Affinity DataKi: 0.0100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Prosidion
Curated by ChEMBL
Prosidion
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Prosidion
Curated by ChEMBL
Prosidion
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of Matrix metalloprotease-8More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of Matrix metalloprotease-9More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Matrix metalloprotease-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Prosidion
Curated by ChEMBL
Prosidion
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Prosidion
Curated by ChEMBL
Prosidion
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Prosidion
Curated by ChEMBL
Prosidion
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Erg by patch clamp assayMore data for this Ligand-Target Pair