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Found 87 with Last Name = 'bezzine' and Initial = 's'
TargetPurine nucleoside phosphorylase(Toxoplasma gondii)
Cnrs Umr 7175

Curated by ChEMBL
LigandPNGBDBM50200328((4S,8R,9aS)-4-benzyl-8-(benzyloxy)-hexahydro-1H-py...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of Toxoplasma gondii purine nucleoside phosphorylaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human group IIA PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  270nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206913((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50:  280nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206912((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  290nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206905((S)-3-(4-(2-(tetradecyloxy)-3-(trityloxy)propoxy)p...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  470nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50:  550nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  660nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human group X PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human group X PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human group IIA PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of human group IIA PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of human group X PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206913((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human group V PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human group IIA PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206918(1,3-O-di[4-(4,5-dihydro-5-oxo-4H-1,2,4-oxadiazol-3...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206917((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Université

Curated by ChEMBL
LigandPNGBDBM50206912((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206914((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206916((+/-)-2,3-O-di[4-(4,5-dihydro-5-oxo-4H-1,2,4-oxadi...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human group IB PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM23770(3-{[4-(tetradecyloxy)phenyl]methyl}-4,5-dihydro-1,...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  4.57E+3nMAssay Description:Inhibition of human group X PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206913((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human group IIA PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human group X PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206913((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human group X PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Université

Curated by ChEMBL
LigandPNGBDBM50206913((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206920((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of human group IB PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human group IIA PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of human group IB PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Université

Curated by ChEMBL
LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206906((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206910((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of human group IB PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Université

Curated by ChEMBL
LigandPNGBDBM50206908((+/-)-1-O-(4-cyanomethylphenyl)-3-O-[4-(4,5-dihydr...)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of pig group IB PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200327((E)-4-(6-Benzyl-1-methyl-4,7-dioxo-[1,3,5]triazepa...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human group 10 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206911((+/+)-1-O-decyl-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human group IB PLA2 in [3H]oleate-labeled Escherichia coli membrane by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200324((4S,7S)-4,7-dibenzyl-5-methyl-1,3,5-triazepane-2,6...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human group 5 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200325((S)-tert-butyl 2-(6-isopropyl-1-methyl-4,7-dioxo-1...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human group 10 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200326(((S)-7-benzyl-3-tert-butoxycarbonylmethyl-5-methyl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human group 5 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGroup 10 secretory phospholipase A2(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200326(((S)-7-benzyl-3-tert-butoxycarbonylmethyl-5-methyl...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human group 10 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50206924((+/-)-3-O-[4-(4,5-dihydro-5-oxo-1,2,4-4H-oxadiazol...)
Affinity DataIC50:  1.16E+4nMAssay Description:Inhibition of human group IIA PLA2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200327((E)-4-(6-Benzyl-1-methyl-4,7-dioxo-[1,3,5]triazepa...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human group 5 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50200325((S)-tert-butyl 2-(6-isopropyl-1-methyl-4,7-dioxo-1...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human group 5 sPLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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