Compile Data Set for Download or QSAR
Report error Found 60 for UniProtKB: P48056
LigandChemical structure of BindingDB Monomer ID 50473314BDBM50473314(CHEMBL553068)
Affinity DataIC50: 51nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50081891BDBM50081891(1-[2-(3,3-Diphenyl-propoxy)-ethyl]-piperidine-3-ca...)
Affinity DataIC50: 55nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473316BDBM50473316(CHEMBL545694)
Affinity DataIC50: 68nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473312BDBM50473312(CHEMBL543108)
Affinity DataIC50: 74nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50080346BDBM50080346((R)-1-(2-Benzhydrylideneaminooxy-ethyl)-piperidine...)
Affinity DataIC50: 82nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50081888BDBM50081888((R)-1-[2-(2-Diphenylamino-ethoxy)-ethyl]-piperidin...)
Affinity DataIC50: 90nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473321BDBM50473321(CHEMBL563076)
Affinity DataIC50: 105nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50437146BDBM50437146(CHEMBL1189315)
Affinity DataIC50: 184nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473306BDBM50473306(CHEMBL556178)
Affinity DataIC50: 248nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473319BDBM50473319(CHEMBL555856)
Affinity DataIC50: 265nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50437144BDBM50437144(CHEMBL1190271)
Affinity DataIC50: 308nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50003634BDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50: 330nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473315BDBM50473315(CHEMBL541561)
Affinity DataIC50: 460nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473313BDBM50473313(CHEMBL545690)
Affinity DataIC50: 561nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473311BDBM50473311(CHEMBL543342)
Affinity DataIC50: 644nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50437145BDBM50437145(CHEMBL1196076)
Affinity DataIC50: 647nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473317BDBM50473317(CHEMBL553053)
Affinity DataIC50: 696nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473320BDBM50473320(CHEMBL545452)
Affinity DataIC50: 770nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473309BDBM50473309(CHEMBL552675)
Affinity DataIC50: 851nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473302BDBM50473302(CHEMBL555631)
Affinity DataIC50: 1.16E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473303BDBM50473303(CHEMBL542641)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50003653BDBM50003653(CHEMBL542610 | 1-(2-Benzhydryloxy-ethyl)-piperidin...)
Affinity DataIC50: 1.37E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24183BDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50226144BDBM50226144(CHEBI:64307 | 2,4-Diamino-Butyric Acid | DL-2,4-di...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24183BDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50078167BDBM50078167(CHEMBL69064)
Affinity DataIC50: 2.02E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473308BDBM50473308(CHEMBL541821)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473305BDBM50473305(CHEMBL71789)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 24183BDBM24183(4-amino-n-[2,3-3H]butyric acid | cid_119 | Gamma-A...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50473318BDBM50473318(CHEMBL539773)
Affinity DataIC50: 5.51E+3nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50003624BDBM50003624(Nipecotic | Piperidine-3-carboxylic acid(nipecotic...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223874BDBM50223874(CHEMBL277372)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473310BDBM50473310(CHEMBL303402)
Affinity DataIC50: 1.36E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473307BDBM50473307(CHEMBL545692)
Affinity DataIC50: 1.46E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50021186BDBM50021186(CHEMBL296263 | S(+)-4-amino-3-hydroxybutanoic acid...)
Affinity DataIC50: 2.90E+4nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50473304BDBM50473304(CHEMBL541556)
Affinity DataIC50: 4.00E+4nMAssay Description:In vitro inhibition of [3H]GABA uptake in rat synaptosomes was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50021187BDBM50021187(R(-)-4-amino-3-hydroxybutanoic acid | CHEMBL290216...)
Affinity DataIC50: 6.70E+4nMAssay Description:In vivo inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50021189BDBM50021189(CHEMBL40804 | 5-Aminomethyl-4,5-dihydro-isoxazol-3...)
Affinity DataIC50: 7.00E+4nMAssay Description:In vivo inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226141BDBM50226141(CHEMBL309688)
Affinity DataIC50: 1.30E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50225363BDBM50225363(CHEMBL40363)
Affinity DataIC50: 1.30E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50021262BDBM50021262(4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-5-ium-3-...)
Affinity DataIC50: 1.60E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226145BDBM50226145(CHEMBL150830)
Affinity DataIC50: 1.60E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223872BDBM50223872(CHEMBL15851)
Affinity DataIC50: 1.73E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223876BDBM50223876(CHEMBL16226)
Affinity DataIC50: 2.03E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50224812BDBM50224812(CHEBI:35010 | CHEMBL170539)
Affinity DataIC50: 2.20E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50224810BDBM50224810(CHEMBL171241)
Affinity DataIC50: 2.30E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223871BDBM50223871(CHEMBL429974)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50223877BDBM50223877(CHEMBL16132)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50000106BDBM50000106(Piperidine-4-carboxylic acid | Piperidine-4-carbox...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50226142BDBM50226142(CHEMBL292757)
Affinity DataIC50: 3.00E+5nMAssay Description:In vitro inhibition of rat neuronal (synaptosomal) GABA uptake.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2018
Entry Details Article
PubMed
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