Compile Data Set for Download or QSAR
Report error Found 114 Enz. Inhib. hit(s) with all data for entry = 1164
TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311486BDBM311486(US10155764, Example 65B | CHEM-US-00192)
Affinity DataIC50: 19nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311498BDBM311498(US10155764, Example 74A | CHEM-US-00210)
Affinity DataIC50: 20nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311480BDBM311480(US10155764, Example 60 | CHEM-US-00186)
Affinity DataIC50: 21nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311495BDBM311495(US10155764, Example 73A | CHEM-US-00207)
Affinity DataIC50: 23nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311483BDBM311483(US10155764, Example 63 | CHEM-US-00189)
Affinity DataIC50: 25nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311512BDBM311512(US10155764, Example 87 | CHEM-US-00232)
Affinity DataIC50: 29nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311511BDBM311511(US10155764, Example 86)
Affinity DataIC50: 30nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311479BDBM311479(US10155764, Example 59 | CHEM-US-00185)
Affinity DataIC50: 33nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311490BDBM311490(US10155764, Example 70A | CHEM-US-00202)
Affinity DataIC50: 36nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311502BDBM311502(US10155764, Example 77)
Affinity DataIC50: 36nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311478BDBM311478(US10155764, Example 58 | CHEM-US-00184)
Affinity DataIC50: 40nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311448BDBM311448(US10155764, Example 34 | CHEM-US-00145)
Affinity DataIC50: 40nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311497BDBM311497(US10155764, Example 74 | CHEM-US-00209)
Affinity DataIC50: 40nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311476BDBM311476(US10155764, Example 56 | CHEM-US-00182)
Affinity DataIC50: 41nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311412BDBM311412(US10155764, Example 8A)
Affinity DataIC50: 42nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311501BDBM311501(US10155764, Example 76)
Affinity DataIC50: 42nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311503BDBM311503(US10155764, Example 78 | CHEM-US-00222)
Affinity DataIC50: 44nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311472BDBM311472(US10155764, Example 54 | US10155764, Example 54A |...)
Affinity DataIC50: 45nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311403BDBM311403(US10155764, Example 1A)
Affinity DataIC50: 45nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311505BDBM311505(US10155764, Example 80 | CHEM-US-00224)
Affinity DataIC50: 46nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311433BDBM311433(US10155764, Example 22A | CHEM-US-00130)
Affinity DataIC50: 47nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311510BDBM311510(US10155764, Example 85 | CHEM-US-00230)
Affinity DataIC50: 50nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311509BDBM311509(US10155764, Example 84 | CHEM-US-00229)
Affinity DataIC50: 56nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311424BDBM311424(US10155764, Example 16A)
Affinity DataIC50: 57nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311507BDBM311507(US10155764, Example 82)
Affinity DataIC50: 59nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311475BDBM311475(US10155764, Example 55)
Affinity DataIC50: 61nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311482BDBM311482(US10155764, Example 62 | CHEM-US-00188)
Affinity DataIC50: 63nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311431BDBM311431(US10155764, Example 21 | CHEM-US-00128)
Affinity DataIC50: 64nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311440BDBM311440(US10155764, Example 28 | CHEM-US-00137)
Affinity DataIC50: 66nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311444BDBM311444(US10155764, Example 32 | US10155764, Example 32A |...)
Affinity DataIC50: 69nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311508BDBM311508(US10155764, Example 83 | CHEM-US-00228)
Affinity DataIC50: 71nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311411BDBM311411(US10155764, Example 7B)
Affinity DataIC50: 72nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311504BDBM311504(US10155764, Example 79 | CHEM-US-00223)
Affinity DataIC50: 73nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311477BDBM311477(US10155764, Example 57 | CHEM-US-00183)
Affinity DataIC50: 75nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311422BDBM311422(US10155764, Example 15A)
Affinity DataIC50: 78nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311513BDBM311513(US10155764, Example 88)
Affinity DataIC50: 80nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311493BDBM311493(US10155764, Example 71B | CHEM-US-00205)
Affinity DataIC50: 83nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311402BDBM311402(US10155764, Example 1)
Affinity DataIC50: 86nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311481BDBM311481(US10155764, Example 61 | CHEM-US-00187)
Affinity DataIC50: 86nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311409BDBM311409(US10155764, Example 6)
Affinity DataIC50: 87nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311455BDBM311455(US10155764, Example 39B | CHEM-US-00152)
Affinity DataIC50: 89nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311506BDBM311506(US10155764, Example 81)
Affinity DataIC50: 98nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311494BDBM311494(US10155764, Example 72 | CHEM-US-00206)
Affinity DataIC50: 99nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311430BDBM311430(US10155764, Example 20)
Affinity DataIC50: 110nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311438BDBM311438(US10155764, Example 26 | CHEM-US-00135)
Affinity DataIC50: 110nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311437BDBM311437(US10155764, Example 25 | CHEM-US-00134)
Affinity DataIC50: 110nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311472BDBM311472(US10155764, Example 54 | US10155764, Example 54A |...)
Affinity DataIC50: 110nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311439BDBM311439(US10155764, Example 27 | CHEM-US-00136)
Affinity DataIC50: 120nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311500BDBM311500(US10155764, Example 75 | CHEM-US-00212)
Affinity DataIC50: 130nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetHistone acetyltransferase KAT2B [719-832](Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 311451BDBM311451(US10155764, Example 37 | CHEM-US-00148)
Affinity DataIC50: 130nMAssay Description:His/Flag epitope tagged PCAF719-832 bromodomain was cloned, expressed and purified to homogeneity in-house. PCAF bromodomain binding and inhibition o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

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