TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity to GluN2B receptor in human cortexMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]Ro 25-6981 from GluN2B receptor in Sprague-Dawley rat forebrain membranes incubated for 1 hr by topcount micro scintillation coun...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Mus musculus)
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at gardiquimod stimulated TRL7 in mouse whole blood assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Antagonist activity at gardiquimod stimulated TRL7 in human PBMC cells assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at gardiquimod stimulated TRL7 in human whole blood assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 2B(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Bristol-Myers Squibb Research And Development
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Binding affinity to GluN2B receptor in human cortexMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at R848 stimulated TRL8 in human whole blood assessed as inhibition of IL-6 production by ELISA analysisMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Antagonist activity at TLR7 (unknown origin) in PBMC cells assessed as reduction of IL-6 productionMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at TLR8 in human whole blood cells assessed as inhibition of IL-6 production by ELISAMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at TLR7 in human whole blood cells assessed as inhibition of gardiquimod induced IL-6 production by ELISAMore data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at gardiquimod stimulated human TRL7 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincuba...More data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Antagonist activity at R848 stimulated human TRL8 overexpressed in HEK293 cells assessed as inhibition of NF kappa B/Ap-1 activation preincubated wit...More data for this Ligand-Target Pair
TargetToll-like receptor 7(Homo sapiens (Human))
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Biocon Bristol Myers Squibb Research Center (Bbrc)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human TLR7 overexpressed in HEK-Blue cells assessed as inhibition of gardiquimod-induced NFkappaB and AP-1 activation preincub...More data for this Ligand-Target Pair