Affinity DataKi: 390nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMpH: 7.0Assay Description:Inhibition assay against beta lactamase enzymes.More data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMpH: 7.0Assay Description:Inhibition assay against beta lactamase enzymes.More data for this Ligand-Target Pair
Affinity DataKi: 6.50E+3nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 1.38E+4nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 1.62E+5nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+6nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+6nMpH: 7.0Assay Description:Enzyme inhibition assay using AmpC or TEM-1 from escherichia coli.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against serine beta-lactamase, PC1 (class A) derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 25.1nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:The compound was evaluated for inhibition against Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 46.4nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 71.8nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against Penicillinase from Staphylococcus aureus TH-14 using piperacillin (40 uM) as a substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of class A beta-lactamase derived from Staphylococcus aureus strain PC1More data for this Ligand-Target Pair
Affinity DataIC50: 104nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 125nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of Staphylococcus aureus Russell beta-lactamase assessed as inhibition of nitrocefin hydrolysis pre-incubated for 5 mins by microtiter pla...More data for this Ligand-Target Pair
Affinity DataIC50: 166nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 181nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 196nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of class A beta-lactamase derived from Staphylococcus aureus strain PC1More data for this Ligand-Target Pair
Affinity DataIC50: 233nMAssay Description:Inhibitory activity against serine beta-lactamase, PC1 (class A) derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Staphylococcus aureus PCIMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibitory activity against Penicillinase from Staphylococcus aureus TH-14 using piperacillin (40 uM) as a substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 289nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:The compound was evaluated for inhibition against Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 297nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of class A beta-lactamase derived from Staphylococcus aureus strain PC1More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibitory activity against serine Beta-lactamase TEM derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 342nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibitory activity against serine Beta-lactamase derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 419nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 461nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Compound was tested for inhibition of Beta-lactamase from Staphylococcus aureus PCIMore data for this Ligand-Target Pair
Affinity DataIC50: 509nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibitory activity against serine beta-lactamase, PC1 (class A) derived from Staphylococcus aureusMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair