Compile Data Set for Download or QSAR
maximum 50k data
Found 69 Enz. Inhib. hit(s) with all data for entry = 10304
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM525977(3-(5-(((1S,2S)-2- hydroxycyclohexyl)amino)-1- oxoi...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM525977(3-(5-(((1S,2S)-2- hydroxycyclohexyl)amino)-1- oxoi...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM525983(3-(5-(methyl((1R,2R)-2- (methylamino)cyclohexyl)am...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM525983(3-(5-(methyl((1R,2R)-2- (methylamino)cyclohexyl)am...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM525983(3-(5-(methyl((1R,2R)-2- (methylamino)cyclohexyl)am...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526006(3-(5-(((1S,2S)-2- (benzylamino)cyclohexyl)amino)-1...)
Affinity DataEC50:  29nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526006(3-(5-(((1S,2S)-2- (benzylamino)cyclohexyl)amino)-1...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526006(3-(5-(((1S,2S)-2- (benzylamino)cyclohexyl)amino)-1...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526020(3-(5-(((1S,2S)-2-(benzyloxy) cyclohexyl)amino)- 1-...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526078(US11185537, Compound I-8 | US11185537, Compound I-...)
Affinity DataEC50:  113nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526078(US11185537, Compound I-8 | US11185537, Compound I-...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526078(US11185537, Compound I-8 | US11185537, Compound I-...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526123(3-(5-(((1S,2S)-2- (benzyl(methyl)amino)cyclohexyl)...)
Affinity DataEC50:  43nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526123(3-(5-(((1S,2S)-2- (benzyl(methyl)amino)cyclohexyl)...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526131(3-(5-(((1S,2S)-2- aminocyclohexyl)amino)-1- oxoiso...)
Affinity DataEC50:  183nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526131(3-(5-(((1S,2S)-2- aminocyclohexyl)amino)-1- oxoiso...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526078(US11185537, Compound I-8 | US11185537, Compound I-...)
Affinity DataEC50:  103nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526078(US11185537, Compound I-8 | US11185537, Compound I-...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526078(US11185537, Compound I-8 | US11185537, Compound I-...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526253(3-(5-(((1S,2S)-2-(ethylamino) cyclohexyl)amino)- 1...)
Affinity DataEC50:  1.67E+3nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526253(3-(5-(((1S,2S)-2-(ethylamino) cyclohexyl)amino)- 1...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526265(3-(5-(((1S,2S)-2- (isopropylamino)cyclohexyl)amino...)
Affinity DataEC50:  100nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526265(3-(5-(((1S,2S)-2- (isopropylamino)cyclohexyl)amino...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526265(3-(5-(((1S,2S)-2- (isopropylamino)cyclohexyl)amino...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526266(3-(5-(ethyl((1S,2S)-2- (ethylamino)cyclohexyl) ami...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526267(3-(5-(((1S,2S)-2- ((cyclohexylmethyl)amino) cycloh...)
Affinity DataEC50:  36nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526267(3-(5-(((1S,2S)-2- ((cyclohexylmethyl)amino) cycloh...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526268(3-(1-oxo-5-(((1S,2S)-2-(piperidin-1- yl)cyclopenty...)
Affinity DataEC50:  730nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526268(3-(1-oxo-5-(((1S,2S)-2-(piperidin-1- yl)cyclopenty...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526269(3-(5-(((1S,2S)-2- (isobutylamino)cyclohexyl)amino)...)
Affinity DataEC50:  940nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526269(3-(5-(((1S,2S)-2- (isobutylamino)cyclohexyl)amino)...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526270(US11185537, Compound Mix)
Affinity DataEC50:  230nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526270(US11185537, Compound Mix)
Affinity DataEC50:  120nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526270(US11185537, Compound Mix)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526271(2-(2,6-dioxopiperidin-3- yl)-5-(methyl((1S,2S)-2- ...)
Affinity DataEC50:  24nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526271(2-(2,6-dioxopiperidin-3- yl)-5-(methyl((1S,2S)-2- ...)
Affinity DataEC50:  290nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526271(2-(2,6-dioxopiperidin-3- yl)-5-(methyl((1S,2S)-2- ...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526272(5-(((1S,2S)-2-aminocyclohexyl) (methyl)amino)- 2-(...)
Affinity DataEC50:  150nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526272(5-(((1S,2S)-2-aminocyclohexyl) (methyl)amino)- 2-(...)
Affinity DataEC50:  5.20E+3nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526272(5-(((1S,2S)-2-aminocyclohexyl) (methyl)amino)- 2-(...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526273(2-(2,6-dioxopiperidin-3-yl)-5-(((1S,2S)-2- (ethyla...)
Affinity DataEC50:  49nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526273(2-(2,6-dioxopiperidin-3-yl)-5-(((1S,2S)-2- (ethyla...)
Affinity DataEC50:  51nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526273(2-(2,6-dioxopiperidin-3-yl)-5-(((1S,2S)-2- (ethyla...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526274(2-(2,6-dioxopiperidin-3- yl)-5-(methyl((1S,2S)-2- ...)
Affinity DataEC50:  230nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526274(2-(2,6-dioxopiperidin-3- yl)-5-(methyl((1S,2S)-2- ...)
Affinity DataEC50: >3.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526274(2-(2,6-dioxopiperidin-3- yl)-5-(methyl((1S,2S)-2- ...)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526270(US11185537, Compound Mix)
Affinity DataEC50:  670nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDNA-binding protein Ikaros(Homo sapiens)
Novartis

US Patent
LigandPNGBDBM526270(US11185537, Compound Mix)
Affinity DataEC50:  630nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM526270(US11185537, Compound Mix)
Affinity DataEC50: >5.00E+4nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetZinc finger protein Helios(Human)
Novartis

US Patent
LigandPNGBDBM526275(5-(((1S,2S)-2- (benzylamino)cyclohexyl) (methyl)am...)
Affinity DataEC50:  450nMAssay Description:The Prolabel system from DiscoverX was used to develop high-throughput and quantitative assays to measure changes in IKZF1, IKZF2, and GSPT1 protein ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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