2nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 19.9nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of COX2-dependent PGE2 production in LPS-stimulated mouse J774 cells by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of COX2-dependent PGE2 production in LPS-stimulated mouse J774 cells by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 22.9nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 24.0nMAssay Description:Inhibitory activity against dihydrofolate reductase of rat liverMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of COX2-dependent PGE2 production in LPS-stimulated mouse J774 cells by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of COX2-dependent PGE2 production in LPS-stimulated mouse J774 cells by RIAMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of COX-2-mediated PGE2 production in LPS-stimulated mouse J774 cells after 24 hrs by radioimmunoassayMore data for this Ligand-Target Pair