9452 SMILES Strings for Replicase polyprotein 1ab

Compound Name
SMILES String
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C |r|
C[C@H](OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CN(C)c1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1cccs1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
CC(C)C(NC(=O)c1cc(C)[o+][n-]1)C(=O)NC(Cc1ccccc1)C(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O
CC(C)[C@H](NC(=O)c1cccs1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
CC(C)[C@H](NC(=O)c1cc(C)on1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C(C)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C(C)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
O[C@@H](CC(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O |r|
c1cc(c(cc1[N+](=O)[O-])Cl)NC(=O)c2cc(ccc2O)Cl
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccc(F)cc1 |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)Cc1ccc(F)cc1 |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccccc1 |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)Cc1ccccc1 |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccc(F)cc1 |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)Cc1ccc(F)cc1 |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccccc1 |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)Cc1ccccc1 |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccc(cc1)-c1ccccc1 |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccc(cc1)N(=O)=O |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccc(cc1)N(C)C |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccc(OC)cc1OC |r|
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccc2OCOc2c1 |r|
Clc1cc(Cl)cc(NC(=O)CSc2nccc(n2)-c2csc(n2)-c2ccccc2)c1
Cn1nc(cc1C(F)(F)F)-c1ccc(s1)-c1ccnc(SCC(=O)Nc2ccc(Cl)cc2)n1
CSc1sc(c(C)c1-c1ccnc(SCC(=O)Nc2ccc(Cl)cc2)n1)-c1nc(C)cs1
CSc1sc(c(C)c1-c1ccnc(SCC(=O)Nc2ccccc2Cl)n1)-c1nc(C)cs1
Cc1nc(cs1)-c1nc(cs1)-c1ccnc(SCC(=O)Nc2ccc(Cl)cc2)n1
Clc1ccc(NC(=O)CSc2nccc(n2)-c2cc(no2)-c2ccccc2)cc1
FC(F)(F)c1ccc(NC(=O)CSc2nccc(n2)-c2cc(no2)-c2ccc(Cl)cc2Cl)cc1
Clc1ccc(NC(=O)CSc2nccc(n2)-c2cc(no2)-c2ccccc2Cl)cc1
CCCc1cc(=O)[nH]c(SCC(=O)Nc2ccc(Cl)cc2)n1
COc1cccc(c1)-c1nc(SCC(=O)Nc2ccc(cc2)S(N)(=O)=O)[nH]c(=O)c1C#N
CC(C)c1ccc(NC(=O)CSc2nccc(n2)-c2cccs2)cc1
COc1ccc(NC(=O)CSc2nc(cc(=O)[nH]2)-c2ccccc2)cc1OC
COc1cccc(c1)-c1nc(SCC(=O)Nc2ccc(cc2)C(C)=O)[nH]c(=O)c1C#N
CCC(Sc1nc(-c2cccc(OC)c2)c(C#N)c(=O)[nH]1)C(=O)Nc1cccc(c1)C(C)=O
Cc1cc(=O)[nH]c(SCC(=O)Nc2cc(Cl)ccc2Oc2ccccc2)n1
Cc1cc(=O)[nH]c(SCC(=O)Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
CC(C)c1ccc(NC(=O)CSc2nccc(n2)-c2csc(COc3ccccc3Cl)n2)cc1
COC(OC)c1cc(=O)[nH]c(SCC(=O)Nc2ccc(cc2)C(F)(F)F)n1
CCCCc1ccc(NC(=O)CSc2nc(C3CCCCC3)c(C#N)c(=O)[nH]2)c(C)c1
FC(F)(F)c1cccc(NC(=O)CSc2nc(-c3ccccc3)c(C#N)c(=O)[nH]2)c1
CCOC(=O)c1cnc(SCC(=O)Nc2ccc(cc2)[N+]([O-])=O)nc1N
CCOc1ccc(cc1)-n1c(O)cc(Sc2nc(C)cc(C)n2)c1O
COc1cccc(c1)-c1nc(SCC(=O)Nc2ccc(cc2)[N+]([O-])=O)[nH]c(=O)c1C#N
CC(Sc1nc(-c2ccccc2)c(C#N)c(=O)[nH]1)C(=O)Nc1ccc(Cl)cc1
CC(C)(C)c1ccc(NC(=O)CSc2nc(C3CCCCC3)c(C#N)c(=O)[nH]2)cc1
COc1ccc(cc1)-c1ccnc(SCC(=O)Nc2ccc(cc2)C(C)C)n1
Cc1cc(nc(SCC(=O)Nc2ccc(Cl)cc2F)n1)C(F)(F)F
Cc1nc(SCC(=O)Nc2ccc(cc2)[N+]([O-])=O)[n-]c(=[OH+])c1C
Cc1cc(c(cc1Cl)Cl)S(=O)(=O)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-]
Cl\[#6](Cl)=[#6](\Cl)-[#6](=O)-[#8]-c1ccc(cc1)S(=O)(=O)c1ccc(-[#8]-[#6](=O)-[#6](\Cl)=[#6](/Cl)Cl)cc1
Nc1ncc(c(N)n1)S(=O)(=O)c1ccc(Cl)cc1
[O-][N+](=O)c1cc(ccc1S(=O)(=O)c1ccc(Cl)cc1)C(F)(F)F
Cc1nc(c(C#N)c(C)c1[N+]([O-])=O)S(=O)(=O)c1ccccc1
Cc1ccc(cc1)S(=O)(=O)c1nc(C)c(c(C)c1C#N)[N+]([O-])=O
[O-][N+](=O)c1ccc([n+]([O-])c1)S(=O)(=O)c1ccc(Cl)cc1
CCOC(=O)C(C=Nc1ccc(cc1)S(=O)(=O)c1ccc(cc1)N=CC(C#N)C(=O)OCC)C#N |w:6.5,23.24|
OC(=O)c1ccc(cc1)S(=O)(=O)c1cc(Br)c(O)c(Br)c1
CC(=O)c1ccccc1S(=O)(=O)c1ccccc1C(O)=O
[O-][N+](=O)c1ccc(cc1)S(=O)(=O)c1ccc(cc1)[N+]([O-])=O
CCOC(=O)C(C=Nc1ccc(cc1)S(=O)(=O)c1ccc(cc1)N=CC(C(=O)OCC)C(=O)OCC)C(=O)OCC |w:7.7,23.24|
FC(F)(F)c1nnc(SC(=O)c2ccc(o2)C#Cc2ccccc2)[nH]1
Cc1[n-][o+]c(NC(=O)c2ccc(s2)-c2cc(nn2C)C(F)(F)F)c1[N+]([O-])=O
Cc1oc(cc1-c1cc(NS(=O)(=O)c2cccs2)[nH]n1)C(C)(C)C
CSc1n[nH]c(NC(=O)c2cccs2)c1S(=O)(=O)c1ccc(Cl)cc1
CC1(C)Cc2c(sc(NCc3ccco3)c2C(=O)C1)C#N
CSc1nn(c(-c2cccs2)c1C#N)-c1c(c(C)nn1C)[N+]([O-])=O |(4.14,6.57,;2.6,6.57,;1.69,5.32,;2.17,3.86,;.92,2.95,;-.32,3.86,;-1.86,3.86,;-2.95,2.76,;-4.32,3.46,;-4.09,4.98,;-2.57,5.23,;.15,5.32,;-.75,6.57,;-1.52,7.9,;.92,1.41,;-.11,.27,;.65,-1.07,;.02,-2.47,;2.16,-.75,;2.33,.78,;3.66,1.54,;-1.64,.44,;-2.56,-.8,;-2.26,1.92,)|
Clc1ccc(s1)-c1csc(CS(=O)(=O)c2cccs2)n1
Cc1nn(C)c(NCc2ccc(s2)-c2cccs2)c1[N+]([O-])=O
O=C(CC1=NCCS1)c1nccs1 |t:3|
O=C(CSc1nc(nc2ccccc12)C1CCCCC1)NCc1ccco1
Cc1ccccc1CCN(Cc1cc2cc(C)c(C)cc2[nH]c1=O)C(=O)NCc1ccccc1
Nc1ccccc1C(=O)On1nnc2ccccc12
CN(C)c1ccc(cc1)C(=O)On1nnc2ccccc12
CNc1ccc(cc1)C(=O)On1nnc2ccccc12
CCN(CC)c1ccc(cc1)C(=O)On1nnc2ccccc12
O=C(On1nnc2ccccc12)c1ccc2nc[nH]c2c1
c1ccc2c(c1)nnn2OC(=O)c3ccc4c(c3)cc[nH]4
O=C(On1nnc2ccccc12)c1cc2ccccc2[nH]1
Fc1ccc2[nH]c(cc2c1)C(=O)On1nnc2ccccc12
O=C(Cn1nnc2ccccc12)c1ccc(cc1)N(=O)=O
CCN(CC)c1ccc(cc1)C(=O)Cn1nnc2ccccc12
Nc1ccc(cc1)C(=O)Cn1nnc2ccccc12
Nc1ccc(cc1)C(O)Cn1nnc2ccccc12
CNc1ccc(cc1)C(=O)Cn1nnc2ccccc12
CN(C)c1ccc(cc1)C(=O)Cn1nnc2ccccc12
CNc1ccc(cc1)C(O)Cn1nnc2ccccc12
CN(C)c1ccc(cc1)C(O)Cn1nnc2ccccc12
CC(C)C[C@H](NC(=O)[C@H](CNC(=O)C(C)(C)C)NC(=O)OCc1ccccc1)C(=O)NC(C[C@@H]1CCNC1=O)=CCC(C)=O |r,w:39.41|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)=CCC(=O)C1CC1 |r,w:38.40|
Cc1cc(no1)C(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=CC(=O)OCc3ccccc3
CCN(CC)C(=S)SSC(=S)N(CC)CC
CCCCCCNC(=O)n1cc(F)c(=O)[nH]c1=O
O=c1n([se]c2ccccc12)-c1ccccc1
[#6]\[#6](-[#6])=[#6]\[#6]-[#6](-[#8])-[#6]-1=[#6]-[#6](=O)-c2c(-[#8])ccc(-[#8])c2-[#6]-1=O |t:7|
O=c1sn(-c2cccc3ccccc23)c(=O)n1Cc1ccccc1
CCC(C)SSc1ncc[nH]1
CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)N[C@H](CC1CCNC1=O)C(O)S([O-])(=O)=O
CC(C)C[C@@H](NC(=O)OC1CCCCC1)C(=O)N[C@H](CC1CCNC1=O)C=O
CCCC1CCC(CC1)OC(=O)N[C@H](CC(C)C)C(=O)N[C@H](CC1CCNC1=O)C(O)S([O-])(=O)=O |wD:21.21,13.13,(-9.14,7.59,;-8.23,6.35,;-6.7,6.51,;-5.8,5.26,;-4.26,5.42,;-3.36,4.18,;-3.98,2.77,;-5.52,2.61,;-6.42,3.86,;-3.08,1.52,;-1.55,1.69,;-.92,3.09,;-.64,.44,;.89,.6,;1.52,2.01,;3.05,2.17,;3.67,3.58,;3.95,.92,;1.79,-.65,;1.17,-2.05,;3.33,-.48,;4.23,-1.73,;5.76,-1.57,;6.67,-2.82,;6.19,-4.28,;7.44,-5.19,;8.68,-4.28,;8.21,-2.82,;9.11,-1.57,;3.6,-3.14,;2.07,-3.3,;4.51,-4.38,;5.41,-5.63,;5.76,-3.48,;3.26,-5.29,)|
CCCC1CCC(CC1)OC(=O)N[C@H](CC(C)C)C(=O)N[C@H](CC1CCNC1=O)C=O |wD:21.21,13.13,(-9.14,7.59,;-8.23,6.35,;-6.7,6.51,;-5.8,5.26,;-4.26,5.42,;-3.36,4.18,;-3.98,2.77,;-5.52,2.61,;-6.42,3.86,;-3.08,1.52,;-1.55,1.69,;-.92,3.09,;-.64,.44,;.89,.6,;1.52,2.01,;3.05,2.17,;3.67,3.58,;3.95,.92,;1.79,-.65,;1.17,-2.05,;3.33,-.48,;4.23,-1.73,;5.76,-1.57,;6.67,-2.82,;6.19,-4.28,;7.44,-5.19,;8.68,-4.28,;8.21,-2.82,;9.11,-1.57,;3.6,-3.14,;2.07,-3.3,)|
CCCCC1CCC(CC1)OC(=O)N[C@H](CC(C)C)C(=O)N[C@H](CC1CCNC1=O)C(O)S([O-])(=O)=O |wD:22.22,14.14,(-10.67,7.43,;-9.14,7.59,;-8.23,6.35,;-6.7,6.51,;-5.8,5.26,;-4.26,5.42,;-3.36,4.18,;-3.98,2.77,;-5.52,2.61,;-6.42,3.86,;-3.08,1.52,;-1.55,1.69,;-.92,3.09,;-.64,.44,;.89,.6,;1.52,2.01,;3.05,2.17,;3.67,3.58,;3.95,.92,;1.79,-.65,;1.17,-2.05,;3.33,-.48,;4.23,-1.73,;5.76,-1.57,;6.67,-2.82,;6.19,-4.28,;7.44,-5.19,;8.68,-4.28,;8.21,-2.82,;9.11,-1.57,;3.6,-3.14,;2.07,-3.3,;4.51,-4.38,;5.41,-5.63,;5.76,-3.48,;3.26,-5.29,)|
CCCCC1CCC(CC1)OC(=O)N[C@H](CC(C)C)C(=O)N[C@H](CC1CCNC1=O)C=O |wD:22.22,14.14,(-10.67,7.43,;-9.14,7.59,;-8.23,6.35,;-6.7,6.51,;-5.8,5.26,;-4.26,5.42,;-3.36,4.18,;-3.98,2.77,;-5.52,2.61,;-6.42,3.86,;-3.08,1.52,;-1.55,1.69,;-.92,3.09,;-.64,.44,;.89,.6,;1.52,2.01,;3.05,2.17,;3.67,3.58,;3.95,.92,;1.79,-.65,;1.17,-2.05,;3.33,-.48,;4.23,-1.73,;5.76,-1.57,;6.67,-2.82,;6.19,-4.28,;7.44,-5.19,;8.68,-4.28,;8.21,-2.82,;9.11,-1.57,;3.6,-3.14,;2.07,-3.3,)|
CC(C)C[C@@H](NC(=O)OC1CCC(F)(F)CC1)C(=O)N[C@H](CC1CCNC1=O)C(O)S([O-])(=O)=O
CC(C)C[C@@H](NC(=O)OC1CCC(F)(F)CC1)C(=O)N[C@H](CC1CCNC1=O)C=O
CC(C)C[C@@H](NC(=O)OCC1CCC(F)(F)CC1)C(=O)N[C@H](CC1CCNC1=O)C(O)S([O-])(=O)=O
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O
Oc1ccccc1-n1[se]c2ccccc2c1=O
COc1ccccc1-n1[se]c2ccccc2c1=O
Oc1ccccc1NC(=O)c1ccccc1[Se][Se]c1ccccc1C(=O)Nc1ccccc1O
COc1ccccc1NC(=O)c1ccccc1[Se][Se]c1ccccc1C(=O)Nc1ccccc1OC
c1ccc2c(c1)cc([nH]2)C(=O)N[C@@H](CC3CCCCC3)C(=O)N[C@@H](C[C@@H]4CCNC4=O)C=O
c1ccc2c(c1)cc([nH]2)C(=O)N[C@@H](Cc3cccc(c3)F)C(=O)N[C@@H](C[C@@H]4CCNC4=O)C=O
CC(NC(=O)c1ccccc1C)c1ccc2ccccc2c1
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1cc(NC(C)=O)ccc1C)c1cccc2ccccc12 |r|
COc1ccc(CNC(=O)C2CCN(Cc3cccc4ccccc34)CC2)cc1
COc1cc(CNC(=O)C2CCN(Cc3ccccc3)CC2)cc(OC)c1OC
Cn1nc(nc2c1nc(=O)n(C)c2=O)-c1ccc(cc1)C(F)(F)F
CC(CNC(=O)CCC1(C)C(CC(N)=O)C2[N-]C1=C(C)C1=NC(=CC3=NC(=C(C)C4=NC2(C)C(C)(CC(N)=O)C4CCC(N)=O)C(C)(CC(N)=O)C3CCC(N)=O)C(C)(C)C1CCC(N)=O)OP([O-])(=O)OC1C(CO)OC(C1O)n1cnc2cc(C)c(C)cc12 |w:23.24,18.19,27.28,t:21,25,30|
Cc1ccc(cc1NC(=O)c1cccc(NC(=O)Nc2cccc(c2)C(=O)Nc2cc(ccc2C)C(=O)Nc2ccc(c3cc(cc(c23)S([O-])(=O)=O)S([O-])(=O)=O)S([O-])(=O)=O)c1)C(=O)Nc1ccc(c2cc(cc(c12)S([O-])(=O)=O)S([O-])(=O)=O)S([O-])(=O)=O
COC(=O)CC[C@H](NC(=O)[C@H](CC(=O)OC)NC(=O)OCc1ccccc1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(=O)OC)C(=O)CF
NS(=O)(=O)c1cccc2C(=O)c3c(O)cccc3C(=O)c12
CC(NC(=O)C(Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)CF
c1cc2c(nc1)C(=O)C(=C(C2=O)Cl)NCCN3CCOCC3
CC1(C)OC2=C(C(NCc3ccccc3)C1O)C(=O)c1ccccc1C2=O |c:4|
O=C1c2ccccc2-[n+]2ccc3c([nH]c4ccccc34)c12
CCCC(NC(=O)C(CC(C)C)NC(=O)C(CC(C)C)NC(=O)OCc1ccccc1)C=O
CC1(C)CCC2=C(O1)c1ccccc1C(=O)C2=O |c:5|
Cc1n(c2c([n+]1Cc3cnccn3)C(=O)c4ccccc4C2=O)CCOC
OCCSC1=C(SCCO)C(=O)c2ccccc2C1=O |c:4|
CC(CNC(=O)CCC1(C)C(CC(N)=O)C2N=C1C(C)=C1N=C(C=C3N=C(C(C)=C4[N-]C2(C)C(C)(CC(N)=O)C4CCC(N)=O)C(C)(CC(N)=O)C3CCC(N)=O)C(C)(C)C1CCC(N)=O)OP([O-])(=O)OC1C(CO)OC(C1O)n1cnc2cc(C)c(C)cc12 |w:23.23,18.19,27.28,c:16,t:22,26|
OC(=O)c1ccc(cc1)N1C(=O)C(=Cc2ccc(o2)-c2ccc(cc2)[N+]([O-])=O)C=C1c1ccccc1 |w:13.14,c:31|
Brc1c(Br)c(Br)c2n[nH]nc2c1Br
Cc1cc(ccc1OCC(=O)O)SCc2c(nc(s2)c3ccc(c(c3)F)C(F)(F)F)C
CCCCCCCCCCCCCCCCC(C(O)=O)C(O)(CC(O)=O)C(O)=O
CNC(CC(C)C)C(=O)NC1C(O)c2ccc(Oc3cc4cc(Oc5ccc(cc5Cl)C(OC5CC(C)(N)C(O)C(C)O5)C5NC(=O)C(NC(=O)C4NC(=O)C(CC(N)=O)NC1=O)c1ccc(O)c(c1)-c1c(O)cc(O)cc1C(NC5=O)C(O)=O)c3OC1OC(CO)C(O)C(O)C1OC1CC(C)(NCc3ccc(cc3)-c3ccc(Cl)cc3)C(O)C(C)O1)c(Cl)c2
COc1ccc2cc(ccc2c1)-c1cc(nn1C(C)c1ccc(cc1)C(=O)NCCC(O)=O)-c1cc(Cl)cc(Cl)c1
Cc1[nH]c(C=C2C(=O)Nc3cc(ccc23)-c2ccccc2)c(C)c1CCC(O)=O |w:4.3|
c1c(cc(c(c1O)O)O)C(=O)OC[C@H]2[C@H]([C@@H]([C@@H]([C@@H](O2)OC(=O)c3cc(c(c(c3)O)O)O)OC(=O)c4cc(c(c(c4)O)O)O)OC(=O)c5cc(c(c(c5)O)O)O)OC(=O)c6cc(c(c(c6)O)O)O
FC(F)(F)c1cc(NC(=O)c2cnc(Cl)nc2C(F)(F)F)cc(c1)C(F)(F)F
CCCCCCCCCCCCCCCc1cccc(O)c1C(O)=O
Cc1cc(OC(CCC(F)(F)F)c2ccc(cc2)C(=O)NCCC(O)=O)cc(C)c1-c1ccc(cc1)C(C)(C)C
Cc1[nH]n(-c2ccc(C)c(C)c2)c(=O)c1N=Nc1cccc(-c2cccc(c2)C(O)=O)c1O |w:16.18|
c1ccc(cc1)C(C[N@](CCCOc2cccc(c2)CC(=O)O)Cc3cccc(c3Cl)C(F)(F)F)c4ccccc4
Oc1c(Br)cc(C=C2C(=O)Nc3ccc(I)cc23)cc1Br
c1c(c(c(c(c1Cl)Cl)Cc2c(c(cc(c2Cl)Cl)Cl)O)O)Cl
CC(C)c1ccc2c(c1)c(c(n2Cc3ccc(cc3)Cl)CC(C)(C)C(=O)O)SC(C)(C)C
CC#CC(CC([O-])=O)c1ccc(OCc2cccc(c2)-c2ccc(cc2)C(F)(F)F)cc1
CCCCCCCc1ccc(CCc2cccc(O)c2C(O)=O)cc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1cccc(F)c1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NCc1cccnc1)c1cccc(F)c1)C(=O)Cn1nnc2ccccc12
COc1ccc(cc1)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C(C)C)cc1)C(=O)NCc1ccccc1
COc1cccc(c1)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C(C)C)cc1)C(=O)NCc1ccccc1
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1cccnc1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1ccc(OCCCN(C)C)cc1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1ccc(Cl)c(F)c1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1cccc(F)c1)C(=O)Cn1cnc2ccccc12
CC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)c1ccsc1
CC(C)(C)NC(=O)C(N(C(=O)Cn1cnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)c1ccsc1
CC(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)c1ccsc1
CC(C)CNC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)c1ccsc1
CC(C)(C)CNC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)c1ccsc1
O=C(Cn1nnc2ccccc12)N(C(C(=O)NC1CC1)c1ccsc1)c1ccc(NC(=O)C2CC2)cc1
O=C(Cn1nnc2ccccc12)N(C(C(=O)NC1CCCC1)c1ccsc1)c1ccc(NC(=O)C2CC2)cc1
O=C(Cn1nnc2ccccc12)N(C(C(=O)NCc1cccnc1)c1ccsc1)c1ccc(NC(=O)C2CC2)cc1
O=C(Cn1nnc2ccccc12)N(C(C(=O)NCc1ccccc1)c1ccsc1)c1ccc(NC(=O)C2CC2)cc1
CC(C)(C)OC(=O)CNC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)c1ccsc1
O=C(Cn1nnc2ccccc12)N(C(C(=O)NC1CCCCC1)c1ccsc1)c1ccc(NC(=O)C2CC2)cc1
CC(C)(C)NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)Cc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1cccnc1)C(=O)c1c[nH]cn1
CC(C)(C)NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C1CC1)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C1CCC1)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C1CCCC1)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C1CCCCC1)c1cccnc1
CC(C)CNC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)CNC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CC1)c1cccnc1)C(=O)c1c[nH]cn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCC1)c1cccnc1)C(=O)c1c[nH]cn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1cccnc1)C(=O)c1c[nH]cn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)c1c[nH]cn1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2ccccc2[nH]1
CCCC[C@H](NC(=O)c1cc2c(OC)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl
CCCC[C@H](NC(=O)c1cc2c(OC)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CCC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CCC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
CC(C)(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)(C)C)NC(=O)c1cc2ccccc2[nH]1
CCOCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)(C)C)NC(=O)c1cc2ccccc2[nH]1
CC(C)(C)C[C@H](NC(=O)[C@H]1CCCO1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)(C)C)NC(=O)[C@H]1CCCO1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
CC(C)C[C@H](N(C)C(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COCc1ccccc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)N(C)[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COCc1ccccc1
COc1cccc2[nH]c(cc12)C(=O)N(C)[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COCc1ccccc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(C)=O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1CC1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C(C)(C)C
CC(C)(C)C[C@H](NC(=O)[C@H]1CCCO1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccccc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccc(C)cc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccc(F)cc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccc(cc1)C#N
COc1ccc(cc1)C(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccc(Cl)cc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)cccc1C
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(F)cccc1F
COc1cccc(OC)c1C(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccc(Cl)cc1O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccc(cc1F)C#N
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CNC(=O)c1ccccc1C#N
CC(C)C[C@H](NC(C)=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CN=[N+]=[N-]
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CNC(C)=O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CNS(C)(=O)=O
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c2ccccc2C#N)NC(=O)c3cc4c([nH]3)cccc4OC
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CN(C)C
CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)C[C@@H]1CCNC1=O
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)CO)NC(=O)c2cc3c([nH]2)cccc3OC
COC(O)[C@@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C(C)=O
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)CO)NC(=O)[C@H](C(C)C)NC(=O)OCc2ccccc2
CC(C)C[C@H](NC(=O)[C@@H](NC(C)=O)C(C)C)C(=O)N[C@H](CO)C[C@@H]1CCNC1=O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(=O)N(C)C)C=O
CON(C)C(=O)[C@H](CCC(=O)N(C)C)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
CCOC(=O)\C=C\[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccc(cc1)[N+]([O-])=O
CCOC(=O)C=CC(CC1CCNC1=O)NC(=O)C(CC(=O)C(NC(=O)c1cc(C)on1)C(C)C)Cc1ccc(F)cc1 |w:5.4|
CCOC(=O)C=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |w:5.4|
CCOC(=O)C=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |w:5.4|
CCOC(=O)C=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C |w:5.4|
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)O)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)O)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
CC(C)C[C@H](NC(=O)C(NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
[O-][N+](=O)c1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)c(Cl)c1
[O-][N+](=O)c1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O
[O-][N+](=O)c1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)cc1
CN(C)c1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1)[N+]([O-])=O
CN(C)c1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1
CN(C)c1ccc(cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1Cl
O=C[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)\C=C\c1ccccc1
CC(OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](CCC(=O)N(C)C)C=O |r|
CC(C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)CF
CCC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)CF
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)CF
CN(C)C(=O)CC[C@H](NC(=O)CNC(=O)OCc1ccccc1)C(=O)CF
C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)CF
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(O)=O)C(=O)CF
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)C(F)(F)F |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)C(F)(F)F
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(=O)N1CCOCC1)C(=O)C(F)(F)F |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc2ccccc2)C(C)C)C(=O)c2nccs2)CCNC1=O |r|
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c2nc3ccccc3s2)NC(=O)c4cc5c([nH]4)cccc5OC
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1cccc(c1)N(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)F
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)F
FC(F)(F)C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C(=O)C(F)(F)F
C[C@H](NC(=O)[C@H](CCC(O)=O)NC(=O)OC(C)(C)C)C(=O)NCC(=O)C(F)(F)F
C[C@H](NC(=O)[C@@H](N)CCC(O)=O)C(=O)NCC(=O)C(F)(F)F
CCCCCCCCCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)F
CCCCCCCCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)F
O[C@H]([C@H](Cc1c[nH]c2ccccc12)NC(=O)OCc1ccccc1)[C@H](O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OCc1ccccc1
CC(C)[C@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)[C@@H](O)[C@H](O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C
CCC(=C)C(=O)c1ccc(c(c1Cl)Cl)OCC(=O)O
CCC(=C)C(=O)c1ccc(OCC(=O)NC(=O)OC(C)(C)C)c(Cl)c1Cl
CCC(=C)C(=O)c1ccc(OCC(=O)NC(=O)OC(C)(C)C(N)=O)c(Cl)c1Cl
Cc1noc(C)c1CC1C(=O)C(=O)c2cc(ccc12)C#N
Fc1ccc(CC2C(=O)C(=O)c3cc(I)ccc23)c(Cl)c1
[O-][N+](=O)c1cccc2C(=O)C(=O)C(Cc3cc4ccccc4s3)c12
Brc1cccc2C(=O)C(=O)C(Cc3cc4ccccc4s3)c12
Fc1ccc2C(Cc3cc4ccccc4s3)C(=O)C(=O)c2c1
Ic1ccc2C(Cc3cc4ccccc4s3)C(=O)C(=O)c2c1
CC1CCN(CC1)S(=O)(=O)c1ccc2C(Cc3ccccc3)C(=O)C(=O)c2c1
c1cc(c(cc1C2=CC(=O)c3c(cc(cc3O2)O)O)O)O
c1cc(c(cc1C2=C(C(=O)c3c(cc(cc3O2)O)O)O)O)O
c1cc(c(cc1C2=C(C(=O)c3c(cc(cc3O2)O)O)O[C@H]4[C@@H]([C@H]([C@H]([C@H](O4)CO)O)O)O)O)O
C[C@H]1O[C@@H](Oc2c(oc3cc(O)cc(O)c3c2=O)-c2ccc(O)c(O)c2)[C@H](O)[C@@H](O)[C@H]1O
Oc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)c(-c3cc(ccc3O)-c3oc4cc(O)cc(O)c4c(=O)c3O)c2o1 |(5.33,1.54,;4,2.31,;2.67,1.54,;1.33,2.31,;1.33,3.85,;2.67,4.62,;4,3.85,;,4.62,;,6.16,;-1.33,6.93,;-1.33,8.47,;-2.67,6.16,;-4,6.93,;-4,8.47,;-5.33,6.16,;-5.33,4.62,;-6.67,3.85,;-4,3.85,;-4,2.31,;-2.67,1.54,;-2.67,,;-4,-.77,;-5.33,,;-5.33,1.54,;-6.67,2.31,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;5.33,,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-2.31,;,-3.08,;,-4.62,;-1.33,-2.31,;-2.67,-3.08,;-2.67,4.62,;-1.33,3.85,)|
COc1ccc(cc1-c1c(O)cc(O)c2c1oc(cc2=O)-c1ccc(O)cc1)-c1oc2cc(O)cc(O)c2c(=O)c1O |(-6.67,3.85,;-6.67,2.31,;-5.33,1.54,;-4,2.31,;-2.67,1.54,;-2.67,,;-4,-.77,;-5.33,,;-6.67,-.77,;-8,,;-8,1.54,;-9.34,-.77,;-9.34,-2.31,;-10.67,-3.08,;-8,-3.08,;-6.67,-2.31,;-5.33,-3.08,;-5.33,-4.62,;-6.67,-5.39,;-8,-4.62,;-9.34,-5.39,;-4,-5.39,;-2.67,-4.62,;-1.33,-5.39,;-1.33,-6.93,;,-7.7,;-2.67,-7.7,;-4,-6.93,;-1.33,-.77,;;1.33,-.77,;2.67,,;4,-.77,;5.33,,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-2.31,;,-3.08,;,-4.62,;-1.33,-2.31,;-2.67,-3.08,)|
COc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)c(-c3cc(ccc3OC)-c3cc(=O)c4c(O)cc(OC)cc4o3)c2o1 |(-13.34,,;-13.34,1.54,;-12,2.31,;-12,3.85,;-10.67,4.62,;-9.34,3.85,;-9.34,2.31,;-10.67,1.54,;-8,4.62,;-8,6.16,;-6.67,6.93,;-6.67,8.47,;-5.33,6.16,;-4,6.93,;-4,8.47,;-2.67,6.16,;-2.67,4.62,;-1.33,3.85,;-4,3.85,;-4,2.31,;-2.67,1.54,;-2.67,,;-4,-.77,;-5.33,,;-5.33,1.54,;-6.67,2.31,;-8,1.54,;-1.33,-.77,;-1.33,-2.31,;,-3.08,;,-4.62,;1.33,-2.31,;2.67,-3.08,;2.67,-4.62,;4,-2.31,;4,-.77,;5.33,,;5.33,1.54,;2.67,,;1.33,-.77,;;-5.33,4.62,;-6.67,3.85,)|
COc1cc(O)c2c(c1)oc(cc2=O)-c1ccc(OC)c(c1)-c1c(O)cc(O)c2c1oc(cc2=O)-c1ccc(O)cc1 |(-10.67,4.62,;-9.34,3.85,;-8,4.62,;-8,6.16,;-6.67,6.93,;-6.67,8.47,;-5.33,6.16,;-5.33,4.62,;-6.67,3.85,;-4,3.85,;-2.67,4.62,;-2.67,6.16,;-4,6.93,;-4,8.47,;-1.33,3.85,;,4.62,;1.33,3.85,;1.33,2.31,;2.67,1.54,;4,2.31,;,1.54,;-1.33,2.31,;;-1.33,-.77,;-2.67,,;-1.33,-2.31,;,-3.08,;,-4.62,;1.33,-2.31,;1.33,-.77,;2.67,,;4,-.77,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;5.33,,;5.33,1.54,;6.67,2.31,;8,1.54,;9.34,2.31,;8,,;6.67,-.77,)|
c1cc(ccc1C2=CC(=O)c3c(cc(cc3O2)O)O)O
CC(C)c1cc2CCC3C(C)(C)CCCC3(C)c2cc1O
CC(C)c1cc2CCC3[C@@](C)(CCC[C@@]3(C)c2cc1O)C=O
CC(C)c1cc2CCC3[C@](C)(CO)CCC[C@@]3(C)c2cc1O
CC1=CC[C@]2(C)CC[C@]3(C)C4=CC=C5C(C)=C(O)C(=O)C=C5[C@]4(C)CC[C@@]3(C)C2C1 |c:20,t:1,10,12,15|
COC(=O)C1(C)CCC2(C)CCC3(C)C4=CC=C5C(C)=C(O)C(=O)C=C5C4(C)CCC3(C)C2C1 |c:24,t:14,16,19|
COC(=O)[C@]1(C)CC[C@]2(C)CC[C@]3(C)C4=CC=C5C(C)=C(O)C(=O)C=C5[C@]4(C)CC[C@@]3(C)C2C1 |r,c:24,t:14,16,19|
CC1=C(O)C(=O)C=C2C1=CC=C1[C@@]2(C)CC[C@@]2(C)C3C[C@@](C)(CC[C@]3(C)CC[C@]12C)C(O)=O |c:1,6,11,t:9|
CC1=C(O)C(O)C=C2C1=CC=C1[C@@]2(C)CC[C@@]2(C)C3C[C@@](C)(CC[C@]3(C)CC[C@]12C)C(O)=O |c:1,6,11,t:9|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)C(CCC4[C@@]5(C)CCC(O)C(C)(C)C5CC[C@@]34C)C12)C(O)=O
O=C1OC[C@H](Cc2ccc3OCOc3c2)C1Cc1ccc2OCOc2c1
CSC1=C(C(C)C(S1)c1nc(C)cs1)c1ccnc(SCC(=O)Nc2ccc(Cl)cc2)n1 |t:2|
CSC1=C(C(C)C(S1)c1nc(C)cs1)c1ccnc(SCC(=O)Nc2ccccc2Cl)n1 |t:2|
CN(C)c1ccc(cc1)C(=O)C(=O)On1nnc2ccccc12
CNc1ccc(cc1)C(=O)C(=O)On1nnc2ccccc12
CCN(CC)c1ccc(cc1)C(=O)C(=O)On1nnc2ccccc12
O=C(On1nnc2ccccc12)C(=O)c1ccc2[nH]cnc2c1
O=C(On1nnc2ccccc12)C(=O)c1ccc2[nH]ccc2c1
O=C(On1nnc2ccccc12)C(=O)c1cc2ccccc2[nH]1
Fc1ccc2cc([nH]c2c1)C(=O)C(=O)On1nnc2ccccc12
Clc1cncc(OC(=O)c2cccs2)c1
Clc1cncc(OC(=O)c2ccco2)c1
Brc1cncc(OC(=O)c2ccco2)c1
Clc1cncc(OC(=O)c2cc3ccccc3[nH]2)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Oc1cncc(Cl)c1
Clc1cncc(OC(=O)c2cccc3[nH]ccc23)c1
CC(=O)n1ccc2c(cccc12)C(=O)Oc1cncc(Cl)c1
Clc1cncc(OC(=O)c2ccc3[nH]ccc3c2)c1
Clc1ccnc(OC(=O)c2ccc3cc[nH]c3c2)c1
Clc1ccnc(OC(=O)c2cccc3cc[nH]c23)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Cc1cc(Br)ccn1
Clc1ccc(cc1)-c1ncc(o1)C(=O)Cc1cc(Br)ccn1
FC(C(=O)c1cnc(o1)-c1ccc(Cl)cc1)c1cc(Br)ccn1
FC(F)(C(=O)c1cnc(o1)-c1ccc(Cl)cc1)c1cc(Br)ccn1
OC(=O)c1cc(Br)ccc1-c1ccc(\C=C2\C(=O)NN(C2=O)c2ccc(Cl)c(Cl)c2)o1
Clc1ccc(cc1)-c1c(c(nn1-c1ccc(Cl)c(Cl)c1)-c1ccc(Br)cc1)-n1ccnc1
OC(=O)c1ccc(\C=C2\C(NN(C2=O)c2ccc(cc2)C#N)c2ccccc2)cc1
OC(=O)c1ccc(\C=C2\C(NN(C2=O)c2ccc(F)cc2)c2ccccc2)cc1
OC(=O)c1ccc(\C=C2\C(NN(C2=O)c2ccc(cc2)[N+]([O-])=O)c2ccccc2)cc1
[O-][N+](=O)c1cccc(c1)-c1nc(SCc2ccccc2)[nH]c(=O)c1C#N
[O-][N+](=O)c1ccc(CSc2nc(-c3cccc(c3)[N+]([O-])=O)c(C#N)c(=O)[nH]2)cc1
[O-][N+](=O)c1ccc(CSc2nc(-c3ccc(Cl)cc3)c(C#N)c(=O)[nH]2)cc1
O=CC(Cc1c[nH]cn1)NC[C@@H]1C[C@H]2CCCC[C@H]2CN1C(=O)c1ccc(cc1)-c1ccccc1
O=CC(Cc1c[nH]cn1)NC[C@H]1C[C@@H]2CCCC[C@@H]2CN1C(=O)c1ccc(cc1)-c1ccccc1
O=CC(Cc1c[nH]cn1)NCC1CC2CCCCC2CN1C(=O)c1ccccc1
Brc1ccc(cc1)C(=O)N1C[C@@H]2CCCC[C@@H]2C[C@H]1CNC(Cc1c[nH]cn1)C=O
Brc1ccc(cc1)C(=O)N1C[C@H]2CCCC[C@H]2C[C@@H]1CNC(Cc1c[nH]cn1)C=O
Fc1ccc(cc1)C(=O)N1CC2CCCCC2CC1CNC(Cc1c[nH]cn1)C=O
CCC(C)c1ccc(cc1)N(C(C(=O)NC1CCCC1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)c1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1cccnc1)C(=O)c1ccco1
CC(C)(C)NC(=O)C(N(C(=O)c1cnco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1cccs1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1ncco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1ccc(Cl)o1)c1ccc(cc1)C(C)(C)C)c1cccnc1
Cn1cnc(c1)C(=O)N(C(C(=O)NC(C)(C)C)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1ccnnc1
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1ccncn1
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1ccncc1
CCC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(C)=O)cc1)c1ccn(C)c1
CCC(C)(C)NC(=O)C(N(C(=O)Cn1cc(nn1)-c1ccccc1)c1ccc(NC(C)=O)cc1)c1ccn(C)c1
CCC(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccn(C)c1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccn(C)c1)C(=O)Cn1nnc2ccccc12
Cn1ccc(c1)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CC2)cc1)C(=O)NC(C)(C)C
Cn1ccc(c1)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CCC2)cc1)C(=O)NC(C)(C)C
CCC(=O)Nc1ccc(cc1)N(Cc1ccn(C)c1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N(Cc1ccn(C)c1)C(=O)Cn1nnc2ccccc12
Cn1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(NC(=O)C3CC3)cc2)c1
Cn1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(NC(=O)C3CCC3)cc2)c1
Cn1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2ccccc2)c1
CC(=O)O[Hg]c1ccccc1
CC[Hg]Sc1ccccc1C([O-])=O
[O-][N+](=O)O[Hg]c1ccccc1
[O-][n+]1ccccc1S[Zn]Sc1cccc[n+]1[O-]
CCN(C(=S)S[Zn]SC(=S)N(CC)c1ccccc1)c1ccccc1
Cc1ccc2S[Zn]Nc2c1
OC(=O)CC1N[Zn]2(NC(CC(O)=O)C(=O)O2)OC1=O
OB(O)c1cccc(COC(=O)c2cc(cc(c2)[N+]([O-])=O)B(O)O)c1
OB(O)c1cc(cc(c1)[N+]([O-])=O)C(=O)OCc1ccccc1COC(=O)c1cc(cc(c1)[N+]([O-])=O)B(O)O
OB(O)c1cc(cc(c1)[N+]([O-])=O)C(=O)Nc1ccc(NC(=O)c2cc(cc(c2)[N+]([O-])=O)B(O)O)cc1
Oc1ccccc1\C=N\c1ccc(cc1)C([O-])=O
CC1=C(C(C2C(CCCC2=O)N1)c1ccccc1[N+]([O-])=O)C(=O)OCCc1ccccc1 |t:1|
Cc1ccc2nc(sc2c1S(O)(=O)=O)-c1ccc(N)cc1
Oc1cc(cc2oc(cc12)C([O-])=O)C(F)(F)F
OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)N1CNc2c1ncnc2Cl
OCC1C(COCc2ccccc2)CC1N1CNc2c1ncnc2Cl
CN(C)CCCNC(=O)C(\NC(=O)c1ccc(C)cc1)=C\c1ccc(o1)-c1cccc(c1)[N+]([O-])=O
CN(C)CCCNC(=O)C(\NC(=O)c1ccc(C)cc1)=C\c1ccc(o1)-c1ccccc1[N+]([O-])=O
Nc1ncnc2[nH]c(nc12)C(F)(F)F
Cn1cnc2cc(NC(=O)c3ccc(Cl)cc3)ccc12
CCOC(=O)C=C[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccc(F)cc1 |w:5.4|
CCOC(=O)C=C[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccccc1 |w:5.4|
CCOC(=O)C=C[C@H](C[C@@H]1CNC(=O)C1)NC(=O)[C@@H](CC(=O)[C@@H](NC(=O)c1cc(C)on1)C(C)C)Cc1ccccc1 |w:5.4|
[#6]-[#6]-[#8]-[#6](=O)-[#6]=[#6]-[#6@H](-[#6]-[#6@@H]-1-[#6]-[#7]-[#6](=O)-[#6]-1)-[#7]-[#6](=O)-[#6@H](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-c1cc(-[#6])on1)-[#6](-[#6])-[#6] |w:5.4|
[#6]-[#6]-[#8]-[#6](=O)-[#6]=[#6]-[#6@H](-[#6]-[#6@@H]-1-[#6]-[#7]-[#6](=O)-[#6]-1)-[#7]-[#6](=O)-[#6@H](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#8])-[#7]-[#6](=O)-[#8]C([#6])([#6])[#6])-[#6](-[#6])-[#6] |w:5.4|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)CC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)CC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C
CC(C)C[C@H](CC(=O)[C@H](C)NC(=O)c1cc(C)on1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)\C=C\C(=O)OCc1ccccc1
CC(OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)C[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
Brc1cccc(\C=C\C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1
Fc1cc(Cl)ccc1\C=C\C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
C[C@H](NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](C1CCCCC1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O
O=C[C@H](Cc1c[nH]cn1)NC[C@@H]1C[C@@H]2CCCC[C@H]2CN1C(=O)c1ccc(cc1)-c1ccccc1
O=C[C@H](Cc1c[nH]cn1)NC[C@@H]1C[C@@H]2CCCC[C@H]2CN1C(=O)c1ccccc1
Brc1ccc(cc1)C(=O)N1C[C@@H]2CCCC[C@H]2C[C@H]1CN[C@@H](Cc1c[nH]cn1)C=O
O=C[C@H](Cc1c[nH]cn1)NC[C@H]1C[C@H]2CCCC[C@@H]2CN1C(=O)c1ccc(cc1)-c1ccccc1
Brc1ccc(cc1)C(=O)N1C[C@H]2CCCC[C@@H]2C[C@@H]1CN[C@@H](Cc1c[nH]cn1)C=O
CC(O)[C@@H](NC(C)=O)C(=O)NCC(=O)NC1CCC[C@H]2CN([C@H](CN[C@@H](Cc3c[nH]cn3)C=O)C[C@H]12)C(=O)c1ccc(Br)cc1
CCCCN(C)C[C@H]1O[C@@H](CN[C@@H](Cc2c[nH]cn2)C=O)C[C@H]2CCCC[C@H]12
CCCCN(C)C[C@H]1O[C@H](CN[C@@H](Cc2c[nH]cn2)C=O)C[C@H]2CCCC[C@H]12
CCCCN(C)C[C@@H]1O[C@@H](CN[C@@H](Cc2c[nH]cn2)C=O)C[C@H]2CCCC[C@H]12
CCCCN(C)C[C@@H]1O[C@H](CN[C@@H](Cc2c[nH]cn2)C=O)C[C@H]2CCCC[C@H]12
CC(C)C[C@H](NC(=O)OC1CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O
CC(C)C[C@H](NC(=O)OC1(Cc2ccccc2)CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O
O=C(N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)\C=C\c1ccccc1
O=C(N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)\C=C\c1ccccc1
O=C(N[C@@H](CC1CCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)\C=C\c1ccccc1
CC(C)(C)OC(=O)Nc1cccn(C(CC2CCCCC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NC2CC2)c1=O
CC(C)(C)OC(=O)Nc1cccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NCc2ccccc2)c1=O
COc1cccc(NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)c1
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)C(C)O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
O[C@H]([C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)[C@H](O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
O=C(On1nnc2ccccc12)c1ccc2[nH]cnc2c1
Clc1cncc(OC(=O)c2ccc3cc[nH]c3c2)c1
Clc1cncc(OC(=O)c2cccc3cc[nH]c23)c1
Cc1ccc(cc1)S(=O)(=O)n1ccc2cc(ccc12)C(=O)Oc1cncc(Cl)c1
Clc1ccc(cc1)-c1ccc(o1)C(=O)Cc1cncc(Br)c1
FC(C(=O)c1ccc(o1)-c1ccc(Cl)cc1)c1cncc(Br)c1
FC(F)(C(=O)c1ccc(o1)-c1ccc(Cl)cc1)c1cncc(Br)c1
Ic1ccc2N(Cc3cc4ccccc4s3)C(=O)C(=O)c2c1
Brc1cccc2C(=O)C(=O)N(Cc3cc4ccccc4s3)c12
NC(=O)c1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
CC1CCN(CC1)S(=O)(=O)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
Clc1ccc(cc1)C1C(C(=NN1c1ccc(Cl)c(Cl)c1)c1ccc(Br)cc1)n1ccnc1 |c:10|
CC(C)c1ccc(cc1)N1NC(\C(=C\C2CCC(O2)c2cc(Cl)ccc2C(O)=O)C1=O)c1ccccc1
OC(=O)c1ccc(Cl)cc1C1CCC(O1)\C=C1\C(NN(C1=O)c1ccccc1)c1ccccc1
CC(C)c1ccc(cc1)N1NC(\C(=C\C2CCC(O2)c2ccccc2C(O)=O)C1=O)c1ccccc1
OC(=O)c1ccc(cc1)N1NC(\C(=C\C2CCC(O2)c2ccccc2)C1=O)c1ccccc1
CC(C)(C)c1ccc(cc1)N([C@H](c2cccnc2)C(=O)NC(C)(C)C)C(=O)c3ccco3
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cnccn1
CC(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccn(C)c1)C(C)=O
CC(C)C(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccsc1)C(=O)Cn1nnc2ccccc12
CC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C2CCC2)cc1)c1ccsc1
CCC(=O)Nc1ccc(cc1)N(Cc2ccsc2)C(=O)Cn3c4ccccc4nn3
CC(C)C(=O)Nc1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cc1ccccc1)Nc1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1cccnc1
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1ccccc1
Oc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)c(-c3cc(ccc3O)-c3cc(=O)c4c(O)cc(O)cc4o3)c2o1 |(-10.67,-4.62,;-9.34,-5.39,;-9.34,-6.93,;-8,-7.7,;-6.67,-6.93,;-6.67,-5.39,;-8,-4.62,;-5.33,-7.7,;-5.33,-9.24,;-4,-10.01,;-4,-11.55,;-2.67,-9.24,;-1.33,-10.01,;-1.33,-11.55,;,-9.24,;,-7.7,;1.33,-6.93,;-1.33,-6.93,;-1.33,-5.39,;,-4.62,;,-3.08,;-1.33,-2.31,;-2.67,-3.08,;-2.67,-4.62,;-4,-5.39,;1.33,-2.31,;1.33,-.77,;2.67,,;2.67,1.54,;4,-.77,;5.33,,;5.33,1.54,;6.67,-.77,;6.67,-2.31,;8,-3.08,;5.33,-3.08,;4,-2.31,;2.67,-3.08,;-2.67,-7.7,;-4,-6.93,)|
CC(C)c1cc2CCC3C(C)(C)CCC[C@]3(C)c2cc1O
CC1=CC[C@]2(C)CC[C@]3(C)C4=CC=C5C(C)=C(O)C(=O)C=C5C4CC[C@@]3(C)C2C1 |c:20,t:1,10,12,15|
C[C@@H]1CC2[C@@](C)(CC[C@]3(C)C4=CC=C5C(C)=C(O)C(=O)C=C5[C@]4(C)CC[C@@]23C)CC1=O |c:20,t:10,12,15|
CC(=C)[C@@H]1CC[C@@]2(CC[C@]3(C)C(CCC4[C@@]5(C)CC[C@H](O)C(C)(C)C5CC[C@@]34C)C12)C(O)=O
O=C1OC[C@H](Cc2ccc3OCOc3c2)\C1=C/c1ccc2OCOc2c1
CN(C)CCCSc1ccccc1NC(=C)\C=C\c1ccccc1
[#6]\[#6](-[#6])=[#6]\[#6]-[#6@@H](-[#8])-[#6]-1-[#6]-[#6](=O)-c2c(-[#8])ccc(-[#8])c2-[#6]-1=O
Nc1nccc2[nH]c(nc12)C(F)(F)F
S=C1NC=NC2NC=NC12 |c:3,7|
NC1=NC2NC=NC2C(=S)N1 |c:5,t:1|
[#6]\[#6](-[#6])=[#6]\[#6]-c1cc(cc(-[#8])c1-[#8])-c1oc2c(-[#6]\[#6]=[#6](\[#6])-[#6])c(-[#8])cc(-[#8])c2c(=O)c1-[#8]
[#6]\[#6](-[#6])=[#6]\[#6]-c1cc(-[#6](=O)\[#6]=[#6]\c2ccc(-[#8])c(-[#8])c2)c(-[#8])cc1-[#8]
CCC(CC)COC(=O)[C@H](C)N[P@](=O)(OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1
c1nc(nn1[C@H]2[C@@H]([C@@H]([C@H](O2)CO)O)O)C(=O)N
NC(=O)c1nc(F)c[nH]c1=O
CC(C)C(=O)OC[C@@H]1[C@H]([C@H]([C@@H](O1)N2C=CC(=NC2=O)NO)O)O
CCN(CC)CCC[C@@H](C)Nc1ccnc2c1ccc(c2)Cl
CN(C)CCCN1c2ccccc2Sc3c1cc(cc3)Cl
CN(C)C(=O)C(CCN1CCC(CC1)(c2ccc(cc2)Cl)O)(c3ccccc3)c4ccccc4
CC(C)[C@H](N1CCCNC1=O)C(=O)N[C@H](C[C@H](O)[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C)Cc1ccccc1
CC[C@H]1CN2CCc3cc(c(cc3[C@@H]2C[C@@H]1C[C@@H]4c5cc(c(cc5CCN4)OC)OC)OC)OC
CCN(CCO)CCCC(C)Nc1ccnc2cc(Cl)ccc12
OC(C1CCCCN1)c1cc(nc2c(cccc12)C(F)(F)F)C(F)(F)F
CCN(CC)Cc1cc(ccc1O)Nc2ccnc3c2ccc(c3)Cl
CCOC(=O)C1OC1C(=O)NC(CC(C)C)C(=O)NCCC(C)C
Nc1ccn([C@@H]2O[C@H](CO)[C@@H](O)C2(F)F)c(=O)n1
CC/C(=C(\c1ccccc1)/c2ccc(cc2)OCCN(C)C)/c3ccccc3
CN(C)CCOc1ccc(cc1)/C(=C(/CCCl)\c2ccccc2)/c3ccccc3
CC(C)N1CCN(CC1)c1ccc(OC[C@H]2CO[C@@](Cn3cncn3)(O2)c2ccc(Cl)cc2Cl)cc1
COc1ccc(C[C@H]2NC[C@H](O)[C@H]2OC(C)=O)cc1
C[C@H]1C[C@@H](C(=O)[C@@H](C1)[C@@H](CC2CC(=O)NC(=O)C2)O)C
CN1[C@H]2CC[C@@H]1CC(C2)OC(c1ccccc1)c1ccccc1 |THB:9:7:1:4.3|
Fc1ccc(cc1)C(CCCN1CCC2(CC1)N(CNC2=O)c1ccccc1)c1ccc(F)cc1
CN(C)S(=O)(=O)c1ccc2Sc3ccccc3\C(=C\CCN3CCN(C)CC3)c2c1
OCCN1CCN(CCCN2c3ccccc3Sc3ccc(cc23)C(F)(F)F)CC1
CC(CN1c2ccccc2Sc2ccccc12)N(C)C
COc1ccc(cc1)CCN2CCC(CC2)Nc3nc4ccccc4n3Cc5ccc(cc5)F
CN(C)CCOC(C)(c1ccccc1)c1ccc(Cl)cc1
CN(C)CCCN1c2ccccc2Sc2ccc(cc12)C(F)(F)F
CN(C)CCCN1c2ccccc2CCc3c1cc(cc3)Cl
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
Cc1cccc(c1NC(=O)c2cnc(s2)Nc3cc(nc(n3)C)N4CCN(CC4)CCO)Cl
C1=CN(C(=O)N=C1NO)[C@H]2[C@@H]([C@@H]([C@H](O2)CO)O)O
[#6]-[#7](-[#6])-[#6](=O)-[#6]-[#8]-[#6](=O)-[#6]-c1ccc(-[#8]-[#6](=O)-c2ccc(cc2)\[#7]=[#6](/[#7])-[#7])cc1
CCN(CC)CCOc1ccc2-c3ccc(OCCN(CC)CC)cc3C(=O)c2c1
CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C |r|
C(C(C1CCCCC1)C1CCCCC1)C1CCCCN1
C[C@@H]1O[C@@H](O[C@H]2CC[C@]3(C)[C@H]4CC[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CCC3=C2)c2ccc(=O)oc2)[C@H](O)[C@H](O)[C@H]1O |c:26|
Nc1ccc(N=Nc2ccccc2)c(N)n1 |w:6.6|
C[C@@H]1[C@H]([C@H](C[C@@H](O1)O[C@@H]2[C@H](O[C@H](C[C@@H]2O)O[C@@H]3[C@H](O[C@H](C[C@@H]3O)O[C@H]4CC[C@]5([C@@H](C4)CC[C@@H]6[C@@H]5CC[C@]7([C@@]6(CC[C@@H]7C8=CC(=O)OC8)O)C)C)C)C)O)O
c1cc(ccc1C(CCCN2CCC(CC2)(c3ccc(c(c3)C(F)(F)F)Cl)O)c4ccc(cc4)F)F
CCN(CC)CCOc1ccc(cc1)C(=C(Cl)c1ccccc1)c1ccccc1 |w:15.16|
C[C@@H]1[C@H]([C@H](C[C@@H](O1)O[C@@H]2[C@H](O[C@H](C[C@@H]2O)O[C@@H]3[C@H](O[C@H](C[C@@H]3O)O[C@H]4CC[C@]5([C@@H](C4)CC[C@@H]6[C@@H]5C[C@H]([C@]7([C@@]6(CC[C@@H]7C8=CC(=O)OC8)O)C)O)C)C)C)O)O
C[C@H]1O[C@H](C[C@H](O)[C@@H]1O[C@H]1C[C@H](O)[C@H](O[C@H]2C[C@H](OC(C)=O)[C@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[C@@H](C)O2)[C@@H](C)O1)O[C@H]1CC[C@@]2(C)[C@H](CC[C@@H]3[C@@H]2C[C@@H](O)[C@]2(C)[C@H](CC[C@]32O)C2=CC(=O)OC2)C1 |t:69|
CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CC[C@]4(C)[C@H]3CC[C@]12C |r,t:11|
CN1CCCC[C@H]1CCN2c3ccccc3Sc4c2cc(cc4)SC
CC[C@H]([C@H]1CC[C@H](C)[C@@H](O1)[C@@H](C)[C@H](O)[C@H](C)C(=O)[C@H](CC)[C@H]1O[C@@]2(O[C@@]3(CC[C@](C)(O3)[C@H]3CC[C@](O)(CC)[C@H](C)O3)[C@H](O)C=C2)[C@H](C)C[C@@H]1C)C(O)=O |c:46|
CCN(CC)CCC[C@@H](C)Nc1c2ccc(cc2nc3c1cc(cc3)OC)Cl
C[C@@H]1O[C@@H](O[C@H]2C[C@@H](O)[C@]3(CO)[C@H]4[C@H](O)C[C@]5(C)[C@H](CC[C@]5(O)[C@@H]4CC[C@]3(O)C2)C2=CC(=O)OC2)[C@H](O)[C@H](O)[C@H]1O |r,t:33|
COc1ccc2C[C@@H]3N(C)CCc4cc(OC)c(Oc5c6OCOc6cc6CCN(C)[C@@H](Cc7ccc(Oc1c2)cc7)c56)cc34 |r|
[H][C@@]12C[C@@]3([H])[C@]4([H])CCC5=CC(=O)C=C[C@]5(C)[C@@]4([H])[C@@H](O)C[C@]3(C)[C@@]1(O[C@@H](O2)C1CCCCC1)C(=O)COC(=O)C(C)C |r,c:13,t:9|
Oc1c(Cl)cc(Cl)cc1NC(=O)c1c(O)c(Cl)cc(Cl)c1Cl
Cc1cc(c(cc1C2CCNCC2)OC(C)C)Nc3ncc(c(n3)Nc4ccccc4S(=O)(=O)C(C)C)Cl
[#6]\[#6](-[#6])=[#6]/[#6]-[#6]C1([#6])[#8]-c2c(-[#6]\[#6]=[#6](\[#6])-[#6])c3-[#8]C45[#6]6-[#6]-[#6](-[#6]=[#6]4-[#6](=O)-c3c(-[#8])c2-[#6]=[#6]1)-[#6](-[#8])C5([#6]\[#6]=[#6](\[#6])-[#6](-[#8])=O)[#8]C6([#6])[#6] |c:22,33,TLB:42:34:19.20:23.22,22:21:18:42.43,24:23:34.32:19.20,33:32:18:42.43,35:34:19.20:23.22,23:18:42.43:32.21.20,THB:17:18:42.43:32.21.20,33:32:19.20:23.22,43:19:34.32:23.22|
COc1cc(N(C)CCN(C)C)c(NC(=O)C=C)cc1Nc1nccc(n1)-c1cn(C)c2ccccc12
CC1(C)CCc2c3OC(C)(C)C=Cc3c3occ(-c4ccc(O)c(O)c4)c(=O)c3c2O1 |c:11|
CCCCCOc1ccc(cc1)-c1ccc(cc1)-c1ccc(cc1)C(=O)N[C@H]1C[C@@H](O)[C@@H](O)NC(=O)[C@@H]2[C@@H](O)[C@@H](C)CN2C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC1=O)[C@@H](C)O)[C@H](O)[C@@H](O)c1ccc(O)cc1)[C@@H](C)O |r|
[#6]\[#6](-[#6])=[#6]\[#6]-c1c(-[#8])c2c(occ(-c3ccc(-[#8])cc3)c2=O)c2-[#6]=[#6]C([#6])([#6])[#8]-c12 |c:25|
CCCCCCO[C@@H](C)c1cccc(-c2csc(NC(=O)c3cc(Cl)c(\C=C(/C)C(O)=O)c(Cl)c3)n2)c1OC
CC1(C)CCc2c3OC(C)(C)C=Cc3c3occ(-c4ccc(O)cc4)c(=O)c3c2O1 |c:11|
CCc1c(nc(c(n1)C(=O)N)Nc2ccc(c(c2)OC)N3CCC(CC3)N4CCN(CC4)C)NC5CCOCC5
COc1cc2CCN(C)[C@H]3Cc4ccc(Oc5cc(C[C@H]6N(C)CCc7cc(OC)c(OC)c(Oc1cc23)c67)ccc5O)cc4 |r|
CC(C)(C)c1ccc(cc1)C(=O)CCCN1CCC(CC1)OC(c1ccccc1)c1ccccc1
[H][C@]12Cc3ccc(Oc4cc(C[C@]5([H])N(C)CCc6cc(OC)c(OC)c(Oc7cc1c(CCN2C)cc7OC)c56)ccc4OC)cc3 |r|
CCN1CCN(Cc2ccc(Nc3ncc(F)c(n3)-c3cc(F)c4nc(C)n(C(C)C)c4c3)nc2)CC1
CC(C)(C)c1cc(c(cc1NC(=O)C2=CNc3ccccc3C2=O)O)C(C)(C)C
Cc1c(-c2ccc(O)cc2)n(Cc2ccc(OCCN3CCCCCC3)cc2)c2ccc(O)cc12
C(C1CN2CCC1CC2)N1c2ccccc2Sc2ccccc12 |THB:0:1:5.4:8.7,(5.33,,;5.33,1.54,;4.2,2.4,;5.55,3.44,;5.66,4.98,;6.77,4.04,;6.64,2.53,;8.13,1.78,;7.37,2.73,;4,-.77,;4,-2.31,;5.33,-3.08,;5.33,-4.62,;4,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;1.33,-.77,;;,1.54,;1.33,2.31,;2.67,1.54,;2.67,,)|
CCN(CC)CCOc1ccc(cc1)C(O)(Cc1ccc(Cl)cc1)c1ccc(C)cc1
CC\C(=C(\c1ccc(OCCN(C)C)cc1)c1cccc(O)c1)c1ccccc1
CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(C)(=O)=O)cc12
COC(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)CN(Cc1ccc(cc1)-c1ccccn1)NC(=O)[C@@H](NC(=O)OC)C(C)(C)C)C(C)(C)C |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccc(Cl)cc1F)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(CN1CCCCC1)C(=O)c1ccc(C)cc1
CC(C)c1ccc2Sc3cc(F)ccc3CC(N3CCN(CCO)CC3)c2c1
O=c1n(CC2CO2)c(=O)n(CC2CO2)c(=O)n1CC1CO1
CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C=O |r|
CCc1cc(c(cc1F)Oc2ccc(cc2F)C(=O)N)O
CCOc1cc2c(cc1NC(=O)/C=C/CN(C)C)c(c(cn2)C#N)Nc3ccc(c(c3)Cl)F
C[C@@H](C(c1ccc(cc1)O)O)N2CCC(CC2)Cc3ccccc3
c1ccc2c(c1)C3(CCN(CC3)CCc4ccc(cc4)C(F)(F)F)OC(=O)N2
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
CN1C(=O)N(C(=O)S1)Cc2ccccc2
c1ccc(cc1)C2=CC(=O)c3c(cc(c(c3O)O)O)O2
c1cc(cc2c1cc3ccc(cc3n2)N)N
OCC(Br)(CO)[N+]([O-])=O
Oc1cc2CC[C@H]3NCc4ccccc4[C@@H]3c2cc1O
Nc1nc2n(cnc2c(=S)[nH]1)C1OC(CO)C(O)C1O
Oc1cc2CCNCC(c3ccccc3)c2cc1O
Cc1cc(C)cc(c1)N1C(=O)CC(Sc2nnc[nH]2)C1=O
CC(C)C[C@@H](C=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1
Cc1ccc(C)c(c1)-n1sc2cc(F)ccc2c1=O
CCOC(=O)Cc1ccc(cc1)-c1ccccc1
Brc1ccc2C(=O)C(=O)C=Cc2c1 |c:9|
Cc1c(ssc1=S)-c1cnccn1
NC(CO)C(=O)NNCc1ccc(O)c(O)c1O
c1c(cc(c(c1O)O)O)C2=C(C(=O)c3c(cc(cc3O2)O)O)O
OC[C@H]1O[C@@H](Oc2cccc3[C@@H]([C@@H]4c5cccc(O[C@@H]6O[C@H](CO)[C@@H](O)[C@H](O)[C@H]6O)c5C(=O)c5c(O)cc(cc45)C(O)=O)c4cc(cc(O)c4C(=O)c23)C(O)=O)[C@H](O)[C@@H](O)[C@@H]1O
CN1CCN(CC1)C(c1ccc(cc1)C(F)(F)F)c1ccc2cccnc2c1O
CN1CCN(CC1)C1=C(Cl)C(=O)N(C1=O)c1ccc(Cl)c(Cl)c1 |c:8|
ClCN1C(=O)c2ccccc2S1(=O)=O
Nc1nc(N)c(SC#N)cc1SC#N
COC(O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(C)=O |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)c1ccc2ccccc2c1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc2ccccc2c1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)CCc1cccc(F)c1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1cc(F)cc(F)c1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(F)c(F)c1 |r|
COc1ccc(OCC(=O)N2C[C@H]3[C@@H]([C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1OC |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(cc1)C(F)(F)F |r|
COc1ccc(OCC(=O)N2C[C@H]3[C@@H]([C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1F |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(OC(F)(F)F)cc1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)c(Br)c1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Br)cc1Cl |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)cc1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)c(Cl)c1 |r|
CC1(C)[C@H]2CN([C@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)cc1Cl |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@H]2CN1C(=O)c1cccnc1 |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@H]2CN1C(=O)c1cc2ccccc2[nH]1 |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@H]2CN1C(=O)c1cc2ccccn2n1 |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@H]2CN1C(=O)\C=C\c1ccccc1 |r|
COc1ccc(\C=C\C(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(OC)c1 |r|
CNc1ccc(\C=C\C(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
Fc1cccc(CCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
Fc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1F |r|
Fc1cc(F)cc(CCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
CN(C)c1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
COc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
COc1ccc(OC(C)C(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc2OCCOc2c1 |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
Fc1cc(Cl)ccc1OCC(=O)N1C[C@@H]2CCC[C@H]2[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(Cl)c1 |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1Cl |r|
Cc1cc(Cl)ccc1OCC(=O)N1C[C@@H]2CCC[C@H]2[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCNC1=O)C(O)S([O-])(=O)=O
c1ccc(cc1)N2C=C(C=C(C2=O)c3ccccc3C#N)c4ccccn4
Clc1cccc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:9|
Clc1cccc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:9|
Clc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:10|
CCCOc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:13|
COCCOc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:14|
Clc1cc(OCc2ccccc2)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:18|
Clc1cc(OCCc2ccccc2)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:19|
CCCOc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cncnc1)c1ccccc1C#N |c:13|
COc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:11|
CCCOc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:13|
CCCCOc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:14|
CCCC(C)Oc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:15|
Clc1cc(OCc2ccccc2)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:18|
Clc1cc(OCCc2ccccc2)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:19|
Cc1ccccc1COc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:19|
Cc1cccc(COc2cc(Cl)cc(c2)C2C=C(C(=O)N(C2=O)c2cccnc2)c2c[nH]c(=O)[nH]c2=O)c1 |c:17|
Fc1ccccc1COc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:19|
Fc1cccc(F)c1COc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:20|
Clc1cc(OCc2ccccc2Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:19|
Fc1ccc(Cl)c(COc2cc(Cl)cc(c2)C2C=C(C(=O)N(C2=O)c2cccnc2)c2c[nH]c(=O)[nH]c2=O)c1 |c:18|
Fc1c(Cl)cc(cc1OCc1ccccc1Cl)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:20|
Clc1cc(OC2CC2)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:14|
FC(F)(F)COc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1c[nH]c(=O)[nH]c1=O |c:15|
Clc1cc(OCC2CC2)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:15|
FC(F)(F)CCOc1cc(Cl)cc(c1)C1C=C(C(=O)N(C1=O)c1cccnc1)c1ccccc1C#N |c:16|
OC[C@H]1O[C@H](C(O)[C@H]1O)n1ccc(NO)nc1=O |r|
CCCCCCCCC(=O)ONc1ccn([C@@H]2O[C@H](CO)[C@H](O)C2O)c(=O)n1 |r|
CCCCCCCOC(=O)ONc1ccn([C@@H]2O[C@H](CO)[C@H](O)C2O)c(=O)n1 |r|
CONc1ccn([C@@H]2O[C@H](CO)[C@H](O)C2O)c(=O)n1 |r|
CC1(O)[C@@H](O)[C@@H](CO)O[C@H]1n1ccc(NO)nc1=O |r|
CNc1nc(N)nc2n(cnc12)[C@@H]1O[C@H](CO[P@@](=O)(N[C@@H](C)C(=O)OC(C)C)Oc2ccccc2)[C@@H](O)[C@@]1(C)F |r|
CNc1nc(N)nc2n(cnc12)[C@@H]1O[C@H](CO[P@](=O)(N[C@@H](C)C(=O)OC(C)C)Oc2ccccc2)[C@@H](O)[C@@]1(C)F |r|
CC(C)OC(=O)[C@H](C)N[P@](=O)(OCC1O[C@@H](n2ccc(=O)[nH]c2=O)[C@](C)(F)[C@@H]1O)Oc1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCC1CC2CCCC(C1)C2)C(=O)NC(CC1CCNC1=O)C=O |r,TLB:9:10:18:13.14.15|
CC(C)C[C@H](NC(=O)OCC1CC2CCCC(C1)C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,TLB:9:10:18:13.14.15|
CC(C)C[C@H](NC(=O)OCC1CC2CC=CC(C1)C2)C(=O)NC(CC1CCNC1=O)C=O |r,c:14,TLB:9:10:18:13.14.15|
CC(C)C[C@H](NC(=O)OCC1CC2CC=CC(C1)C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,c:14,TLB:9:10:18:13.14.15|
CC(C)C[C@H](NC(=O)OCC1CC2CC1C=C2)C(=O)NC(CC1CCNC1=O)C=O |r,c:16,THB:9:10:15.16:13|
CC(C)C[C@H](NC(=O)OCC1CC2CC1C=C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,c:16,THB:9:10:15.16:13|
CC(C)C[C@H](NC(=O)OCC1CC2CCC1C2)C(=O)NC(CC1CCNC1=O)C=O |r,TLB:9:10:14.13:16|
CC(C)C[C@H](NC(=O)OCC1CC2CCC1C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,TLB:9:10:14.13:16|
CC(C)C[C@H](NC(=O)OC1CC2CCC(C1)N2C(C)(C)C)C(=O)NC(CC1CCNC1=O)C=O |r,THB:8:9:16:12.13|
CC(C)C[C@H](NC(=O)OC1CC2CCC(C1)N2C(C)(C)C)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1CC2CCC(C1)N2C(=O)OCc1ccccc1)C(=O)NC(CC1CCNC1=O)C=O |r,THB:8:9:16:12.13|
CC(C)C[C@H](NC(=O)OC1CC2CCC(C1)N2C(=O)OCc1ccccc1)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r|
CCCCCC12CCC(COC(=O)N[C@@H](CC(C)C)C(=O)NC(CC3CCNC3=O)C=O)(CC1)CC2 |r|
CCCCCC12CCC(COC(=O)N[C@@H](CC(C)C)C(=O)NC(CC3CCNC3=O)C(O)S([O-])(=O)=O)(CC1)CC2 |r|
CC(C)C[C@H](NC(=O)OCC12CC3CC(CC(C3)C1)C2)C(=O)NC(CC1CCNC1=O)C=O |r,TLB:9:10:13:17.16.15,THB:15:14:11:17.16.18,15:16:11:13.14.19,18:16:13:11.19.10,18:10:13:17.16.15|
CC(C)C[C@H](NC(=O)OCC12CC3CC(CC(C3)C1)C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,TLB:9:10:13:17.16.15,THB:18:16:13:11.19.10,18:10:13:17.16.15,15:14:11:17.16.18,15:16:11:13.14.19|
CC(C)C[C@H](NC(=O)OCCC12CC3CC(CC(C3)C1)C2)C(=O)NC(CC1CCNC1=O)C=O |r,TLB:10:11:14:18.17.16,THB:19:17:14:12.20.11,19:11:14:18.17.16,16:15:12:18.17.19,16:17:12:14.15.20|
CC(C)C[C@H](NC(=O)OCCC12CC3CC(CC(C3)C1)C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,THB:16:15:12:18.17.19,16:17:12:14.15.20,19:17:14:12.20.11,19:11:14:18.17.16|
CC(C)C[C@H](NC(=O)OCC12CC3CC(CC(O)(C3)C1)C2)C(=O)NC(CC1CCNC1=O)C=O |r,TLB:20:10:18:15.13.14,THB:9:10:18:15.13.14,11:12:15:19.10.20,11:10:15:18.12.13,20:14:18:19.10.11|
CC(C)C[C@H](NC(=O)OCC12CC3CC(CC(O)(C3)C1)C2)C(=O)NC(CC1CCNC1=O)C(O)S([O-])(=O)=O |r,TLB:20:10:18:15.13.14,THB:20:14:18:19.10.11,9:10:18:15.13.14,11:12:15:19.10.20,11:10:15:18.12.13|
CC(C)C[C@H](NC(=O)OCc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(C)=O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)C(C)(C)C
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)C(C)(C)C#N
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)C(C)(C)C(F)(F)F
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)C1(C)OCCCO1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)C1(CCCCC1)C(F)(F)F
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1ccccc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1c(cccc1C(F)(F)F)C(F)(F)F
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1ccccn1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1cccnc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1ccncc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1c(C)cc(C)nc1C
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1c(C)nc(C)cc1C(F)(F)F
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1c(C)nc(C)nc1C
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C(=O)COC(=O)c1c(C)nn(C)c1C
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c2nc3ccccc3s2)NC(=O)[C@H](C(C)C)NC(=O)OCc4ccccc4
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)N(C)C
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)NC(CC1CCC1)C(=O)C(N)=O)C2(C)C)C(C)(C)C |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCNC1=O)C=O
CCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C=O
CCC[C@H](NC(=O)[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)c1cnccn1)C1CCCCC1)C(C)(C)C)C(=O)C(=O)NC1CC1 |r|
CC(OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](CC1CCNC1=O)C=O
c1ccc2c(c1)nnn2CC(=O)N(Cc3ccsc3)c4ccc(cc4)NC(=O)C5CC5
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccccc1
NC(=O)c1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)C(=O)NC1CC1
CS(=O)(=O)Nc1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(NS(=O)(=O)C2CC2)cc1
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1ccccn1
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1ccncc1
COc1ncccc1-c1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1ccc[nH]c1=O
Cn1cc(cn1)-c1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1cn[nH]c1
Cn1cnc(c1)-c1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)-c1c[nH]cn1
CC(C)CCN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1cccnc1
O=C(Cn1nnc2ccccc12)N(CC1CC1)c1ccc(cc1)-c1cccnc1
O=C(Cn1nnc2ccccc12)N(CC1CCC1)c1ccc(cc1)-c1cccnc1
O=C(Cn1nnc2ccccc12)N(CC1CCCC1)c1ccc(cc1)-c1cccnc1
O=C(Cn1nnc2ccccc12)N(CC1CCOC1)c1ccc(cc1)-c1cccnc1
O=C(Cn1nnc2ccccc12)N(Cc1cscn1)c1ccc(cc1)-c1cccnc1
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)c1
Fc1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)cc1Cl
Fc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)c1
Clc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)c1
Cc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)c1
Clc1cncc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)c1
c1ccc2c(c1)nnn2CC(=O)N(Cc3cccc(c3)Cl)c4ccc(cc4)C5=CC=CNC5=O
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cn[nH]c2)c1
COc1cc(ccc1-c1cn[nH]c1)N(Cc1cccc(Cl)c1)C(=O)Cn1nnc2ccccc12
COc1cc(ccc1N(Cc1cccc(Cl)c1)C(=O)Cn1nnc2ccccc12)-c1cn[nH]c1
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(nc2)-c2cn[nH]c2)c1
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cn2)-c2cn[nH]c2)c1
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Clc1cccc(CN(C(=O)Cc2cccnc2)c2ccc(cc2)-c2cn[nH]c2)c1
Clc1cccc(CN(C(=O)Cc2cncnc2)c2ccc(cc2)-c2cn[nH]c2)c1
CCCOc1cc(cc(c1)Cl)C2=CC(=CN(C2=O)c3cccnc3)c4ccccc4C#N
c1ccc(c(c1)C#N)C2=CN(C(=O)C(=C2)c3cc(cc(c3)Cl)OCC4CC4)c5cccnc5
FC(F)(F)CCOc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1ccccc1C#N
CCCOc1cc(cc(c1)Cl)C2=CC(=CN(C2=O)c3cccnc3)C4=CNC(=O)NC4=O
Clc1cc(OCC2CC2)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
c1cc(cnc1)N2C=C(C=C(C2=O)c3cc(cc(c3)Cl)OCCC(F)(F)F)C4=CNC(=O)NC4=O
Clc1cc(OCC2CCCC2)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1ccccc1C#N
Cc1ocnc1COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1ccccc1C#N
Cc1ocnc1COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
Cc1ncoc1COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
Clc1sccc1COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
Cc1c(ncs1)COc2cc(cc(c2)Cl)C3=CC(=CN(C3=O)c4cccnc4)C5=CNC(=O)NC5=O
FC(F)(F)c1ncoc1COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
FC(F)(F)c1ncsc1COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
Cn1cc(-c2cc(-c3cc(Cl)cc(OCC4CC4)c3)c(=O)n(c2)-c2cccnc2)c(=O)[nH]c1=O
Cn1cc(-c2cc(-c3cc(Cl)cc(OCCC(F)(F)F)c3)c(=O)n(c2)-c2cccnc2)c(=O)[nH]c1=O
c1ccc(c(c1)COc2cc(cc(c2F)Cl)C3=CC(=CN(C3=O)c4cccnc4)C5=CNC(=O)NC5=O)Cl
CN1C=C(C(=O)NC1=O)C2=CN(C(=O)C(=C2)c3cc(c(c(c3)Cl)F)OCc4ccccc4Cl)c5cccnc5
Cn1cc(-c2cc(-c3cc(Cl)cc(OCc4ocnc4C(F)(F)F)c3)c(=O)n(c2)-c2cccnc2)c(=O)[nH]c1=O
Cn1cc(-c2cc(-c3cc(Cl)cc(OCc4scnc4C(F)(F)F)c3)c(=O)n(c2)-c2cccnc2)c(=O)[nH]c1=O
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)OCc1ccccc1
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)OCc1ccccc1
COc1cc(cc(CO)c1OCC(=O)N1CCC(C1)Oc1cccc(c1)C(=O)N(C)C)-c1cccc2[nH]ncc12
COc1cc(cc(C=O)c1OCC(=O)N(C)C)-c1cccc2[nH]ncc12
CN(C)C(=O)COc1ccc(cc1C=O)-c1cccc2[nH]ncc12
CNCc1cc(cc(OC)c1OCC(=O)N(C)C)-c1cccc2[nH]ncc12
COC(=O)CN(C)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CN(Cc4c3cc(cc4)Cl)S(=O)(=O)CC5(CC5)C#N
Clc1ccc2CN(C[C@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Fc1ccc2c(NC(=O)[C@H]3CCS(=O)(=O)c4ccc(Cl)cc34)cncc2c1
CC(C)(O)c1ccc2cncc(NC(=O)C3CCNc4ccc(Cl)cc34)c2c1
Clc1ccc2OCCC(C(=O)Nc3cncc4ccc(CN5CC6(CNC6)C5)cc34)c2c1
Cc1nccn1Cc1ccc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2c1
CS(=O)(=O)c1ccc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2c1
Clc1ccc2OCCC(C(=O)Nc3cncc4cc(CN5CC6(CNC6)C5)ccc34)c2c1
Cc1c(N)cncc1NC(=O)C1CCOc2ccc(Cl)cc12
c1ccc2c(c1)cncc2N3CC[C@](C3=O)(c4cccc(c4)Cl)O
Clc1ccc2OCCC(C(=O)Nc3cncc4ccc(CN5CCNCC5)cc34)c2c1
O[C@@]1(CCN(C1=O)c1cncc2ccccc12)c1cccc(Cl)c1
Cc1cc(N)ncc1NC(=O)C1CCOc2ccc(Cl)cc12
Cc1ccnc(NC(=O)C2CCOc3ccc(Cl)cc23)c1N
Clc1cc2NCCC(C(=O)Nc3cnc4ccccn34)c2cc1Cl
Cc1cc(NC(=O)C2CCOc3ccc(Cl)cc23)ncc1N
Cc1ccnc(N)c1NC(=O)C1CCOc2ccc(Cl)cc12
CC1(CNC(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(cc12)S(C)(=O)=O
Clc1ccc2OCCC(C(=O)Nc3cnc4ccccn34)c2c1
Cn1ncc(NC(=O)C2CCOc3ccc(Cl)cc23)c1C(F)F
Clc1cccc(CC(=O)N2CC(=O)Cc3ccccc23)c1
CS(=O)(=O)c1ccc2cncc(NC(=O)C3CNC(=O)c4ccc(Cl)cc34)c2c1
Clc1ccc2C(=O)NCC(C(=O)Nc3cnc4ccccn34)c2c1
Cc1cc(O)ncc1NC(=O)C1CCOc2ccc(Cl)cc12
Clc1cccc(c1)C(NC(=O)[C@H]1CC[C@@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
FC(F)(F)c1ccc2cncc(NC(=O)C3CCOc4ccc(Cl)cc34)c2c1
Clc1cccc(c1)C(NC(=O)[C@@H]1CC[C@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)[C@H]1CC[C@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
CNC(=O)CN1CC(C(=O)Nc2cncc3ccc(cc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
Clc1ccc2c(c1)C1CCC2(O1)C(=O)Nc1cncc2ccccc12 |TLB:6:5:9.8:11,THB:3:4:9.8:11|
COC(=O)c1cc(\C=c2/s\c(=C(\C#N)C(=O)NC(C)C)n(-c3ccc(OC)c(F)c3)c2=O)oc1C
CC(C(=O)NS(=O)(=O)c1cnn(c1)-c1cccc(c1)C(F)(F)F)n1cnc(n1)C#N
COC(=O)c1cc(\C=c2/sc(=C(C#N)C#N)n(-c3cccc(c3)C(F)(F)F)c2=O)oc1C |(.52,-3.37,;.52,-4.91,;1.85,-5.68,;3.18,-4.91,;1.85,-7.22,;3.1,-8.12,;2.62,-9.59,;3.52,-10.84,;5.06,-10.67,;5.83,-9.34,;7.33,-9.66,;8.48,-8.63,;8.16,-7.12,;7.84,-5.62,;9.94,-9.11,;11.41,-9.58,;7.49,-11.19,;8.83,-11.96,;10.16,-11.19,;11.49,-11.96,;11.49,-13.5,;10.16,-14.27,;8.83,-13.5,;10.16,-15.81,;10.16,-17.35,;8.62,-15.81,;11.7,-15.81,;6.09,-11.82,;5.77,-13.32,;1.08,-9.59,;.6,-8.12,;-.86,-7.65,)|
CC1(CCS(=O)(=O)C1)n1cc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cn1
Clc1ccc2OCCC(CNCc3cnn(c3)C3CCS(=O)(=O)C3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CNCc3cnc4OCC(=O)Nc4c3)(C(=O)Nc3cncc4ccccc34)c2c1
COc1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1OCC(N)=O
OC1(CCN(C1=O)c1cncc2ccccc12)c1cccc(Cl)c1
COC(=O)[C@H]1CC[C@@H](CNC(C(=O)Nc2cncc3ccccc23)c2cccc(Cl)c2)O1
Clc1cc2nccc(C(=O)Nc3cncc4ccccc34)c2cc1Cl
CC(C(=O)OC1CCCN(Cc2cccc(c2)C(F)(F)F)C1=O)n1cnc(n1)C#N
FC(F)(F)c1ccnn1-c1cccc(c1)C(=O)NNC(=O)OCc1ccccc1
OC1CCCC1C(=O)NC[C@@H]1C[C@H](F)CN1C(=O)c1ccc([nH]1)C#N
Fc1ccc(cc1)S(=O)(=O)N1CCCN(CC1)C(=O)CCl
Clc1cccc(CC(=O)Nc2cncc3cnoc23)c1
OCc1ccc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2c1
COc1ccc2cncc(NC(=O)[C@]3(CCOc4ccc(Cl)cc34)OC)c2c1
CS(=O)(=O)N1C[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CS(=O)(=O)N1C[C@@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2OCCC(CNCc3cn(CC4CCCO4)nn3)(C(=O)Nc3cncc4ccccc34)c2c1
Cc1nc(CN2CC(C(=O)Nc3cncc4ccc(F)cc34)c3cc(Cl)ccc3C2)cs1
Clc1ccc2OCCC(CNCc3c(nc4ccccn4c3=O)N3CCOCC3)(C(=O)Nc3cncc4ccccc34)c2c1
CNC(=O)COc1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1OC
NC(=O)c1ccn(n1)-c1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cn1
NS(=O)(=O)c1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1F
Cn1cc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)n2ncc(C#N)c12
Clc1ccc2OCCC(NC(=O)C3CCC(O3)C(=O)N3CCCC3)(C(=O)Nc3cncc4ccccc34)c2c1
NS(=O)(=O)c1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1
CNS(=O)(=O)c1cc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)ccc1F
CN1CCN(C(=O)C1c1cccc(Cl)c1)c1cncc2ccccc12
Clc1ccc2OCCC(CNCc3ccc(cc3)N3CCNC(=O)C3)(C(=O)Nc3cncc4ccccc34)c2c1
Cn1ccc(CN2CC(C(=O)Nc3cncc4ccc(F)cc34)c3cc(Cl)ccc3C2)n1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cc(=O)[nH]c2ccccc12)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cc(=O)[nH]c2ccccc12)C(=O)c1c[nH]cn1
CN(C)S(=O)(=O)N1CC(C(=O)Nc2cnccc2C(F)(F)F)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CNC1)C#N
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)N1CCOCC1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)N1CCC1
COC1CN(C1)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)N1CC(C1)C#N
CN1CCN(CC1)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(Cc3ncn[nH]3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Cc1n[nH]c(CN2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)n1
COCc1csc(CNC(=O)c2ncc(Cl)cc2Cl)c1
NS(=O)(=O)c1cc(CN2CCN(CC2)C(c2ccccc2)c2ccccc2)co1
Cc1nc(C)c(s1)S(=O)(=O)NCC1CCCC2CC12
Cc1nc(sc1S(N)(=O)=O)N1CCN(CC1)S(=O)(=O)c1ccccc1
Cc1csc2ncc(C(=O)N3C4CCC3c3ccccc43)c(=O)n12 |TLB:16:15:10:12.13,19:20:10:12.13|
CCS(=O)(=O)c1c(Cl)cccc1CNC(C1CC1)c1cccc(F)c1
COCc1csc(c1)-c1nnc(o1)-c1sc(nc1C)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)NCC(=O)N1CCC(CC1)NS(N)(=O)=O
CCS(=O)(=O)c1cc(Cl)cc(CNS(=O)(=O)c2cccs2)c1
Cc1ccc(cc1)S(=O)(=O)NCCNC(=O)N1CCN(CC1)S(=O)(=O)N1CCCC1
COCc1ccccc1CNS(=O)(=O)c1c(C)sc(C)c1C
CN(C)S(=O)(=O)N1CCN(CC1)C(=O)C1Nc2ccccc2S(=O)(=O)N1
CCS(=O)(=O)c1ccc(CNS(=O)(=O)c2cnc(s2)-c2ccccc2)s1
Cc1nc2scc(C)n2c1CN1CCN(Cc2ccsc2)CC1
NS(=O)(=O)NCCNS(=O)(=O)c1ccccc1[N+]([O-])=O
COc1cc(OC)cc(c1)-c1nc(no1)-c1c(C)nc2sccn12
NS(=O)(=O)C1CN(CCNS(=O)(=O)c2ccccc2)c2ccccc2C1
CCN(CC)S(=O)(=O)c1ccc(cc1)S(=O)(=O)N1CCN(CC1)S(N)(=O)=O
CNc1cncc(NC(=O)C2CCOc3ccc(Cl)cc23)c1C
CN(C)c1cncc(NC(=O)C2CCOc3ccc(Cl)cc23)c1C
Nc1cncc(NC(=O)C2CCOc3ccc(Cl)cc23)c1C1CC1
CC(C)(C)OC(=O)NC(CCO)CNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
O[C@@H]1CCC[C@H]1S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2OCCC(CNCCN3C(=O)c4ccccc4C3=O)(C(=O)Nc3cncc4ccccc34)c2c1
Cn1nnc(CNC(=O)OC(C)(C)C)c1CNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Cn1cc(CN2CC(C(=O)Nc3cncc4ccc(F)cc34)c3cc(Cl)ccc3C2)nn1
COc1cc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc(OC)c1OCC(N)=O
Clc1ccc2OCCC(CNCc3cn(CC4CCOC4)nn3)(C(=O)Nc3cncc4ccccc34)c2c1
Cc1nn(C)c(N2CCOCC2)c1CNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(CNCc3cnc(nc3)N3CCOCC3)(C(=O)Nc3cncc4ccccc34)c2c1
COC(=O)c1cnc(Cn2ccc(CNCC3(CCOc4ccc(Cl)cc34)C(=O)Nc3cncc4ccccc34)n2)cn1
COC(=O)CCc1nocc1CNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2CN(CC#N)CC(C(=O)Nc3cncc4ccccc34)c2c1
Cc1nc(CN2CC(C(=O)Nc3cncc4ccc(F)cc34)c3cc(Cl)ccc3C2)c[nH]1
Fc1ccc2cncc(N3C(=O)NC4(COc5ccc(Cl)cc45)C3=O)c2c1
Cn1c(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)nc2n(C)c(=O)[nH]c(=O)c12
CO[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4
CO[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cc(cc4)F
Cc1cc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2s1
NC(=O)c1cc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2s1
CNC(=O)c1cc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2s1
Clc1cc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2s1
CS(=O)(=O)N1CC(C(=O)Nc2cncc3CCCCc23)c2cc(Cl)ccc2C1
Fc1ccc2c(NC(=O)C3CCS(=O)(=O)c4ccc(Cl)cc34)cncc2c1
Clc1ccc2c(c1)C(CCS2(=O)=O)C(=O)Nc1cncc2cc(Cl)ccc12
CS(=O)(=O)c1ccc2c(NC(=O)C3CCS(=O)(=O)c4ccc(Cl)cc34)cncc2c1
Cn1cc(cn1)N1CCC(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)C1
CN(CCO)c1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cn1
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(NS(C)(=O)=O)cc12
CNS(=O)(=O)c1ccc2cncc(NC(=O)C3(CCOc4ccc(Cl)cc34)OC)c2c1
Clc1ccc2OCC[C@]3(OC(=O)N(C3=O)c3cncc4ccccc34)c2c1
Clc1ccc2OCC[C@@]3(OC(=O)N(C3=O)c3cncc4ccccc34)c2c1
Fc1cc2OCC[C@H](C(=O)Nc3cncc4ccncc34)c2cc1Cl
CO[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(F)cc12
Fc1ccc2cncc(NC(=O)[C@H]3CCNc4cc(Cl)c(Cl)cc34)c2c1
COc1ccc2cncc(NC(=O)[C@H]3CCNc4cc(Cl)c(Cl)cc34)c2c1
Fc1ccc2cncc(NC(=O)[C@H]3CCOc4cc(F)c(Cl)cc34)c2c1
CN(C)C(=O)COCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)c(F)cc2C1
CS(=O)(=O)N1CC(C(=O)Nc2cncc3cccc(F)c23)c2cc(Cl)ccc2C1
Clc1ccc2C3CCC(O3)(C(=O)Nc3cncc4ccccc34)c2c1 |TLB:3:4:7.6:9,THB:24:23:7.6:9|
COC1(CCN(C1=O)c1cncc2ccccc12)c1cccc(Cl)c1
COC1(CCCN(C1=O)c1cncc2ccccc12)c1cccc(Cl)c1
Fc1cc2OCCC(C(=O)Nc3cncc4ccncc34)c2cc1Cl
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(F)cc12
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccncc12
CNS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CN(C)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)C1CC1
COCCS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
OCCS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CCS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)C1COC1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)C1CCOC1
CC1CCN(C1)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCC1)C#N
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1CNC1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)C1CNC1
OCC1CCCN1S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)C(=O)C1CC1
CN(C)C(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
OC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
COC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CNC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CN(C)C(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
NC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
FC(F)(F)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
COCCN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)c1ncc[nH]1
Cn1ncc(n1)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)C(=O)CC#N
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)C(=O)c1cnco1
Cn1nncc1C(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)C(=O)c1ncco1
Cc1nocc1C(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Cn1nccc1C(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Cn1cncc1C(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CS(=O)(=O)NCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CN(C)S(=O)(=O)NCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
COC(=O)NCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(CNC(=O)C=C)(C(=O)Nc3cncc4ccccc34)c2c1
CC(=O)NCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CN(C)C(=O)CNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
COc1ccc2cncc(NC(=O)C3(CCOc4ccc(Cl)cc34)OC)c2c1
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(cc12)S(C)(=O)=O
COc1ccc2cncc(NC(=O)C3CCOc4cc(F)c(Cl)cc34)c2c1
CS(=O)(=O)c1ccc2cncc(NC(=O)C3CCOc4cc(F)c(Cl)cc34)c2c1
Fc1ccc2cncc(NC(=O)C3CCOc4cc(F)c(Cl)cc34)c2c1
COc1ccc2cncc(NC(=O)C3CCNc4cc(Cl)c(Cl)cc34)c2c1
COC(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CCOC(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CN(C)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CNC(=O)COCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
OC(=O)CCc1cc2OCOc2cc1S(=O)(=O)N1CCN(CC1)c1ccccc1
CCCc1cc2OCOc2cc1S(=O)(=O)N1CCN(CC1)c1ncccn1
CCCc1cc2OCOc2cc1S(=O)(=O)N1CCN(CC1)c1cccc(Cl)c1Cl
CCCc1cc2OCOc2cc1S(=O)(=O)N1CCN(CC1)c1ccccc1OC
Cc1cc2OCOc2cc1S(=O)(=O)N1CCN(CC1)c1ccccc1
CNS(=O)(=O)c1cc2OCOc2cc1OCc1ccccc1
O=S(=O)(Nc1ccccc1)c1cc2OCOc2cc1OCc1ccccc1
O=S(=O)(Nc1cc2OCOc2cc1OCc1ccccc1)c1ccccc1
O=S(=O)(N1CCOCC1)c1cc2OCOc2cc1OCc1ccccc1
CO[C@@]1(CCOc2cc(F)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
CO[C@]1(CCOc2c1cc(c(c2)F)Cl)C(=O)Nc3cncc4c3cccc4
OC(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cc(=O)[nH]c2ccccc12)C(=O)c1cocn1
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CNCc4c3cc(cc4)Cl
Clc1ccc2CNC[C@H](C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc(OCc2ccccn2)c2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc(OCc2cccnc2)c2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc(OCc2ccncc2)c2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Cc1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
Cc1cccc2c(NC(=O)Cc3cccc(Cl)c3)cncc12
Clc1cccc(CC(=O)NC2C(=O)NCc3ccccc23)c1
Clc1cccc(CC(=O)Nc2cncc3cn[nH]c23)c1
Clc1cccc(CC(=O)Nc2cncc3[nH]ncc23)c1
Cn1c2c(cncc2NC(=O)Cc3cccc(c3)Cl)cn1
Clc1cccc(CC(=O)NC2COCc3ccccc23)c1
Clc1cccc(CC(=O)NC2CS(=O)(=O)Cc3ccccc23)c1
Clc1cccc(CC(=O)NC2=NC(=O)c3ccccc23)c1 |t:10|
CC1(C)Nc2ccccc2C1NC(=O)Cc1cccc(Cl)c1
Clc1cccc(CC(=O)Nc2noc3ncccc23)c1
COc1ccncc1NC(=O)Cc1cccc(Cl)c1
Clc1cccc(CC(=O)Nc2c[nH]c3ccccc23)c1
CC(C)(C)Oc1ccncc1NC(=O)Cc2cccc(c2)Cl
Clc1cccc(CC(=O)Nc2ncnc3ccccc23)c1
Clc1cccc(CC(=O)Nc2noc3ccccc23)c1
Clc1cccc(CC(=O)Nc2cnn3ccccc23)c1
Clc1cccc(CC(=O)Nc2cncc3nccnc23)c1
Fc1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
Fc1cccc2c(NC(=O)Cc3cccc(Cl)c3)cncc12
Clc1cccc(CC(=O)Nc2cncc3cc[nH]c23)c1
Clc1cccc(CC(=O)Nc2cncc3CCCNc23)c1
Oc1cnc2ccccc2c1NC(=O)Cc1cccc(Cl)c1
Clc1cccc(CC(=O)Nc2cncc3sccc23)c1
COc1ncc(NC(=O)Cc2cccc(Cl)c2)c2ccccc12
Clc1cccc(CC(=O)Nc2cnc(C#N)c3ccccc23)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1nnn[nH]1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1c[nH]cn1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)N1CCC(CC1)c1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccns1
Cc1cnnn1-c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccon1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccc(O)c(=O)o1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)N2CCCC2=O)c2cccnc2)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1coc(CS(C)(=O)=O)n1
CC(C)(C)c1cnc(o1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CN1CCCN(C1=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1cc(no1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(O)cc(=O)o1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccnc(n1)N1CCOCC1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccno1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nnn[nH]1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cscn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnsn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnon1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2cnn(c2)-c2ccccc2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)C2CC(=O)NC(=O)C2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)N2CCCS2(=O)=O)c2cccnc2)c1
Cc1nnn(n1)-c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)C2CCC(=O)N2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)-n2cc[nH]c2=O)c2cccnc2)c1
CC(C)(c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1)S(C)(=O)=O
CC(C)(O)c1cccc(c1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)-c2nnc3CCCn23)c2cccnc2)c1
FC(F)(F)CN1CCOCC1C(=O)NCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CO[C@@]1(CCOc2c(F)cc(F)cc12)C(=O)Nc1cncc2ccccc12
CO[C@]1(CCOc2c1cc(cc2F)F)C(=O)Nc3cncc4c3cccc4
COC[C@@]1(CCOc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
COC[C@]1(CCOc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
CCC(CC)COC(=O)[C@H](C)NP(=O)(OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1
CC(C)C(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc\c(=N\O)[nH]c1=O
Clc1ccc2C(CCOc2c1)C(=O)N(Cc1c[nH]c(=O)[nH]c1=O)c1cncc2ccccc12
Clc1ccc2c(OCCC2(CNc2c[nH]c(=O)[nH]c2=O)C(=O)Nc2cncc3ccccc23)c1
Clc1cc2NCCC(C(=O)Nc3cnccc3C3CC3)c2cc1Cl
Clc1cc2NCCC(C(=O)Nc3cncc4CCCCc34)c2cc1Cl
Clc1cc2NCCC(C(=O)Nc3cncc4cnccc34)c2cc1Cl
Clc1cc2NCCC(C(=O)Nc3cncc4ccncc34)c2cc1Cl
CS(=O)(=O)c1ccc2cncc(NC(=O)C3CCNc4cc(Cl)c(Cl)cc34)c2c1
Fc1ccc2cncc(NC(=O)C3CCNc4cc(Cl)c(Cl)cc34)c2c1
Clc1cccc(c1)C(NC(=O)COCC(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC[C@@H]1CC[C@@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)[C@@H]1CCCO1)C(=O)Nc1cncc2ccccc12
CC(=O)NC(C(=O)Nc1cncc2ccccc12)c1cccc(Cl)c1
CN(C)C(=O)COCC(=O)NC(C(=O)Nc1cncc2ccccc12)c1cccc(Cl)c1
Clc1cccc2C(COCc12)C(=O)Nc1cncc2ccccc12
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)CCC#N
CC(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
NC(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CNC(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2OCCC3(OC(=O)N(C3=O)c3cncc4ccccc34)c2c1
c1cc2cncc(c2cc1F)NC(=O)[C@@H]3CCNc4c3cc(c(c4)Cl)Cl
c1cc2cncc(c2cc1F)NC(=O)[C@@H]3CCOc4c3cc(c(c4)F)Cl
COc1ccc2cncc(NC(=O)[C@@]3(CCOc4ccc(Cl)cc34)OC)c2c1
COc1ccc2cncc(NC(=O)[C@@H]3CCNc4cc(Cl)c(Cl)cc34)c2c1
Fc1cc2OCC[C@@H](C(=O)Nc3cncc4ccncc34)c2cc1Cl
Cc1nc2CCC(Cn2n1)C(=O)NC(C(=O)Nc1cncc2ccccc12)c1cccc(Cl)c1
Fc1cc2OCC[C@H](C(=O)Nc3cncc4ccccc34)c2cc1Cl
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(c(c4)F)Cl
Clc1cccc(c1)C(NC(=O)[C@@H]1CC[C@@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
CS(=O)(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
FC(F)(F)CCOc1cc(Cl)cc2C(CCOc12)C(=O)Nc1cncc2ccccc12
CCCOc1cc(Cl)cc2C(CCOc12)C(=O)Nc1cncc2ccccc12
Clc1cc(OCC2CC2)c2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc(OCc2ccccc2)c2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
CCc1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cccc3
FC(F)(F)Oc1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
CCCc1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
CC(C)(C)c1ccc(cc1)N([C@@H](C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)C=C
CCOC(=O)C1OC1C(=O)N(CCC(N)=O)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)CCCC#C)C(C)(C)C
COC(=O)\C=C\C(=O)N(CCC(N)=O)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)CCCC#C)C(C)(C)C
CC(C)C[C@@H](NC(=O)[C@@H](NC(=O)CCCC#C)C(C)(C)C)C(=O)NN(CCC(N)=O)C(=O)CCl
CC[C@H](NC(=O)CCCC#C)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)COC(=O)c1c(C)cccc1C)C(C)(C)C
CC[C@H](NC(=O)CCCC#C)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)COC(=O)c1c(C)cccc1C)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)N1CCOCC1)c1cccnc1)C(=O)c1ccco1
N[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Cc1ccncc1C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
Cc1cc(O)c(C(N(C(=O)c2cocn2)c2ccc(cc2)C(C)(C)C)C(=O)NCCc2cccc(F)c2)c(=O)[nH]1
Cn1cc(ccc1=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
COc1nc2ncc(cn2n1)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1ccnnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1ccc[nH]c1=O)C(=O)c1cocn1
Cn1cccc(C(N(C(=O)c2cocn2)c2ccc(cc2)C(C)(C)C)C(=O)NCCc2cccc(F)c2)c1=O
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cnc(nc1)N1CCOCC1)C(=O)c1cocn1
CN(C)c1ncc(cn1)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
COc1nccnc1C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cncnc1)C(=O)c1cocn1
COc1ncncc1C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cnccn1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1c(nc2ccccn2c1=O)N1CCOCC1)C(=O)c1cocn1
CN1CCN(CC1)c1ncc(cn1)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
Clc1ccc2SCCC(C(=O)Nc3cncc4ccccc34)c2c1
CNC(=O)C1(CC(=O)Nc2cncc3ccccc23)CCOc2ccc(Cl)cc12
COC(OC)C(=O)N1CCN(Cc2cccc(Cl)c2)CC1
Clc1cccc(CN2CCN(CC2)C(=O)C=O)c1
CC(C)C[C@H]1CN(CCN1Cc1cccc(Cl)c1)C(=O)C(C)=O
CC(C)C[C@H]1CN(CCN1Cc1cccc(Cl)c1)C(=O)CCl
COc1cc(Cl)nc(Nc2cc(Cl)cc(CC(=O)Nc3cncc4ccccc34)c2)n1
FC(F)(F)c1ccc(Nc2cc(Cl)cc(CC(=O)Nc3cncc4ccccc34)c2)nc1
COc1cc(Br)ccc1Nc1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
CCN(Cc1ccc(F)cc1)c1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
Cc1ccc2nc(Nc3cc(Cl)cc(CC(=O)Nc4cncc5ccccc45)c3)sc2c1
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)N4CCN(CC4)C(=O)c5ccco5
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(NCc2ccc(Br)cc2)c1
CN(Cc1cccc2ccccc12)c1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
CCS(=O)(=O)N1CCN(CC1)c2cc(cc(c2)Cl)CC(=O)Nc3cncc4c3cccc4
COc1ncc(Br)cc1Nc1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
Clc1ccc2CCNC(C(=O)Nc3cncc4ccccc34)c2c1
CN1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(CNC(=O)Cn3ccnc3)(C(=O)Nc3cncc4ccccc34)c2c1
CN(C)CC(=O)NCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
COCC1(CCOc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
COC1(CCOc2c(F)cc(F)cc12)C(=O)Nc1cncc2ccccc12
Clc1cc(C#N)c2NCCC(C(=O)Nc3cncc4ccccc34)c2c1
COC1(CCOc2cc(F)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1cc2NC(=O)CC(C(=O)Nc3cncc4ccccc34)c2cc1Cl
OCCN1CCCC2C1CCN2C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(CC(=O)N3CCN(CCC#N)CC3)(C(=O)Nc3cncc4ccccc34)c2c1
OCCCN1CCN(CC1)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
OCC(F)(F)CN1CCN(CC1)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
NS(=O)(=O)c1ccc(CNC(=O)CC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1
COCCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1cccnc1)c1cccnc1)C(=O)c1cocn1
COC(=O)C(C)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COC(=O)[C@@H]1CC[C@@H](C1)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1ccncc1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCOCC1)c1cccnc1)C(=O)c1cocn1
CN(C)C(=O)CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)OC(=O)NCCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COC(=O)C1CC(C1)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1 |(-.94,.5,;-.17,-.84,;1.37,-.84,;2.14,.5,;2.14,-2.17,;3.63,-2.57,;3.23,-4.06,;1.74,-3.66,;4,-5.39,;5.54,-5.39,;6.31,-4.06,;6.31,-6.72,;7.85,-6.72,;8.62,-5.39,;7.85,-4.06,;10.16,-5.39,;11.07,-4.14,;12.53,-4.62,;12.53,-6.16,;11.07,-6.64,;8.62,-8.06,;10.16,-8.06,;10.93,-9.39,;10.16,-10.72,;8.62,-10.72,;7.85,-9.39,;10.93,-12.06,;11.7,-13.39,;9.6,-12.83,;12.26,-11.29,;5.54,-8.06,;6.31,-9.39,;5.54,-10.72,;4,-10.72,;3.23,-9.39,;4,-8.06,)|
CSCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CCOC(=O)CCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)OC(=O)NCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCC(=O)Nc1cccc(c1)[N+]([O-])=O)c1cccnc1)C(=O)c1cocn1
COC(=O)[C@@H]1C[C@H](CN1C(=O)OC(C)(C)C)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COC(=O)[C@H]1C[C@@H](CN1C(=O)OC(C)(C)C)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)OC(=O)N1CCC(C1)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCC1CCOC1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCC1CCCO1)c1cccnc1)C(=O)c1cocn1
COC(CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1)OC
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCOC1)c1cccnc1)C(=O)c1cocn1
COCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CCOC(=O)CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COC(=O)CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1COC1)c1cccnc1)C(=O)c1cocn1
COC(=O)C1(CCCC1)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COC(=O)[C@H]1C[C@H](CN1C(=O)OC(C)(C)C)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)OC(=O)CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CC(F)(F)C1)c1cccnc1)C(=O)c1cocn1
COC(=O)[C@@H]1C[C@@H](CN1C(=O)OC(C)(C)C)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COc1ccc(NC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)C(C)(C)C)c2cccnc2)cn1
Cc1ccc(cc1)S(=O)(=O)CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)OC(=O)N1CC(C1)NC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCC(=O)OCc1ccccc1)c1cccnc1)C(=O)c1cocn1
CSCCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCN1CCOCC1)c1cccnc1)C(=O)c1cocn1
CCOC(=O)CCCNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CCOC(=O)c1ncoc1CNC(=O)C(N(C(=O)c1cocn1)c1ccc(cc1)C(C)(C)C)c1cccnc1
COCCCNCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Cn1ccc(CNCC2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)n1
Cn1c(=O)ccn(CC(=O)NC(C(=O)Nc2cncc3ccccc23)c2cccc(Cl)c2)c1=O
Cn1ncc2c1ncn(CC(=O)NC(C(=O)Nc1cncc3ccccc13)c1cccc(Cl)c1)c2=O
CC(NC(=O)C1CCC1)C(=O)NC(C(=O)Nc1cncc2ccccc12)c1cccc(Cl)c1
Clc1cccc(c1)C(NC(=O)CNC(=O)c1ccc(cc1)C#N)C(=O)Nc1cncc2ccccc12
Cn1cc(cn1)C1=NOC(C1)C(=O)NC(C(=O)Nc1cncc2ccccc12)c1cccc(Cl)c1 |t:7|
Clc1cccc(c1)C(NC(=O)Cn1cc(C#N)c(=O)[nH]c1=O)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)Cn1nnc(n1)-c1ccccc1)C(=O)Nc1cncc2ccccc12
FC(F)(F)c1ncn(CC(=O)NC(C(=O)Nc2cncc3ccccc23)c2cccc(Cl)c2)n1
NC(=O)c1ccc(OCC(=O)NC(C(=O)Nc2cncc3ccccc23)c2cccc(Cl)c2)cc1
Clc1cccc(c1)C(NC(=O)Cn1nc2CCCn2c(=O)c1=O)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)Cc1ccc(cc1)-n1cnnn1)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)Cn1cc(Cl)c(=O)[nH]c1=O)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)Cn1ncn2nccc2c1=O)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)C(NC(=O)CN1CCN(C2CC2)C1=O)C(=O)Nc1cncc2ccccc12
O[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
OCC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
COC(=O)\C=C\C(=O)N(C(=O)[C@H]1CCOc2ccc(Cl)cc12)c1cncc2ccccc12
Clc1ccc2OCCC(CC(=O)N3CCCCC3c3nc[nH]n3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CC(=O)N3CCCCC3c3cc[nH]n3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CC(=O)N3CCCCC3c3cn[nH]c3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CC(=O)N3CCCC3c3nnn[nH]3)(C(=O)Nc3cncc4ccccc34)c2c1
CN1C[C@@H]2C[C@H]1CN2C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12 |THB:0:1:4:6.7,8:7:1.2:4|
CC1CN(C)CCN1C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Cn1cncc1CN(C1CC1)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Cn1ccnc1CN(C1CC1)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CC1Cn2nccc2CN1C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CC1N(CCn2cnnc12)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
FC(F)CC1COCCN1C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(CC(=O)N3CCCC3Cn3ccnc3)(C(=O)Nc3cncc4ccccc34)c2c1
NC(=O)C1Cc2[nH]cnc2CN1C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
FC(F)CN1C[C@@H]2C[C@H]1CN2C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12 |TLB:11:10:7:5.4,3:4:10.9:7|
CC1CN(CCN1CCO)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CC1CN(CCO)CCN1C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CN(CCO)C1CCN(CC1)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CC(=O)N5CCN(CC5)CCCO
CN1C(=O)CCc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C2CC3CCCC3C2)C(=O)c2cocn2)c2cccnc2)c1
Fc1ccc2C(CCc2c1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C2COc3ccccc3C2)C(=O)c2cocn2)c2cccnc2)c1
CC(C)S(=O)(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
COC1CC2(C1)CC(C2)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1 |(-8.11,12.44,;-6.59,12.73,;-5.59,11.57,;-4.05,11.46,;-4.16,9.92,;-5.7,10.03,;-2.62,9.81,;-2.73,8.28,;-4.27,8.39,;-1.73,7.11,;-.21,7.4,;.79,6.24,;.29,4.78,;2.31,6.53,;3.31,5.37,;4.83,5.66,;5.84,4.49,;7.35,4.78,;8.36,3.62,;7.85,2.16,;6.34,1.87,;5.84,.42,;5.33,3.04,;.29,8.86,;-.72,10.02,;-.21,11.48,;1.3,11.77,;2.31,10.6,;1.8,9.15,;-2.23,5.66,;-1.22,4.49,;-3.74,5.37,;-4.4,3.97,;-5.92,4.16,;-6.22,5.67,;-4.87,6.42,)|
Cn1ncc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CS(=O)(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Cn1cnc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CS(=O)(=O)Cc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC(C)Oc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C2CCCCC2)C(=O)c2cocn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCCOC2)C(=O)c2cocn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(Cn3cccn3)cc2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)S(=O)(=O)C2CCCC2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc3nc([nH]c3c2)C(F)(F)F)c2cccnc2)c1
COc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Cn1ccc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Cc1nc2ccc(cc2o1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C2CCCCCC2)C(=O)c2cocn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCc3ccccc23)C(=O)c2cocn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc3ncsc3c2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc3c(CCCS3(=O)=O)c2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCN(C2)c2ccccc2F)C(=O)c2cocn2)c2cccnc2)c1
Cc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccccc2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2Cc3ccccc23)C(=O)c2cocn2)c2cccnc2)c1
FC(F)CN1C(=O)CCc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C2CCN(C2)c2ccccc2)C(=O)c2cocn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(OC3CCOC3)cc2)c2cccnc2)c1
Fc1ccc2C(COc2c1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
COCc1csc(n1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2cn(Cc3ccccc3)cn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc3scnc3c2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(nc2)C(F)(F)F)c2cccnc2)c1
COc1ccccc1CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Cc1ccccc1CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CN1CCCC(C1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc3COCCc3c2)c2cccnc2)c1
COc1cc(C)ccc1CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CCOc1ccc(cn1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
COc1cc(ccc1S(=O)(=O)N(C)C)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N([C@H]2C[C@@H](C2)Oc2ccccc2)C(=O)c2cocn2)c2cccnc2)c1 |r,wU:13.12,wD:15.17,(-6.9,-5.86,;-7.4,-7.32,;-8.91,-7.61,;-9.42,-9.06,;-8.41,-10.23,;-6.9,-9.93,;-5.89,-11.1,;-4.37,-10.81,;-3.37,-11.97,;-1.85,-11.68,;-1.35,-10.23,;-.85,-12.85,;.67,-12.55,;1.67,-13.72,;3.21,-13.83,;3.1,-15.36,;1.56,-15.25,;4.11,-16.53,;5.62,-16.24,;6.12,-14.78,;7.64,-14.49,;8.64,-15.66,;8.14,-17.11,;6.63,-17.4,;1.17,-11.1,;.16,-9.93,;2.68,-10.81,;3.34,-9.41,;4.86,-9.6,;5.15,-11.12,;3.81,-11.86,;-1.35,-14.3,;-.34,-15.46,;-.85,-16.92,;-2.36,-17.21,;-3.37,-16.05,;-2.86,-14.59,;-6.39,-8.48,)|
Fc1cccc(CCNC(=O)C(N(C2CCC3(CCO3)CC2)C(=O)c2cocn2)c2cccnc2)c1 |(10.44,.99,;9.93,-.47,;8.42,-.76,;7.92,-2.21,;8.93,-3.38,;10.44,-3.08,;11.45,-4.25,;12.96,-3.96,;13.97,-5.12,;15.48,-4.83,;15.98,-3.38,;16.49,-6,;18,-5.7,;19.01,-6.87,;20.52,-6.58,;21.53,-7.74,;21.02,-9.2,;22.56,-9.31,;22.45,-10.84,;20.91,-10.73,;19.51,-9.49,;18.5,-8.32,;18.5,-4.25,;17.5,-3.08,;20.02,-3.96,;20.67,-2.56,;22.2,-2.75,;22.49,-4.27,;21.14,-5.01,;15.98,-7.45,;16.99,-8.61,;16.49,-10.07,;14.98,-10.36,;13.97,-9.2,;14.47,-7.74,;10.94,-1.63,)|
Fc1cccc(CCNC(=O)C(N(C2COC3(CCCC3)C2)C(=O)c2cocn2)c2cccnc2)c1
CC(N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1)c1ccccc1C
Fc1cccc(CCNC(=O)C(N(C2CCC3OCCC3C2)C(=O)c2cocn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2cnc(nc2)C2CCC2)c2cccnc2)c1
CCOc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC1CN(CCC1NC(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12)S(C)(=O)=O
Cn1nnnc1C1=CCN(CC1)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12 |t:7|
Clc1ccc2OCCC(CC(=O)N3CCN(CC3)C3CCOC3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCC[C@](CC(=O)N3CCN(CC3)C3CCOC3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc(Cl)c2NC(=O)CC(C(=O)Nc3cncc4ccccc34)c2c1
CN1C(=O)CC(O)(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
CN(C)C(=O)C[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CN(C)C(=O)C[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4
CNC(=O)C[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CNC(=O)C[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4
COc1ccc2cncc(NC(=O)C3CCOc4ccc(Cl)cc34)c2c1
Clc1cc2NCC[C@@H](C(=O)Nc3cncc4ccccc34)c2cc1Cl
Clc1cc2NCC[C@H](C(=O)Nc3cncc4ccccc34)c2cc1Cl
Clc1ccc2OCC[C@@](CC(=O)N3CCN(CC3)C3CCOC3)(C(=O)Nc3cncc4ccccc34)c2c1
c1cc2cncc(c2cc1F)NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl
Fc1ccc2cncc(NC(=O)[C@H]3CCOc4ccc(Cl)cc34)c2c1
CC(=O)N1CC[C@H](c2c1ccc(c2)Cl)C(=O)Nc3cncc4c3cccc4
CC(=O)N1CC[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
CN1CC[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
CN1CC[C@H](c2c1ccc(c2)Cl)C(=O)Nc3cncc4c3cccc4
c1ccc2c(c1)cncc2N3CC[C@@H](C3=O)c4cccc(c4)Cl
c1ccc2c(c1)cncc2N3CC[C@H](C3=O)c4cccc(c4)Cl
Clc1ccc2OCC[C@@]3(NC(=O)N(C3=O)c3cncc4ccccc34)c2c1
CC1(C(=O)Nc2cncc3ccccc23)C(=O)Nc2ccc(Cl)cc12
CO[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CO[C@@]1(CCOc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
CO[C@]1(CCOc2c1cc(c(c2)Cl)Cl)C(=O)Nc3cncc4c3cccc4
COC1(CCOc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
c1cc(c(cc1CC(=O)Nc2cncc3c2ccnc3)Cl)Cl
Clc1ccc(CC(=O)Nc2cncc3ccncc23)cc1Cl
CC1(CNc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCC(C(=O)N(C(=O)C=C)c3cncc4ccccc34)c2c1
Cn1c2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2[nH]c1=O
Clc1ccc2OCCC(C(=O)Nc3cncc4[nH]c(=O)[nH]c34)c2c1
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2NCCC3(CCCN(C3=O)c3cncc4ccccc34)c2c1
NC(=O)C12CC(CNC(=O)CC3(CCOc4ccc(Cl)cc34)C(=O)Nc3cncc4ccccc34)(C1)OC2
CC(=O)N1CC2CC1CN2C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12 |THB:1:3:6:8.9,10:9:3.4:6|
Clc1ccc2OCCC(CC(=O)N3CCC4CS(=O)(=O)CC4C3)(C(=O)Nc3cncc4ccccc34)c2c1
NC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CN(C)C(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(=O)NC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
Clc1ccc(cc1Cl)C(NCC1CC1)C(=O)Nc1cncc2ccccc12
Clc1ccc(cc1Cl)C1NC(=O)N(C1=O)c1cncc2ccccc12
CC(C)N1CCOC(C1)C(=O)NC(C)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(NC(=O)C1CCC(=O)NC1)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
Cn1nc(cc1C#N)C(=O)NC(C)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(NC(=O)c1cc2OCCn2n1)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(NC(=O)CN1CCN(C2CC2)C1=O)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(NC(=O)Cc1ccc(cc1)-n1cnnn1)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
Cc1nc2CCC(Cn2n1)C(=O)NC(C)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(NC(=O)COc1ccc(cc1)C(N)=O)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CC(NC(=O)CN)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
COCC(=O)NC(C)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CN1CCC(C1)C(=O)NC(C)(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
COC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
COCCOC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
Clc1ccc2OCCC(COCC(=O)Nc3ncc[nH]3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CC(=O)Nc3nnco3)(C(=O)Nc3cncc4ccccc34)c2c1
C[C@]1(CCNc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
C[C@@]1(CCNc2cc(Cl)c(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(C(=O)N(C(=O)C=C)c3cncc4ccccc34)c2c1
CCOc1c(Cl)cccc1CC(=O)Nc1cncc2ccccc12
Clc1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
CC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
OC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
CNC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
c1ccc2c(c1)cncc2NC(=O)C(c3ccc(c(c3)Cl)Cl)(F)F
Clc1ccc(cc1Cl)C(C#N)C(=O)Nc1cncc2ccccc12
OCC(C(=O)Nc1cncc2ccccc12)c1ccc(Cl)c(Cl)c1
c1ccc2c(c1)cncc2NC(=O)[C@]3(CCOc4c3cc(cc4)Cl)CN
Cn1cnc2cncc(NC(=O)C3CCOc4ccc(Cl)cc34)c12
OCC(F)(F)CN1CCN(CC1)C(=O)C[C@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CC(=O)C(=O)N1CCN(Cc2cccc(Cl)c2)CC1
OC(=O)c1ccncc1NC(=O)Cc1cccc(Cl)c1
OC(=O)c1ccncc1NC(=O)Cc1cccc(c1)C(F)(F)F
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2ccc(Cl)cc2)c2cccnc2)c1
CN(C)C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CNC(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Fc1cc2OCCC(C(=O)Nc3cncc4ccccc34)c2cc1Cl
c1ccc(cc1)CC(=O)Nc2cncc3c2cccc3
Clc1ccc(CC(=O)Nc2cncc3ccccc23)cc1
Cc1ccc(CC(=O)Nc2cncc3ccccc23)cc1
COc1ccc(CC(=O)Nc2cncc3ccccc23)cc1
O=C(Cc1ccc(cc1)C#N)Nc1cncc2ccccc12
c1ccc2c(c1)cncc2NC(=O)Cc3ccc(c(c3)Cl)F
c1ccc2c(c1)cncc2NC(=O)Cc3ccc(cc3)F
Cc1ccc(CC(=O)Nc2cncc3ccccc23)cc1Cl
Fc1cc(CC(=O)Nc2cncc3ccccc23)ccc1Cl
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)F
COc1cccc(CC(=O)Nc2cncc3ccccc23)c1
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)C#N
Cc1cccc(c1)CC(=O)Nc2cncc3c2cccc3
Fc1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)F)F
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cc(c3)Cl)C#N
Fc1c(Cl)cccc1CC(=O)Nc1cncc2ccccc12
Fc1cccc(CC(=O)Nc2cncc3ccccc23)c1F
c1ccc2c(c1)cncc2NC(=O)Cc3cc(ccc3F)F
c1ccc2c(c1)cncc2NC(=O)Cc3cc(cnc3)Cl
FC(F)(F)c1cccc(CC(=O)Nc2cncc3ccccc23)c1
FC(F)(F)c1ccc(CC(=O)Nc2cncc3ccccc23)cc1
c1ccc2c(c1)cncc2NC(=O)Cc3ccc(cn3)Cl
Clc1cnccc1CC(=O)Nc1cncc2ccccc12
Clc1ccccc1CC(=O)Nc1cncc2ccccc12
Fc1ccccc1CC(=O)Nc1cncc2ccccc12
Cc1ccccc1CC(=O)Nc1cncc2ccccc12
COc1ccccc1CC(=O)Nc1cncc2ccccc12
Clc1ccc(cc1Cl)C1CCCN(C1=O)c1cncc2ccccc12
Clc1cc(Cl)c2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc2NCCC(C(=O)Nc3cncc4ccccc34)c2cc1Cl
OC1(CC(=O)Nc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1cc2OCCC(C(=O)Nc3cncc4ccccc34)c2cc1Cl
Clc1ccc2C(CCOc2c1Cl)C(=O)Nc1cncc2ccccc12
CN(C)c1ccc(nc1)N(Cc2cccc(c2)Cl)C(=O)Cc3cncc4c3cccc4
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(on1)C1(O)COC1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]c(=O)s1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1scnc1Cl
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc(o1)C(C)(C)CF
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nc2CCCc2s1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nc(=O)[nH][nH]1
Cc1nc(oc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C)C1CC1
Cc1nc(nn1-c1nnc[nH]1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CN1CCn2nc(cc2S1(=O)=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cn(CCN2CCOCC2)nn1
Cn1cnc(cc1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1c2nc(ccc2c(=O)[nH]c1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]nn1
CCc1nc(sc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C)-c1nnc[nH]1
CC(O)Cc1c([nH][nH]c1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nc2cnccc2s1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(=O)c2c(O)cccc2o1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ocnc1C(F)(F)F
CCOC(=O)Cn1cc(nn1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1sc(nc1Cl)N1CCOCC1
COc1cc(sn1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1c(cc2c1n(C)c(=O)n(C)c2=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1nc2CCS(=O)(=O)Cc2c1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1nc(cc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C)C(=O)N1CCOCC1
Cn1nncc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccc(=O)[nH]n1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc(s1)C1CCOC1
Cn1cc(cn1)-c1cc(on1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(=O)n2ncnc2[nH]1
Cc1cn2nnc(C(=O)N(C(C(=O)NCCc3cccc(F)c3)c3cccnc3)c3ccc(cc3)C(C)(C)C)c2c(=O)[nH]1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]c(=O)cn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nc2ncc(CCO)cn2n1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1n[nH]c(=O)[nH]c1=O
COCc1nc(C)c(s1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cn(nn1)C1COCC1=O
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(CO)[nH]n1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(=O)[nH]c(=O)[nH]1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nnc(O)cc1O
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cncs1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nnc(S)[nH]c1=O
CO[C@@H]1COC[C@H]1n1cc(nn1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cc1cnoc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
COc1c([nH]c(=O)[nH]c1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1ncc(n1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnco1
Cn1cc(ncc1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1[nH]nc(O)c1CCO
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]c(=O)[nH]1
COCCn1nc(ccc1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1cnc(n1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cn1cc(C(=O)N(C(C(=O)NCCc2cccc(F)c2)c2cccnc2)c2ccc(cc2)C(C)(C)C)n(C)c1=O
Cn1c(c[nH]c1=O)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nc(CN2CCOCC2)cs1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(=O)[nH][nH]1
CC(=O)N1CCN(CC1)CC(=O)Nc2cnccc2C3CC3
CC(=O)N1CCN(CC(=O)Nc2cnccc2-c2ccccc2)CC1
Cc1ccncc1NC(=O)CN2CCC(CC2)C
c1ccc2c(c1)cncc2NC(=O)[C@@H]3COc4c3cc(cc4)Cl
Clc1ccc2OC[C@H](C(=O)Nc3cncc4ccccc34)c2c1
NS(=O)(=O)c1[nH]ncc1C(=O)NC[C@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
O[C@]1(CCSC1)C(=O)NC[C@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
O=C(NCc1cccs1)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
O=C(N1CCC(CC1)C1CCNC1)c1cccc(CN2CCCC2=O)c1
Cc1ccc(Nc2ccccc2C(=O)N2CCC(CC2)C2CCNC2)cc1
CS(=O)(=O)Nc1ccc(Cl)cc1C(=O)N1CCC(CC1)C1CCNC1
O=C(N1CCC(CC1)C1CCNC1)c1ccc2NC(=O)CCc2c1
CN(C)S(=O)(=O)c1cc(cc(C)c1C)C(=O)N1CCC(CC1)C1CCNC1
Cc1c(cccc1-c1ccccn1)C(=O)N1CCC(CC1)C1CCNC1
CCCOc1c(Cl)cc(cc1OCC)C(=O)N1CCC(CC1)C1CCNC1
CC(C)OCc1cc(ccc1F)C(=O)N1CCC(CC1)C1CCNC1
O=C(N1CCC(CC1)C1CCNC1)c1cccc(c1)N1CCCNC1=O
CN1CCN(CC1)c1ccc(F)cc1C(=O)N1CCC(CC1)C1CCNC1
Cc1cc(cc(C)c1OC(F)F)C(=O)N1CCC(CC1)C1CCNC1
CS(=O)(=O)c1ccccc1C(=O)N1CCC(CC1)C1CCNC1
CCc1ccc(cc1C(=O)N1CCC(CC1)C1CCNC1)S(C)(=O)=O
FC(F)c1nc2cc(ccc2[nH]1)C(=O)N1CCC(CC1)C1CCNC1
O=C(Nc1ccccc1)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
Clc1ccc(NC(=O)[C@H](N2Cc3ccccc3C2=O)c2ccccc2)cc1
Cc1cccc(NC(=O)[C@H](N2Cc3ccccc3C2=O)c2ccccc2)n1
O=C(Nc1ccncc1)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
Fc1ccc(NC(=O)[C@H](N2Cc3ccccc3C2=O)c2ccccc2)cc1
COCCNC(=O)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
O=C(NCCc1ccccc1)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
O=C(Nc1ccccc1C#N)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
Fc1cccc(NC(=O)[C@H](N2Cc3ccccc3C2=O)c2ccccc2)c1
O=C(Nc1cccnc1)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
CNCC1CCCN(C1)C(=O)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
CN(C)C(=O)C(CNC(=O)[C@H](N1Cc2ccccc2C1=O)c1ccccc1)c1ccccc1
FC(F)(F)c1cccc(Cc2nc3cnccc3c(=O)[nH]2)c1
FS(F)(F)(F)(F)c1cccc(Cc2nc3cnccc3c(=O)[nH]2)c1
CC(C(N)=O)c1cc(Cl)cc(CC(=O)Nc2cncc3ccccc23)c1
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(c1)-c1nnn[nH]1
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCNc4c3cc(cc4)Cl
Clc1ccc2NCC[C@H](C(=O)Nc3cncc4ccccc34)c2c1
Fc1cccc(CCNC(=O)C(N(C2CCN(C2)c2ccccc2F)C(=O)c2cnc[nH]2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCN(C2)c2ccccc2)C(=O)c2cnc[nH]2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc(OC3CCOC3)cc2)c2cccnc2)c1
CC(N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1)c1ccccc1
CC(N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1)c1ccccc1C
Fc1cccc(CCNC(=O)C(N(C2CCCC3(CCC3)C2)C(=O)c2cnc[nH]2)c2cccnc2)c1
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)O
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)N
c1ccc2c(c1)cncc2NC(=O)[C@@]3(CCOc4c3cc(cc4)Cl)CN
Oc1cc(Cl)cc2C(CCOc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCC[C@H](C(=O)Nc3cncc4cnccc34)c2c1
Clc1ccc2OCC[C@H](C(=O)Nc3cncc4ccncc34)c2c1
[O-][n+]1cc(NC(=O)[C@H]2CCOc3ccc(Cl)cc23)c2ccccc2c1
Clc1ccc(cc1)C1CCCN(C1=O)c1cncc2ccccc12
Clc1ccc2OCCC3(NC(=O)N(C3=O)c3cncc4ccccc34)c2c1
COc1ccccc1OCCNC(=O)c1cc(=O)cc[nH]1
Clc1cccc(c1)N1CCN(CC1)C(=O)c1cc(=O)cc[nH]1
Clc1ccc(CC(=O)Nc2cncc3ccccc23)cc1Cl
Clc1cccc(c1)N1CCN(CC1)C(=O)C1CC(=O)Nc2ccccc12
COc1ccccc1OCCNC(=O)c1cc(=O)ccn1C
COC(=O)\C=C\C(=O)N(C(=O)[C@@H]1CCOc2ccc(Cl)cc12)c1cncc2ccccc12
Fc1ccc2cncc(NC(=O)C3CCOc4ccc(Cl)cc34)c2c1
CCN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Fc1cccc(CCNC(=O)C(N(Cc2ccccc2)C(=O)c2c[nH]cn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(Cc2cccnc2)C(=O)c2c[nH]cn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCCCCC2)C(=O)c2c[nH]cn2)c2cccnc2)c1
CC(C)S(=O)(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
FC(F)Oc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
CC(C)Oc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
COc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
CS(=O)(=O)Cc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
COCc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
COc1ccccc1CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
CCOc1ccc(cn1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
COc1cc(ccc1S(=O)(=O)N(C)C)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
Fc1cccc(CCNC(=O)C(N(C2CCC3OCCC3C2)C(=O)c2c[nH]cn2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCC3(CCO3)CC2)C(=O)c2c[nH]cn2)c2cccnc2)c1 |(10.44,.99,;9.93,-.47,;8.42,-.76,;7.92,-2.21,;8.93,-3.38,;10.44,-3.08,;11.45,-4.25,;12.96,-3.96,;13.97,-5.12,;15.48,-4.83,;15.98,-3.38,;16.49,-6,;18,-5.7,;19.01,-6.87,;20.52,-6.58,;21.53,-7.74,;21.02,-9.2,;22.56,-9.31,;22.45,-10.84,;20.91,-10.73,;19.51,-9.49,;18.5,-8.32,;18.5,-4.25,;17.5,-3.08,;20.02,-3.96,;20.67,-2.56,;22.2,-2.75,;22.49,-4.27,;21.14,-5.01,;15.98,-7.45,;16.99,-8.61,;16.49,-10.07,;14.98,-10.36,;13.97,-9.2,;14.47,-7.74,;10.94,-1.63,)|
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2ccc3ncsc3c2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2ccc3CCOCc3c2)c2cccnc2)c1
Cn1ncc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
Cn1cnc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
Cn1ccc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
Cc1nc2ccc(cc2o1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2cnc(nc2)C2CCC2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2ccc3c(CCCS3(=O)=O)c2)c2cccnc2)c1
FC(F)CN1C(=O)CCc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
CN1C(=O)CCc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2cccc(c2)C2COC2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2ccc(cc2)C2COC2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2ccc(Cn3cccn3)cc2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2c[nH]cn2)c2cccc(Oc3cccnn3)c2)c2cccnc2)c1
Clc1ccc2NC(=O)CC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2N(Cc3ccccc3)CCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2N(Cc3ncc[nH]3)CCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2N(Cc3ccn[nH]3)CCC(C(=O)Nc3cncc4ccccc34)c2c1
CN(C)C(=O)CN1CCC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
Clc1ccc2N(Cc3ncn[nH]3)CCC(C(=O)Nc3cncc4ccccc34)c2c1
NC(=O)N1CCC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
COCCN1CCC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
COc1ccccc1OCCNC(=O)C1CC(=O)Nc2ccccc12
Clc1cccc(c1)N1CCN(CC1)C(=O)c1cncc2ccccc12
CC1CN(CCN1c1cccc(Cl)c1)C(=O)c1cc(=O)[nH]c2ccccc12
COc1ccc(Cl)cc1OCCNC(=O)c1cc(=O)[nH]c2cccc(OC)c12
COc1cccc2[nH]c(=O)cc(C(=O)N3CCN(CC3)c3cccc(Cl)c3)c12
CC(=O)N1CCC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
Clc1ccc2OCCN(C(=O)Cc3cncc4ccccc34)c2c1
c1ccc2c(c1)c[n+](cc2NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl)[O-]
Clc1ccc2OCCC(C(=O)Nc3cncc4ccc(cc34)C#N)c2c1
Oc1ccc2cncc(NC(=O)C3CCOc4ccc(Cl)cc34)c2c1
CS(=O)(=O)c1ccc2cncc(NC(=O)C3CCOc4ccc(Cl)cc34)c2c1
Clc1ccc2OCCC(C(=O)Nc3cncc4CCNCc34)c2c1
Clc1ccc2OCCN(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2COCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2CNCC(C(=O)Nc3cncc4ccccc34)c2c1
CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
c1cc2c(cc1Cl)[C@@H](CCO2)C(=O)Nc3cncc4c3ccnc4
Clc1ccc2OCC[C@@H](C(=O)Nc3cncc4ccncc34)c2c1
COc1cccc2[nH]c(=O)cc(C(=O)NCCOc3ccccc3OCC3CC3)c12
COc1cc(Cl)cc2[C@H](CCOc12)C(=O)Nc1cncc2ccccc12
Cc1ccc(cc1)N(Cc1cscn1)C(=O)Cc1cncc2ccccc12
Cc1ccc(nc1)N(Cc1cscn1)C(=O)Cc1cncc2ccccc12
CC(=O)Nc1ccc(cn1)N(Cc2cccc(c2)Cl)C(=O)Cc3cncc4c3cccc4
CCC(=O)Nc1ccc(cc1)N(Cc1ccccc1)C(=O)n1nnc2ccccc12
Clc1cccc(NC(=O)Cc2cncc3ccccc23)c1
Oc1ccc(Cl)c2C(CCOc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(C(=O)Nc3c[nH]c(=O)c4ccccc34)c2c1
Clc1ccc2OCCC3(CC(=O)N(C3=O)c3cncc4ccccc34)c2c1
CN1C(=O)N(C(=O)C11CCOc2ccc(Cl)cc12)c1cncc2ccccc12
Brc1ccc2NC(=O)CC(C(=O)Nc3cncc4ccccc34)c2c1
c1ccc2c(c1)C(=CC(=O)N2)C(=O)N3CCN(C(=O)C3)c4cccc(c4)Cl
c1ccc2c(c1)cncc2C(=O)N3CCN(C(=O)C3)c4cccc(c4)Cl
Fc1cccc2cncc(NC(=O)Cc3cccc(Cl)c3)c12
Cc1cccc2cncc(NC(=O)Cc3cccc(Cl)c3)c12
Cc1cc(nc2n(nc(N)c12)C(=O)C1CCOc2ccc(Cl)cc12)C(F)(F)F
Nc1nn(C(=O)Cc2cccc(Cl)c2)c2cccnc12
COc1ccc2c(N)nn(C(=O)C3CCOc4ccc(Cl)cc34)c2c1
Cc1cc(nc2n(nc(N)c12)C(=O)Cc1cccc(Cl)c1)C(F)(F)F
Clc1ccc(NC(=O)C(N(C(=O)C=C)c2ccc(I)cc2)c2cncnc2)cc1
Nc1nn(C(=O)Cc2cccc(Cl)c2)c2cc(F)ccc12
Nc1nn(C(=O)C2CCOc3ccc(Cl)cc23)c2ccncc12
CC(=O)c1ccccc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1snc2ccccc12)C(=O)c1ccco1
Nc1ccc2[nH]c(cc2c1)C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccccc1
COc1cncc(C(N(C(=O)c2ccco2)c2ccc(cc2)C(C)(C)C)C(=O)NCCc2cccc(F)c2)c1C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)C1CCCO1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1coc2ccccc12)C(=O)c1ccco1
Cn1cncc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccncc1
Cn1nc(C(N(C(=O)c2ccco2)c2ccc(cc2)C(C)(C)C)C(=O)NCCc2cccc(F)c2)c2ccccc12
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc2ccccc12)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cccc(c1)C#N
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cnc2ccccn12)C(=O)c1ccco1
COc1ccccc1C(=O)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)c1ccc(cc1)C(C)(C)C
Cc1ccncc1C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cn2ccccc2n1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ncc[nH]1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1n[nH]c2ccccc12)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1nccs1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)C1CCCN1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccn[nH]1
CN(C)C(=O)CNC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCN1CCOCC1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)Nc1ccccc1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1cccnc1)C(=O)c1ccco1
CC1CC(CCN(C(C(=O)NCCc2cccc(F)c2)c2cccnc2)C(=O)c2ccco2)CC(C)(C)C1
Fc1cccc(CCNC(=O)C(N(Cc2ccccc2)C(=O)c2ccco2)c2cccnc2)c1
CCOC1CC2(CC2N(C(C(=O)NCCc2cccc(F)c2)c2cccnc2)C(=O)c2ccco2)C1 |(-7.63,-3.95,;-6.11,-3.65,;-5.61,-2.2,;-4.1,-1.91,;-3.23,-.63,;-1.96,-1.5,;-.8,-.49,;-.5,-2,;.5,-3.16,;2.02,-2.87,;3.02,-4.04,;2.52,-5.49,;4.54,-3.75,;5.54,-4.91,;7.06,-4.62,;8.07,-5.78,;9.58,-5.49,;10.59,-6.66,;10.08,-8.11,;8.57,-8.4,;8.07,-9.86,;7.56,-7.24,;2.52,-1.42,;1.51,-.25,;2.02,1.2,;3.53,1.49,;4.54,.33,;4.03,-1.13,;,-4.62,;1.01,-5.78,;-1.51,-4.91,;-2.17,-6.31,;-3.69,-6.12,;-3.98,-4.6,;-2.64,-3.86,;-2.82,-2.77,)|
Fc1cccc(CCNC(=O)C(N(C(=O)c2ccco2)c2ccc(cc2)C2CCCC2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(Cc2cc(cs2)C(F)(F)F)C(=O)c2ccco2)c2cccnc2)c1
COc1ccccc1N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Fc1cccc(CCNC(=O)C(N(Cc2ccccc2C2CCC2)C(=O)c2ccco2)c2cccnc2)c1
CC(C)c1cc(ccc1C(F)(F)F)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1cnc(s1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Fc1cccc(CCNC(=O)C(N(C(=O)c2ccco2)c2cccc(CSC3CCOCC3)c2)c2cccnc2)c1
COc1ccc(cc1NC(=O)C1CCCCC1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Fc1cccc(CCNC(=O)C(N(C(=O)c2ccco2)c2ccc(cc2)-c2n[nH]c3CCOCc23)c2cccnc2)c1
COC(=O)CCSc1cc(Cl)ccc1N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
COc1ccc(cc1OCCO)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Oc1ccc2CCCCc2c1CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CSc1ccc(CN(C(C(=O)NCCc2cccc(F)c2)c2cccnc2)C(=O)c2ccco2)cc1C#N
Fc1cccc(CCNC(=O)C(N([C@H]2C[C@@H](C2)c2cc(F)cc(F)c2)C(=O)c2ccco2)c2cccnc2)c1 |r,wU:13.12,wD:15.17,(4.33,-6.18,;3.82,-7.63,;2.31,-7.93,;1.81,-9.38,;2.81,-10.54,;4.33,-10.25,;5.33,-11.42,;6.85,-11.13,;7.86,-12.29,;9.37,-12,;9.87,-10.54,;10.38,-13.16,;11.89,-12.87,;12.9,-14.04,;14.43,-14.15,;14.32,-15.68,;12.79,-15.57,;15.33,-16.85,;16.84,-16.56,;17.85,-17.72,;19.36,-17.43,;17.35,-19.18,;15.83,-19.47,;15.33,-20.92,;14.83,-18.3,;12.39,-11.42,;11.38,-10.25,;13.9,-11.13,;14.56,-9.73,;16.09,-9.92,;16.38,-11.44,;15.03,-12.18,;9.87,-14.62,;10.88,-15.78,;10.38,-17.24,;8.86,-17.53,;7.86,-16.37,;8.36,-14.91,;4.83,-8.8,)|
COc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CC(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Fc1cccc(CCNC(=O)C(N(C(=O)c2ccco2)c2ccc(cc2)C#N)c2cccnc2)c1
COc1cc(C)ccc1N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
Fc1cccc(CCNC(=O)C(N(C2CCCC(C2)c2ccc(F)c(F)c2)C(=O)c2ccco2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2ccco2)c2ccc(Oc3ccc(cc3)C(F)(F)F)c(c2)C#N)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCN(CC2)c2ccccc2)C(=O)c2ccco2)c2cccnc2)c1
COC(=O)C(C)(CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1)c1ccccc1F
Nc1nn(C(=O)C2CCOc3ccc(Cl)cc23)c2cc(F)ccc12
Nc1nn(C(=O)Cc2cccc(Cl)c2)c2ccc(F)cc12
c1cc(cc(c1)Cl)CC(=O)N2CCCc3c2cncc3N
c1ccc2c(c1)cncc2N3C(=O)[C@@]4(CCOc5c4cc(cc5)Cl)NC3=O
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)C=C
Clc1ccc2CCC=C(C(=O)Nc3cncc4ccccc34)c2c1 |t:7|
COc1ccc2n(nc(N)c2c1)C(=O)Cc1cccc(Cl)c1
Nc1nn(C(=O)Cc2cccc(Cl)c2)c2ccccc12
Nc1nn(C(=O)Cc2cccc(Cl)c2)c2cccc(F)c12
COc1ccc2c(N)nn(C(=O)Cc3cccc(Cl)c3)c2c1
CC(C)Oc1cc(Cl)cc(c1)N(CCC1CCCCC1)C(=O)Nc1cnccc1C
Clc1cc(OC2CC(=O)N2)cc(c1)N(CCC1CCCCC1)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(C(=O)Nc3cncc4cc(CN5CCNCC5)ccc34)c2c1
Cc1nc(CN2C(=O)C(=O)c3cc(Br)ccc23)cs1
CCCCN1C(=O)C(=O)c2cc(Br)cc(C)c12
CC(C)CCN1C(=O)C(=O)c2cc(Br)ccc12
CCc1ccc2N(CC(O)=O)C(=O)C(=O)c2c1
OC(=O)CN1C(=O)C(=O)c2cc(ccc12)[N+]([O-])=O
[O-][N+](=O)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
Clc1ccc2C(=O)NCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2c(c1)C(CCS2(=O)=O)C(=O)Nc1cncc2ccccc12
CN1CCC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc12
Cc1ccc(cc1)N(Cc1cccc(Cl)c1)C(=O)Cn1nnc2ccccc12
COc1ccc(cc1)N(Cc2cccc(c2)Cl)C(=O)Cn3c4ccccc4nn3
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)N2CCOCC2)c1
Clc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)N2CCCCC2)c1
c1ccc2c(c1)cncc2CC(=O)N(CCC3CCCCC3)Cc4cccs4
CN(C)CCCN(Cc1cccs1)C(=O)Cc1cncc2ccccc12
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2CCC3
Clc1cccc2C(COc12)C(=O)Nc1cncc2ccccc12
c1ccn2c(c1)nnc2NC(=O)Cc3cccc(c3)Cl
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(c1)-c1nnc[nH]1
COc1ccc2c(NC(=O)Cc3cccc(Cl)c3)noc2c1
COc1ccc2n[nH]c(NC(=O)Cc3cccc(Cl)c3)c2c1
COc1ccc2c(NC(=O)Cc3cccc(Cl)c3)[nH]nc2c1
Cc1ccn2cnnc2c1NC(=O)Cc1cccc(Cl)c1
Cc1cc(nc2n[nH]c(NC(=O)Cc3cccc(Cl)c3)c12)C(F)(F)F
Cc1nn(C)c2[nH]nc(NC(=O)Cc3cccc(Cl)c3)c12
Fc1ccc2[nH]nc(NC(=O)Cc3cccc(Cl)c3)c2c1
Fc1ccc2c(NC(=O)Cc3cccc(Cl)c3)[nH]nc2c1
Clc1cccc(CC(=O)Nc2n[nH]c3ccccc23)c1
Clc1cccc(CC(=O)Nc2cccc3cn[nH]c23)c1
Fc1cccc2n[nH]c(NC(=O)Cc3cccc(Cl)c3)c12
Clc1cccc(CC(=O)Nc2[nH]nc3cccnc23)c1
Clc1cccc(CC(=O)Nc2n[nH]c3ccnc(Br)c23)c1
Clc1cccc(CC(=O)Nc2n[nH]c3ccncc23)c1
Clc1ccc2OCCC(C(=O)NC3CCNC(=O)C3)c2c1
Clc1cccc(CC(=O)NC2CC(=O)c3ccccc23)c1
Fc1cccc2n[nH]c(NC(=O)C3CCOc4ccc(Cl)cc34)c12
Clc1ccc2OCCC(C(=O)Nc3[nH]nc4ccccc34)c2c1
Clc1ccc2OCCC(C(=O)Nc3[nH]nc4cccnc34)c2c1
COc1ccc2n[nH]c(NC(=O)C3CCOc4ccc(Cl)cc34)c2c1
Fc1ccc2c(NC(=O)C3CCOc4ccc(Cl)cc34)[nH]nc2c1
COc1ccc2c(NC(=O)C3CCOc4ccc(Cl)cc34)noc2c1
Cc1ccn2cnnc2c1NC(=O)C1CCOc2ccc(Cl)cc12
COc1ccc2c(NC(=O)C3CCOc4ccc(Cl)cc34)[nH]nc2c1
Clc1ccc2OCCC(C(=O)Nc3cccc4cn[nH]c34)c2c1
Clc1ccc2OCCC(C(=O)Nc3n[nH]c4ccnc(Br)c34)c2c1
Clc1ccc2OCCC(C(=O)Nc3n[nH]c4ccncc34)c2c1
Cc1cc(nc2n[nH]c(NC(=O)C3CCOc4ccc(Cl)cc34)c12)C(F)(F)F
Clc1ccc2OCCC(C(=O)Nc3cc[nH]c(=O)c3)c2c1
Fc1ccc(Cl)cc1CC(=O)Nc1cncc2ccccc12
Clc1ccc(Cl)c(CC(=O)Nc2cncc3ccccc23)c1
CC1COCCN1CCOc1cc(Cl)cc(CC(=O)Nc2cnccc2C)c1
Clc1cccc(CC(=O)N[C@H]2CCNC2=O)c1
Cn1cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)N2CCCCC2)cn1
Clc1ccc2OCC[C@@H](C(=O)N(C(=O)C=C)c3cncc4ccccc34)c2c1
Clc1cc(CC2CC(=O)N2)cc(CC(=O)Nc2cncc3ccccc23)c1
C[C@@H]1C[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2O1
C[C@H]1C[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2O1
C[C@H]1COc2ccc(Cl)cc2[C@H]1C(=O)Nc1cncc2ccccc12
C[C@@H]1COc2ccc(Cl)cc2[C@H]1C(=O)Nc1cncc2ccccc12
C[C@@H]1COc2ccc(cc2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl
Clc1ccc2N(Cc3cnc[nH]3)CCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(C(=O)Oc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(C(=O)NC3N=Nc4ccccc34)c2c1 |c:13|
COc1ccccc1OCCNC(=O)c2cncc3c2cccc3
COc1ccccc1OCCC(=O)Nc1cncc2ccccc12
COc1ccccc1NCCNC(=O)c1cc(=O)[nH]c2ccccc12
c1ccc(cc1)N2CCN(CC2)C(=O)c3cncc4c3cccc4
Clc1cccc(c1)N1CCN(CC1)C(=O)c1cc(=O)[nH]c2ccccc12
c1ccc2c(c1)C(=CC(=O)N2)C(=O)N3CCN(CC3)c4cccc(c4)C(F)(F)F
COc1ccccc1OC1CCN(C1)C(=O)c1cc(=O)[nH]c2ccccc12
COc1ccccc1NC2CN(C2)C(=O)C3=CC(=O)Nc4c3cccc4
COc1ccccc1OC2CN(C2)C(=O)C3=CC(=O)Nc4c3cccc4
COc1cccc(CN2CCN(CC2)C(=O)c2cc(=O)[nH]c3ccccc23)c1
Clc1cccc(CN2CCN(CC2)C(=O)c2cc(=O)[nH]c3ccccc23)c1
FC(F)(F)c1cccc(CN2CCN(CC2)C(=O)c2cc(=O)[nH]c3ccccc23)c1
Clc1ccc2OCC[C@H](C(=O)N(C(=O)C=C)c3cncc4ccccc34)c2c1
Clc1cccc(c1)N(CCC1CCCCC1)C(=O)Cc1cncc2ccccc12
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2n[nH]c3ccccc23)c1
c1ccc2c(c1)cncc2NC(=O)Cc3cc(ccn3)Cl
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(Cc2ccn[nH]2)c1
C[C@@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OC[C@@H](Cc2c1)C(=O)Nc1cncc2ccccc12
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2CCCN3
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(n3)Cl
CNC(=O)Nc1ccc(cc1)N(Cc2ccsc2)C(=O)Cn3c4ccccc4nn3
CN(C)c1ccc(cc1)N(Cc2ccsc2)C(=O)Cc3cncc4c3cccc4
Clc1ccc2CCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2NCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CCC3CC3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC3(CCCN(C3=O)c3cncc4ccccc34)c2c1
C[C@@H]1C[C@@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2O1
C[C@H]1C[C@@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2O1
COc1cc(Cl)cc2[C@@H](CCOc12)C(=O)Nc1cncc2ccccc12
Cc1c(Cl)ccc2OCC[C@@H](C(=O)Nc3cncc4ccccc34)c12
C[C@H]1COc2ccc(cc2[C@@H]1C(=O)Nc3cncc4c3cccc4)Cl
Clc1ccc2OC[C@H](Cc2c1)C(=O)Nc1cncc2ccccc12
C[C@]1(CCOc2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4
Brc1ccc2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Cc1ccncc1NC(=O)[C@@H](C)OC(F)F
Clc1cc2CCOc2c(CC(=O)Nc2cncc3ccccc23)c1
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CCOc4c3cc(cc4)Cl
Clc1ccc2OCC[C@H](C(=O)Nc3cncc4ccccc34)c2c1
Cc1ccncc1NC(=O)[C@H]1CCOc2ccc(Cl)cc12
Cc1ccncc1NC(=O)[C@@H]2CCOc3c2cc(cc3)Cl
c1ccc2c(c1)nnn2NC(=O)Cc3cccc(c3)Cl
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N([C@H](c2cccnc2)C(=O)NCCc3cccc(c3)F)C(=O)c4ccco4
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1c[nH]cn1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccc(Cl)o1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cn[nH]c1
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCNC1=O)C(O)S(O)(=O)=O
COc1ccc(OC)c(CNC(=O)Nc2cn(C)c(=O)c3ccccc23)c1
Fc1ccc(cc1)-c1nc(c(o1)S(=O)(=O)Cc1ccccc1F)S(=O)(=O)c1ccccc1
CC(C)N(C(C)C)C(=O)Cc1c(O)c2ccccc2[nH]c1=O
CC(C)Cn1cc(NC(=O)Nc2ccc(C)cc2Br)c2ccccc2c1=O
COc1ccc(NC(=O)Nc2cn(C)c(=O)c3ccccc23)cc1OC
CC(=O)c1cccc(NC(=O)Nc2cn(C)c(=O)c3ccccc23)c1
CCOC(=O)c1c(C)n(c2ccc(cc12)N(C(=O)c1ccco1)S(C)(=O)=O)S(C)(=O)=O
CC(C)Cn1cc(NC(=O)Nc2cc(C)on2)c2ccccc2c1=O
Clc1cnc(nc1C(=O)NCc1ccc2OCOc2c1)S(=O)(=O)Cc1ccccc1
COC(=O)c1c(C)n(c2ccc(cc12)N(C(=O)c1ccco1)S(C)(=O)=O)S(C)(=O)=O
CCOC(=O)c1ccc(NC(=O)Nc2cn(C)c(=O)c3ccccc23)cc1
CC(C)Cn1cc(NC(=O)NCC2CCCO2)c2ccccc2c1=O
COc1ccc(NC(=O)Nc2cn(C)c(=O)c3ccccc23)c(OC)c1
OC(=O)[C@H](N1Cc2ccccc2C1=O)c1ccccc1
CC(C)Cn1cc(NC(=O)NCCc2c[nH]c3ccccc23)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)Nc2ncccc2C)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)Nc2cccnc2)c2ccccc2c1=O
CCOC(=O)c1cc(sc1NC(=O)Cc1csc(n1)-c1ccccc1)-c1ccccc1
CCCc1c(C)[nH]c2[nH]n(-c3ccccc3)c(=O)c2c1=O
CC(C)Cn1cc(NC(=O)NC2CCCCCC2)c2ccccc2c1=O
COc1ccc(OC)c(CNC(=O)Nc2cn(CC(C)C)c(=O)c3ccccc23)c1
CCOC(=O)Cc1csc(NC(=O)Nc2cn(CC(C)C)c(=O)c3ccccc23)n1
CC(C)Cn1cc(NC(=O)Nc2nc3ccccc3s2)c2ccccc2c1=O
N#Cc1ccc(CN2CCC(CC2)C2CCNC2)cc1
COc1cc2CCN(C(C)c2cc1OC)C(=O)Nc1cn(C)c(=O)c2ccccc12
COc1cc(Cl)c(C)cc1NC(=O)Nc1cn(C)c(=O)c2ccccc12
CCN(CC)S(=O)(=O)c1ccc(NC(=O)Nc2cn(C)c(=O)c3ccccc23)cc1
CC(CCc1ccco1)NC(=O)Nc1cn(C)c(=O)c2ccccc12
CC(C)Cn1cc(NC(=O)NCCC2=CCCCC2)c2ccccc2c1=O |t:13|
COc1ccc(cc1S(=O)(=O)Nc1cccc2cccnc12)N1C(=O)CCS1(=O)=O
CC(C)Cn1cc(NC(=O)NC2CCCc3ccccc23)c2ccccc2c1=O
COc1cc(Cl)c(C)cc1NC(=O)Nc1cn(CC(C)C)c(=O)c2ccccc12
CC(C)Cn1cc(NC(=O)NCc2ccco2)c2ccccc2c1=O
COc1ccc(OC)c(CCNC(=O)Nc2cn(CC(C)C)c(=O)c3ccccc23)c1
Cn1cc(NC(=O)NCc2ccccn2)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCCc2c(C)noc2C)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCc2ccc3OCOc3c2)c2ccccc2c1=O
COC(=O)c1sccc1NC(=O)Nc1cn(CC(C)C)c(=O)c2ccccc12
COc1ccc2nc(NC(=O)Nc3cn(CC(C)C)c(=O)c4ccccc34)sc2c1
[O-][N+](=O)c1cnc(Sc2nnc(-c3ccco3)n2-c2ccc(OCc3ccccc3)cc2)s1
Nc1n[nH]c2cc(O)nc(O)c12
COC(=O)c1c(C)nn(c1-c1cc(C)on1)-c1ccccc1
Fc1c(Cl)cccc1CSc1ccccc1NS(=O)(=O)c1cc(Cl)sc1Cl
CC(C)(C)c1ccc(cc1)-c1nnc(Sc2cnc(s2)[N+]([O-])=O)o1
COC(=O)c1c(C)nn(C(=O)c2cccs2)c1-c1snnc1C |(3.68,1.97,;3.68,.43,;2.35,-.34,;1.01,.43,;2.35,-1.88,;3.59,-2.78,;5.06,-2.31,;3.12,-4.25,;1.58,-4.25,;.67,-5.49,;1.3,-6.9,;-.86,-5.33,;-1.89,-6.48,;-3.3,-5.85,;-3.14,-4.32,;-1.63,-4,;1.1,-2.78,;-.37,-2.31,;-1.61,-3.21,;-2.86,-2.31,;-2.38,-.84,;-.84,-.84,;.06,.4,)|
[O-][N+](=O)c1cnc(Sc2nnc(o2)-c2ccc(Cl)cc2)s1
[O-][N+](=O)c1cnc(Sc2ccccc2NC(=O)Nc2cccc(c2)C(F)(F)F)s1
O=C(c1cccs1)n1ncc(C#N)c1C1CC1
[O-][N+](=O)c1cnc(Sc2nccc(n2)-c2cccnc2)s1
Cc1cc(C)c(C#N)c(Sc2ncnc3n(Cc4ccccc4)nnc23)n1
CCOC(=O)c1ccc(NC(=O)CC2SC(=O)N(C2=O)c2ccccc2)cc1
Cc1ccccc1NC(=O)CC1SC(=O)N(C1=O)c1ccccc1
S(c1nnc(o1)-c1cccs1)c1cc(nc2ncnn12)-c1ccccc1
CN(C)c1ccc(cc1)N(Cc2ccn[nH]2)C(=O)Cn3c4ccccc4nn3
Cc1ccncc1NC(=O)Cc2cc(cc(c2)Cl)OCc3nc(no3)C
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2nnc(o2)C2CCCCC2)c1
COc1cc(COc2cc(Cl)cc(CC(=O)Nc3cnccc3C)c2)ccc1OC(F)F
CCOC(=O)c1c(COc2cc(Cl)cc(CC(=O)Nc3cnccc3C)c2)oc2ccccc12
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2cc(no2)-c2ccc(Cl)cc2)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2ccc(OCc3ccccc3F)cc2)c1
COc1ccc(cc1)-c1cc(COc2cc(Cl)cc(CC(=O)Nc3cnccc3C)c2)on1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2nn(C(=O)OC(C)(C)C)c3ccccc23)c1
CN(C)c1ccc(cc1)N(Cc2cscn2)C(=O)Cn3c4ccccc4nn3
CCC(=O)Nc1ccc(cc1)N(Cc1cscn1)C(=O)Cn1nnc2ccccc12
O=C1OC(=N\C1=C/c1ccc(s1)N1CCOCC1)c1cccs1 |c:3|
CCC(=O)Nc1ccc(cc1)N(Cc1ccccc1)C(=O)Nn1nnc2ccccc12
COc1ccc(cc1)C(Cc1ccsc1)C(=O)Nc1n[nH]c2ccccc12
Cc1ccc(cc1)C(Cc1cnn(C)c1)C(=O)Nc1n[nH]c2ccccc12
Cc1ccc(cc1)C(Cc1ccccc1)C(=O)Nc1nnn2ccccc12
CN(C)c1ccc(cc1)C(Cc1ccsc1)C(=O)Nn1cnc2ccccc12
CN(C)c1ccc(cc1)C(Cc1ccsc1)C(=O)Nc1nnc2ccccn12
Clc1cccc(CC(C(=O)Nn2cnc3ccccc23)c2ccc(cc2)N2CCOCC2)c1
Clc1cccc(CC(C(=O)Nn2nnc3ccccc23)c2ccc(cc2)N2CCCCC2=O)c1
COc1ccc(cc1)C(Cc1cnn(C)c1)C(=O)Nc1c[nH]c2ccccc12
COc1ccc(cc1)N(Cc1ccccc1)C(=O)Cc1c[nH]c2ccccc12
O=C(Cc1n[nH]c2ccccc12)N(Cc1ccccc1)c1ccc(cc1)N1CCCCC1=O
O=C(Cc1nnn2ccccc12)N(Cc1ccccc1)c1ccc(cc1)N1CCCCC1
CC(=O)N1CCN(CC1)CC(=O)Nc2cncc3c2cccc3
COC(=O)C(C(=O)Nc1cnccc1C)c1cccc(Cl)c1
Clc1ccc2OCC(C(=O)Nc3cncc4ccccc34)c2c1
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cncc3
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2[nH]cn3
CN(C)c1ccc(cc1)N(Cc2ccccc2)C(=O)Cn3c4ccccc4nn3
CN(C)c1ccc(cc1)N(Cc2cccc(c2)Cl)C(=O)Cn3c4ccccc4nn3
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)N1CCCCC1
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(cc1)N1CCOCC1
O=C(Cn1nnc2ccccc12)N(Cc1ccccc1)c1ccc(cc1)N1CCOCC1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)-c1ccc(cc1)C1CC1(F)F
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)-c1ccc(cc1Cl)S(C)(=O)=O
COC(=O)c1ccc(c(OC)c1)-c1cc(Cl)cc(CC(=O)Nc2cnccc2C)c1
CCc1cc(F)ccc1-c1cc(Cl)cc(CC(=O)Nc2cnccc2C)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)-c1ccc(cc1)C1(C)CCO1
Cc1ccc(c(F)c1F)-c1cc(Cl)cc(CC(=O)Nc2cnccc2C)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)-c1cnn(C)c1C(F)F
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(\C=C(\c2ccccc2)C(F)(F)F)c1
CCOC(=O)c1cc(n[nH]1)-c1cc(Cl)cc(CC(=O)Nc2cnccc2C)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(NC2CCCC2O)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(NC2CCC(F)(F)C2O)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(NC2CC2C(F)(F)F)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(NC2(C)CCC(F)(F)CC2)c1
Cc1ccncc1NC(=O)Cc2cc(cc(c2)Cl)NCC(C)(C)C#N
Cc1cc(C)[n+](C)c(n1)C#N
COc1cc(OC)[n+](C)c(n1)C#N
Clc1cccc(OCC(=O)Nc2cncc3ccccc23)c1
Clc1cccc(CCC(=O)Nc2cncc3ccccc23)c1
Cc1ccncc1NC(=O)CCc2cccc(c2)Cl
Cn1cc(NC(=O)Cc2cccc(Cl)c2)c2ccccc2c1=O
OCCn1c(CSc2nc3ccccc3o2)nc2ccc(Cl)cc12
Clc1cc(Br)ccc1NC(=O)Cn1cnc(n1)C#N
C[n+]1ccn(CCCc2cccc(Cl)c2)c1C#N
C[n+]1ccn(CCc2cccc(Cl)c2)c1C#N
Clc1cccc(CCCn2ccnc2C#N)c1
CC(Cn1ccnc1C#N)c1cccc(Cl)c1
CC1(C)OB(OC1(C)C)c1cnc(nc1)C#N
Clc1ccnc(n1)C#N
Clc1cnc(nc1)C#N
Fc1cnc(nc1)C#N
Cc1cc(C)nc(n1)C#N
Clc1cccc(CCn2ccnc2C#N)c1
Brc1cnc(nc1)C#N
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2ccnc3
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2nccc3
CC(C)c1ccncc1NC(=O)Cc1cccc(Cl)c1
Clc1cccc(CC(=O)Nc2c[nH]c(=O)c3ccccc23)c1
CN(c1cncc2c1cccc2)C(=O)Cc3cccc(c3)Cl
Clc1cccc(CC(=O)Nc2cncc3c(Cl)cccc23)c1
Cc1cc2OCC(C(=O)N3CCCCC3c3cn[nH]c3)c2cc1C
OC(Cc1cccc(Cl)c1)Cn1cncn1
COc1cccc(n1)Oc2cc(cc(c2)Cl)NC(=O)Cc3cncc4c3cccc4
Clc1cccc(CC(=O)NC2C(=O)Nc3ccccc23)c1
Clc1ccc2OCCC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(OC2CCC(=O)N2)c1
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(Oc2cccc(=O)[nH]2)c1
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(Oc2cccnc2)c1
CNC(=O)C(N(Cc1ccccc1Cl)C(=O)C=C)c1cncc2ccccc12
CC(C)(C)NC(=O)C(N(Cc1ccccc1Cl)C(=O)C=C)c1cccnc1
CNC(=O)C(N(Cc1ccccc1Cl)C(=O)C=C)c1cccnc1
CC(C)(C)NC(=O)C(N(Cc1ccccc1Cl)C(=O)C=C)c1cncc2ccccc12
COc1cc(OC)nc(n1)C#N
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1ccccc1)C(=O)c1ccco1
O=C(Nc1cccnc1)NC1(CC1)C#Cc1c[nH]cn1
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cccn3
CC1CCNC(=O)C1NC(=O)Cc1cccc(Cl)c1
CC1(CCNC1=O)NC(=O)Cc1cccc(Cl)c1
c1ccn2c(c1)ncc2NC(=O)Cc3cccc(c3)Cl
Cn1cncc1NC(=O)Cc2cccc(c2)Cl
Clc1cccc(c1)N(CCC1CCCCC1)C(=O)Nc1cncc2ccccc12
Clc1cccc(CC(=O)Nc2cncc3CCCOc23)c1
CC(NC(C)=O)c1cc(Cl)cc(c1)-c1ccc(cc1)S(N)(=O)=O
CCC(=O)Nc1ccc(cc1)N(C)C(=O)Cn1nnc2ccccc12
CN(Cc1cccc(c1)Cl)C(=O)Cn2c3ccccc3nn2
C#Cc1cccc(c1)CC(=O)Nc2cncc3c2cccc3
Clc1cccc(c1)C1CCCN(C1=O)c1cncc2ccccc12
Clc1cccc(c1)C1CCN(C1=O)c1cncc2ccccc12
COc1ccc(cc1CC(=O)Nc2cncc3c2cccc3)Cl
Clc1cc(CC(=O)Nc2cc(=O)[nH]c3ccccc23)cc(OC2CC(=O)N2)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2ncc[nH]2)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OCc2ncn[nH]2)c1
Cc1ccncc1NC(=O)Cc2cc(cc(c2)Cl)CNC(=O)C
CNC(=O)c1cc(Cl)cc(CC(=O)Nc2cnccc2C)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)-c1ncc[nH]1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(CNS(C)(=O)=O)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)S(N)(=O)=O
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2CCCC3
Cn1cc(NC(=O)NCCc2ccc(Cl)cc2)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCCc2ccc(Cl)cc2)c2ccccc2c1=O
Cn1cc(NC(=O)NCCc2ccsc2)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCCCN2CCC(C)CC2)c2ccccc2c1=O
CCCCN(CCNC(=O)Nc1cn(C)c(=O)c2ccccc12)Cc1ccco1
Cn1cc(NC(=O)N2CCN(CC2)C(=O)c2ccco2)c2ccccc2c1=O
Cn1cc(NC(=O)N(CC2CCCO2)Cc2ccco2)c2ccccc2c1=O
CC(C)OCCCN(Cc1ccco1)C(=O)NC2=CN(C(=O)c3c2cccc3)C
CCN(C(=O)Nc1cn(C)c(=O)c2ccccc12)c1ccccc1CC
COC(=O)c1c(NCCCc2ccccc2)c2cc(F)ccc2[nH]c1=O
CCOC(=O)N1CCC(CC1)NC(=O)Nc1cn(C)c(=O)c2ccccc12
Cn1cc(NC(=O)NCCCN2CCc3ccccc3C2)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCCCN2CCCC2=O)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)N2CCC(C2)c2ccccc2)c2ccccc2c1=O
CCCCN(CCCNC(=O)Nc1cn(CC(C)C)c(=O)c2ccccc12)c1ccccc1
CC(C)Cn1cc(NC(=O)N2CCC(Cc3ccccc3)CC2)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCC2CCN(Cc3ccc(C)cc3)C2)c2ccccc2c1=O
CC(C)Cn1cc(NC(=O)NCCN2CCOCC2)c2ccccc2c1=O
COc1cccc(c1)C1=N\C(=C\c2sccc2C)C(=O)O1 |t:9|
COc1cccc(c1)C(=O)Nc1n[nH]c(SCc2ccc(Cl)cc2)n1
O=c1oc(Nc2ccccc2)nc2ccccc12
O=C(Cc1ccsc1)N1CCN(CC1)c1cc(n[nH]1)-c1cccs1
CCCCc1nc(c[nH]1)-c1nccn1CC(F)(F)F
CCCCc1nc(c[nH]1)-c1nccn1CCc1ccccn1
CCCCc1nc(c[nH]1)-c1nccn1Cc1ccoc1
c1ccc2c(c1)cnnc2NC(=O)Cc3cccc(c3)Cl
Clc1cccc(CC(=O)Nc2cnnc3ccccc23)c1
c1ccn2cnc(c2c1)NC(=O)Cc3cccc(c3)Cl
COc1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
Clc1cccc(CC(=O)Nc2cnccc2-c2ccccc2)c1
Clc1cc(CC(=O)Nc2cncc3ccccc23)cc(OC2CC(=O)N2)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cccnc1
CNc1ccc(cc1)N(C(=O)Cn1nnc2ccccc12)c1cccc(Cl)c1
COC(=O)C(N1CCC(S)\C(C1)=C\C(O)=O)c1ccccc1Cl
O=C(Nc1nncn1C1CC1)C1CCOc2ccccc12
Cc1ccncc1C(N(Cc1cccc(Cl)c1)C(=O)C=C)C(=O)NCCc1cccc(F)c1
COc1ccc(Cl)cc1OCCNC(=O)c1cc(=O)[nH]c2ccccc12
Cc1ccncc1OCCNC(=O)C(C)(C)c1cccc(Cl)c1
Cc1ccncc1NC(=O)C(C(=O)c1cc(=O)[nH]c2ccccc12)c1cccc(Cl)c1
CN(C)c1cncc(CN(C(=O)c2cc(=O)[nH]c3ccccc23)c2cccc(Cl)c2)c1
COc1cccc(CCN(C(=O)c2cc(=O)[nH]c3ccccc23)c2cccc(Cl)c2)c1
Cn1c(nc2ccccc12)C(NC(=O)Cc1cc2ccccc2[nH]1)c1cccc(Cl)c1
COc1cccc(c1)C(NC(=O)Cc1cccc(Cl)c1)c1nc2ccccc2[nH]1
Clc1cccc(CC(=O)NC2CC(=O)NC2=O)c1
Clc1cccc(CC(=O)NC2CCCNC2=O)c1
Clc1cccc(CC(=O)NC2CNC(=O)C2)c1
Clc1ccc2OCCC(C(=O)NC3CNC(=O)C3)c2c1
Cc1cccc(COC(=O)c2cccc3C(=O)C(=O)Nc23)c1
Cc1ccc(OCCN2C(=O)C(=O)c3cccc(Cl)c23)cc1
CCOc1ccccc1CN1C(=O)C(=O)c2cc(Br)ccc12
COc1ccc(CN2C(=O)C(=O)c3cc(Br)cc(C)c23)cc1OC
Cc1cccc(NC(=O)CN2C(=O)C(=O)c3ccccc23)c1
Fc1cc(ccc1CN1C(=O)C(=O)c2cccc(Br)c12)C#N
Brc1cccc2C(=O)C(=O)N(Cc3cccc(c3)C#N)c12
FCCOc1ccc2NC(=O)C(=O)c2c1
COC(=O)c1cc(Br)cc2C(=O)C(=O)Nc12
Brc1ccc2N(Cc3ncon3)C(=O)C(=O)c2c1
Clc1cc(CC(=O)Nn2cnc3ccccc3c2=O)cc(OC2CC(=O)N2)c1
Clc1cc(CC(=O)Nn2cnc3ccccc23)cc(OC2CC(=O)N2)c1
Cc1ccncc1NC(=O)Cc2cc(cc(c2)Cl)OC
Fc1ccccc1OCC(=O)Nc1ncnc2[nH]cnc12
O=C1C(CCN1Cc1ccccc1)Nc1ncnc2[nH]cnc12
Cn1c(nc2ccccc12)-c1ccc(NC(=O)C2CCCCC(=O)N2)cc1
Cc1[nH]c2ncnc(NC(=O)c3cc4ccccc4c(=O)o3)c2c1C
Fc1cc(ccc1NC(=O)C1CCCCC(=O)N1)-c1nc[nH]n1
O=C(Nc1c[nH]nc1-c1ccccn1)c1cccc2nccn12
Cc1[nH]c2ncnc(NC(=O)C3CCN(CC3)c3ccc(Cl)cn3)c2c1C
COc1c(Cl)cccc1OCCNC(=O)c1cc(=O)[nH]c2ccccc12
Cc1noc(C)c1S(=O)(=O)N1CCN(CC1)C(=O)CCl
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(c1)C1COC1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OC2COC2)c1
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(NS(C)(=O)=O)c1
Cc1ccncc1NC(=O)Cc2cc(cc(c2)Cl)NS(=O)(=O)N
c1cc2c(cc1Cl)[C@@H](CCO2)C(=O)Nc3nncn3C4CC4
c1cc2c(cc1Cl)[C@H](CCO2)C(=O)Nc3nncn3C4CC4
Fc1cccc2C(CCOc12)C(=O)Nc1nncn1C1CC1
Clc1ccc2OCCC(C(=O)Nc3cc(=O)[nH]c4ccccc34)c2c1
CN(C)S(=O)(=O)c1cccc(c1)C(=O)Nc1c(nc2sccn12)-c1ccccc1
Cc1c(C(=O)CCl)c2ccccn2c1C(=O)c1ccc(F)cc1
CSC1=C(C#N)C2(CCCCC2)C(C#N)=C(NC(=O)CCl)N1 |c:2,t:15|
Cc1cc(C(=O)CCl)c(C)n1CC1COc2ccccc2O1
CCN(c1ccccc1)S(=O)(=O)c1ccc(OC)c(NC(=O)CCl)c1
Cc1cc(C(=O)CCl)c(C)n1NC(=O)c1n[nH]c(=O)c2ccccc12
CN(CC(=O)Nc1ccccc1Br)C(=O)CCl
CS(=O)(=O)Nc1cccc(c1)C1=NN(C(C1)c1ccccc1)C(=O)CCl |t:12|
Cc1ccncc1NC(=O)C1CCOc2ccc(Cl)cc12
OCc1ccncc1NC(=O)C1CCOc2ccc(Cl)cc12
O=C(Nc1nncn1C1CC1)C1CCS(=O)(=O)c2ccccc12
c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl
Cc1ccncc1CC(=O)Nc2cccc3c2CNCC3
COc1ccc(Cl)cc1N1C(=O)CN(Cc2cc(=O)[nH]c3ccccc23)C1=O
Clc1cc(NC(=O)Cc2cncc3ccccc23)cc(OC2CCC(=O)N2)c1
Clc1cc(OCCNC(=O)c2cc(=O)[nH]c3ccccc23)cc(OC2CC(=O)N2)c1
Cc1ccncc1NC(=O)Cc1ccc2[nH]ncc2c1
c1cc(cc(c1)Cl)CC(=O)Nc2cccc3c2cn[nH]3
Cc1ccncc1N(CC#N)C(=O)Cc1cccc(Cl)c1
CS(=O)(=O)c1ncc(Cl)c(n1)C(=O)Nc1ccccc1Cc1ccccc1
CCOC(=O)c1nc(ncc1Cl)S(C)(=O)=O
CCn1c(CSc2nc(C)c(C)n2CC2CCCO2)nc2cc(ccc12)S(=O)(=O)N(C)C
CN(C)c1ccc(cc1)N(Cc2ccsc2)C(=O)Cn3c4ccccc4nn3
c1cc(cc(c1)Cl)CC(=O)Nc2c[nH]nc2
Cc1[nH]ncc1CC(=O)Nc1cccc(Cl)c1
CCCc1cc2OCOc2cc1S(=O)(=O)N1CCN(CC1)c1ccccc1
Cc1cc2c(N)nc(=O)n(CC(=O)Nc3cccc(Cl)c3)c2s1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc(Cl)c1)C(=O)C=C
Cc1cncc(c1)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)C(=O)NCCc1cccc(F)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc(c1)C#N)C(=O)C=C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc(O)c1)C(=O)C=C
Fc1cccc(CCNC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(F)(F)F)c2cncc(Cl)c2)c1
Cc1cncc(c1)C(N(C(=O)C=C)c1ccc(cc1)C(F)(F)F)C(=O)NCCc1cccc(F)c1
Fc1cccc(CCNC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(F)(F)F)c2cncc(c2)C#N)c1
Oc1cncc(c1)C(N(C(=O)C=C)c1ccc(cc1)C(F)(F)F)C(=O)NCCc1cccc(F)c1
Fc1cccc(CCNC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(F)(F)F)c2cccnc2)c1
CC(C)(C)c1cc(no1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)C=C
CC(C)(C)c1cc(no1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc(Cl)c1)C(=O)C=C
CC(C)(C)c1cc(no1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc(O)c1)C(=O)C=C
CC(C)(C)c1cc(no1)N(C(C(=O)NCCc1cccc(F)c1)c1cncc(c1)C#N)C(=O)C=C
COc1ccccc1OCCNC(=O)c1cc(N)cc2ccccc12
Cc1ccc(NC2=C(C(=O)N(Cc3cccnc3)C2=O)c2ccccc2)cc1C |t:6|
Cc1ccc(NC2=C(C(=O)N(Cc3cccnc3)C2=O)c2ccccc2)c(C)c1 |t:6|
Cc1ccc(NC2=C(C(=O)N(Cc3cccnc3)C2=O)c2ccccc2)cc1Cl |t:6|
CC(=O)N(CC(=O)Nc1ccc(F)c(Cl)c1)c1cccc(Cl)c1
CC(=O)N(CC(=O)Nc1ccc(F)c(Cl)c1)c1cccc(c1)C#N
CC(=O)N(CC(=O)Nc1ccc(F)c(Cl)c1)c1cccc(c1)C(F)(F)F
Cc1ccc(cc1C)-n1ncc2c1ncn(CC(N)=O)c2=O
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C(F)(F)F
Oc1ccc(cc1)-c1nnc2CCC(Cn12)C(=O)NCc1coc2ccccc12
Cc1nc(n[nH]1)-c1cccc(CNC(=O)Nc2cccc(CN3CCCC3=O)c2)c1
CNc1ccc(cc1)N(Cc2ccsc2)C(=O)Cn3c4ccccc4nn3
COc1ccc2c(c1)n(nn2)CC(=O)N(Cc3ccccn3)c4ccc(cc4)C5CCNCC5
O=C(Cn1nnc2ccccc12)N(CC(=O)N1CCNCC1)c1ccc(cc1)-c1ccccc1
NCc1cn(CC(=O)N(Cc2cscn2)c2ccc(nc2)-c2ccccc2)nn1
NCc1cn(CC(=O)N(Cc2ccsc2)c2ccc(cc2)-c2ccccc2)nn1
CC(C)(C(N)=O)c1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
NCc1cn(CC(=O)N(CC(=O)N2CCNCC2)c2ccc(cc2)-c2ccccc2)nn1
Cn1cnc(CN(C(=O)c2cnnn2-c2ccccc2)c2ccc(OCc3ccccc3)cc2)c1
O=C(Cc1cccnc1)N(CC(=O)N1CCNCC1)c1ccc(cc1)-c1ncccn1
NCc1cn(CC(=O)N(Cc2ccsc2)c2ccc(cc2)-n2cnnc2)nn1
O=C(Cn1nnc2ccccc12)N(CC1CCOC1)c1ccc(cc1)C1CCNCC1
Cn1ccc(CN(C(=O)Cc2cccnc2)c2ccc(cc2)-c2ccccn2)n1
O=C(Cn1nnc2ccccc12)N(Cc1ccccn1)c1cnc(nc1)-c1ccccc1
O=C(Cn1nnc2ccccc12)N(Cc1ccccn1)c1ccc(cc1)-n1cnnc1
O=C(Cn1ccnn1)N(CC(=O)N1CCNCC1)c1ccc(cc1)-c1ccccn1
Clc1cccc(CN2CCN(C2=O)c2nccc3[nH]ncc23)c1
ClCC(=O)N1CCN(CC1)S(=O)(=O)c1ccccc1
COc1ccc(cc1)S(=O)(=O)N1CCN(CC1)C(=O)CCl
Cc1cccc2c1C(=CC(=O)N2)C(=O)NCCOc3ccccc3OC
COc1ccccc1OCCNC(=O)C2=CC(=O)Nc3c2c(ccc3)F
COc1ccccc1OCCNC(=O)C2=CC(=O)Nc3c2c(ccc3)OC
O=C(Cc1ccc2[nH]c(=O)[nH]c2c1)NC1(CNC(=O)c2cnc[nH]2)CC1
ClCC(=O)N1CCN(Cc2cccc(c2)C#N)CC1
ClCC(=O)N1CCN(CC1)S(=O)(=O)c1ccsc1
Fc1ccc(CNc2ccc3N(CCCc3c2)C(=O)CCl)c(Cl)c1
Brc1cccc2C(=O)C(=O)Nc12
Brc1ccc(CN2C(=O)C(=O)c3cccc(Br)c23)cc1
Brc1ccc2NC(=O)C(=O)c2c1
Brc1ccc(CN2C(=O)C(=O)c3ccccc23)cc1
Cc1cc(Br)cc2C(=O)C(=O)N(CCBr)c12
OC(=O)C12CC(CNCc3ccc4CCOc4c3)(C1)OC2c1ccccc1 |TLB:21:20:4:18,(-5.38,-6.97,;-3.9,-6.54,;-4.58,-7.93,;-2.36,-6.44,;-2.71,-7.94,;-1.33,-5.39,;,-4.62,;,-3.08,;1.33,-2.31,;1.33,-.77,;;,1.54,;1.33,2.31,;1.65,3.82,;3.19,3.98,;3.81,2.57,;2.67,1.54,;2.67,,;-.35,-6.63,;-1.9,-3.96,;-2.88,-5.09,;-4.39,-4.82,;-5.38,-6,;-6.9,-5.73,;-7.43,-4.29,;-6.44,-3.11,;-4.92,-3.37,)|
Cc1ccncc1NC(=O)Cc1ccccc1N
NC(=O)c1ccncc1NC(=O)Cc1cccc(Cl)c1
Cc1ccncc1NC(=O)C[C@@H](N1CCC(O)CC1)c1ccccc1
Cc1ccncc1NC(=O)Cn2ccc3c2cc(cc3)Cl
Cc1ccncc1NC(=O)CN2c3cc(ccc3OCC2=O)Cl
CC(C)C(C)CC(=O)Nc1cnccc1C
Cc1ccncc1NC(=O)[C@H](C)OC(F)F
Cc1ccncc1NC(=O)CCc1ccn[nH]1
COc1ccccc1OCCNC(=O)C2=CC(=O)Nc3c2ccc(c3)F
COc1ccccc1OC(C)CNC(=O)c1cc(=O)[nH]c2cc(F)ccc12
COc1ccccc1OCC(C)NC(=O)c1cc(=O)[nH]c2cc(F)ccc12
COc1ccccc1OCC(C)NC(=O)c1cc(=O)[nH]c2ccc(F)cc12
CC1(C)Cc2cccc(OCCNC(=O)c3cc(=O)[nH]c4cc(F)ccc34)c2O1
Cc1ccc(c(C)c1)S(=O)(=O)N1CCN(CC1)C(=O)c1cc(=O)[nH]c2cc(F)ccc12
Fc1ccc2[nH]c(=O)cc(C(=O)N3CCN(CC3)S(=O)(=O)c3cccc(Cl)c3)c2c1
c1cc2c(cc1Cl)[C@@H](CO2)C(=O)Nc3cnccc3CO
Clc1ccc2OCCC(C(=O)Nc3nncn3C3CC3)c2c1
Cc1ccncc1N1CCN(C1=O)c1cccc(Cl)c1
O=C(Cc1cccnc1)Nc1cccc(OC2CC(=O)N2)c1
Cc1cc(NC(=O)Cc2cncnc2)cc(OC2CC(=O)N2)c1
Fc1cc(NC(=O)Cc2cncnc2)cc(OC2CC(=O)N2)c1
ClCC(=O)N1CCCN(CC1)S(=O)(=O)Cc1ccccc1
Fc1ccc(F)c(c1)S(=O)(=O)N1CCCN(CC1)C(=O)CCl
Fc1ccccc1S(=O)(=O)N1CCCN(CC1)C(=O)CCl
Fc1cccc(F)c1S(=O)(=O)N1CCCN(CC1)C(=O)CCl
ClCC(=O)N1CCCN(CC1)S(=O)(=O)c1cccs1
Fc1cccc(c1)S(=O)(=O)N1CCCN(CC1)C(=O)CCl
Cc1ccncc1CC(=O)Nc2cccc(c2)Cl
Cc1ccncc1N1CCC(c2cccc(Cl)c2)S1(=O)=O
c1ccc(cc1)NCCNC(=O)C2=CC(=O)Nc3c2cccc3
O=C(NCCOc1ccccc1)c1cc(=O)[nH]c2ccccc12
O=C(N1CCN(Cc2ccccc2)CC1)c1cc(=O)[nH]c2ccccc12
COc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(=O)[nH]c2ccccc12
COc1cccc(c1)N1CCN(CC1)C(=O)c1cc(=O)[nH]c2ccccc12
COc1ccccc1N1CCN(CC1)C(=O)c1cc(=O)[nH]c2ccccc12
Fc1ccc(cc1)N1CCN(CC1)C(=O)c1cc(=O)[nH]c2ccccc12
c1ccc2c(c1)C(=CC(=O)N2)C(=O)N3CCN(CC3)c4ccccc4F
Cc1ccncc1NC(=O)CCc2cccc(c2)F
Cc1ccncc1NC(=O)CN2CCN(CC2)C(=O)C
Cc1ccncc1NC(=O)CN2CCCCC2
Cc1ccncc1NC(=O)Cc1cccc(c1)-c1cn[nH]c1
COc1ccc2CC(N(Cc2c1)C(=O)CCl)c1ccccc1
Cc1nnc(o1)C1Cc2ccccc2CN1C(=O)CCl
Cc1ccncc1N1CCC(C1=O)c1cccc(Cl)c1
Oc1cc(Cl)cc(CN2CCN(CC2)C(=O)CCl)c1
c1cc(cc(c1)Cl)CC(=O)Nc2cccnc2
CN(C(=O)Nc1cnccc1C)c1cccc(Cl)c1
Cc1ccncc1NC(=O)C(CO)c1cccc(Cl)c1
CCCCOc1ccc(cc1CC(=O)Nc2cnccc2C)Cl
Cc1ccnnc1NC(=O)Cc2cccc(c2)Cl
Cc1cc(N)ncc1NC(=O)Cc1cccc(Cl)c1
Cc1ccncc1NC(=O)N(Cc1ccccc1)c1cccc(Cl)c1
Cc1[nH]ncc1NC(=O)Cc1cccc(Cl)c1
COc1cnc(nc1)C#N
Clc1cccc(NC(=O)Cn2nnc3ccccc23)c1
Clc1cccc(NC(=O)Cn2cnc3ccccc23)c1
Cc1nnn(NC(=O)Cc2cccc(Cl)c2)c1C
c1ccc2c(c1)ncn2NC(=O)Cc3cccc(c3)Cl
Clc1cccc(CC(=O)Nn2cnc3ccccc3c2=O)c1
Clc1cccc(CC(=O)Nc2nnn[nH]2)c1
Cc1ccncc1NC(=O)Cc2cc(cnc2)Cl
Cc1ccncc1NC(=O)Cc1cc(OC2CC(=O)N2)cc(c1)C#N
Cc1ccncc1NC(=O)Cc1cc(Cl)cc(OC2CC(=O)N2)c1
CC(C(=O)Nc1cnccc1C)c1cc(Cl)cc(OC2CC(=O)N2)c1
Cc1ccncc1NC(=O)Cc2cccc(c2)F
c1cc(cc(c1)Cl)CC(=O)Nc2cnccc2C3CC3
CCCC(C(=O)Nc1cnccc1C)c1cccc(Cl)c1
Cc1ccncc1NC(=O)Cc2cccc(c2)Br
Cc1ccncc1NC(=O)Cc2cccc(c2)I
Clc1cccc(c1)N1C(=O)NC(C1=O)c1cccnc1
Cc1ccncc1NC(=O)C2(CC2)c3cccc(c3)Cl
Cc1ccncc1NC(=O)C(C)(C)c2cccc(c2)Cl
CS(=O)(=O)c1ccc(cc1)N2CCNCC2
Cc1ccc(cc1)S(=O)(=O)N1CCN(CC1)C(=O)CCl
Cn1ccc(n1)C(=O)NC[C@@H]2CCCO2
COc1ccc(NC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(C)(C)C)c2cccnc2)c(C)c1
CCc1cccc(NC(=O)C(N(C(=O)C=C)c2ccc(cc2)C2(C)CC2)c2cccnc2)c1
CC1(CC1)c1ccc(cc1)N(C(C(=O)Nc1ccc(Br)cc1)c1cccnc1)C(=O)C=C
CN(C(=O)Cn1nnc2ccccc12)c1ccc(Oc2ccc(cn2)C(F)(F)F)cc1
CNC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cccnc1
CSCCCNC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cccnc1
CSCCNC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1ccc(F)cc1)c1cccnc1)C(=O)C=C
COCCNC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1cccnc1)c1cccnc1)C(=O)C=C
CCNC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCC1CCCO1)c1cccnc1)C(=O)C=C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCc1ccccc1)c1cccnc1)C(=O)C=C
CC(C)(C)c1ccc(cc1)N(C(C(=O)Nc1ccc2OCOc2c1)c1cccnc1)C(=O)C=C
COc1ccc(NC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(C)(C)C)c2cccnc2)c(OC)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)C=C
CC(C)(C)NC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cncc(Cl)c1
CC(C)(C)NC(=O)C(N(C(=O)C=C)c1ccc(CCC#N)cc1)c1cccnc1
Cc1cc(O)c2C(=O)C3CC(O)(C4=C3C(=O)c3cccc(O)c3C4=O)c2c1 |c:12,TLB:26:25:9:13.12,7:6:9:13.12,THB:23:12:9:5.25.6,14:13:9:5.25.6|
Cc1cc(O)c2C(=O)C=CC(=O)c2c1-c1c(C)cc2C(=O)C=CC(=O)c2c1O |c:8,23,(4.47,.97,;5.81,1.74,;5.81,3.28,;7.14,4.05,;7.14,5.59,;8.47,3.28,;9.85,4.1,;9.83,5.64,;11.25,3.31,;11.25,1.71,;9.85,.92,;9.85,-.58,;8.47,1.74,;7.14,.97,;7.14,-.57,;8.47,-1.34,;9.81,-2.11,;8.47,-2.88,;7.14,-3.65,;7.16,-5.25,;8.51,-6.01,;5.78,-6.07,;4.39,-5.26,;4.4,-3.66,;3.08,-2.88,;5.81,-2.88,;5.81,-1.34,;4.47,-.57,)|
CC(C)(C)N1C=CN(C1[Au]Cl)C(C)(C)C |c:5|
CCP(CC)(CC)=[Au]S[C@@H]1O[C@H](COC(C)=O)[C@@H](OC(C)=O)[C@H](OC(C)=O)[C@H]1OC(C)=O
OC[C@H]1O[C@H](S[Au])[C@H](O)[C@@H](O)[C@@H]1O
O\C(=C(\C#N)C(=O)Nc1ccc(F)cc1)c1ccc(Cl)cc1
Oc1ccccc1CN(C[C@@H]1CCCO1)C(=O)CNC(=O)C=C
CC(C)(C)NS(=O)(=O)c1ccccc1CNC(=O)C=C
CNS(=O)(=O)c1ccccc1CNC(=O)C=C
O[C@]1(CN(Cc2ccccc2)C(=O)CNC(=O)C=C)CN2CCC1CC2 |wU:1.1,wD:1.0,TLB:2:1:21.22:24.25,0:1:21.22:24.25,(3.43,-1,;3.1,-2.51,;4.64,-2.52,;5.42,-1.19,;6.96,-1.21,;7.72,-2.55,;9.26,-2.56,;10.02,-3.9,;9.24,-5.23,;7.7,-5.22,;6.94,-3.88,;4.67,.15,;5.45,1.47,;3.13,.16,;2.37,1.5,;.83,1.52,;.05,.19,;.07,2.86,;-1.47,2.87,;3.39,-3.93,;1.99,-3.28,;2.25,-1.34,;1.79,-.21,;1.72,-1.89,;.22,-2.54,;.42,-3.95,)|
C=CC(=O)NCCC(=O)N(Cc1ccccc1)Cc1nc2ccccc2c(=O)[nH]1
CN(C)CCNC(=O)[C@@H](Cc1ccccc1)NC(=O)C=C
O[C@H](CNC(=O)c1cc(NC(=O)C=C)ccc1O)c1ccc2ccccc2c1
ClCC(=O)Nc1cccc(c1)N1CCCC1=O
Fc1cccc(F)c1S(=O)(=O)N1CCN(CC1)C(=O)CCl
ClCC(=O)N1CCN(CC1)S(=O)(=O)c1cccs1
Fc1cccc(c1)S(=O)(=O)N1CCN(CC1)C(=O)CCl
ClCC(=O)N1CCN(Cc2cccs2)CC1
ClCC(=O)N1CCN(Cc2ccsc2)CC1
CC(C)(C)NC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(C)(C)C)c1cccnc1
ClCC(=O)N1CCN(CC1)S(=O)(=O)c1ccc(Cc2cccc3ccccc23)cc1
ClCC(=O)N1CCN(CC1)C1(CC1)c1cccc(Cl)c1
CC1CN(Cc2cccc(Cl)c2)CCN1C(=O)CCl
ClCC(=O)N1CCN(Cc2cccc(Cl)c2)CC1
ClCC(=O)N1CCN(Cc2cnc(Cc3ccccc3)s2)CC1
COc1ccc(cc1OC)C1CC(=NN1C(=O)CCl)c1ccccc1 |c:13|
ClCC(=O)N1CCN(Cc2cccc3ccccc23)CC1
COCc1cc(Cl)cc(CN2CCN(CC2)C(=O)CCl)c1
COCCc1ccc(Cl)cc1CN1CCN(CC1)C(=O)CCl
CCc1cccc(NC(=O)C(N(C(=O)C=C)c2cc(on2)C(C)(C)C)c2cccnc2)c1
CCc1cccc(NC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(C)OC)c2cccnc2)c1
CC(C)(C)NC(=O)C(N(C(=O)C=C)c1cc(on1)C(C)(C)C)c1cccnc1
COc1ccc(NC(=O)C(N(C(=O)C=C)c2ccc(cc2)C(F)(F)F)c2cccnc2)cc1
CCc1cccc(NC(=O)C(N(C(=O)C=C)c2ccc3ncsc3c2)c2cccnc2)c1
CCc1cccc(C)c1NC(=O)C(N(C(=O)C=C)c1ccc(cc1)C(F)(F)F)c1cccnc1
COc1ccc(cc1OC)C1CC(=NN1C(=O)CCl)c1cccs1 |c:13|
COc1ccccc1OCCNC(=O)C2=CC(=O)Nc3c2cccc3
Cc1cc(C)c(C)c(c1C)S(=O)(=O)N1CCN(CC1)C(=O)c1cc(=O)[nH]c2ccccc12
c1ccc(cc1)N2CCN(CC2)C(=O)C3=CC(=O)Nc4c3cccc4
O[C@@H](CN(Cc1ccccc1)C(=O)CNC(=O)C=C)c1cccs1
Cc1[nH]c2c(CNC(=O)c3ccc(CNC(=O)C=C)cc3)cc(C)cc2c1C
Brc1ccsc1CN(CCN1CCOCC1)C(=O)CNC(=O)C=C
OC[C@@H](NC(=O)c1ccc(CNC(=O)C=C)cc1)c1ccc(Br)c(F)c1
Oc1ccc(cc1NC(=O)C=C)C(=O)NC[C@H](Cc1ccccc1)c1ccccn1
Oc1ccc(O)c(CN2CCN(CC2)C(=O)CCl)c1
NS(=O)(=O)CCc1ccccc1CN1CCN(CC1)C(=O)CCl
Cc1ccc(cc1)S(=O)(=O)NC1CCN(CC1)C(=O)CCl
Cc1ccc(C)c(c1)S(=O)(=O)N1CCN(CC1)C(=O)CCl
Cc1ccnc2[nH]c(CC3CCN(CC3)C(=O)CCl)nc12
ClCC(=O)N1CCC(CC1)c1nc(nc2ccccc12)-c1cccnc1
ClCC(=O)N1CCN(CC1)C(c1ccccc1)c1ccccc1
NS(=O)(=O)c1ccc2CCN(CC3CCN(CC3)C(=O)CCl)Cc2c1
ClCC(=O)N1CCN(Cc2cc(Cl)ccc2CNC(=O)[C@@H]2CCCOC2)CC1
ClCC(=O)N1CCN(Cc2cc(Cl)ccc2CNC(=O)N2CCOCC2)CC1
ClCC(=O)N1CCN(Cc2cc(Cl)cc(Cl)c2)CC1
CS(=O)(=O)N1CCc2ccc(CN3CCN(CC3)C(=O)CCl)cc2C1
ClCC(=O)N1CCN(Cc2cccc(CNC(=O)N3CCOCC3)c2)CC1
CC(=O)Nc1ccc(cc1CN1CCN(CC1)C(=O)CCl)C#N
CC(CCc1ccccc1)N1CCN(CC1)C(=O)CCl
Cc1cccc(CC2CCN(CC2)C(=O)CCl)c1
ClCC(=O)N1CCN(CC1)C(C1CCOCC1)c1ccccc1
ClCC(=O)N1CCN(CC1)C(C1CCCCC1)c1ccccc1
CCNc1ncc(cc1CN1CCN(CC1)C(=O)CCl)C#N
ClCC(=O)N1CCN(Cc2cc(cc3ccccc23)C#N)CC1
COc1cc(CN2CCN(CC2)C(=O)CCl)c2ccccc2c1
NS(=O)(=O)c1ccc(cc1)N1CCC(CC1)Nc1ccc(F)cc1
NS(=O)(=O)c1ccc(cc1)N1CCC(CC1)N1CCCCCC1
NS(=O)(=O)c1ccc(cc1)N1CCC(CC1)[C@@H]1CCCO1
Cn1nncc1CC(=O)NC(c1nc2ccccc2n1C)c1ccccc1
Cc1ccncc1NC(=O)CN(C)S(=O)(=O)c2cccc3c2nccc3
Cc1ccn2c(c(nc2c1)-c1ccc(F)cc1)-c1ccc2[nH]ncc2c1
CC(NC(=O)CCl)c1cc(Cl)cc(c1)-c1ccc(cc1)S(N)(=O)=O
OCC(NC(=O)CCl)c1cccc(Cl)c1
CC(NC(=O)CCl)c1cc(F)cc(Cl)c1
CC1C(O)CCCN1Cc1ccccc1
CCC(C)(C)CCN(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
Cc1cc(C)nc(NC2CCN(CC2)C(=O)CCl)n1
Cc1cc(Cl)cc(CC2CCN(CC2)C(=O)CCl)c1
Nc1cccc(c1)C1CN(Cc2ccccc12)C(=O)CCl
ClCC(=O)N1CC(c2cccc(c2)C#N)c2ccccc2C1
Cc1cccc(c1)C1CN(Cc2ccccc12)C(=O)CCl
CC(C)C[C@@H]1CN(CCN1Cc1cccc(Cl)c1)C(=O)CCl
ClCC(=O)N1CC2CC1CN2Cc1cccc(Cl)c1 |THB:2:4:7:9.10,11:10:4.5:7|
ClCC(=O)N1CCN(Cc2cccc(Cl)c2)C[C@@H]1Cc1ccccc1
CC(=O)NCCc1c[nH]c2ccc(O)cc12
Oc1ccc(Cl)cc1C(=O)Nc1cnccc1Cl
Clc1ccc(-c2ccccc2)c(c1)C(=O)Nc1cccnc1
CS(=O)(=O)N1CCN(CC1c1ccccc1)C(=O)CCl
ClCC(=O)Nc1nc2c(cccc2s1)S(=O)(=O)NCCc1ccccc1
CC(=O)NCCc1c[nH]c2c(CN3CCN(CC3)C(=O)CCl)cccc12
CS(=O)(=O)N(CCc1ccccc1)CC1CCN(CC1)C(=O)CCl
COc1cc(Cl)cc(OC(=O)Nc2cccnc2)c1
c1cc(cc(c1)Cl)N(CCN2CCOCC2)C(=O)Nc3cccnc3
c1cc(cc(c1)Cl)N(CCC2CCCCC2)C(=O)Nc3cccnc3
Cc1c(cncc1NC(=O)Cc2cccc(c2)Cl)N
Cc1ccncc1NC(=O)Cc2cccc(c2)Cl
Cc1ccncc1NC(=O)Nc2cccc(c2)Cl
CC(C(=O)Nc1cnccc1C)c1cccc(Cl)c1
Cc1c(cncc1NC(=O)Cc2cccc(c2)C#N)N
Cc1ccncc1NC(=O)Cc2cccc(c2)C#N
CC(C(=O)Nc1cnccc1C)c1cccc(c1)C#N
Cc1ccncc1NC(=O)Nc1cccc(c1)C#N
Clc1cc(NC(=O)Nc2cccnc2)cc(c1)C#N
Nc1cncc(NC(=O)Nc2cccc(c2)C#N)c1
O=C(Nc1c[nH]c2ncccc12)Nc1cccc(c1)C#N
O=C(Cc1cncc2ccccc12)Nc1cccc(c1)C#N
c1ccc(cc1)NC(=O)Cc2cncc3c2cccc3
C[C@@H](NC(=O)c1cc(NC2CN(C2)C(=O)OC(C)(C)C)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CCN(CC2)C(=O)OC(C)(C)C)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC(=O)C2CN(C2)C(=O)OC(C)(C)C)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC(=O)C2CCN(CC2)C(=O)OC(C)(C)C)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CCNCC2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC(=O)C2CNC2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC(=O)C2CCNCC2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CCN(C)CC2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CN(C)C1)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CN(C)C2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(CNCC(O)=O)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(CNC2CNC2)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(CN2CC(C2)C(O)=O)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(CN2CCC(CC2)C(O)=O)ccc1C)c1cccc2ccccc12
C[C@@H](NCc1cccc(N)c1)c1cccc2ccccc12
C[C@@H](NS(=O)(=O)c1cc(N)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1F)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1Cl)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1C(F)(F)F)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1C=C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1Br)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ncc1Br)c1cccc2ccccc12
C[C@@H](NC(=O)c1c[nH]c2ccccc12)c1cccc2ccccc12
C[C@@H](NC(=O)c1cccc2[nH]ccc12)c1cccc2ccccc12
C[C@@H](NC(=O)c1ccc2cc[nH]c2c1)c1cccc2ccccc12
C[C@@H](NC(=O)c1c(C)ccc2[nH]ccc12)c1cccc2ccccc12
C[C@@H](NC(=O)c1c(C)ccc2n(CC3CNC3)ccc12)c1cccc2ccccc12
C[C@@H](NC(=O)c1nc(N)ccc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CNC2)ncc1C)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(ncc1C)N(C)C1CNC1)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1Cl)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1Cl)N(C)C1CNC1)c1cccc2ccccc12
Cc1ccc(N)cc1C(=O)NC(CO)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1C)c1c(O)ccc2ccccc12
Cc1ccc(N)cc1C(=O)N[C@H](CCO)c1cccc2ccccc12
CC[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1c(O)ccc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1c(OC2CNC2)ccc2ccccc12
CN(C1CNC1)c1ccc(C)c(c1)C(=O)NC(CO)c1cccc2ccccc12
CN(C)C(=O)C[C@@H](NC(=O)c1cccc(c1)N(C)C1CNC1)c1cccc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1C)c1csc2ccccc12
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cn(C)c2ccccc12
CC(NC(=O)c1cc(ccc1C)[N+]([O-])=O)c1cccc2cc[nH]c12
CC(NC(=O)c1cc(N)ccc1C)c1cccc2cc[nH]c12
CC(NC(=O)c1cc(N)ccc1C)c1c[nH]c2ccccc12
CC(NC(=O)c1cc(N)ccc1C)c1cccc2ccn(C)c12
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cccc2cccnc12
CC(NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1cccc2cc[nH]c12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1ccc2sccc2c1
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1cccc2n(CC3CCC3)ccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1csc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1Cl)c1csc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1Cl)N(C)C1CNC1)c1csc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1cccc2[nH]c3ccccc3c12
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1csc2ccccc12
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc2[nH]c3ccccc3c12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1nccc2ccccc12
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C1CNC1)c1ccccc1-c1cccs1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1Cl)c1cccc(c1)-c1cccs1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1cccs1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccsc1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1cc[nH]c1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CCNCC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CCOCC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC2CCN(C)CC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNCC2CCNCC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC2CCCC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CCCC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(C)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(s1)C(O)=O
COC(=O)c1ccc(s1)-c1cccc(c1)[C@@H](C)NC(=O)c1cc(NC2CNC2)ccc1C
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(s1)C(=O)NC[C@H]1CCCO1
CNC(=O)c1ccc(s1)-c1cccc(c1)[C@@H](C)NC(=O)c1cc(NC2CNC2)ccc1C
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(s1)C(=O)NCC1CCO1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CC[C@@H](O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CC[C@@H](C)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CCC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CC[C@H](O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(Br)c1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@@H]2CCOC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@H]2CCOC2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC2CCC(O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC(C)=O)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC2CCNC2=O)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC2CNC(=O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@@H]2CC[C@H](O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@@H]2CC[C@@H](O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@H]2CC[C@@H](O)C2)s1
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@H]2CC[C@H](O)C2)s1
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cccc(c1)-c1ccc(CNC(=O)OC(C)(C)C)s1
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cccc(c1)-c1ccc(CN)s1
C[C@@H](NC(=O)c1cc(N)ccc1C)c1cccc(c1)-c1ccc(CNC(=O)C2CCCC2)s1
C[C@@H](NC(=O)c1cc(NC(C)=O)ccc1C)c1cccc(c1)-c1ccc(CNC(C)=O)s1
C[C@@H](NC(=O)c1cc(NC(C)=O)ccc1C)c1cccc(c1)-c1ccc(CN[C@H]2CC[C@@H](O)C2)s1
c1cc(c2c(c1)NCC2)C(=O)Oc3cc(cnc3)Cl
c1cc(cc(c1)S(=O)(=O)n2ccc3c2ccc(c3)C(=O)Oc4cc(cnc4)Cl)[N+](=O)[O-]
COc1cccc2[nH]c(cc12)C(=O)Oc1cncc(Cl)c1
Clc1cncc(OC(=O)c2cccc3n(CC=C)ccc23)c1
Clc1cncc(OC(=O)c2cccc3n(CC=C)cc(CC=C)c23)c1
Cc1c[nH]c2cccc(C(=O)Oc3cncc(Cl)c3)c12
Cc1ccc2[nH]ccc2c1C(=O)Oc1cncc(Cl)c1
Cc1cc(C(=O)Oc2cncc(Cl)c2)c2cc[nH]c2c1
Fc1cc(C(=O)Oc2cncc(Cl)c2)c2cc[nH]c2c1
Clc1cncc(OC(=O)c2cccc3[nH]cnc23)c1
Cc1nc2c(cccc2[nH]1)C(=O)Oc1cncc(Cl)c1
Clc1cncc(OC(=O)c2cccc3ncoc23)c1
Clc1cncc(OC(=O)c2cccc3NCCOc23)c1
Clc1cncc(NC(=O)c2cccc3[nH]ccc23)c1
Clc1cccc(OC(=O)c2cccc3[nH]ccc23)c1
Cc1ncc(Cl)cc1OC(=O)c1cccc2[nH]ccc12
Cc1c(cncc1Cl)OC(=O)c2cccc3c2cc[nH]3
Cc1ncc(OC(=O)c2cccc3[nH]ccc23)cc1Cl
Cc1ncc(OC(=O)c2cccc3[nH]cnc23)cc1Cl
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](c2nc3ccccc3s2)O)NC(=O)c4cc5c([nH]4)cccc5OC
OB(O)c1cc(cc(c1)[N+]([O-])=O)C(=O)Oc1ccc(OC(=O)c2cc(cc(c2)[N+]([O-])=O)B(O)O)cc1
Nc1cc(cc(c1)C(=O)OCc1cccc(c1)B(O)O)B(O)O
OB(O)c1cc(O)cc(c1)C(O)=O
OB(O)c1cc(cc(c1)[N+]([O-])=O)C(=O)Oc1c(Cl)cc(Cl)cc1[N+]([O-])=O
CCOC(=O)\C=C\[C@@H](C[C@H]1CCNC1=O)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)\C=C\C(=O)OC1CC1
COC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)NC(=O)C(C)(C)C
Cl\[#6](Cl)=[#6](\Cl)-[#6](=O)-[#8]-c1ccc(cc1)S(=O)(=O)c1ccc(-[#8]-[#6](=O)-[#6](\Cl)=[#6](\Cl)Cl)cc1Cl
FC(F)(F)c1nnc(SC(=O)C2CCC(O2)C#Cc2ccccc2)[nH]1
Cc1noc(NC(=O)c2ccc(s2)-c2cc(nn2C)C(F)(F)F)c1[N+]([O-])=O
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)c1cc(C)on1)C(C)C
O[C@H]1CO[C@@H](OC[C@H]2O[C@@H](Oc3c(oc4cc(O)cc(O)c4c3=O)-c3ccc(O)c(O)c3)[C@H](O)[C@@H](O)[C@@H]2O)[C@H](O)[C@H]1O
OC[C@H]1OC(Oc2c(oc3cc(O)cc(O)c3c2=O)-c2ccc(O)c(O)c2)[C@H](O)[C@H](O)[C@H]1O
CC1CCN(CC1)C(=O)c1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
O=C(N1CCCC1)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
CN1C(=O)C(=O)c2cc(ccc12)C(=O)N1CCOCC1
O=C(N1CCCC1)c1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
O=C(N1CCCCC1)c1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
CC(C)C[C@@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](CC1CCNC1=O)C=O
CC(C)C[C@@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](CC1CCNC1=O)C(O)S([O-])(=O)=O
CC(C)C[C@@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](CC1CCNC1=O)C(=O)C(=O)NC(C)C
CC(C)C[C@@H](NC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)OCc1ccccc1)C(=O)N[C@H](CC1CCNC1=O)C=O
CC(C)C[C@@H](NC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)OCc1ccccc1)C(=O)N[C@H](CC1CCNC1=O)C(=O)C(=O)NC(C)C
c1cc(c(cc1[C@H]2[C@@H](C(=O)c3c(cc(cc3O2)O)O)O)O)O
CC(C)C[C@@H]1[C@@H](CC(=O)OCc2ccccc2)Cc2cn(CCCNC(=O)CC[C@H](NC1=O)C=O)nn2
Cc1ccc(SSc2nccs2)cc1
CC(=O)Nc1cnc(SSc2ccccc2[N+]([O-])=O)s1
[O-][N+](=O)c1ccccc1SSc1nccs1
COC(=O)c1c[nH]c(SSc2ccccc2[N+]([O-])=O)n1
Fc1ccc(SSc2nccs2)cc1
O=C[C@H](CC1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc2ccccc2[nH]1
CC(C)[C@H](NC(=O)c1cncc(F)c1)C(=O)N[C@@H](Cc1ccccc1)C(=C)N[C@@H](CC1CCNC1=O)C=O
CC(C)[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC1CCNC1=O)C=O
O=C[C@H](CC1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2OCOc2c1
Fc1ccc2[nH]c(cc2c1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC1CCNC1=O)C=O
CC(C)C(=O)Nc1ccc(cc1)N([C@H](C(=O)NCc1ccccc1)c1ccc(Cl)c(F)c1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N([C@H](C(=O)NCc1ccccc1)c1ccc(O)cc1)C(=O)Cn1nnc2ccccc12
CC(C)C(=O)Nc1ccc(cc1)N([C@H](C(=O)NCc1ccccc1)c1cccc(F)c1)C(=O)Cn1nnc2ccccc12
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NC1CCCC1)c1cccnc1)C(=O)c1c[nH]cn1
O=C(Cn1nnc2ccccc12)N([C@H](C(=O)NCc1ccccc1)c1ccsc1)c1ccc(NC(=O)C2CC2)cc1
CC(C)C[C@H](NC(=O)OC1CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O
CC(C)C[C@H](NC(=O)OC1CCN(CC1)S(C)(=O)=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O
CC(C)C[C@H](NC(=O)OC1(Cc2ccccc2)CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O
CC(C)C[C@H](NC(=O)OCCc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O
CC(C)(C)NC(=O)C(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@H](Cc1cccc2ccccc12)NC(=O)OCc1ccc(OCN2CCOCC2)cc1
COC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC(C)C
CC(C)C[C@H](NC(=O)[C@H](CN(C)C)NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC(C)(C)C
CC(C)C[C@H](NC(=O)[C@H](CN1CCOCC1)NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC(C)C
CC(C)C[C@H](NC(=O)[C@H](CN1CCC(F)CC1)NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC(C)C
O=C(N[C@@H](C[C@@H]1CCCNC1=O)C(=O)C(=O)NC1CCCCC1)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2o1
O=C(N[C@@H](C[C@@H]1CCCNC1=O)C(=O)C(=O)NCc1ccccc1)[C@H](Cc1ccccc1)NC(=O)c1cc2ccccc2[nH]1
O=C(N[C@@H](C[C@@H]1CCCNC1=O)C(=O)C(=O)NCc1ccccc1)[C@H](Cc1ccccc1)NC(=O)c1cnc2ccccc2n1
O=C(N[C@@H](C[C@@H]1CCCNC1=O)C(=O)C(=O)NCc1ccccc1)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1
O=C(N[C@@H](C[C@@H]1CCCNC1=O)C(=O)C(=O)NCc1ccccc1)[C@H](CC1CCCCC1)NC(=O)c1cnc2ccccc2n1
Cc1c(cccc1O)C(=O)N[C@@H](CSc2ccccc2)[C@@H](C[N@@]3C[C@H]4CCCC[C@H]4C[C@H]3C(=O)NC(C)(C)C)O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1cccc2[nH]c(cc12)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C
CC(C)[C@H](NS(C)(=O)=O)C(=O)N1C[C@@H]2[C@H]([C@@H]1C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@@H]2[C@H]([C@@H]1C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C
CC1([C@@H]2[C@H]1[C@H](N(C2)C(=O)[C@H](C(C)(C)C)NC(=O)C(F)(F)F)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)C
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NC(CC1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1nc2cccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1nc2ccncc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1nc2ncccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(O)C#N
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NC(CC1CCNC1=O)C(O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC(C)C)C(=O)NC(CC1CCNC1=O)C(O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@H](O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)\C=C\S(C)(=O)=O |r|
CC(C)C[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2nc([nH]c12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H]([C@@H]1Cc2ccccc2O1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](C1Cc2ccccc2C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](Cc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)OC(C)(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C1CCCCC1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)c1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1CCC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@H]2C([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC#C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
Fc1cc(Cl)ccc1\C=C\C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)c1ccccc1 |r|
Fc1cc(Cl)ccc1\C=C\C(=O)N1NCCC[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](Cc1cnc[nH]1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1cnc[nH]1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1cncn1C)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1cn(C)cn1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1cccnc1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](Cc1cc(=O)[nH]c2ccccc12)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1cc[nH]n1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1n[nH]c2ccccc12)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NC(CC1CC(=O)Nc2ccccc12)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc[nH]c1=O)C#N |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)n1ccc2cc[nH]c2c1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)N1CCc2cc[nH]c2C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@@H](CC1CC1)N1CCc2cc[nH]c2C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)n1ccc2[nH]cnc2c1=O |r|
CN1CCCC11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC11CCN([C@@H](CC2CC2)C(=O)N[C@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC11CCN([C@@H](CC2CC2)C(=O)N[C@H](C[C@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC[C@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC[C@@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC[C@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@]1(CCc2cccnc2C1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2CCCC2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](NC(C)(C)C)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@H](NC(C)(C)C)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NCC(F)(F)F)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(Nc1ccccc1)C#N |r,w:31.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(N[C@@H](C)c1ccccc1)C#N |r,w:31.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@H](C#N)N1CCCC1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](C#N)N1CCCC1 |r|
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C=O
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC1CCNC1=O)C(N)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](CC1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)c1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)C#N)c1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)C#N)c1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@H](O)C#N)c1ccccc1 |r|
CCCN1C(=O)OC([C@H](C[C@@H]2CCNC2=O)NC(=O)[C@H](CC(C)C)NC(=O)c2cc3c(OC)cccc3[nH]2)C1=N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C1OC(=O)N(C(C)C)C1=N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C1OC(=O)N(C1=N)c1ccccc1 |r|
CC(C)C[C@H](NC(=O)c1cc2c(OC(F)(F)F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1nc2c(OC(F)(F)F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)C[C@@](C)(O)c1ccc(Cl)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)C[C@](C)(O)c1ccc(Cl)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)C[C@](O)(c1ccccc1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)C[C@@](O)(c1ccccc1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)NC(=O)c1cc2c(cccc2[nH]1)C1CC1 |r|
CCOc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CCCOc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)OCC1CCC(F)(F)CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C12CC(C1)C2 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C12CC(C1)C2 |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CC1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)CCOCC2 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@]2(CC1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)CCCCC2 |r|
CC[C@H]1CN([C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC(C)(C)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC(C)(C)C[C@H]1C(=O)N[C@@H](C[C@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@]2(CCC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CCCC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@]2(CCCC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CO[C@@H]1C[C@H](N(C1)C(=O)c1cc2c(OC)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NC(C#N)c1cccnc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccn1)C#N |r|
Cc1ccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1N |r|
Cc1ccn([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1N |r|
Cc1ccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1NCC(F)(F)F |r|
Cc1ccn([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1NCC(F)(F)F |r|
FC(F)(F)CN[C@H]1CC[C@@H]2SC[C@H](N2C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
O=C(N[C@H]1CC[C@@H]2SC[C@H](N2C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)OCc1ccccc1 |r|
Cc1cc(no1)C(=O)N[C@H]1CC[C@@H]2SC[C@H](N2C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
Nc1cccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c1=O |r|
Nc1cccn([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c1=O |r|
FC(F)(F)CNc1cccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c1=O |r|
CC(C)(C)OC(=O)N1CCCC11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCC[C@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCC[C@@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCC[C@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCC[C@@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)N1CCC2(CCCN2)C1=O |r|
CC(C)(C)OC(=O)N1CCCC[C@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCCC[C@@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)N1CC[C@@]2(CCCCN2)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)N1CC[C@]2(CCCCN2)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@@H](CC1CC1)N1CC[C@@]2(CCCCN2)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@@H](CC1CC1)N1CC[C@]2(CCCCN2)C1=O |r|
O=C(N[C@H]1CC[C@@H]2SC[C@H](N2C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)OCC1c2ccccc2-c2ccccc12 |r|
N[C@H]1CC[C@@H]2SC[C@H](N2C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
C[Si](C)(C)CCOCn1cnc2ccn([C@H](CC3CC3)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(=O)c12 |r|
C[Si](C)(C)CCOCn1cnc2ccn([C@@H](CC3CC3)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(=O)c12 |r|
O=C(CNc1ccc2CC[C@@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)n2c1=O)Oc1ccccc1 |r|
O=C(CNc1ccc2CC[C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)n2c1=O)Oc1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@]1(C[C@H]2CC[C@@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@]1(C[C@H]2CC[C@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N |r,TLB:30:29:22.23:25.26,33:28:22.23:25.26|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
O=C(N[C@@H](CC1CC1)C(=O)N[C@@]1(C[C@H]2CC[C@@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N)OCc1ccccc1 |r|
O=C(N[C@@H](CC1CC1)C(=O)N[C@]1(C[C@H]2CC[C@@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N)OCc1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](C1CC2CC2C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
OC(=O)CNc1ccc2CCC(C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)n2c1=O |r,w:11.11|
CC(C)(C)OC(=O)Nc1cccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c1=O |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](NCc1ccccc1)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@H](NCc1ccccc1)C#N |r|
CC(C)C[C@H](NC(=O)c1cc2c(OC(F)F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CCNC(C#N)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
CCN[C@H](C#N)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
CCN[C@@H](C#N)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2N[C@H](Cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2N[C@@H](Cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)NC(=O)c1cc2c(OCCN3CCOCC3)cccc2[nH]1 |r|
Clc1ccc2[nH]c(cc2c1)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
Clc1cccc2cc([nH]c12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CCO[C@@H]1C[C@H](N(C1)C(=O)c1cc2c(OC)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)SC |r|
COc1cccc2[nH]c(cc12)C(=O)N1CCc2ccccc2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CCCNC(=O)OC(C#N)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(OC(=O)NC(C)C)C#N |r|
Cc1ccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1NC(=O)OC(C)(C)C |r|
Cc1ccn([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1NC(=O)OC(C)(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)O[Na] |r|
CC(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1nccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
O=C(N[C@@H](C[C@@H]1CCCNC1=O)C#N)[C@H](CC1CC1)NC(=O)c1cc2cnccc2[nH]1 |r|
Clc1ccc2cc([nH]c2c1)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1ccc(Cl)c2[nH]c(nc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1cccc2cc([nH]c12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](CC1CCCNC1=O)C#N |r|
Fc1cc(F)cc(CCC(=O)N[C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NCC(O)=O)C#N |r,w:31.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CN[C@@H](C[C@@H]1CCNC1=O)C#N)CC(C)(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CC1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)CCCCC2 |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)NC(=O)c1cc2CCCCc2[nH]1 |r|
Clc1nccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1cc2cc([nH]c2cn1)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CCC2)CC1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
CC(C)(C)C[C@H](NC(=O)c1cc2cccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CC(F)(F)C2)CC1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
CC(C)(C)C[C@H](NC(=O)c1cc2ccc(Cl)c(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1cccc2cc([nH]c12)C(=O)N1CC2(CCC2)CC1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1cccc2cc([nH]c12)C(=O)N1CC2(CC1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)CCCCC2 |r|
Clc1ccc2cc([nH]c2c1)C(=O)N1CC2(C[C@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)CCCCC2 |r|
CC(C)(C)C[C@H](NC(=O)c1cc2c(Cl)ccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1ccc(Cl)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1c(Cl)ccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
FC1(F)CC2(C1)CC(N(C2)C(=O)c1cc2cccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
CC(C)(C)C[C@H](NC(=O)c1cc2ccc(Cl)cc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O)c1ccccc1 |r|
CCCCC1CCC(CC1)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |wU:22.22,24.24,wD:14.14,(-2.6,-5.27,;-1.26,-6.04,;.07,-5.27,;1.41,-6.04,;2.74,-5.27,;2.74,-3.73,;4.07,-2.96,;5.41,-3.73,;5.41,-5.27,;4.07,-6.04,;6.73,-2.93,;8.07,-3.67,;8.1,-5.21,;9.39,-2.88,;10.74,-3.62,;10.77,-5.16,;12.12,-5.91,;12.15,-7.45,;13.44,-5.11,;12.06,-2.83,;12.03,-1.29,;13.41,-3.57,;14.73,-2.78,;14.7,-1.24,;16.01,-.44,;17.41,-1.09,;18.46,.03,;17.72,1.38,;16.2,1.09,;15.08,2.14,;16.07,-3.52,;16.1,-5.06,)|
CC(C)C[C@H](NC(=O)OCC1CCC(F)(F)CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
C[C@H](NC(=O)C(N(C(=O)CN=[N+]=[N-])c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)CF)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C=CC(=O)N(C(C(=O)NCc1ccccc1)c1cccnc1)c1ccc(cc1)-c1ccccc1
C[C@H](NC(=O)C(N(C(=O)C=C)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
CC#CC(=O)N(C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1)c1ccc(cc1)-c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccccc1)c1cnccn1)c1ccccc1 |r|
ClCC(=O)N(C(C(=O)NC1CCCCC1)c1cccnc1)c1ccc(cc1)-c1ccccc1
C[C@H](NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1ccccc1)c1cnccn1)c1ccccc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-n1cccc1)c1cccnc1)c1ccccc1 |r|
ClCC(=O)N(C(C(=O)NC1CC1)c1cccnc1)c1ccc(cc1)-c1ccccc1
ClCC(=O)N(C(C(=O)NC1CCCC1)c1cccnc1)c1ccc(cc1)-c1ccccc1
CCOC(=O)\C=C\C(=O)N(C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1)c1ccc(cc1)-c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)\C=C\CN(C)C)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)C(Cl)=C)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](Cl)C(=O)N(C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1)c1ccc(cc1)-c1ccccc1 |r|
C[C@H](NC(=O)[C@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccc(Br)cc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccc(Br)cc1 |r|
C[C@@H](CCc1ccccc1)NC(=O)[C@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1 |r|
C[C@@H](CCc1ccccc1)NC(=O)[C@@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1 |r|
C[C@H](NC(=O)[C@H](N(C(=O)C(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccc(Br)cc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)C(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccc(Br)cc1 |r|
C[C@H](NC(=O)C(N(C(=O)C(C)(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)C(Cl)(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)C(F)(F)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)C(Cl)(Cl)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@H](N(C(=O)C(Cl)(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)C(Cl)(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@H](N(C(=O)C(Br)(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)C(Br)(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)CN(C)C |r|
CCC(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1CCCCC1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1(C)CCCCC1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1(C)CCC1 |r|
COc1ccccc1CC(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1ccccc1Cl |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1(C)CCN(C)CC1 |r|
CC[C@H](C)C(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
CC[C@@H](C)C(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1(C)CC1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cnccc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cccnc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)[C@@H]1CCCN1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)[C@H]1CCCN1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cccnc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)C1CCN(C)CC1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccncc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccccn1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)[C@H]1CCCCN1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cn(C)nc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cnn(C)c1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccnn1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1ccn(C)n1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cnn(C)c1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cncn1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)nn(C)c1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1cn(C)cn1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1ccccc1CN(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)ccnc1CN(C)C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)ccnc1C |r|
CCOc1nccc(C)c1C(=O)OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1c(C)cc(cc1C)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1c(C)cccc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1c(C)cccc1Cl |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)cncc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)nc(C)nc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1c(C)ncnc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1c(C)cccc1F |r|
COc1cc(C)c(CC(=O)OCC(=O)[C@H](C[C@@H]2CCNC2=O)NC(=O)[C@H](CC(C)C)NC(=O)c2cc3c(OC)cccc3[nH]2)c(C)c1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)Cc1c(C)cc(F)cc1C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(C)nc(nc1C)C1CCOCC1 |r|
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COP(=O)(O)O)NC(=O)c2cc3c([nH]2)cccc3OC
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
CC(C)(C)C[C@H](NC(=O)CN1CCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1c(Cl)cccc1Cl)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1cccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F
COc1ccc(c2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
Cc1c(sc2nccn12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COC(C1CCCCC1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COC(C1CCCCC1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@H](C[C@@H]1CCNC1=O)C#N
CCn1nc(C)c(Br)c1C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)CC1CC(F)(F)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CCC(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1ccc(F)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1c(F)ccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1cccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(F)c12
COc1c(F)cc(F)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1c(F)ccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(F)c12
COc1ccc(F)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1cccc2[nH]c(C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(F)c12
COc1c(F)cc(F)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1csc(n1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)C1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)C1CCCCC1)C(=O)N[C@H](C[C@@H]1CCNC1=O)C#N
CC(C)OCC(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)COC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(CC(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
CN(C)[C@H](C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)c1ccccc1
CC(C)(C)C[C@H](NC(=O)[C@H]1CC[C@@H](CC1)C#N)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |wU:20.20,12.15,wD:22.22,5.5,9.8,(-3.99,-2.03,;-3.99,-.49,;-2.65,.28,;-3.99,1.05,;-5.32,.28,;-5.32,1.82,;-6.65,2.59,;-7.99,1.82,;-7.99,.28,;-9.32,2.59,;-9.32,4.13,;-10.65,4.9,;-11.99,4.13,;-11.99,2.59,;-10.65,1.82,;-13.32,4.9,;-14.66,5.67,;-3.99,2.59,;-3.99,4.13,;-2.65,1.82,;-1.32,2.59,;-1.32,4.13,;.01,4.9,;.18,6.43,;1.68,6.75,;2.45,5.42,;1.42,4.27,;1.74,2.77,;.01,1.82,;1.35,1.05,)|
CC(OC1CCCCC1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2c(O)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1c(O)ccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
Cc1nn(C)c(C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c1Cl
CN(C)[C@@H](C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)c1ccccc1
COc1cccc2[nH]c(C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F
COc1ccc(c2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
COc1ccc(c2[nH]c(C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F)C(F)(F)F
COc1c(ccc2[nH]c(C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F)C(F)(F)F
COc1cc(cc2[nH]c(C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F)C(F)(F)F
CN(C)[C@@H](C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)c1cccc(c1)C(F)(F)F
CN(C)[C@@H](C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)c1ccc(cc1)C(F)(F)F
CC(C)C[C@H](NC(=O)c1cc2ccc(cc2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2ccc(cc2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1ccc(c2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F)C(F)(F)F
COc1cc(c(c2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F)C(F)(F)F)C(F)(F)F
COc1c(cc(c2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(c12)C(F)(F)F)C(F)(F)F)C(F)(F)F
CC(C)(C)C[C@H](NC(=O)c1cc2c(OC(F)(F)F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2cc(ccc2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2cccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1ccc(C)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2ccc(Cl)cc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2c(Cl)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2cc(Cl)ccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2cccc(c2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2c(Cl)cc(Cl)cc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)(C)C[C@H](NC(=O)c1cc2c(cccc2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2cc(ccc2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2cccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1ccc(C)c2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2cc(Cl)ccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2c(Cl)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2cccc(c2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2c(Cl)cc(Cl)cc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1cc2c(cccc2[nH]1)C(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
Cc1c(sc2ncc(n12)C(F)(F)F)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
Cc1sc(nc1C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
Cc1nc(sc1C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
CCn1nc(C)c(Br)c1C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(C)C[C@H](NC(=O)c1c(Cl)c(C)nn1C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
COc1cccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)c(C(C)=O)c12
CC(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1CC[C@H](C[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(C)(C)C
CC(C)(C)C(NC(=O)C(F)(F)F)C(=O)N1CC(C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
CNC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(C)(C)C
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(F)(F)F
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CC(O)NC1=O)C#N)C2(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@@]2(C)CO
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@]2(C)CO
CC(C)(CO)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
CC(C)(CO)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CC(=O)NC1=O)C#N)C2(C)C
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@H](CCC(F)(F)F)NC(=O)C(F)(F)F
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](NS(=O)(=O)C(F)(F)F)C1CCCCC1
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@H](CC1CCC1)NC(=O)C(F)(F)F
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](CC1CCC1)NC(=O)C(F)(F)F
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](Cc1ccccn1)NC(=O)C(F)(F)F
CC(C)(C)[C@H](NC(=O)COc1ccc(F)cc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
Cc1ccc(CC(=O)N[C@H](C(=O)N2C[C@H]3[C@@H]([C@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C3(C)C)C(C)(C)C)cc1
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@H](Cn1cccn1)NC(=O)C(F)(F)F
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@H](CC(F)F)NC(=O)C(F)(F)F
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
CC[C@@H]([C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(F)(F)F
CC[C@H]([C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(F)(F)F
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)CO
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1cccc(c1)N(C)C)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)(C)C)C(=O)NC(CC1CCNC1=O)C(=O)CO
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccc(O)cc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1ccccc1C#N
CCCCC(NC(=O)c1cc2c(OC)cccc2[nH]1)C(=O)NC(CC1CCNC1=O)C(=O)CO
CC(C)(C)CC(NC(=O)c1cc2ccccc2[nH]1)C(=O)NC(CC1CCNC1=O)C(=O)CO
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@H](NC(=O)c1cc2c(O)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@H](NC(=O)c1cc2cc(Cl)ccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1cccc2[nH]c(cc12)C(=O)NC(CCC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)CO
COCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
CC(C)CC(NC(=O)c1cc2ccccc2[nH]1)C(=O)NC(CC1CCNC1=O)C(=O)CO
CC(C)C[C@H](NC(=O)[C@H](CNC(=O)C(C)(C)C)NC(=O)OCc1ccccc1)C(=O)N[C@H](CCC(C)=O)C[C@@H]1CCNC1=O
COc1cccc2[nH]c(cc12)C(=O)NC(CC1CCCCC1)C(=O)NC(CC1CCNC1=O)C(=O)CO
NC(=O)c1ccc2N(Cc3ccc4cc(Br)ccc4c3)C(=O)C(=O)c2c1
CC(C)C[C@H](NC(=O)c1cc2cc(OC(C)C)ccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CNC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1ccc(cc1)C#N
COCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
NC(=O)c1ccc2N(Cc3cc4ccccc4s3)C(=O)C(=O)c2c1
[O-][N+](=O)c1ccc(cc1)-c1ccc(o1)C(=O)Oc1cncc(Cl)c1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1ncc(s1)-c1ccccc1
CC(C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](Cc1c[nH]c[nH+]1)C=O
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1ccc2[nH]c(cc2c1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C(NC(=O)C(C)NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)[C@@H](O)[C@H](O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(NC(=O)C(C)NC(=O)OCc1ccccc1)C(C)C
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1c(C)cccc1C
COc1ccc(cc1)C(=O)OCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1ccc(F)cc1
COc1cccc2[nH]c(cc12)C(=O)N(C)C(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)CO
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1ccccc1
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1ccc(C)cc1
c1cc(cc(c1)S(=O)(=O)n2ccc3c2ccc(c3)C(=O)Oc4cc(cnc4)Cl)[N+](=O)[O-]
CC(C)(C)CC(NC(=O)C1CCCO1)C(=O)NC(CC1CCNC1=O)C(=O)CO
Clc1cncc(OC(=O)c2cc3ccccc3s2)c1
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1ccc(Cl)cc1
CC(C)[C@H](NC(=O)[C@@H](NC(C)=O)[C@@H](C)O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](Cc1c[nH]c[nH+]1)C=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)OC(C)(C)C)C(=O)N[C@H](CCC(=O)C1CC1)C[C@@H]1CCNC1=O
COc1cccc2[nH]c(cc12)C(=O)NC(Cc1ccccc1)C(=O)NC(CC1CCNC1=O)C(=O)CO
COCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)(C)C)NC(=O)c1cc2ccccc2[nH]1
Clc1cncc(OC(=O)c2cc3ccccc3oc2=O)c1
CCOCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)(C)C)NC(=O)c1cc2ccccc2[nH]1
CC(C)C[C@H](NC(=O)C1Cc2ccccc2N1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
[O-][N+](=O)c1cc(Cl)ccc1-c1ccc(o1)C(=O)Oc1cncc(Cl)c1
Clc1cncc(OC(=O)c2cccc3ccccc23)c1
COCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)C(CCC(C)C)N(C)C(=O)c1cc2ccccc2[nH]1
CC(=O)N1Cc2ccccc2CC1C(=O)Oc1cncc(Cl)c1
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)S(=O)(=O)O)NC(=O)OCc2ccccc2
CC(C)C[C@H](NC(=O)c1cc2cc(O)ccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
Clc1cncc(OC(=O)c2ccncc2)c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)c1ccc2ccccc2c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc2ccccc2c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)CCc1cccc(F)c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1cc(F)cc(F)c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(F)c(F)c1
COc1ccc(OCC(=O)N2CC3C([C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1OC
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1cccc(c1)C(F)(F)F
COc1ccc(OCC(=O)N2CC3C([C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1F
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(OC(F)(F)F)cc1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)c(Br)c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Br)cc1Cl
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)cc1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)c(Cl)c1
CC1(C)C2CN([C@H](C12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)cc1Cl
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1C2CCCC2CN1C(=O)c1cccnc1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1C2CCCC2CN1C(=O)c1cc2ccccc2[nH]1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1C2CCCC2CN1C(=O)c1cc2ccccn2n1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1C2CCCC2CN1C(=O)C=Cc1ccccc1 |w:23.25|
COc1ccc(C=CC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(OC)c1 |w:6.5|
CN(C)c1ccc(C=CC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |w:7.6|
Fc1cccc(CCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1
Fc1ccc(CCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1F
Fc1cc(F)cc(CCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1
CN(C)c1ccc(CCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1
COc1ccc(OCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1
COc1ccc(OC(C)C(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H]1C2CCCC2CN1C(=O)COc1ccc2OCCOc2c1
Clc1ccc(OCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1
Fc1cc(Cl)ccc1OCC(=O)N1CC2CCCC2[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
Clc1ccc(OCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(Cl)c1
Clc1ccc(OCC(=O)N2CC3CCCC3[C@@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1Cl
Cc1cc(Cl)ccc1OCC(=O)N1CC2CCCC2[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
Clc1cncc(OC(=O)c2cc3ccccc3o2)c1
O=n1ccccc1S[Zn]Sc1ccccn1=O
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1cccc(c1)N(C)C)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1ncc(s1)-c1ccccc1
O=C(N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:34.36|
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)C1CC1
CC(C)CC(NC(=O)C(NC(=O)c1ccncc1)C(C)C)C(=O)NC(CC1CCCNC1=O)C=O
Fc1cc(Cl)ccc1C=CC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |w:9.10|
CCCCC1CCC(CC1)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)S(O)(=O)=O |wU:14.14,22.22,24.24,wD:30.32,(-6.67,3.85,;-8,4.62,;-8,6.16,;-6.67,6.93,;-5.33,6.16,;-4,6.93,;-2.67,6.16,;-2.67,4.62,;-4,3.85,;-5.33,4.62,;-1.33,3.85,;,4.62,;,6.16,;1.33,3.85,;2.67,4.62,;2.67,6.16,;4,6.93,;4,8.47,;5.33,6.16,;4,3.85,;4,2.31,;5.33,4.62,;6.67,3.85,;8,4.62,;9.34,3.85,;9.5,2.32,;11,2,;11.77,3.33,;10.74,4.48,;11.06,5.98,;6.67,2.31,;5.33,1.54,;8,1.54,;7.23,.21,;8.77,2.87,;9.34,.77,)|
COc1cccc(OC)c1C(=O)OCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1
[O-][N+](=O)c1ccccc1-c1ccc(o1)C(=O)Oc1cncc(Cl)c1
Cc1cc(ccc1N=Nc1ccc2c(cc(c(N)c2c1O)S([O-])(=O)=O)S([O-])(=O)=O)-c1ccc(N=Nc2ccc3c(cc(c(N)c3c2O)S([O-])(=O)=O)S([O-])(=O)=O)c(C)c1 |w:34.37,7.7|
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(C)=O
COc1cccc2[nH]c(cc12)C(=O)NC(CC(C)C)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)C(C)(C)C
CCCC1CCC(CC1)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)S(O)(=O)=O |wU:13.13,21.21,23.23,wD:29.31,(-8,4.62,;-8,6.16,;-6.67,6.93,;-5.33,6.16,;-4,6.93,;-2.67,6.16,;-2.67,4.62,;-4,3.85,;-5.33,4.62,;-1.33,3.85,;,4.62,;,6.16,;1.33,3.85,;2.67,4.62,;2.67,6.16,;4,6.93,;4,8.47,;5.33,6.16,;4,3.85,;4,2.31,;5.33,4.62,;6.67,3.85,;8,4.62,;9.34,3.85,;9.5,2.32,;11,2,;11.77,3.33,;10.74,4.48,;11.06,5.98,;6.67,2.31,;5.33,1.54,;8,1.54,;9.34,.77,;7.23,.21,;8.77,2.87,)|
O=C(N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:31.33|
CC(C)[C@H](NC(=O)[C@H](C)NC(C)=O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
Clc1cncc(OC(=O)c2cscn2)c1
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2ncc(s2)-c2ccccc2)cc1
CCCC1CCC(CC1)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |wU:13.13,21.21,wD:23.23,(-7.56,2,;-8.07,3.46,;-7.06,4.62,;-5.54,4.33,;-4.54,5.49,;-3.02,5.2,;-2.52,3.75,;-3.53,2.58,;-5.04,2.87,;-1.01,3.46,;,4.62,;-.5,6.08,;1.51,4.33,;2.52,5.49,;2.02,6.95,;3.02,8.11,;2.52,9.57,;4.54,7.82,;4.03,5.2,;4.54,3.75,;5.04,6.37,;6.55,6.08,;7.56,7.24,;9.07,6.95,;10.2,8,;11.55,7.26,;11.26,5.74,;9.73,5.55,;8.98,4.21,;7.06,4.62,;6.05,3.46,)|
O=N(=O)O[Hg]c1ccccc1
c1ccc(cc1)C[C@@H](C(=O)CCl)NC(=O)OCc2ccccc2
COc1ccccc1NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1ccc2cc([nH]c2c1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@H](NC(=O)C=Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1 |w:8.7|
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1cccc(c1)N(C)C)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1ncc(C)s1
[O-][N+](=O)c1ccccc1C(=O)Oc1cncc(Cl)c1
CC(C)[C@H](NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
COc1cccc(c1)C(=O)Oc1cncc(Cl)c1
Cc1ccc(cc1)S(=O)(=O)N1C=CC2C=C(C=CC12)C(=O)Oc1cncc(Cl)c1 |c:12,15,17|
ClCC(=O)[C@H](Cc1ccc2ccccc2c1)NC(=O)OCc1ccccc1
Fc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)CCl)cc1
CC(C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CC(=O)n1ccc2cc(ccc12)C(=O)Oc1cncc(Cl)c1
CC(C)(C)OC(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)CBr
CC(C)C[C@H](NC(=O)OC1CCC(F)(F)CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)S(O)(=O)=O
OCCn1[se]c2ccccc2c1=O
OC(=O)Cn1[se]c2ccccc2c1=O
OC(=O)CCn1[se]c2ccccc2c1=O
OC(=O)c1ccc(cc1)-n1[se]c2ccccc2c1=O
O=c1n([se]c2ccccc12)-c1cccc(c1)N(=O)=O
O=c1n([se]c2ccccc12)-c1ccc(cc1)N(=O)=O
O=c1n(CCN2CCOCC2)[se]c2ccccc12
CC(C)(C)OC(=O)NCn1[se]c2ccccc2c1=O
O=c1n(Cc2ccco2)[se]c2ccccc12
O=c1[nH]sc2ccccc12
Cn1sc2ccccc2c1=O
CCCn1sc2ccccc2c1=O
OCCn1sc2ccccc2c1=O
CC(C)Cn1sc2ccccc2c1=O
C=CCn1sc2ccccc2c1=O
Nc1ccccc1-n1sc2ccccc2c1=O
O=c1n(Cc2ccccc2)sc2ccccc12
Cc1ccc(cc1)-n1sc2ccccc2c1=O
Clc1ccc(cc1)-n1sc2ccccc2c1=O
O=c1n(Cc2ccco2)sc2ccccc12
O=c1n(CCCc2ccccc2)sc2ccccc12
O=c1n(sc2ccccc12)-c1ccccc1
COC(=O)c1ccc(cc1)-n1sc2ccccc2c1=O
CCCNC(=O)c1ccc(cc1)-n1sc2ccccc2c1=O
CCCCNC(=O)c1ccc(cc1)-n1sc2ccccc2c1=O
O=C(NCc1ccco1)c1ccc(cc1)-n1sc2ccccc2c1=O
COc1ccc(CC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
CC(C)C[C@H](NC(=O)OC1CCC(F)(F)CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
Clc1ccc(cc1)C(=O)Oc1cncc(Cl)c1
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)O)NC(=O)OCC2CCC(CC2)(F)F
CCCC(NC(=O)C(CC(C)C)NC(=O)OCc1ccccc1)C(=O)C(=O)NCc1ccccn1
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2ncc(s2)-c2ccccc2OC)cc1
CN(C)c1ccc(C=CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |w:8.8|
Brc1cncc(OC(=O)c2cccs2)c1
[O-][N+](=O)c1cccc(c1)-c1ccc(o1)C(=O)Oc1cncc(Cl)c1
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)/C=C/c2ccccc2
COC(=O)CC(NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)CF
Clc1ccc(SSc2nnco2)cc1
CCOC(=O)\C=C\C(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)C=Cc1ccc(cc1)N(C)C |w:29.30|
CC(C)C[C@H](NC(=O)COc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C(NC(=O)[C@@H](C)NC(=O)OCc1ccccc1)C(=O)N[C@H](Cc1ccccc1)C(O)C(O)[C@@H](Cc1ccccc1)NC(=O)C(NC(=O)[C@@H](C)NC(=O)OCc1ccccc1)C(C)C
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(C)=O)C(C)C)[C@H](C)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)[N+]([O-])=O
COc1ccc(CCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccc(cc1)N(C)C)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CCOC(=O)C=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C |w:5.4|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1ncc(s1)-c1ccccc1
COC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C
CC(C)C[C@H](NC(=O)OC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)[C@@H](O)S(O)(=O)=O
CC(C)(C)OC(=O)NC1=CC=CN(C1=O)[C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]3CCNC3=O)[C@H](C(=O)NCc4ccccc4)O
CC(C)C[C@H](NC(=O)c1c[nH]c2ccccc12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
[O-][N+](=O)c1cccc(c1)C(=O)Oc1cncc(Cl)c1
Clc1ccc(SSc2ncccn2)cc1
CC(C)C[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
Clc1cncc(OC(=O)c2cccnc2)c1
Brc1ccc(SSc2ncccn2)cc1
Brc1cccc(C=CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |w:7.7|
c1c(c(cc(c1C(=O)O)C(=O)O)C(=O)O)C(=O)O
COc1ccc(\C=C\C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
COc1cccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)c1
CC(C)C[C@H](NC(=O)c1nc2ccccc2s1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
[H][C@@]12CC(C)=CC[C@]1(C)CC[C@]1(C)C3=CC=C4C(C)=C(O)C(=O)C=C4[C@]3(C)CC[C@@]21C |r,c:4,24,t:14,16,19|
CC(C)C[C@H](NC(=O)OC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)CC(NC(=O)\C=C\c1ccccc1)C(=O)NC(CC1CCNC1=O)C=O
CC(C)CC(NC(=O)COc1ccc(cc1)N(C)C)C(=O)NC(CC1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@H](NC(=O)COc1cccc(c1)N(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
[O-][N+](=O)c1ccccc1SSc1ncccn1
Cc1cc(C)nc(SSc2ccccc2[N+]([O-])=O)n1
CSCCC(NC(=O)C(CC(C)C)NC(=O)C(CC(C)C)NC(C)=O)C=O
CCNCCc1ccc(cc1)C(=O)Cn1nnc2ccccc12
CC(C)CC(NC(C)=O)C(=O)NC(CC1CCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
CC1CCN(CC1)S(=O)(=O)c1ccc2N(C)C(=O)C(=O)c2c1
COCC(=O)C(CC1CCNC1=O)NC(=O)C(CC(C)(C)C)NC(=O)C1CCCO1
Ic1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
COC(=O)c1ccccc1SSc1nnco1
Cc1cc(C)nc(SSc2ccc(Br)cc2)n1
CC1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1
O=C(N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)OCc1ccccc1
COC(=O)c1ccccc1SSc1nc(C)co1
O=C(N[C@@H](CC1CCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:33.35|
COc1cc(ccc1N=Nc1ccc2c(cc(c(N)c2c1O)S([O-])(=O)=O)S([O-])(=O)=O)-c1ccc(N=Nc2ccc3c(cc(c(N)c3c2O)S([O-])(=O)=O)S([O-])(=O)=O)c(OC)c1 |w:9.10,34.36|
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2ncc(s2)-c2ccc(Cl)cc2)cc1
COc1ccc(\C=C\C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1OC
CN(C)c1ccc(cc1)C(=O)O
Cc1ccc2S[Zn]Sc2c1
Oc1cc(cc(O)c1O)C(=O)Oc1cc(cc(O)c1O)C(=O)OC[C@H]1O[C@@H](OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)[C@H](OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)[C@@H](OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)[C@@H]1OC(=O)c1cc(O)c(O)c(OC(=O)c2cc(O)c(O)c(O)c2)c1
Cc1ccc(c(c1)S)S
Cc1cc(C)nc(SSc2ccc(Cl)cc2)n1
O=C(N[C@@H](CC1CCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:32.34|
CCCCCCCCCC(=O)N[C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1Oc1c2Oc3ccc(C[C@H]4NC(=O)[C@H](N)c5ccc(O)c(Oc6cc(O)cc(c6)[C@H](NC4=O)C(=O)N[C@@H]4c(c2)cc1Oc1ccc(cc1Cl)[C@@H](O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1NC(C)=O)[C@@H]1NC(=O)[C@H](NC4=O)c2ccc(O)c(c2)-c2c(OC4O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]4O)cc(O)cc2[C@H](NC1=O)C(O)=O)c5)cc3Cl
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2ncc(s2)-c2ccc(C)cc2)cc1
Cc1ccc(SSc2nc(C)cc(C)n2)cc1
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(NCc2ccccc2)cc1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)CNc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(=O)Nc1cnc(SSc2ccccc2)s1
Cc1ccc(SSc2ncccn2)cc1
CCOC(=O)c1ccccc1SSc1nnc(C)o1
COc1ccc(OCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
CCCC[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(=O)Nc1cnc(SSc2ccc(Br)cc2)s1
COC(=O)c1ccccc1SSc1nnc(C)o1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccc(cc1)C(O)=O)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@H](NC(=O)c1ccc[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
Cc1nnc(SSc2ccccc2[N+]([O-])=O)o1
CC(=O)n1nc(SSc2ccccc2[N+]([O-])=O)nc1-c1cccnc1
Clc1ccc(SSc2nccs2)cc1
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)c1cc(C)on1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=CC(=O)OCc1ccccc1 |w:38.40|
COc1ccccc1OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
O=C(N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:34.36|
Cc1cc(C)nc(SSc2ccccc2)n1
[O-][N+](=O)c1cccc2C(=O)C(=O)N(Cc3cc4ccccc4s3)c12
Nc1ccc(cc1N)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O
CC(O)C(NC(=O)CCC(=O)NC(C(C)O)C(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)N(=O)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O
CC(O)C(NC(=O)CC(O)C(=O)NC(C(C)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O)C(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)N(=O)=O
CC(O)C(NC(=O)C(O)C(O)C(=O)NC(C(C)O)C(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)N(=O)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O
COc1c(Sc2nnnn2-c2ccc(OCc3ccccc3)cc2)c(=O)[nH]c2ccccc12
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc(C)c(C)s1
COC(=O)c1nc(SSc2ccccc2[N+]([O-])=O)[nH]c1C
C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)CCO
OC[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)C=Cc1ccccc1 |w:24.25|
CC1CCCCN1S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1
CC(C)(C)OC(=O)Nc1cccn(C(CC2CCCCC2)C(=O)NC(CC2CCNC2=O)C(=O)C(=O)NC2CC2)c1=O
CC[Hg]Sc1ccccc1C(=O)O[Na]
CCOC(=O)c1ccccc1SSc1nc(C)cs1
CCOC(=O)C=CC(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)C=Cc1ccc(cc1)N(=O)=O |w:5.4,29.30|
CC1=C(C(C2=C(CCCC2=O)N1)c1ccccc1[N+]([O-])=O)C(=O)OCCc1ccccc1 |t:1,4|
COc1ccccc1-c1cnc(s1)C(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1
Cc1csc(SSc2ccccc2[N+]([O-])=O)n1
CC(=O)Nc1cnc(SSc2ccc(F)cc2)s1
Nc1nc2nc3nc(N)sc3cc2s1
CC(=O)Nc1cnc(SSc2ccc(Cl)cc2)s1
CC(C)C[C@H](NC(=O)C1CCC(=O)N1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(=O)Nc1cnc(SSc2ccc(C)cc2)s1
CC1CC(C)CN(C1)S(=O)(=O)c1ccc2N(C)C(=O)C(=O)c2c1
CC1OC(OC2C(O)C(OCCc3ccc(O)c(O)c3)OC(COC3OCC(O)(CO)C3O)C2OC(=O)C=Cc2ccc(O)c(O)c2)C(O)C(O)C1O |w:37.39|
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1cccnc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
Oc1cc(cc(O)c1O)C(=O)Oc1cc(cc(O)c1O)C(=O)OCC1OC(OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)C(OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)C(OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)C1OC(=O)c1cc(O)c(O)c(OC(=O)c2cc(O)c(O)c(O)c2)c1
Oc1ccc(cc1)-c1cc(=O)c2c(O)c(O)c(O)cc2o1
CCOC(=O)C=CC(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)C=Cc1ccc2OCOc2c1 |w:5.4,29.30|
[H][C@@]12C[C@@](C)(CC[C@]1(C)CC[C@]1(C)C3=CC=C4C(C)=C(O)C(=O)C=C4[C@]3(C)CC[C@@]21C)C(=O)OC |r,c:24,t:14,16,19|
CC(=O)n1nc(SSc2ccccc2[N+]([O-])=O)nc1C
CC1OC(OCC2OC(OCCc3ccc(O)c(O)c3)C(O)C(O)C2OC(=O)C=Cc2ccc(O)c(O)c2)C(O)C(O)C1O |w:28.29|
CC(C)C[C@H](NC(=O)Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1ccc(NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
C[C@H](CNC(=O)CC[C@]1(C)[C@@H](CC(N)=O)[C@H]2[N-]\C1=C(C)/C1=N/C(=C\C3=N\C(=C(C)/C4=N[C@]2(C)[C@@](C)(CC(N)=O)[C@@H]4CCC(N)=O)\[C@@](C)(CC(N)=O)[C@@H]3CCC(N)=O)/C(C)(C)[C@@H]1CCC(N)=O)OP([O-])(=O)O[C@@H]1[C@@H](CO)O[C@@H]([C@@H]1O)n1cnc2cc(C)c(C)cc12 |c:18,23,t:21,25,27,30|
COc1ccccc1N=Cc1nc(oc1OC(C)=O)-c1ccccc1 |w:8.8|
Brc1ccc(SSc2nccs2)cc1
CC(C)CC(NC(=O)C(NC(=O)C(NC(C)=O)C(C)C)C(C)O)C(=O)NC(CC1CCNC1=O)C(=O)CN1NC(=O)C2C(C=CC=C2[N+]([O-])=O)C1=O |c:44,46|
COCCC(=O)Nc1ccc(cc1)N(C(C)c1ccsc1)C(=O)Cn1nnc2ccccc12
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccc(cc1)N(=O)=O)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CCOC(=O)c1c[nH]c(SSc2ccc(Cl)cc2)n1
COC(=O)c1nc(SSc2ccccc2C(=O)OC)[nH]c1C
OSC(CC(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)N(=O)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc(cc1Cl)[N+]([O-])=O
C[C@@H]1C[C@@H]2[C@@](C)(CC[C@]3(C)C4=CC=C5C(C)=C(O)C(=O)C=C5[C@]4(C)CC[C@@]23C)CC1=O |c:20,t:10,12,15|
ClC1=C(Cl)C(=O)C(Cl)=C(Cl)C1=O |c:1,t:7|
COc1ccc(SSc2nc(-c3ccccc3)n(n2)C(C)=O)cc1
COC(=O)c1nc(SSc2ccc(Cl)cc2)[nH]c1C
CC(=O)n1nc(SSc2ccc(C)cc2)nc1-c1ccccc1
CC1=C(C(=O)C=C2C1=CC=C3[C@]2(CC[C@@]4([C@@]3(CC[C@@]5([C@H]4C[C@](CC5)(C)C(=O)O)C)C)C)C)O
CC1CC(C)CN(C1)S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1
O=C1Nc2ccc(cc2C1=O)S(=O)(=O)N1CCCCC1
CCOC(=O)c1ccccc1SSc1nc(-c2ccncc2)n(n1)C(C)=O
OB(O)c1cc(cc(c1)N(=O)=O)C(=O)Oc1ccc(OC(=O)c2cc(cc(c2)N(=O)=O)B(O)O)cc1
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(N)=O)C#N |r|
COc1cc(ccc1O)C(=S)N1CCOCC1
OC1O[C@@H]2COC(=O)c3cc(O)c(O)c(O)c3-c3c(O)c(O)c4oc(=O)c5c(c(O)c(O)c6oc(=O)c3c4c56)-c3c(O)c(O)c(O)cc3C(=O)O[C@H]2[C@@H]2OC(=O)c3c(O)c(O)c(O)cc3-c3c(O)c(O)c(O)cc3C(=O)O[C@@H]12
CC1CC(C)CN(C1)S(=O)(=O)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
Fc1ccc2N(Cc3cc4ccccc4s3)C(=O)C(=O)c2c1
CN(C)CCCSc1ccccc1NC(=O)\C=C\c1ccccc1
CC1OC(OCC2OC(OCCc3ccc(O)c(O)c3)C(O)C(OC(=O)C=Cc3ccc(O)c(O)c3)C2O)C(O)C(O)C1O |w:26.26|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(cc2)C#N)cc1 |c:12|
CN1C(=O)C(=O)c2cc(ccc12)S(=O)(=O)N1CCN(CC1)c1ccccn1
CCOc1cccc(c1)C(=O)c1ccc(O)c(O)c1O
CCOC(=O)c1ccccc1SSc1nc(-c2cccnc2)n(n1)C(C)=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](Cc1c[nH]c[nH+]1)C=O
CCCCC(NC(=O)C1[C@@H]2[C@H](CN1C(=O)C(NC(=O)NC1(CS(=O)(=O)C(C)(C)C)CCCCC1)C(C)(C)C)C2(C)C)C(=O)C(=O)NC1CC1
COc1ccc(SSc2nc(-c3cccnc3)n(n2)C(C)=O)cc1
C[C@@H]1O[C@H](OC[C@H]2O[C@@H](OCCc3ccc(O)c(O)c3)[C@H](O)[C@@H](OC(=O)\C=C\c3ccc(O)c(O)c3)[C@@H]2O)[C@H](O)[C@H](O)[C@H]1O
CC(C)C[C@H](NC(=O)CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(O)c1c(C)c2cc3[nH]c(cc4nc(cc5nc(cc1[nH]2)c(C)c5CCC(O)=O)c(CCC(O)=O)c4C)c(C)c3C(C)O
CCOC(=O)c1ccccc1SSc1nc(C(=O)OC)c(C)[nH]1
ClCC(=O)N1N=C(CC1c1cccs1)c1cccs1 |c:5|
ClCC(=O)N1CCc2sccc2C1c1cccs1
ClCC(=O)N1CCc2sccc2C1c1ccccc1
ClCC(=O)N1N=C(CC1c1cccs1)c1ccco1 |c:5|
ClCC(=O)Nc1cc(nn1-c1ccccc1)-c1ccccc1
O=N(=O)C=Cc1ccc(cc1)C#N |w:3.2|
COc1ccc(C=CN(=O)=O)cc1 |w:6.5|
COc1cc(C=CN(=O)=O)cc(OC)c1OC |w:5.4|
Brc1cccc(C=CN(=O)=O)c1 |w:6.5|
Cc1ccc(cc1)S(=O)(=O)C(=Cc1cccnc1)C#N |w:11.12|
CN(C#N)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N(C)N(C)C#N |r|
CN(N(CCc1ccccc1)C#N)C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1 |r|
CCCCCN(C#N)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1 |r|
CN(N(Cc1ccccc1)C#N)C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1 |r|
CC(C)C[C@H](NC(=O)NCc1ccc(cc1)-c1noc(C)n1)C(=O)N(C)N(C)C#N |r|
CC(C)C[C@H](NC(=O)NCc1ccc(cc1)-c1noc(n1)-c1cccs1)C(=O)N(C)N(C)C#N |r|
CC(C)C[C@H](NC(=O)Nc1ccc(cc1)-c1noc(n1)-c1cccs1)C(=O)N(C)N(C)C#N |r|
CC(C)C[C@H](NC(=O)NCc1ccccc1)C(=O)N(C)N(C)C#N |r|
CC(C)C[C@H](NC(=O)c1ccc(cc1)-c1noc(n1)-c1cccs1)C(=O)N(C)N(C)C#N |r|
CC(C)C[C@H](N(C)C(=O)c1ccc(cc1)-c1noc(n1)-c1cccs1)C(=O)N(C)N(C)C#N |r|
CN1N(CCC(NC(=O)OCc2ccccc2)C1=O)C#N
CC(C)(C)OC(=O)NN(CC(=O)N(Cc1ccccc1)Cc1ccccc1)C#N
CN(Cc1ccccc1)C(=O)CN(NC(=O)OC(C)(C)C)C#N
S=c1sc(SC#N)nc2ccccc12
CC(C)CC(NC(=O)OCc1ccccc1)C(=O)N(C)N(CCC(N)=O)C#N
CN(N(CCC(N)=O)C#N)C(=O)C(Cc1ccccc1)NC(=O)OCc1ccccc1
CC(C)CC(NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C)C(=O)N(C)N(CCC(N)=O)C#N
CN(N(CCC(N)=O)C#N)C(=O)C(Cc1ccccc1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C
CCC(NC(=O)OCc1ccccc1)C(=O)NC(C(=O)NC(CC(C)C)C(=O)N(C)N(CCC(N)=O)C#N)C(C)(C)C
CCC(NC(=O)OCc1ccccc1)C(=O)NC(C(=O)NC(Cc1ccccc1)C(=O)N(C)N(CCC(N)=O)C#N)C(C)(C)C
NC(=N)Nc1ccc(cc1Cl)-c1ccc(o1)-c1ccc(NC(N)=N)c(Cl)c1
CC(=O)OCC1O[C@@H](CS[Au])[C@@H](OC(C)=O)C(OC(C)=O)[C@H]1OC(C)=O
Cn1c2nc3n(CC#Cc4ccc(Cl)c(Cl)c4)ccn3c2c(=O)n(C)c1=O
Clc1cncc(OC(=O)c2c[nH]c3ccccc23)c1
Clc1cncc(OC(=O)c2cc3cc(Cl)ccc3[nH]2)c1
Brc1cncc(OC(=O)c2cccc3[nH]ccc23)c1
Clc1cncc(OC(=O)c2ccc3[nH]c4CCCCc4c3c2)c1
Clc1cncc(OC(=O)c2cc3c(Cl)cc(Cl)cc3[nH]2)c1
CC(C)(C)NC(=O)C(N(C(=O)C1=NC=NC1)c1ccc(cc1)C(C)(C)C)c1cccnc1 |c:13,t:11|
OB(O)c1cc(cc(c1)N(=O)=O)C(=O)OCc1ccccc1COC(=O)c1cc(cc(c1)N(=O)=O)B(O)O
CCC(C)(C)NC(=O)[C@@H](c1cccn1C)N(c2ccc(cc2)NC(=O)C)C(=O)Cn3c4ccccc4nn3
O=C(N[C@@H](C1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:30.32|
c1ccc(cc1)C2=CC(=O)c3c(cc(c(c3O)O)O[C@H]4[C@@H]([C@H]([C@@H]([C@H](O4)C(=O)O)O)O)O)O2
CCOC(=O)C=CC(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)C=Cc1ccc(cc1)-c1ccccc1 |w:5.4,29.30|
CC1OC(OCC2OC(OCCc3ccc(O)c(O)c3)C(O)C(O)C2O)C(O)C(O)C1O
COc1ccc2[nH]c(C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)c3nc4ccccc4s3)c(C)c2c1
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)c1ccoc1)C(C)C)C(C)C
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CCC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)c1ccco1)C(C)C)C(C)C
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
COC(=O)CCC(NC(=O)C(CC(=O)OC)NC(=O)OCc1ccccc1)C(=O)NC(C(C)C)C(=O)NC(CC(=O)OC)C(=O)CF
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2ccc(F)cc2)cc1 |w:7.6,c:12|
COc1ccc(cc1)N1C(=O)NC(=O)C(=Cc2cc(Cl)c(OCc3cccc(c3)C(O)=O)c(Cl)c2)C1=O |w:15.16|
CCC(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccsc1)C(=O)Cn1nnc2ccccc12
COC(=O)c1cc2c(O)cc(nc2o1)C(F)(F)F
O[C@@H]1Cc2c(O)cc(O)cc2OC1c1cc(O)c(=O)c2c(O)c(O)cc(C3Oc4cc(O)cc(O)c4C[C@@H]3OC(=O)c3cc(O)c(O)c(O)c3)c2c1
O=C1C=CC(=O)c2cn(Cc3ccccc3)cc12 |c:2|
Cc1c(sc2ccc(Cl)cc12)C(=O)CC1OC(=O)C(Cl)=C1Cl |c:21|
COc1cc(CS(=O)c2nc3cccnc3s2)oc(=O)c1
Cc1noc(C)c1CN1C(=O)C(=O)c2cc(ccc12)C#N
CC(C)C[C@H](NC(=O)CCc1cccnc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
c1nc2c(nc(nc2n1[C@@H]3C[C@@H](C=C3)CO)N)NC4CC4
C[C@H](Cn1cnc2c1ncnc2N)OCP(=O)(O)O
CC(C)(C)NC(=O)[C@@H]1CN(Cc2cccnc2)CCN1C[C@@H](O)C[C@@H](Cc1ccccc1)C(=O)N[C@@H]1[C@H](O)Cc2ccccc12 |r|
CCCc1c2c(n(n1)C)C(=O)NC(=N2)c3cc(ccc3OCC)S(=O)(=O)N4CCN(CC4)C
N[C@@H](CC(=O)N1CCn2c(C1)nnc2C(F)(F)F)Cc1cc(F)c(F)cc1F |r|
CCc1c([nH]c2ccc(OC)cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)CNCc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(=O)Oc1c(Cl)cc(Cl)c(Cl)c1Sc1c(Cl)c(Cl)cc(Cl)c1OC(C)=O
CC(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccsc1)C(=O)Cn1nnc2ccccc12
O=C(Oc1cccnc1)C1CCCO1
CC1=CC(=O)c2ccccc2C1=O
CCCn1c(NCc2ccc(cc2)N2N=C(CC2c2ccccc2)c2ccccc2)nc2ccccc12 |c:15|
CCCCn1c(NCc2ccc(cc2)N2N=C(CC2c2ccccc2)c2ccccc2)nc2ccccc12 |c:16|
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(NC(=O)C2CCC2)cc1
CC(=C)C1CCC2(CCC3(C)C(CCC4C5(C)CCC(O)C(C)(C)C5CCC34C)C12)C(O)=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCC(O)=O)NC(C)=O)[C@@H](C)O)C(=O)N[C@H](CO)CCC(N)=O
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2cccc(c2)[N+]([O-])=O)cc1 |w:7.6,c:12|
CC(C)C[C@H](NC(=O)COc1ccc(O)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CCn1c(NCc2ccc(cc2)N2N=C(CC2c2ccccc2)c2ccccc2)nc2ccccc12 |c:14|
CCCC[C@H](NC(=O)C=Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1 |w:8.7|
CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(C)=O)C=O |r|
S=C=NCCc1ccccc1
CCOc1ccc(cc1)C(=O)c1ccc(O)c(O)c1O
CCOC(=O)C=CC(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)C=Cc1ccc(OC)cc1OC |w:5.4,29.30|
OC1C2C(CC(O)=O)C(=O)OC3C4COC(=O)c5cc(O)c(O)c(O)c5-c5c(O)c(O)c(O)cc5C(=O)OC3C(OC(=O)c3cc(O)c(O)c(OC1=O)c23)C(OC(=O)c1cc(O)c(O)c(O)c1)O4
O=C1OC[C@H](Cc2ccc3OCOc3c2)C1=Cc1ccc2OCOc2c1 |w:16.19|
OC(=O)c1cc(Br)ccc1-c1ccc(C=C2C(=O)NN(C2=O)c2ccc(Cl)c(Cl)c2)o1 |w:14.14|
CC1(C)OC2=C([C@H](NCc3ccccc3)[C@@H]1O)C(=O)c1ccccc1C2=O |r,c:4|
Oc1c(Sc2cc(Cl)cc(c2O)N(=O)=O)cc(Cl)cc1N(=O)=O
CSCCC(NC(=O)OCc1ccccc1)C(=O)NC(CC1CCNC1=O)C(=O)c1nc2ccccc2s1
Fc1ccc(CN2C(=O)C(=O)c3cc(I)ccc23)c(Cl)c1
Oc1cc(O)c2C[C@H](OC(=O)c3cc(O)c(O)c(O)c3)C(Oc2c1)c1cc(O)c(O)c2c1cc(cc(O)c2=O)C1Oc2cc(O)cc(O)c2C[C@@H]1OC(=O)c1cc(O)c(O)c(O)c1
COc1ccc(cc1)C(c1c(O)c2cc(C)ccc2oc1=O)c1c(O)c2cc(C)ccc2oc1=O
CC1=C(CCC(O)=O)C2=NC1=Cc1c(C)c(C=C)c3C=C4N=C(C=c5c(C)c(CCC(O)=O)c(=C2)n5[Fe](Cl)n13)C(C=C)=C4C |w:34.35,11.12,23.23,19.19,c:1,8,46,t:22,(9.94,.88,;8.64,1.95,;7.12,2.05,;6.53,.63,;6.92,-.86,;8.44,-1.14,;9.33,-2.3,;8.99,.44,;6.75,3.52,;8.03,4.33,;9.2,3.36,;10.93,2.4,;11.69,1.09,;13.1,.52,;14.39,1.43,;13,-.99,;14.27,-1.96,;15.8,-1.64,;11.53,-1.37,;10.57,-3.09,;9.25,-3.85,;8.09,-2.88,;6.8,-3.69,;5.07,-2.73,;4.31,-1.42,;2.9,-.86,;1.71,-1.89,;3,.66,;1.77,1.65,;.25,1.27,;-.98,2.24,;-2.41,1.64,;-.75,3.79,;4.47,1.03,;5.43,2.76,;5.28,-.25,;8,-.17,;7.76,1.26,;10.72,-.08,;7.17,-5.17,;6.2,-6.43,;6.53,-7.97,;8.69,-5.26,;9.59,-6.57,)|
COC(=O)[C@@]1(C)CCCc2c1ccc1-c3occ(C)c3C(=O)C(=O)c21 |r|
COc1ccc2C3=NN(C(C3CCc2c1)c1cccc(I)c1)C(C)=O |t:6|
CN1C(=O)C(=O)c2cc(ccc12)S(=O)(=O)N1CCOCC1
CN(C)CCCNC(=O)C(\NC(=O)c1ccc(C)cc1)=C/c1ccc(o1)-c1ccc(cc1)[N+]([O-])=O
CC(C)[C@H](NC(=O)[C@H](CC(N)=O)NC(C)=O)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)OC(C)(C)C)C(C)C)\C=C\C(=O)OCC)CCNC1=O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C)C(=O)NC(Cc1ccccc1)C(=O)C(F)(F)F
Oc1c(Sc2nnnn2-c2ccc(OCc3ccccc3)cc2)c(=O)[nH]c2ccccc12
Oc1ccc(cc1)-n1nnnc1Sc1c(O)c2c(Cl)cc(Cl)cc2[nH]c1=O
O=C(N1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1)c1ccco1
CC1OC(OCC2OC(OCCc3ccc(O)c(O)c3)C(OC(=O)C=Cc3ccc(O)c(O)c3)C(O)C2O)C(O)C(O)C1O |w:24.24|
CCCN1C(=O)C(=O)c2cc(ccc12)C(N)=O
CC(C)COC(=O)Nc1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
CC[C@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C=O |r|
CCCCC(NC(=O)C(CC(C)C)NC(=O)OCc1ccccc1)C=O
O=C(N[C@@H](CC#C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NCc1ccccc1)C=Cc1ccccc1 |w:30.31|
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2cccc(Cl)c2)cc1 |w:7.6,c:12|
O=N(=O)c1ccccc1C1N(CCN1c1ccccc1)c1ccccc1
CC1OC(OCC2OC(Oc3c(oc4cc(O)cc(O)c4c3=O)-c3ccc(O)c(O)c3)C(O)C(O)C2O)C(O)C(O)C1OCC(=O)Nc1ccc(cc1)N([C@H](C(=O)NC(C)(C)C)c1ccsc1)C(=O)n1cc(nn1)-c1ccccc1
CC(=O)Nc1ccc(cc1)N(C(C(=O)NC(C)(C)C)c1ccsc1)C(=O)Cn1cc(nn1)-c1ccccc1
OC(=O)c1c(O)cccc1CCCCCCCC=CCC=CCC=C |w:21.22,18.19|
Clc1cccc2N(Cc3cc4ccccc4s3)C(=O)C(=O)c12
CN1C(=O)C(=O)c2cc(ccc12)S(=O)(=O)N1CCN(C)CC1
COc1ccc(cc1)N1N=C(C(=Cc2ccc(cc2)C(O)=O)C1=O)c1ccccc1 |w:12.13,c:10|
COc1ncc(cn1)-c1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
NC(=O)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
Clc1ccc(NC(=O)c2ccc(CN3C(=O)C(=O)c4cc(I)ccc34)s2)cc1
O=C1Nc2ccc(cc2C1=O)S(=O)(=O)N1CCOCC1
CCOC(=O)C=CC(Cc1ccccc1)NC(=O)C(CC(=O)C(NC(=O)c1cc(C)on1)C(C)C)Cc1ccccc1 |w:5.4|
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)CCc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
Cc1ccc(cc1)C1=CC=C(C1)C(=C)Cc1cccc(C)c1 |c:10,t:8|
O=C1N(Cc2cc3ccccc3s2)c2ccccc2C1=O
CC(C)(C)C(=O)Nc1ccc(cc1)N(Cc1ccsc1)C(=O)Cn1nnc2ccccc12
Ic1ccc2N(CC3COc4ccccc4O3)C(=O)C(=O)c2c1
COc1ccc2c(O[C@@H]3C[C@@H]4[C@@H](C3)C(=O)N(C)CCCCC=C[C@H]3C[C@]3(NC4=O)C(=O)NS(=O)(=O)C3CC3)cc(nc2c1C)-c1nc(cs1)C(C)C |w:21.21|
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2ccc(Cl)cc2)cc1 |w:7.6,c:12|
O=C1N(Cc2ccccc2)c2ccc(cc2C1=O)S(=O)(=O)N1CCOCC1
CN1C(=O)C(=O)c2cc(ccc12)S(=O)(=O)N1CCN(CCc2ccccc2)CC1
O=C1N(Cc2ccccc2)c2ccc(cc2C1=O)S(=O)(=O)N1CCCCC1
CC(C)C[C@H](NC(=O)c1cc2ccccc2o1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
Cc1csc(n1)-c1nc(cs1)-c1ccnc(SCC(=O)Nc2ccc(Cl)cc2)n1
Cc1cccc2c1ccc3c2C(=O)C(=O)C4=C3OC[C@@H]4C
[H][C@@]1(C[C@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)OC(C)(C)C)C(C)C)\C=C\C(=O)OCC)CCNC1=O
CSc1[nH]nc(NC(=O)c2cccs2)c1S(=O)(=O)c1ccccc1
CC(C)CC(NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccccc1)C(=O)C(F)(F)F
O=C(ON1C(=O)CCC1=O)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
CCOC(O)=C(\C=N\c1ccc(cc1)S(=O)(=O)c1ccc(N\C=C(/C#N)C(=O)OCC)cc1)C#N |w:3.3|
OB(O)c1cccc(COC(=O)c2cc(cc(c2)N(=O)=O)B(O)O)c1
Clc1ccc(cc1)-c1nc(SCCc2ccccc2)[nH]c(=O)c1C#N
CC1=CC(=O)c2c(cccc2O)C1=O
CCOC(=O)c1ccc(cc1)N1NC(=O)C(=Cc2ccc(o2)[N+]([O-])=O)C1=O |w:16.17|
Ic1ccc2N(Cc3ccc(s3)C(=O)N3CCCCC3)C(=O)C(=O)c2c1
CCCCN1C(=O)C(=O)c2cc(ccc12)C(N)=O
CC1CCN(CC1)S(=O)(=O)c1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
Clc1ccc(s1)-c1c[s+]c(CS(=O)(=O)c2cccs2)[nH]1
CCOC(=O)C1OC1C(=O)N(CCC(N)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)C(CC(C)C)NC(=O)OCc1ccccc1
CSc1nn(c(-c2cccs2)c1C#N)-c1c(c(C)nn1C)N(=O)=O |(1.01,.43,;2.35,-.34,;2.35,-1.88,;3.59,-2.78,;3.12,-4.25,;1.58,-4.25,;.67,-5.49,;1.15,-6.96,;-.1,-7.86,;-1.35,-6.96,;-.87,-5.49,;1.1,-2.78,;-.37,-2.31,;-1.83,-1.83,;4.02,-5.49,;5.56,-5.49,;6.04,-6.96,;7.5,-7.43,;4.79,-7.86,;3.54,-6.96,;2.08,-7.43,;6.47,-4.25,;8,-4.41,;5.84,-2.84,)|
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2ccccc2)cc1 |w:7.6,c:12|
CC(CNC(=O)CCC1(C)C(CC(N)=O)C2[N-]C1=C(C)C1=NC(=CC3=NC(=C(C)C4=NC2(C)C(C)(CC(N)=O)C4CCC(N)=O)C(C)(CC(N)=O)C3CCC(N)=O)C(C)(C)C1CCC(N)=O)OP(O)(=O)OC1C(CO)OC(C1O)n1cnc2cc(C)c(C)cc12 |w:23.24,18.19,27.28,t:21,25,30|
Cc1nn(C)c(NCc2ccc(s2)-c2cccs2)c1N(=O)=O
FC(F)(F)C(=O)C(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)OCc1ccccc1
COc1ccc(cc1)-c1nc(SCCc2ccccc2)[nH]c(=O)c1C#N
COc1ccc2c(O[C@@H]3C[C@@H]4N(C3)C(=O)[C@H](CCCCCC=C[C@@H]3C[C@]3(NC4=O)C(O)=O)NC(=O)OC3CCCC3)cc(nc2c1)-c1csc(NC(C)C)n1 |w:21.21|
CC(C)C1=Cc2ccc3c(CCCC3(C)C)c2C(=O)C1=O |t:3|
COc1cc(C=C2SC(=Nc3ccccc3)N(C2=O)c2ccccc2)ccc1OCc1cccc(c1)C(O)=O |w:5.4,9.9|
[H][C@@]12C[C@@](C)(CC[C@]1(C)CC[C@]1(C)C3=CCc4c(C)c(O)c(O)cc4[C@]3(C)CC[C@@]21C)C(O)=O |r,t:14|
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2ncc(s2)-c2ccc3ccccc3c2)cc1
O=C(Cn1nnc2ccccc12)N(Cc1ccsc1)c1ccc(NC(=O)C2CCCCC2)cc1
Cc1coc-2c1C(=O)C(=O)c1c3CCCC(C)(CO)c3ccc-21
CC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)C(C)(C)C)cc1)c1ccsc1
Cc1c(CCC(O)=O)c2cc3[nH]c(cc4nc(cc5[nH]c(cc1n2)c(C)c5C=C)c(C)c4C=C)c(C)c3CCC(O)=O
CC(C)C[C@H](NC(=O)CN1C(=O)CSC1=S)C(=O)N[C@@H](Cc1ccccc1)[C@@H](O)C[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
Ic1ccc2N(C\C=C\c3cc4ccccc4s3)C(=O)C(=O)c2c1
COc1c(ccc(c1)/C=C/C(=O)CC(=O)/C=C/c2cc(c(cc2)O)OC)O
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](Cc1ccccc1)C(O)C[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
COc1ccc(C=CC(=O)NC(CC(C)C)C(=O)N[C@H](Cc2ccccc2)C(O)C[C@@H](Cc2ccccc2)NC(=O)COc2c(C)cccc2C)cc1 |w:6.5|
CC(C)C[C@@H](NC(=O)[C@H](NC(C)=O)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
CC1OC(Oc2c(oc3cc(O)cc(O)c3c2=O)-c2ccc(O)c(O)c2)C(O)C(O)C1O
CN[C@H](CC(C)C)C(=O)N[C@@H]1[C@H](O)c2ccc(Oc3cc4cc(Oc5ccc(cc5Cl)[C@@H](O[C@H]5C[C@](C)(N)[C@@H](O)[C@H](C)O5)[C@@H]5NC(=O)[C@H](NC(=O)[C@@H]4NC(=O)[C@H](CC(N)=O)NC1=O)c1ccc(O)c(c1)-c1c(O)cc(O)cc1[C@H](NC5=O)C(O)=O)c3O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O[C@H]1C[C@](C)(NCc3ccc(cc3)-c3ccc(Cl)cc3)[C@@H](O)[C@H](C)O1)c(Cl)c2
CC#C[C@@H](CC(O)=O)c1ccc(OCc2cccc(c2)-c2ccc(cc2)C(F)(F)F)cc1 |r|
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2ccc(Cl)c(Cl)c2)cc1 |w:7.6,c:12|
COc1ccc2cc(ccc2c1)-c1cc(nn1[C@@H](C)c1ccc(cc1)C(=O)NCCC(O)=O)-c1cc(Cl)cc(Cl)c1 |r|
NC(=O)c1ccc2N(Cc3ccc4cc(ccc4c3)-c3ccccc3)C(=O)C(=O)c2c1
CC(C)C[C@H](NC(=O)c1ccc(o1)N(=O)=O)C(=O)N[C@@H](Cc1ccccc1)C(O)C[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
CC(C)C[C@H](NC(=O)c1cccc(C)c1)C(=O)N[C@@H](Cc1ccccc1)C(O)C[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
CC(C)CC(NC(=O)c1ccc(cc1)C(F)(F)F)C(=O)N[C@H](Cc1ccccc1)C(O)C[C@@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
CC(C)CC(NC(=O)C1=CCOc2ccc(CCl)cc12)C(=O)N[C@H](Cc1ccccc1)C(O)C[C@@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C |t:8|
CC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NS(C)(=O)=O)cc1)c1ccsc1
CC(NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)CF
CC(C)(C)NC(=O)C(N(C(=O)Cn1nnc2ccccc12)c1ccc(NC(=O)c2ccno2)cc1)c1ccsc1
COc1ccc(cc1)-c1nc(SCc2ccc(cc2)[N+]([O-])=O)[nH]c(=O)c1C#N
Oc1cc(cc(O)c1O)C(=O)OC[C@H]1O[C@@H](OC(=O)c2cc(O)c(O)c(O)c2)[C@H](OC(=O)c2cc(O)c(O)c(O)c2)[C@@H](OC(=O)c2cc(O)c(O)c(O)c2)[C@@H]1OC(=O)c1cc(O)c(O)c(O)c1 |r|
CC(C)CC(NC(=O)C(NC(=O)C(NC(C)=O)C(C)C)C(C)O)C(=O)NC(CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
CC(C)c1ccc(cc1)N([C@@H](C(=O)NC(C)(C)C)c1cccnc1)C(=O)c1ccco1
CC[C@@H](C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CCCc1cc(O)nc(SCC(=O)Nc2ccc(Cl)cc2)n1
OC1COC(Oc2c(oc3cc(O)cc(O)c3c2=O)-c2ccc(O)c(O)c2)C(O)C1O
Clc1cccc(CN2CCN(CC2)S(=O)(=O)c2ccc3NC(=O)C(=O)c3c2)c1
[#6]-[#6]-[#8]-[#6](-[#8])=[#6](\[#6]=[#7]\c1ccc(cc1)S(=O)(=O)c1ccc(-[#7]\[#6]=[#6](\[#6](=O)-[#8]-[#6]-[#6])-[#6](=O)-[#8]-[#6]-[#6])cc1)-[#6](=O)-[#8]-[#6]-[#6] |w:3.3|
COc1cc(CN2CCN(CC2)S(=O)(=O)c2ccc3NC(=O)C(=O)c3c2)cc(OC)c1OC
O=C1Nc2ccc(cc2C1=O)S(=O)(=O)N1CCN(CCc2ccccc2)CC1
CC(C)C[C@H](NC(=O)CSc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)C(O)C[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
O=c1[nH]c(SCc2ccc(cc2)N(=O)=O)nc(-c2ccccc2)c1C#N
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)OCc1ccc(cc1)N(=O)=O)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
CCC(=C)C(=O)c1ccc(OCC(=O)NC(C)(C)C(N)=O)c(Cl)c1Cl
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1ncc(s1)-c1ccc(C)cc1
CN(C)CCCNC(=O)C(NC(=O)c1ccc(C)cc1)=Cc1ccc(o1)-c1cccc(c1)[N+]([O-])=O |w:20.21|
CCOC(=O)C=CC(Cc1ccccc1)NC(=O)C(Cc1ccc(F)cc1)NC(=O)C(NC(=O)c1cc(C)on1)C(C)C |w:5.4|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)C(CO)NC(=O)C(NC(=O)OCc1ccccc1)C(C)O)C(C)C)C(=O)N[C@@H](CCC(N)=O)C=N
Cc1coc-2c1C(=O)C(=O)c1c-2ccc2c(C)cccc12
NC(=O)Cc1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
O[C@@H]1C[C@](O)(C[C@@H](OC(=O)C=Cc2ccc(O)c(O)c2)[C@@H]1O)C(O)=O |w:10.9|
O=C1N(Cc2ccc3ccccc3c2)c2ccc(cc2C1=O)S(=O)(=O)N1CCOCC1
O=C(Cc1nccs1)c1nccs1
CC(C)CC(NC(=O)OC(C)(C)C)C(=O)NC(C)C(=O)C(F)(F)F
CC(C)C[C@H](NC(=O)Cc1ccc2ccccc2c1)C(=O)N[C@@H](Cc1ccccc1)C(O)C[C@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
CC(C)CC(NC(=O)CCNC(=O)OC(C)(C)C)C(=O)N[C@H](Cc1ccccc1)C(O)C[C@@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
CC(C)CC(NC(=O)COc1ccc2ccccc2c1)C(=O)N[C@H](Cc1ccccc1)C(O)C[C@@H](Cc1ccccc1)NC(=O)COc1c(C)cccc1C
c1cc(c(cc1[N+](=O)[O-])Cl)NC(=O)c2cc(ccc2O)Cl
C[C@@H](O)[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(C)=O)C(=O)N[C@@H](CO)C(=O)N[C@H](CO)CCC(N)=O
CC(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@H](CO)CCC(N)=O
CN(C)CCCNC(=O)C(NC(=O)c1ccc(C)cc1)=Cc1ccc(o1)-c1ccccc1[N+]([O-])=O |w:20.21|
CCCCN1C(=O)C(=O)c2cc(I)ccc12
OC(=O)c1ccc(C=C2C(=O)N(N=C2c2ccccc2)c2ccc(OC(F)(F)F)cc2)cc1 |w:7.6,c:12|
OC(=O)C(NC(=O)C(NC(=O)c1ccc(Br)cc1)=C\C=C\c1ccccc1)Nc1ccccc1 |w:18.19|
OCC1OC(Oc2c(oc3cc(O)cc(O)c3c2=O)-c2ccc(O)c(O)c2)C(O)C(O)C1O
COc1ccc(NC(=O)CSc2nc(O)cc(n2)-c2ccccc2)cc1OC
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(=O)c1nccs1)C(=O)c1nccs1 |r|
CCC(=C)C(=O)c1ccc(OCC(=O)NC(C)(C)C)c(Cl)c1Cl
CCOC(=O)c1cc(=O)oc2cc(O)c(O)cc12
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](Cc1cccs1)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](CCC(N)=O)C=N
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)c1cc(C)on1)C(C)C)C(=O)N[C@@H](CCC(N)=O)C=N
[H][C@@]12CCc3cc(C(C)C)c(O)cc3[C@@]1(C)CCCC2(C)C |r|
CCN(CC)C(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)c1nc2ccccc2s1 |r|
CC(=O)CCC(=O)N1N=C(CC1c1ccc(Br)cc1)c1c(O)nc2ccc(C)cc2c1-c1ccccc1 |c:8|
Ic1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
O=C1Nc2ccc(cc2C1=O)S(=O)(=O)N1CCN(CC1)c1ccccn1
COc1ccc(cc1)-c1cnc(s1)C(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1
CC(C)CC(NC(=O)C(NC(=O)C(NC(C)=O)C(C)C)C(C)O)C(=O)NC(CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)N(=O)=O
O[C@H]1Cc2c(O)cc(O)cc2OC1c1cc(O)c(O)c2c1cc(cc(O)c2=O)C1Oc2cc(O)cc(O)c2C[C@H]1O
COc1ccc(OCC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]2CCNC2=O)C(=O)c2ncc(s2)-c2ccc(OC)cc2)cc1
Cc1ccc(N2C(=O)CC(Sc3ccccc3C(O)=O)C2=O)c(Br)c1
Fc1ccc(cc1)C(=O)N1C[C@H]2CCCC[C@@H]2C[C@H]1CN[C@@H](Cc1c[nH]cn1)C=O
Nc1nc(CSc2nnc(-c3cccc4ccccc34)n2-c2ccccc2)cs1
OCC1OC(Oc2cc(O)c3c(c2)oc(-c2ccc(O)c(O)c2)c(OC2OC(CO)C(O)C(O)C2O)c3=O)C(O)C(O)C1O
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](CC1CCCCC1)C=O |r|
c1cc(ccc1C(=O)N2C[C@H]3CCCC[C@@H]3C[C@H]2CN[C@@H](Cc4cnc[nH]4)C=O)Br
COc1cc(ccc1O)C1N(CCN(C)C)C(=O)C(O)=C1C(=O)c1ccc(OCC(C)C)cc1C |c:20|
CC(C)CC(NC(=O)C(NC(=O)C(NC(C)=O)C(C)C)C(C)Oc1ccccc1)C(=O)NC(CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2ccccc2c1=O
C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)CF |r|
CN1CCN(CC1)S(=O)(=O)c1ccc2N(Cc3ccccc3)C(=O)C(=O)c2c1
O=C[C@H](Cc1c[nH]cn1)NC[C@@H]1C[C@H]2CCCC[C@@H]2CN1C(=O)c1ccccc1
CC(C)CC(NC(=O)C(NC(=O)C(NC(C)=O)C(C)C)C(C)Oc1ccccc1)C(=O)NC(CCC(=O)N(C)C)C(=O)Cn1[nH]c(=O)c2c(cccc2c1=O)N(=O)=O
[#6]-[#6]-[#8]-[#6](=O)\[#6]=[#6]\[#6@H](-[#6]-[#6@@H]-1-[#6]-[#6]-[#7]-[#6]-1=O)-[#7]-[#6](=O)-[#6@H](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-c1cc(-[#6])on1)-[#6](-[#6])-[#6]
CN1C(=O)C(=O)c2cc(ccc12)C(N)=O
COc1ccc(cc1-c1c(O)cc(O)c2c1oc(cc2=O)-c1ccc(O)cc1)-c1cc(=O)c2c(O)cc(O)cc2o1 |(6.67,-5.39,;5.33,-4.62,;4,-5.39,;4,-6.93,;2.67,-7.7,;1.33,-6.93,;1.33,-5.39,;2.67,-4.62,;2.67,-3.08,;1.33,-2.31,;,-3.08,;1.33,-.77,;2.67,,;2.67,1.54,;4,-.77,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;5.33,1.54,;8,-3.08,;9.34,-2.31,;10.67,-3.08,;10.67,-4.62,;12,-5.39,;9.34,-5.39,;8,-4.62,;,-7.7,;,-9.24,;-1.33,-10.01,;-1.33,-11.55,;-2.67,-9.24,;-4,-10.01,;-4,-11.55,;-5.33,-9.24,;-5.33,-7.7,;-6.67,-6.93,;-4,-6.93,;-2.67,-7.7,;-1.33,-6.93,)|
CC(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CO)C(=O)N[C@H](CO)CCC(N)=O
c1cc(c(cc1Cl)O)Oc2ccc(cc2Cl)Cl
Clc1ccc(cc1)-c1ncc(o1)C(=O)Cc1cncc(Br)c1
CN1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1
COc1cc(C=NNC(=O)C(NC(=O)c2ccccc2)=Cc2ccccc2)cc(OC)c1O |w:5.4,20.21|
[#6]-[#6]-[#8]-[#6](=O)-[#6]-[#6]-[#6@H](-[#6]-[#6@H]-1-[#6]-[#6]-[#7]-[#6]-1=O)-[#7]-[#6](=O)-[#6@H](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#8])-[#7]-[#6](=O)-[#8]C([#6])([#6])[#6])-[#6](-[#6])-[#6]
[#6]-[#6]-[#8]-[#6](=O)-[#6]=[#6]-[#6](-[#6]-[#6]-1-[#6]-[#6]-[#7]-[#6]-1=O)-[#7]-[#6](=O)-[#6](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6](-[#7]-[#6](=O)-[#6](-[#6]-[#8])-[#7]-[#6](=O)-[#8]C([#6])([#6])[#6])-[#6](-[#6])-[#6] |w:5.4|
COC(=O)C1=C(C)N(Cc2cccnc2)C(=O)C1=Cc1ccc(OCC(=O)NCC2=CCCO2)cc1 |w:18.20,c:4,t:31|
CN1CCN(CC1)S(=O)(=O)c1ccc2N(Cc3ccc4ccccc4c3)C(=O)C(=O)c2c1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)Oc1ccccc1)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
Cc1coc-2c1C(=O)C(=O)c1c3CCCC(C)(C)c3ccc-21
O=C(CSc1ncnc2c1sc1nc(N3CCOCC3)c3CCCCc3c21)NCc1ccco1
CCCCN(C)C[C@H]1O[C@H](CN[C@@H](Cc2c[nH]cn2)C=O)CC2CCCCC12
c1c(cc(c(c1O)O)O)[C@@H]2[C@@H](Cc3c(cc(cc3O2)O)O)O
Cn1cnc2c1C(=O)N(C(=O)N2C)C
c1cc(c(cc1[C@@H]2[C@H](Cc3c(cc(cc3O2)O)O)O)O)O
c1cc(c(cc1[C@@H]2[C@H](Cc3c(cc(cc3O2)O)O)OC(=O)c4cc(c(c(c4)O)O)O)O)O
c1c(cc(c(c1O)O)O)[C@@H]2[C@@H](Cc3c(cc(cc3O2)O)O)OC(=O)c4cc(c(c(c4)O)O)O
Cn1c2nc[nH]c2c(=O)n(C)c1=O
Cc1nc(C)c(s1)C(=O)C1=C(O)C(=O)N(CCCN2CCOCC2)C1c1cccc(c1)[N+]([O-])=O |c:10|
CC(C)COC(=O)N[C@@H](C(C)C)C(=O)CCl
C[C@@]1(C(=O)N2[C@H](C(=O)N3CCC[C@H]3[C@@]2(O1)O)Cc4ccccc4)NC(=O)[C@@H]5C[C@@H]6c7cccc8c7c(c[nH]8)C[C@H]6N(C5)C
O=C[C@H](Cc1cnc[nH]1)NC[C@@H]1C[C@H]2CCCC[C@@H]2CN1C(=O)c1ccc(cc1)-c1ccccc1
CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)[C@H](O)CCl
[H][C@@]12CCc3cc(C(C)C)c(OC(C)=O)cc3[C@@]1(C)CCC[C@@]2(C)CO |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(C)=O)C(C)=O
O=C[C@H](Cc1c[nH]cn1)NC[C@@H]1C[C@H]2CCCC[C@@H]2CN1C(=O)c1cccc(c1)-c1ccccc1
O=C[C@H](Cc1c[nH]cn1)NC[C@@H]1C[C@H]2CCCC[C@@H]2CN1C(=O)c1ccccc1-c1ccccc1
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)C(F)(F)F |r|
CC(CC[C@H]1C(=C)CC[C@H]2[C@](C)(CO)CCC[C@]12C)=CCO |w:19.21|
CCN(CC)C(=O)CC[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)c1nc2ccccc2s1 |r|
[H][C@@]12CCc3cc(C(C)C)c(O)cc3[C@@]1(C)CCC[C@@]2(C)C=O |r|
Brc1ccc(cc1)C(=O)N1C[C@H]2CCCC[C@@H]2C[C@@H]1CN[C@@H](Cc1cnc[nH]1)C=O
CC(C)C1=CC2=CC[C@@H]3[C@@]([C@H]2CC1)(CCC[C@@]3(C)C(=O)O)C
CCOC(=O)C=CC(CC1CCNC1=O)NC(=O)C(CC(C)C)NC(=O)C(NC(=O)c1cc(C)on1)C(C)C |w:5.4|
Cc1cc(O)nc(SCC(=O)Nc2ccc(Oc3ccc(Cl)cc3)cc2)n1
COC(OC)c1cc(O)nc(SCC(=O)Nc2ccc(cc2)C(F)(F)F)n1
[H][C@@]12CCc3cc(ccc3[C@@]1(C)CCC[C@@]2(C)C(=O)OC)C(C)C |r|
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)COc1ccccc1)C(C)C)C(=O)N[C@H](Cc1c[nH]cn1)C(=O)c1nccs1
[H][C@@]12CCc3cc(C(C)C)c(O)cc3[C@@]1(C)CCC[C@@]2(C)CO
C[C@H]1COC2=C1C(=O)C(=O)c1c3CCCC(C)(C)c3ccc21 |c:4|
[H][C@@]12CCc3cc(C(C)C)c(O)cc3[C@@]1(C)CC[C@H](O)C2(C)C |r|
O=C[C@H](Cc1cnc[nH]1)NC[C@H]1C[C@@H]2CCCC[C@H]2CN1C(=O)c1ccc(cc1)-c1ccccc1
CCOC(=O)c1cnc(SCC(=O)Nc2ccc(cc2)N(=O)=O)nc1N
CC(C)COC(=O)N[C@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
COc1c2c(cc(c1N3C[C@@H]4CCCN[C@@H]4C3)F)C(=O)C(=CN2C5CC5)C(=O)O
CCCCN(C)C[C@H]1O[C@@H](CN[C@@H](Cc2c[nH]cn2)C=O)CC2CCCCC12
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@H](Cc1c[nH]cn1)C(=O)c1nccs1
CC(C)C[C@@H](NC(=O)[C@H](NC(=O)OCC(C)(C)C)C(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(=O)c1nccs1
[H][C@]12CC[C@@](C)(CC1=CC[C@@]1([H])[C@@](C)(CCC[C@]21C)C(O)=O)C=C |r,c:8|
CC(C)CC(NC(=O)C(NC(=O)C(CCC(=O)OCc1ccccc1)NC(=O)OC(C)(C)C)C(C)C)C(N)=O
CCCN(CCC)C(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(C)C)C(=O)C(F)(F)F |r|
CCOC(=O)C=CC(CC1CCNC1=O)NC(=O)C(Cc1ccccc1)NC(=O)C(NC(=O)c1cc(C)on1)C(C)C |w:5.4|
CCOc1ccc(cc1)N1C(=O)CC(Sc2nc(C)cc(C)n2)C1=O
COc1cccc(c1)-c1nc(SCC(=O)Nc2ccc(cc2)N(=O)=O)[nH]c(=O)c1C#N
c1c(cc(c(c1F)CNC(=O)C2=CN3C[C@@H]4N([C@H]5CC[C@H](C5)O4)C(=O)C3=C(C2=O)O)F)F
CCCN(CCC)C(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)C(F)(F)F |r|
Cc1ccc(cc1)C(NC(=O)OCc1ccccc1)NC(=O)OCc1ccccc1
CC(C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(O)=O)C(=O)CCl
CCCCN(C)C[C@@H]1O[C@@H](CN[C@@H](Cc2c[nH]cn2)C=O)CC2CCCCC12
CCN(CC)C(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C(=O)c1nccs1 |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(=O)N1CCOCC1)C(=O)c1nccs1 |r|
CC(C)CN(C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)O[C@H]1CO[C@H]2OCC[C@@H]12)S(=O)(=O)c1ccc(N)cc1 |r|
CCCN(CCC)C(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C(=O)C(F)(F)F |r|
CCN(CC)C(=O)CC[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)c1nccs1 |r|
[#6]-[#6]-[#8]-[#6](=O)-[#6]=[#6]-[#6@@H](-[#6]-[#6@@H]-1-[#6]-[#6]-[#7]-[#6]-1=O)-[#7]-[#6](=O)-[#6](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6@H](-[#7]-[#6](=O)-c1cc(-[#6])on1)-[#6](-[#6])-[#6] |w:5.4|
C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)C(=O)C(F)(F)F
CCOC(=O)C=CC(CC1CCNC1=O)NC(=O)C(CC(=O)C(NC(=O)c1cc(C)on1)C(C)C)Cc1ccccc1 |w:5.4|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(C)=O)C(C)C)C(=O)N[C@@H](Cc1ccccc1)C=O |r|
[#6]-[#7]-[#6]-1-[#6](-[#8])-[#6](-[#8])-[#6](-[#6]-[#8])-[#8]-[#6]-1-[#8]-[#6]1-[#6](-[#8]-[#6]-2-[#6](-[#8])-[#6](-[#8])-[#6](\[#7]=[#6](\[#7])-[#7])-[#6](-[#8])-[#6]-2\[#7]=[#6](/[#7])-[#7])-[#8]-[#6](-[#6])C1([#8])[#6]=O
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
CC(C)(C)c1ccc(cc1)N([C@H](c2cccnc2)C(=O)NC3CCCCC3)C(=O)CCl
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl |r|
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)C=C
CC(C)(C)c1ccc(cc1)N([C@@H](C(=O)NC1CCCCC1)c1cccnc1)S(=O)(=O)C=C |r|
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NC1CCCCC1)c1cccnc1)S(=O)(=O)C=C |r|
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NC1CCCCC1)c1cccnc1)C(=O)C=O |r|
ClCC(=O)N(C(C(=O)NC1CCCCC1)c1cccnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CCCCC1)c1cncnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CCS(=O)(=O)CC1)c1cncnc1)c1ccc(cc1)-c1cnco1
CC(NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1)S(=O)(=O)c1ccc(C)cc1
Cc1ccc(cc1)S(=O)(=O)CNC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
ClCC(=O)N(C(C(=O)NCCc1ccccc1)c1cncnc1)c1ccc(cc1)-c1cnco1
Cc1cc(ccc1N(C(C(=O)NC1CCCCC1)c1cncnc1)C(=O)CCl)-c1cnco1
Cc1ncoc1-c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cncnc1)C(=O)CCl
ClCC(=O)N(C(C(=O)NC1CCN(CC1)S(=O)(=O)C1CC1)c1cncnc1)c1ccc(cc1)-c1cnco1
CCS(=O)(=O)N1CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
ClCC(=O)N([C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCOCC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N(C(C(=O)NC1CCCCC1)c1cnccn1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CCS(=O)(=O)CC1)c1cnccn1)c1ccc(cc1)-c1cnco1
Cc1ccc(cc1)S(=O)(=O)CNC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cnccn1
ClCC(=O)N([C@H](C(=O)NCCc1ccccc1)c1cnccn1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N([C@H](C(=O)NC1CCN(CC1)S(=O)(=O)C1CC1)c1cnccn1)c1ccc(cc1)-c1cnco1 |r|
CCS(=O)(=O)N1CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cnccn1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cnccn1 |r|
Cc1ccc(CN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)cc1
ClCC(=O)N(CCc1ccccc1)C(C(=O)NC1CCCCC1)c1cccnc1
Cc1ccccc1CCN(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
Cc1cccc(CCN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c1
Cc1ccc(CCN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)cc1
ClCC(=O)N(CCc1ccccc1Cl)C(C(=O)NC1CCCCC1)c1cccnc1
ClCC(=O)N(CCc1cccc(Cl)c1)C(C(=O)NC1CCCCC1)c1cccnc1
ClCC(=O)N(CCc1ccc(Cl)cc1)C(C(=O)NC1CCCCC1)c1cccnc1
Fc1ccccc1CCN(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
Fc1ccc(CN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)cc1
COc1ccccc1CN(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
Fc1cc(Br)ccc1N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
COc1cccc(c1)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
Cc1ccc(cc1C)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
CC(C)(C)c1ccc(N(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c(Br)c1
ClCC(=O)N(CCc1c[nH]c2ccncc12)C(C(=O)NC1CCCCC1)c1cccnc1
FC(F)(F)Oc1ccc(N(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c(c1)C#N
FC(F)(F)Oc1ccc(N([C@@H](C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c(c1)C#N |r|
FC(F)(F)Oc1ccc(N([C@H](C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c(c1)C#N |r|
FC(F)(F)Oc1ccc(N(C(C(=O)NC2CCC(F)(F)CC2)c2cncnc2)C(=O)CCl)c(c1)C#N
FC(F)(F)Oc1ccc(N([C@@H](C(=O)NC2CCC(F)(F)CC2)c2cncnc2)C(=O)CCl)c(c1)C#N |r|
FC(F)(F)Oc1ccc(N([C@H](C(=O)NC2CCC(F)(F)CC2)c2cncnc2)C(=O)CCl)c(c1)C#N |r|
FC(F)(F)Oc1ccc(N(C(C(=O)NC2CCC(F)(F)CC2)c2cnccn2)C(=O)CCl)c(c1)C#N
FC(Cl)C(=O)N(C(C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(OC(F)(F)F)cc1C#N
F[C@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(OC(F)(F)F)cc1C#N |r|
F[C@@H](Cl)C(=O)N([C@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(OC(F)(F)F)cc1C#N |r|
F[C@@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(OC(F)(F)F)cc1C#N |r|
F[C@H](Cl)C(=O)N([C@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(OC(F)(F)F)cc1C#N |r|
CN1CCC(CCN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)CC1
ClCC(=O)N(C(C(=O)NC1CCCCC1)c1cccnc1)c1ccc(cc1)N1CCCC1
CC(NC(=O)C(N(C(=O)CCl)c1ccc(cc1)C(C)(C)C)c1cccnc1)S(=O)(=O)c1ccc(C)cc1
CC(C)(C)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cncc(O)c1)C(=O)CCl
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cncnc1)C(=O)CCl
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1ccnnc1)C(=O)CCl
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1ccnnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccno1)c1ccnnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)C1CO1)c1ccc(cc1)-c1ccno1)c1ccnnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cnccn1)C(=O)CCl
CC(C)(C)c1ccc(cc1)N(C(=O)CCl)C(C)(C(=O)NC1CCCCC1)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(=O)CCl)[C@@](C)(C(=O)NC1CCCCC1)c1cccnc1 |r|
CC(C)(C)c1ccc(cc1)N(C(=O)CCl)[C@](C)(C(=O)NC1CCCCC1)c1cccnc1 |r|
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cncc(c1)C#N)C(=O)CCl
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1ccc(nc1)C#N)C(=O)CCl
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1c[nH]c2ncccc12)C(=O)CCl
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1cccc2n(ccc12)C1CC1)c1cncnc1
Fc1cccc(CCN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c1
Fc1cccc(CCN(C(C(=O)NC2CCC(F)(F)CC2)c2cccnc2)C(=O)CCl)c1
CC(C)(C)OC(=O)CNC(=O)C(N(CCc1cccc(F)c1)C(=O)CCl)c1cccnc1
Fc1ccc(CCN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)cc1
COc1ccccc1CCN(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
CC(Cl)C(=O)N(C(C(=O)NC1CCCCC1)c1cccnc1)c1ccc(cc1)C(C)(C)C
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)C#C
CC(C)(C)c1ccc(cc1)N([C@H](C(=O)NC1CCCCC1)c1ccnnc1)C(=O)CCl |r|
FC1(F)CCC(C1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cncnc1 |r|
COC(=O)c1ccc(NC(=O)[C@H](N(C(=O)CCl)c2ccc(cc2)-c2cncs2)c2cncnc2)[nH]1 |r|
FC(Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
F[C@@H](Cl)C(=O)N([C@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
F[C@@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
F[C@@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1ccno1 |r|
F[C@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1ccno1 |r|
F[C@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)C1CN=CS1 |r,c:35|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CS)c1ccc(cc1)-c1cncs1)c1cncnc1
FC(F)(F)c1cccc(CN(C(C(=O)NC2CCCCC2)c2cccnc2)C(=O)CCl)c1
FC(F)(F)c1ccccc1CN(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
Cc1oc2ccc(cc2c1C)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)CCl
ClCC(=O)N(C(C(=O)NC1CCCCC1)c1cccnc1)c1ccc2ccoc2c1
ClCC(=O)N(C(C(=O)NC1CCOCC1)c1ccnnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CCOCC1)c1cccnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CCOCC1)c1cncnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CCOCC1)c1cnccn1)c1ccc(cc1)-c1cnco1
FC1(F)CCC(C1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
FC1(F)CC[C@H](C1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CC[C@H](C1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CC[C@H](C1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CC[C@@H](C1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CC[C@@H](C1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CC[C@@H](C1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
ClCC(=O)N(C(C(=O)NC1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)N[C@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N([C@H](C(=O)N[C@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N([C@@H](C(=O)N[C@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N(C(C(=O)N[C@@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N([C@@H](C(=O)N[C@@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
ClCC(=O)N([C@H](C(=O)N[C@@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cnco1 |r|
FC1(F)CC(C1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
CC1(COC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
FC1(F)CC2(CC(C2)NC(=O)C(N(C(=O)CCl)c2ccc(cc2)-c2cnco2)c2cncnc2)C1
ClCC(=O)N(C(C(=O)NC1CC2(COC2)C1)c1cncnc1)c1ccc(cc1)-c1cnco1
ClCC(=O)N(C(C(=O)NC1CC2(C1)CS(=O)(=O)C2)c1cncnc1)c1ccc(cc1)-c1cnco1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnc[nH]1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccno1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1ccno1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccncn1)c1cncnc1
CN1CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
Cc1cc(F)cc(F)c1NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
CNC(=O)c1cc(C)c(NC(=O)C(N(C(=O)CCl)c2ccc(cc2)-c2cnco2)c2cncnc2)c(Cl)c1
Fc1cccc(CCN(C(C(=O)NC2CCC(F)(F)CC2)c2cncnc2)C(=O)C2CO2)c1
Fc1cccc(CCN([C@H](C(=O)NC2CCC(F)(F)CC2)c2cncnc2)C(=O)C2CO2)c1 |r|
Fc1cccc(CCN([C@@H](C(=O)NC2CCC(F)(F)CC2)c2cncnc2)C(=O)C2CO2)c1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)C1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)[C@@H]1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)[C@@H]1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)[C@@H]1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)[C@H]1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)[C@H]1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)[C@H]1CO1)c1ccc(cc1)-c1cnco1)c1cncnc1 |r|
Cc1cc(cc(F)c1NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1)-c1cccnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)C1CO1)c1ccc(cc1)-c1ccno1)c1cncnc1
CN(C)C(=O)C1CCCC(C1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cnco1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1ccnnc1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cnccn1
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cnccn1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cnccn1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccno1)c1cnccn1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1cnccn1
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1cnccn1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1cnccn1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1ccnnc1
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1ccnnc1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1cncnc1
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-c1ccccc1)c1cncnc1 |r|
CC(=O)c1ccc(NC(=O)[C@H](N(C(=O)CCl)c2ccc(cc2)-c2ccns2)c2cnccn2)[nH]1 |r|
CC(N(C(=O)CCl)c1ccc(cc1)-c1ccns1)(C(=O)NC1CCC(F)(F)CC1)c1cnccn1
C[C@@](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)(C(=O)NC1CCC(F)(F)CC1)c1cnccn1 |r|
C[C@](N(C(=O)CCl)c1ccc(cc1)-c1ccns1)(C(=O)NC1CCC(F)(F)CC1)c1cnccn1 |r|
CC(C)c1cc(F)c(NC(=O)[C@H](N(C(=O)CCl)c2ccc(cc2)-c2ccns2)c2cncnc2)c(F)c1 |r|
CC(N(C(=O)CCl)c1ccc(cc1)-c1ccno1)(C(=O)NC1CCC(F)(F)CC1)c1cncnc1
C[C@@](N(C(=O)CCl)c1ccc(cc1)-c1ccno1)(C(=O)NC1CCC(F)(F)CC1)c1cncnc1 |r|
C[C@](N(C(=O)CCl)c1ccc(cc1)-c1ccno1)(C(=O)NC1CCC(F)(F)CC1)c1cncnc1 |r|
ClCC(=O)N(C(C(=O)N[C@H]1CCOC1)c1cnccn1)c1ccc(cc1)-c1ccno1 |r|
ClCC(=O)N([C@@H](C(=O)N[C@H]1CCOC1)c1cnccn1)c1ccc(cc1)-c1ccno1 |r|
ClCC(=O)N([C@H](C(=O)N[C@H]1CCOC1)c1cnccn1)c1ccc(cc1)-c1ccno1 |r|
ClCC(=O)N(C(C(=O)N[C@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
ClCC(=O)N([C@@H](C(=O)N[C@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
ClCC(=O)N([C@H](C(=O)N[C@H]1CCOC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
FC1(F)CC[C@@H](C1)NC(=O)C(N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cncnc1 |r|
FC1(F)CC[C@@H](C1)NC(=O)[C@@H](N(C(=O)CCl)c1ccc(cc1)-c1cncs1)c1cncnc1 |r|
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)CC#N)c1ccc(cc1)-c1cncs1)c1cncnc1
F[C@H](Cl)C(=O)N([C@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
F[C@H](Cl)C(=O)N([C@@H](C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1cncs1 |r|
FCC(=O)N(C(C(=O)NC1CCC(F)(F)CC1)c1cncnc1)c1ccc(cc1)-c1cncs1
FC1(F)CCC(CC1)NC(=O)C(N(C(=O)C=C)c1ccc(cc1)-c1cncs1)c1cncnc1
CC1(C)OCc2cc(cnc12)N(C(C(=O)Nc1cncc2ccccc12)c1ccno1)C(=O)CCl
CNC(=O)Cn1c(=O)[nH]\c(=N/c2ccc(OC(F)F)cc2C)n(Cc2cc(F)c(F)c(F)c2)c1=O
CNC(=O)Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)c(F)c2)c1=O
Cn1cnc(Cn2c(=O)[nH]\c(=N/c3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
CCC(CC)COC(=O)[C@@H](C)NP(=O)(OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1 |r|
CC(C)OC(=O)[C@@H](C)NP(=O)(OC[C@@]1(F)O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1 |r|
CC(C)OC(=O)[C@H](C)NP(=O)(OC[C@@]1(F)O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1 |r|
CC(C)CCOC(=O)C[C@H](NP(=O)(OC[C@@]1(F)O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1)C(=O)OCCC(C)C |r|
C[C@H](NP(=O)(OC[C@@]1(F)O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1)C(=O)OCC(C)(C)C |r|
CCC(CC)COC(=O)[C@@H](C)NP(=O)(OC[C@@]1(F)O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1 |r|
CCCOC(=O)[C@H](C)NP(=O)(N[C@@H](C)C(=O)OCCC)OC[C@@]1(F)O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CC(C)OC(=O)[C@@H](C)NP(=O)(OC[C@]1(O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N=[N+]=[N-])Oc1ccccc1 |r|
NC(=O)CCN(NC(=O)CNC(=O)OCc1ccccc1)C(=O)CCl
CC(C)C[C@@H](C(=O)NN(CCC(=O)N)C(=O)CCl)NC(=O)OCc1ccccc1
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CCC(N)=O)C(=O)C(Cl)c1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CCC(N)=O)C(=O)C(C)Cl |r|
CCC(Cl)C(=O)N(CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CCC(N)=O)C(=O)CBr |r|
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)OCc1ccccc1)C(=O)CCl |r|
NC(=O)CCN(NC(=O)[C@H](CC1CCCC1)NC(=O)OCc1ccccc1)C(=O)CCl |r|
NC(=O)CCN(NC(=O)[C@H](CC1CC1)NC(=O)OCc1ccccc1)C(=O)CCl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)OCc1ccccc1)C(=O)CF |r|
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)OCc1ccccc1)C(=O)C(F)Cl |r|
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)OCc1ccccc1)C(=O)[C@@H](F)Cl |r|
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)OCc1ccccc1)C(=O)[C@H](F)Cl |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CC1CCNC1=O)C(=O)CCl |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(CC1CCCNC1=O)C(=O)CCl
CCCN(NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C(=O)CCl
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(Cc1cc[nH]n1)C(=O)CCl
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)NN(Cc1c[nH]cn1)C(=O)CCl
CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)NN(CCC(N)=O)C(=O)CCl
COc1cccc2[nH]c(OC(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)CCl)cc12
CC(C)C[C@H](NC(=O)Oc1cc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)Oc1cc(C)on1)C(=O)NN(CCC(N)=O)C(=O)CCl
COc1cccc2[nH]c(OC(=O)NC(CC(C)C)C(=O)NN(CCC(N)=O)C(=O)CF)cc12
CC(C)C[C@H](NC(=O)Oc1cc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CF
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)\C=C\c1ccc(Cl)cc1F)C(=O)CCl
CC(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1F)C(=O)NN(CCC(N)=O)C(=O)CCl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1)C(=O)CCl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1)C(=O)CF
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)CF
FCC(=O)N(CC1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1
FCC(=O)N(C[C@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1
FCC(=O)N(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1
CN([C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)CCl)C(=O)c1cc2ccccc2[nH]1
CC(C)C[C@H](N(C)C(=O)c1cc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1ccon1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2cccnc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1coc(C)n1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cnoc1C)C(=O)NN(CCC(N)=O)C(=O)CCl
COc1cc2cc(nc2c[nH]1)C(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)CCl
Cc1cc(no1)C(=O)N[C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)CCl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CNC(=O)CCN(NC(=O)[C@H](CC(C)C)N(C)C(=O)c1cc2ccccc2[nH]1)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)NN(CC1CCNC1=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)NN(C[C@H]1CCNC1=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2cnccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CCl
CC(C)C[C@H](NC(=O)c1cc2c(Cl)cccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)c1cc2c(Cl)cccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
CC(C)C[C@H](NC(=O)c1cc2cc(F)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](N(C)C(=O)c1cc2cc(F)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
CC(C)C[C@H](NC(=O)c1cc2cc(Cl)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)c1cc2cc(Cl)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1)C(=O)[C@@H](F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1)C(=O)[C@H](F)Cl
CC(C)C[C@H](NC(=O)c1nc2cc(Cl)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)c1nc2cc(Cl)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
CC(C)C[C@H](NC(=O)c1nc2cc(F)ccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CC1)NC(=O)c1cc2ccccc2[nH]1)C(=O)C(F)Cl
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
CC(C)(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)(C)C[C@H](NC(=O)c1nc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CCC1)NC(=O)c1nc2ccccc2[nH]1)C(=O)C(F)Cl
NC(=O)CCN(NC(=O)[C@H](CC12CC(C1)C2)NC(=O)c1nc2ccccc2[nH]1)C(=O)C(F)Cl
Cc1cc(no1)C(=O)N[C@@H](CC1(C)CC1)C(=O)NN(C[C@H]1CCNC1=O)C(=O)C(F)Cl
Cc1cc(no1)C(=O)N[C@@H](CC12CC(C1)C2)C(=O)NN(C[C@H]1CCNC1=O)C(=O)[C@H](F)Cl
Cc1cc(no1)C(=O)N[C@@H](CC1CCC1)C(=O)NN(C[C@H]1CCNC1=O)C(=O)[C@H](F)Cl
Cc1cc(no1)C(=O)N[C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
Cc1cc(no1)C(=O)N[C@@H](CC1CC1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC(C)(C)CC(NC(=O)c1cnccn1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CCC1)NC(=O)c1cnccn1)C(=O)C(F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cn2ccccc2n1)C(=O)C(F)Cl
COc1cccc(NCC(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl)c1
COc1cccc(NCC(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl)c1
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NS(=O)(=O)Cc1ccccc1)C(=O)[C@H](F)Cl
NC(=O)CCN(NC(=O)[C@H](CC1CCCCC1)NS(=O)(=O)Cc1ccccc1)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)\C=C\c1ccccc1)C(=O)NN(CCC(N)=O)C(=O)[C@@H](F)Cl
CC(C)C[C@H](NC(=O)\C=C\c1ccccc1)C(=O)NN(CCC(N)=O)C(=O)[C@H](F)Cl
CC(C)C[C@H](NC(=O)c1cc2ccncc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
COc1cc2cc([nH]c2cn1)C(=O)N[C@@H](CC(C)C)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC(C)C[C@H](NC(=O)c1cc2ccccn2n1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC(C)C[C@H](NC(=O)c1cc2ncccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC(C)C[C@H](NC(=O)c1cn2ccccc2n1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC(C)C[C@H](NC(=O)c1ncc[nH]1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC(C)C[C@H](NC(=O)c1cc(C)on1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
CC1(C[C@H](NC(=O)c2cc(on2)C(F)(F)F)C(=O)NN(C[C@@H]2CCNC2=O)C(=O)[C@H](F)Cl)CC1
F[C@H](Cl)C(=O)N(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC12CC(C1)C2)NC(=O)c1cc(on1)C(F)(F)F
FC(F)c1cc(no1)C(=O)N[C@@H](CC12CC(C1)C2)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)[C@H](F)Cl
CC(C)CC[C@H](NC(=O)c1cc(C)on1)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)[C@H](F)Cl
Cc1cc(no1)C(=O)N[C@@H](CC1CCCC1)C(=O)NN(CCC(N)=O)C(=O)C(F)Cl
N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)c1nc2ccccc2s1 |r|
N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)c1nc2ccccc2s1 |r|
CC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)c1nc2ccccc2s1 |r|
CS(=O)(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)c1nc2ccccc2s1 |r|
CS(=O)(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](Cc1ccccc1)C(=O)N[C@H](CCCNC(N)=N)C(O)c1nc2ccccc2s1 |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(cc2)[N+]([O-])=O)[C@@H](O)[C@H]1O
COc1cc(ccc1S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)[N+]([O-])=O
COc1ccc(c(c1)[N+]([O-])=O)S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(cc2[N+]([O-])=O)C(F)(F)F)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(Cl)c(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(cc1[N+]([O-])=O)C(F)(F)F
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2cccc(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(F)c(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(Br)c(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O
Cc1ccc(cc1[N+]([O-])=O)S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
CCc1ccc(cc1[N+]([O-])=O)S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
COc1ccc(cc1[N+]([O-])=O)S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1cccc(c1)[N+]([O-])=O
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(Br)c(c1)[N+]([O-])=O
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(C)c(c1)[N+]([O-])=O
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(OC)c(c1)[N+]([O-])=O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2cccc(c2)C#N)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(F)c(c2)C#N)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(Cl)c(c2)C#N)[C@@H](O)[C@H]1O
COc1ccc(cc1C#N)S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1cccc(c1)C#N
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(OC)c(c1)C#N
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(Cl)cc2)[C@@H](O)[C@H]1O
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(Cl)c(Cl)c2)[C@@H](O)[C@H]1O
Cc1ccc(cc1Cl)S(=O)(=O)NC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1cccc(Cl)c1
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(Cl)c(Cl)c1
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(C)c(Cl)c1
CCOC(=O)CCCCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)S(=O)(=O)c1ccc(OC)c(c1)[N+]([O-])=O
COc1ccc(cc1[N+]([O-])=O)S(=O)(=O)N(CCCCOC(C)=O)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
COc1ccc(cc1[N+]([O-])=O)S(=O)(=O)N(CCCCN1C(=O)c2ccccc2C1=O)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12
c1nc(c2c(n1)n(cn2)[C@H]3[C@@H]([C@@H]([C@H](O3)C[C@H](CC[C@@H](C(=O)O)N)N)O)O)N
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N1Cc2ccccc2C1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N(C)Cc1ccccc1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N(C)Cc1ccc(F)c(Cl)c1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N(C)C(=O)c1ccc(F)c(Cl)c1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccccc1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N(C)Cc1cc(F)cc(c1)C#N |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)SCc1ccccc1 |r|
CCCCCCCCCCCCCCCCCCO[C@H](C)[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)SCc1ccccc1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N1Cc2cc(Cl)c(Cl)cc2C1 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N(Cc1ccc(F)c(Cl)c1)C(C)=O |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N1Cc2ccccc2C1=O |r|
CCCCCCCCCCCCCCCCCCOC[C@@H](OCc1ccccc1)C(C)OP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOC[C@@H](OCc1ccccc1)[C@@H](C)OP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OC(=O)c1ccccc1C(O)=O |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)N1C(=O)c2ccccc2C1=O |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Nc1cccc(c1)C#C |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OC(=O)c1ccccc1 |r|
CCCCCCCCCCCCCCCCCCOC[C@@H](COc1ccccc1)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCSCCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCOCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCO[C@H](COCc1ccccc1)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCO[C@H](COCc1ccccc1)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCO[C@H](COCc1ccccc1)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCO[C@H](COCc1ccccc1)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCO[C@H](COCc1ccccc1)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCOCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCO[C@@H](CO[P@](S)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccccc1 |r|
CCCCCCCCCCCCCCCCOC[C@@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1c(cc(C)cc1C#N)C#N |r|
CCCCCCCCCCCCCCCCOC[C@@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)NC(=O)c1ccccc1 |r|
CCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Nc1ccccc1C(O)=O |r|
CCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cc(F)cc(c1)S(C)(=O)=O |r|
CCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1cc(OC)c(C#N)c(OC)c1 |r|
CCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cc(F)cc(c1)C#N |r|
CCCCCCCCCCCCCCCCOC[C@@H](COCc1cc(F)cc(c1)C#N)COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Nc1ccccc1C(O)=O |r|
CCCCCCCCCCCCCCCCCCOC[C@H](Cc1cc(F)cc(c1)C#N)OP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COc1ccc(cn1)C#N)OP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Nc1cc(ccn1)C#N |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cncc(c1)S(C)(=O)=O |r|
CCCCCCCCCCCCCCCCCC(=O)NC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cc(F)cc(c1)C(O)=O |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COc1ccc(nn1)C#N)OP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCNC(=O)[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cc(F)cc(c1)C#N |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)NC(=O)c1cccc(c1)C#N |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)NC(=O)c1ccccc1C#N |r|
CCCCCCCCCCCCCCOCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCOCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCSCCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCSCCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCSCCCOP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccc(F)c(Cl)c1F |r|
CCCCCCCCCCCCCCCCCCOC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cc(F)cc(c1)C#N |r|
CCCCCCCCCCCCCCCCCCC[C@H](COCc1ccc(cc1F)C#N)OP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12 |r|
CCCCCCCCCCCCCCCCCC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccc(cc1F)C#N |r|
CCCCCCCCCCCCCCCCCC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccc(C#N)c(F)c1 |r|
CCCCCCCCCCCCCCCCCCC[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccccc1 |r|
CCCCCCCCCCCCCCC#C[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccccc1 |r|
CCCCCCCCCCCCCCC#C[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1cc(F)cc(c1)C#N |r|
CCCCCCCCCCCCCCC#C[C@H](COP(O)(=O)OC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)OCc1ccc(C#N)c(F)c1 |r|
CC(C)[C@H](NS(C)(=O)=O)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)C(=O)c1cc2ccccc2[nH]1 |r|
CC(C)[C@H](NS(C)(=O)=O)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)[C@H](NS(C)(=O)=O)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3c(cccc3s1)C(F)(F)F)C2(C)C |r|
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)[C@H](NS(C)(=O)=O)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3cccc(c3s1)C(F)(F)F)C2(C)C |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)C(=O)[C@@H]1CCCO1 |r|
CC(C)[C@H](NS(=O)(=O)C1CC1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)(C)[C@H](NS(=O)(=O)C(C)(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)[C@H](NS(=O)(=O)C(C)(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)C(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C)C(C)(C)C |r|
CCC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C)C(C)(C)C |r|
CCS(=O)(=O)N[C@@H](C(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(C)(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(C)(C)[C@H](NS(C)(=O)=O)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C |r|
CC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3ccccc3s1)C2(C)C)C(C)(C)C |r|
CC1(C)C[C@H](N(C1)C(=O)[C@H]1CCCO1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
COC(=O)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)c1cc2ccccc2[nH]1)C(=O)CF |r|
COC(=O)C[C@H](NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)\C=C\c1ccccc1)C2(C)C)C(=O)CF |r|
FCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)C1[C@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl)C(=O)CF |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@H]2CCC[C@H]2CN1C(=O)COc1cccc(c1)-c1ccccc1)C(=O)CF |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2[C@H](CN1C(=O)COc1ccc(Cl)cc1Cl)C2(C)C)C(=O)CF |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2[C@H](CN1C(=O)COc1ccc(Cl)c(Cl)c1)C2(C)C)C(=O)CF |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2[C@H](CN1C(=O)COc1cccc(c1)-c1ccc(Cl)cc1)C2(C)C)C(=O)CF |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](Cc1ccccc1)C=O)C(=O)c1ccc2ccccc2n1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](Cc1ccccc1)C=O)C(=O)c1ccc2ccccc2c1 |r|
CCC[C@@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)c1cc2ccccc2[nH]1)C(=O)C(=O)NC1CC1 |r|
CCC[C@@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)[C@H](C(C)C)c1ccccc1)C(=O)C(=O)NC1CC1 |r|
CCC[C@@H](NC(=O)C1C2[C@H](CN1C(=O)[C@H](C(C)C)c1ccccc1)C2(C)C)C(=O)C(=O)NC1CC1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(OC(F)(F)F)cc1 |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(Cl)c1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)c1ccc2ccccc2c1 |r|
COc1ccc(OCC(=O)N2C[C@@H]3CCC[C@@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
C[C@H](OCc1ccccc1)C(=O)N1C[C@@H]2CCC[C@@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
Fc1cc(F)cc(CCC(=O)N2C[C@@H]3CCC[C@@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
COc1ccc(OCC(=O)N2C[C@H]3[C@@H](C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1OC |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc2OCOc2c1 |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc2OCCOc2c1 |r|
COc1cccc(OCC(=O)N2C[C@H]3[C@@H](C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)c1 |r|
Cc1cc(Cl)ccc1OCC(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
Fc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1F |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc2ccccc2c1 |r|
COc1ccc(OCC(=O)N2C[C@H]3[C@@H](C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1F |r|
COc1ccc(OC(C)C(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)c(Br)c1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Br)cc1Cl |r|
COc1ccc(OCC(=O)N2C[C@H]3[C@@H](C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(F)c(F)c1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1cc(F)cc(F)c1 |r|
COc1cc(OCC(=O)N2C[C@H]3[C@@H](C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)C3(C)C)cc(OC)c1OC |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)CCc1cccc(F)c1 |r|
Fc1cccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
CC(C)(Oc1ccc(Cl)cc1Cl)C(=O)N1Cc2ccccc2CC1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
CC(C)(Oc1ccc(Cl)cc1Cl)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl)C=O |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)C(C)(C)Oc1ccc(Cl)cc1Cl)C=O |r|
ClCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)cc1 |r|
CC1(C)[C@H]2CN(C([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(=O)COc1ccc(Cl)cc1Cl |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1Cl |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1cccc(c1)-c1ccccc1 |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1cccc(c1)-c1ccccc1)C=O |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2[C@H](CN1C(=O)COc1ccc(Cl)c(Cl)c1)C2(C)C)C=O |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2[C@H](CN1C(=O)COc1cccc(c1)-c1ccc(Cl)cc1)C2(C)C)C=O |r|
CC(C)(C)NC(=O)C(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NCc2ccccc2)c(Cl)c1 |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NC2CC2)c(Cl)c1 |r|
Clc1ccc(OCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NCc2ccccn2)c(Cl)c1 |r|
CC1(C)CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl)C=O |r|
CC1(C)[C@H]2CN(C([C@H]12)C(=O)N[C@@H](C[C@H]1C(=O)NCC1(C)C)C=O)C(=O)COc1ccc(Cl)cc1Cl |r|
CC1(C)[C@H]2CN(C([C@H]12)C(=O)N[C@@H](C[C@H]1C(=O)NCC1(F)F)C=O)C(=O)COc1ccc(Cl)cc1Cl |r|
COc1ccc(CNC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
Fc1ccc(CNC(=S)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
Fc1cccc(CNC(=S)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
CC(C)(C)C(NC(=O)Cc1ccc(Cl)cc1Cl)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)C(NCc1ccc(Cl)cc1Cl)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(OCc1ccc(F)cc1F)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(CCc1ccc(Cl)c(F)c1)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
Clc1cc(Cl)cc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
Clc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
Clc1cccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
Clc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(Cl)c1 |r|
Clc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1Cl |r|
CC(Oc1ccc(Cl)cc1Cl)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
Clc1ccc(\C=C\C(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(Cl)c1 |r|
FC(F)(Oc1ccc(Cl)cc1Cl)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
FC(Oc1ccc(Cl)cc1Cl)C(=O)N1C[C@@H]2CCC[C@H]2C1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
Oc1cccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
Oc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
Oc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1O |r|
COc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)cc1 |r|
COc1ccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c(Cl)c1 |r|
COc1cccc(CCC(=O)N2C[C@@H]3CCC[C@H]3C2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@H]2[C@H](CN1C(=O)COc1ccc(OC(F)(F)F)cc1)C2(C)C)C(=O)CF |r|
CC1CNC(=O)[C@@H]1C[C@H](NC(=O)C1[C@@H]2CCC[C@H]2CN1C(=O)COc1ccc(OC(F)(F)F)cc1)C(=O)CF |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C[C@@H]1CCNC1=O)[C@H](O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](Cc1cccc(Cl)c1)C(=O)N[C@@H](CC1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](Cc1cnc[nH]1)C#N |r|
CN1CCC[C@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCC[C@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCC[C@@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCC[C@@]11CCN([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(Nc1ccccc1)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(N[C@@H](C)c1ccccc1)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(C[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)CCCCC2 |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC(C)(C)C[C@@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
Cc1ccn(C(CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)c(=O)c1N |r|
CC(C)(C)OC(=O)N1CCCC11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@]1(C[C@@H]2CC[C@@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N |r,TLB:30:29:22.23:25.26,33:28:22.23:25.26|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NCC(O)=O)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(C[C@@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)CCCCC2 |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CCC2)C[C@@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CC(F)(F)C2)C[C@@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1cccc2cc([nH]c12)C(=O)N1CC2(CCC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
Clc1cccc2cc([nH]c12)C(=O)N1CC2(C[C@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)CCCCC2 |r|
FC1(F)CC2(C1)C[C@@H](N(C2)C(=O)c1cc2cccc(Cl)c2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)O[K])c1ccccc1 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc(F)cc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc(F)cc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc(F)c(F)c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1cc(F)c(F)c(F)c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc2ccccc2c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1cccc2ccccc12)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)N(C)c1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)N(C)c1ccc(F)cc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc2cccnc2c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc2cnccc2c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc2ccccc2n1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1ccc2ncccc2c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1cnc2ccccc2c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1nn(C)c2ccccc12)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1nc2ccccc2s1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1nc2ccccc2n1C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1n[nH]c2ccccc12)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)cc1F |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)cc1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)c(F)c1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)NC1CCC1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)NC1CCCCC1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccccn1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)NC1CC1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)N1CCCCC1 |r|
CN([C@@H](Cc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)cc1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)NC1CCCC1 |r|
CN([C@@H](Cc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccccc1 |r|
CN([C@@H](Cc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccccn1 |r|
CN([C@@H](Cc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)NC1CC1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1c(C)cccc1C |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)N(C)c1ccccc1 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc2ncccc2c1 |r|
CN([C@@H](CC1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)c(F)c1 |r|
CN([C@@H](CC1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)cc1 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)NC1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)c1ccc(F)cc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)N(C)C1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)C1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)NC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CN([C@@H](Cc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)c(F)c1 |r|
CN([C@@H](Cc1ccc(F)cc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(F)c(F)c1 |r|
CCCC[C@H](N(C)C(=O)C(=O)Nc1ccc(F)c(F)c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CCCC[C@H](N(C)C(=O)C(=O)C(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CCCC[C@H](N(C)C(=O)C(=O)NC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CCCC[C@H](N(C)C(=O)C(=O)Nc1cnc2ccccc2c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CN([C@@H](CC1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1cnc2ccccc2c1 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1nc2ccccc2[nH]1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(=O)Nc1nc2ccccc2o1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CN([C@@H](CC1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C(=O)Nc1ccc(cc1C(F)(F)F)C(F)(F)F |r|
CC(C)(C)C[C@H](NC(=O)C(=O)NC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)(C)C[C@H](NC(=O)C(=O)NC1CC1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)(C)C[C@H](NC(=O)C(=O)Nc1c(F)cccc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)(C)C[C@H](NC(=O)C(=O)NC1(CC1)c1ccc(F)cc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
NC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccc(Cl)cc1F
NC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccccc1
NC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)OCc1ccccc1
NC(=O)C(=N/O)\C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccccc1
CC(C)(C)NC(=O)C(=O)C(CC1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccc(Cl)cc1F
NC(=O)C(=O)C(CC1CC1)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccccc1
NC(=O)C(=O)C(CC1CCCC1)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccccc1
CC(C)(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1Cl)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)C#N
CC(C)(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1Cl)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1
CC(C)(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1F)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1
C[C@@H](CC(=O)N[C@@H](CC(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)c1ccccc1
C[C@H](CC(=O)N[C@@H](CC(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)c1ccccc1
CC[C@@H](CC(=O)N[C@@H](CC(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)c1ccccc1
CC[C@H](CC(=O)N[C@@H](CC(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)c1ccccc1
CC(C)(C)C[C@H](NC(=O)C[C@@H](c1ccccc1)C(F)(F)F)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1
CC(C)(C)C[C@H](NC(=O)C[C@H](c1ccccc1)C(F)(F)F)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1
CC(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1F)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(N)=O
CCNC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccc(Cl)cc1F
NC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccc(Cl)cc1Cl
Fc1cc(Cl)ccc1\C=C\C(=O)N[C@@H](CC1CC1)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1
CC(C)(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1F)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(N)=O
CCNC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)(C)C)NC(=O)\C=C\c1ccc(Cl)cc1F
CCNC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccc(Cl)cc1Cl
Clc1ccc(\C=C\C(=O)N[C@@H](CC2CC2)C(=O)NC(C[C@@H]2CCNC2=O)C(=O)C(=O)NC2CC2)c(Cl)c1
CCNC(=O)C(=O)C(C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)(C)C)NC(=O)\C=C\c1ccc(Cl)cc1Cl
CC(C)(C)C[C@H](NC(=O)\C=C\c1ccc(Cl)cc1Cl)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(N)=O
O=C(N[C@@H](CC1CC1)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)OCc1ccccc1
Clc1ccc(CCC(=O)N[C@@H](CC2CC2)C(=O)NC(C[C@@H]2CCNC2=O)C(=O)C(=O)NC2CC2)c(Cl)c1
Fc1cc(Cl)ccc1\C=C\C(=O)N[C@@H](CC1CCC1)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1
CC[C@@H](CC(=O)N[C@@H](CC1CC1)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)c1ccccc1
CC[C@H](CC(=O)N[C@@H](CC1CC1)C(=O)NC(C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)c1ccccc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C[C@H]1CCNC1=O)C(O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1cnc[nH]1)C#N |r|
CN1CCCC11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CN1CCCC11CCN([C@H](CC2CC2)C(=O)N[C@H](C[C@H]2CCNC2=O)C#N)C1=O |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NC(C)(C)C)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NC(C)(C)C)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)C#N)c1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CC1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)CCCCC2 |r|
COc1cccc2[nH]c(cc12)C(=O)N1CC2(CCC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)(C)OC(=O)N1CCCC11CCN([C@H](CC2CC2)C(=O)N[C@H](C[C@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCCC11CCN([C@@H](CC2CC2)C(=O)N[C@H](C[C@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCCC[C@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
CC(C)(C)OC(=O)N1CCCC[C@@]11CCN([C@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C#N)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@@H](CC1CC1)N1CCC2(CCCCN2)C1=O |r|
O=C(N[C@@H](C[C@@H]1CCNC1=O)C#N)[C@H](CC1CC1)N1CCC2(CCCCN2)C1=O |r|
O=C(N[C@H](C[C@H]1CCNC1=O)C#N)[C@@H](CC1CC1)N1CCC2(CCCCN2)C1=O |r|
O=C(N[C@H](C[C@H]1CCNC1=O)C#N)[C@H](CC1CC1)N1CCC2(CCCCN2)C1=O |r|
[H]C12CCC([H])([C@@H]3[C@H]1C(=O)NC3=O)[C@](C2)(NC(=O)[C@@H](CC1CC1)NC(=O)c1cc2c(OC)cccc2[nH]1)C#N |r|
[H]C12CCC([H])([C@@H]3[C@H]1C(=O)NC3=O)[C@](C2)(NC(=O)[C@H](CC1CC1)NC(=O)c1cc2c(OC)cccc2[nH]1)C#N |r|
O=C(N[C@H](CC1CC1)C(=O)NC1(C[C@H]2CC[C@@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N)OCc1ccccc1 |r,w:11.11,TEB:10:11:18.17:14.15|
O=C(N[C@@H](CC1CC1)C(=O)NC1(C[C@H]2CC[C@@H]1[C@@H]1[C@H]2C(=O)NC1=O)C#N)OCc1ccccc1 |r,w:11.11,TEB:10:11:18.17:14.15|
COc1cccc2[nH]c(cc12)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NCc1ccccc1)C#N |r,w:30.33|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(NCc1ccccc1)C#N |r,w:30.33|
CCNC(C#N)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H](CC(C)C)NC(=O)c1cc2c(OC)cccc2[nH]1 |r|
COc1cccc2NC(Cc12)C(=O)N[C@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2NC(Cc12)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O)c1ccccc1 |r|
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
CC(C)(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
CC(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(c1)C(F)(F)F)C2(C)C |r|
Cn1nc(cc1OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NS(C)(=O)=O)C(C)(C)C)C2(C)C)C(F)(F)F |r|
CC(C)(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(c1)C(F)(F)F)C2(C)C |r|
CC(C)(C)[C@H](NS(C)(=O)=O)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
COC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(Cl)c1)C2(C)C)C(C)(C)C |r|
COC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(c1)C(F)(F)F)C2(C)C)C(C)(C)C |r|
CC(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(c1)C(F)(F)F)C2(C)C |r|
COC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C)C(C)(C)C |r|
COC(=O)N[C@@H](C(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(Cl)c1)C2(C)C |r|
CCn1nc(C)cc1OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C2(C)C |r|
CC(C)(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(Cl)c1)C2(C)C |r|
Cn1nc(cc1OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NS(=O)(=O)C(F)(F)F)C(C)(C)C)C2(C)C)C(F)(F)F |r|
COC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccccc1)C2(C)C)C(C)(C)C |r|
CC[C@H]([C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C)C(F)(F)F |r|
CCn1nc(C)cc1OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C)C2(C)C |r|
Cn1nc(cc1OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C2(C)C)C(F)F |r|
CC(C)(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CC(O)NC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CC(O)NC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
CC(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1cccc(Cl)c1)C2(C)C |r|
CC(C)[C@H](NS(C)(=O)=O)C(=O)N1CCC(C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1ccc(F)cc1F)C(F)(F)F |r|
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CC(=O)NC1=O)C(=O)COc1ccc(F)cc1F)C2(C)C |r|
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CC(=O)NC1=O)C(=O)COc1ccccc1F)C2(C)C |r|
Fc1cc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2cc1C(F)(F)F |(-6.29,2.29,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,;-4.96,-.02,;-6.29,-.79,;-7.63,-.02,;-6.29,-2.33,;-4.96,-1.56,)|
FC(F)(F)c1ccc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
FC(F)(F)c1ccc2n(CC#N)c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;-.96,3.83,;-2.29,4.6,;-3.62,5.37,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
FC(F)(F)Oc1ccc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-8.96,-.79,;-7.63,-.02,;-7.63,1.52,;-7.63,-1.56,;-6.29,-.79,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
FC(F)(F)c1cnc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
Nc1cccc2c(cncc12)-n1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F |(7.04,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;.38,-.02,;.38,1.52,;1.71,2.29,;-.96,2.29,;-2.29,1.52,;-3.63,2.29,;-4.96,1.52,;-4.96,-.02,;-3.63,-.79,;-2.29,-.02,;-.96,-.79,;-.96,-2.33,;-6.29,-.79,;-7.63,-.02,;-6.29,-2.33,;-4.96,-1.56,)|
FC(F)(F)c1ccc2[nH]c(=O)n(-c3cncc4CCCCc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
FC(F)(F)c1ccc2C[c](=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
Brc1ccc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-6.29,-.79,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
CC1(C)c2ccc(cc2c(=O)n(-c2cncc3ccccc23)[c]1=O)C(F)(F)F |(-.19,3.62,;-.96,2.29,;-1.73,3.62,;-2.29,1.52,;-3.62,2.29,;-4.96,1.52,;-4.96,-.02,;-3.62,-.79,;-2.29,-.02,;-.96,-.79,;-.96,-2.33,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;.38,1.52,;1.71,2.29,;-6.29,-.79,;-7.63,-.02,;-6.29,-2.33,;-4.96,-1.56,)|
Fc1cc(cc2c1[nH]c(=O)n(-c1cncc3ccccc13)c2=O)C(F)(F)F |(-3.63,3.83,;-3.62,2.29,;-4.96,1.52,;-4.96,-.02,;-3.62,-.79,;-2.29,-.02,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-6.29,-.79,;-7.63,-.02,;-6.29,-2.33,;-4.96,-1.56,)|
COc1ccc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-4.96,-.02,;-4.96,1.52,;-3.63,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.63,-.79,)|
Cc1ccncc1-n1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F |(3.04,1.52,;3.04,-.02,;4.38,-.79,;4.38,-2.33,;3.04,-3.1,;1.71,-2.33,;1.71,-.79,;.38,-.02,;.38,1.52,;1.71,2.29,;-.96,2.29,;-2.29,1.52,;-3.63,2.29,;-4.96,1.52,;-4.96,-.02,;-3.63,-.79,;-2.29,-.02,;-.96,-.79,;-.96,-2.33,;-6.29,-.79,;-7.63,-.02,;-6.29,-2.33,;-4.96,-1.56,)|
FC(F)(F)c1ccc2oc(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,)|
NC(=O)c1cncc(c1)-n1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
FC(F)(F)c1ccc2n(CCC#N)c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;-.96,3.83,;-2.29,4.6,;-2.29,6.14,;-2.29,7.68,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,)|
FC(F)(F)c1ccc2n(C3CC3)c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;-.96,3.83,;-1.73,5.16,;-.19,5.16,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,)|
FS(F)(F)(F)(F)c1ccc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2c1 |(-7.63,-.02,;-6.29,-.79,;-6.29,-2.33,;-4.96,-1.56,;-6.29,.75,;-7.63,-1.56,;-4.96,-.02,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,)|
Cc1cc2[nH]c(=O)n(-c3cncc4ccccc34)c(=O)c2cc1C(F)(F)F |(-6.29,2.29,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;.38,1.52,;1.71,2.29,;.38,-.02,;1.71,-.79,;1.71,-2.33,;3.04,-3.1,;4.38,-2.33,;4.38,-.79,;5.71,-.02,;5.71,1.52,;4.38,2.29,;3.04,1.52,;3.04,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,;-4.96,-.02,;-6.29,-.79,;-6.29,-2.33,;-6.29,.75,;-7.63,-1.56,)|
Fc1cccc2cncc(-n3c(=O)n(CCC#N)c4ccc(cc4c3=O)C(F)(F)F)c12 |(2.14,2.77,;3.04,1.52,;4.38,2.29,;5.71,1.52,;5.71,-.02,;4.38,-.79,;4.38,-2.33,;3.04,-3.1,;1.71,-2.33,;1.71,-.79,;.38,-.02,;.38,1.52,;1.71,2.29,;-.96,2.29,;-.96,3.83,;.38,4.6,;.38,6.14,;.38,7.68,;-2.29,1.52,;-3.62,2.29,;-4.96,1.52,;-4.96,-.02,;-3.62,-.79,;-2.29,-.02,;-.96,-.79,;-.96,-2.33,;-6.29,-.79,;-6.29,-2.33,;-6.29,.75,;-7.63,-1.56,;3.04,-.02,)|
Fc1cccc2cncc(-n3c(=O)c4C[C@H](CCc4n(CC#N)c3=O)C(F)(F)F)c12 |r,wU:15.26,(2.14,2.77,;3.04,1.52,;4.38,2.29,;5.71,1.52,;5.71,-.02,;4.38,-.79,;4.38,-2.33,;3.04,-3.1,;1.71,-2.33,;1.71,-.79,;.38,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,;-4.96,-.02,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;-.96,3.83,;.38,4.6,;1.71,5.37,;.38,1.52,;1.71,2.29,;-6.29,-.79,;-6.29,-2.33,;-6.29,.75,;-7.63,-1.56,;3.04,-.02,)|
Fc1cccc2cncc(-n3c(=O)c4C[C@@H](CCc4n(CC#N)c3=O)C(F)(F)F)c12 |r,wD:15.26,(2.14,2.77,;3.04,1.52,;4.38,2.29,;5.71,1.52,;5.71,-.02,;4.38,-.79,;4.38,-2.33,;3.04,-3.1,;1.71,-2.33,;1.71,-.79,;.38,-.02,;-.96,-.79,;-.96,-2.33,;-2.29,-.02,;-3.62,-.79,;-4.96,-.02,;-4.96,1.52,;-3.62,2.29,;-2.29,1.52,;-.96,2.29,;-.96,3.83,;.38,4.6,;1.71,5.37,;.38,1.52,;1.71,2.29,;-6.29,-.79,;-6.29,-2.33,;-6.29,.75,;-7.63,-1.56,;3.04,-.02,)|
COc1cc(cc(C=O)c1OCC(=O)N1CCC(C1)Oc1cccc(c1)C(=O)N(C)C)-c1cccc2[nH]ncc12
COc1cc(cc(C(=O)CO)c1OCC(=O)N(C)C)-c1cccc2[nH]ncc12
CCC[C@H](NC(=O)c1cccc2nc(-c3cncc4ccccc34)n([C@H]3C[C@@H](C3)C(=O)NC)c12)c1ccc(cc1)C(F)(F)F |wU:25.26,wD:27.31,3.3,(11.14,1.24,;10.37,2.58,;8.83,2.58,;8.06,3.91,;6.52,3.91,;5.75,5.24,;6.52,6.58,;4.21,5.24,;3.44,6.58,;1.9,6.58,;1.13,5.24,;1.9,3.91,;1.42,2.45,;2.67,1.54,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;3.91,2.45,;5.38,1.97,;6.75,2.67,;7.45,1.3,;6.08,.6,;8.91,.82,;10.06,1.85,;9.23,-.69,;10.7,-1.16,;3.44,3.91,;8.83,5.24,;8.06,6.58,;8.83,7.91,;10.37,7.91,;11.14,6.58,;10.37,5.24,;11.14,9.24,;11.91,10.58,;12.47,8.47,;9.8,10.01,)|
CNC(=O)[C@H]1C[C@@H](C1)n1c(nc2cccc(C(=O)N[C@@H](C)c3ccc(cc3)C(F)(F)F)c12)-c1cncc2ccccc12 |wU:6.8,wD:4.3,19.20,(10.7,-1.16,;9.23,-.69,;8.91,.82,;10.06,1.85,;7.45,1.3,;6.75,2.67,;5.38,1.97,;6.08,.6,;3.91,2.45,;2.67,1.54,;1.42,2.45,;1.9,3.91,;1.13,5.24,;1.9,6.58,;3.44,6.58,;4.21,5.24,;5.75,5.24,;6.52,6.58,;6.52,3.91,;8.06,3.91,;8.83,2.58,;8.83,5.24,;8.06,6.58,;8.83,7.91,;10.37,7.91,;11.14,6.58,;10.37,5.24,;11.14,9.24,;11.91,10.58,;12.47,8.47,;9.8,10.01,;3.44,3.91,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,)|
CCC[C@H](NC(=O)c1cccc2nc(-c3cncc4ccccc34)n([C@H]3C[C@@H](C3)C(=O)NC)c12)c1ccc(OC(F)F)cc1 |wU:25.26,wD:27.31,3.3,(11.14,1.24,;10.37,2.58,;8.83,2.58,;8.06,3.91,;6.52,3.91,;5.75,5.24,;6.52,6.58,;4.21,5.24,;3.44,6.58,;1.9,6.58,;1.13,5.24,;1.9,3.91,;1.42,2.45,;2.67,1.54,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;3.91,2.45,;5.38,1.97,;6.75,2.67,;7.45,1.3,;6.08,.6,;8.91,.82,;10.06,1.85,;9.23,-.69,;10.7,-1.16,;3.44,3.91,;8.83,5.24,;8.06,6.58,;8.83,7.91,;10.37,7.91,;11.14,9.24,;10.37,10.58,;8.83,10.58,;11.14,11.91,;11.14,6.58,;10.37,5.24,)|
CCC[C@H](NC(=O)c1cccc2nc(-c3cncc4ccccc34)n([C@H]3C[C@@H](C3)C(=O)NC)c12)c1cccc(c1)C(F)(F)F |wU:25.26,wD:27.31,3.3,(11.14,1.24,;10.37,2.58,;8.83,2.58,;8.06,3.91,;6.52,3.91,;5.75,5.24,;6.52,6.58,;4.21,5.24,;3.44,6.58,;1.9,6.58,;1.13,5.24,;1.9,3.91,;1.42,2.45,;2.67,1.54,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,;3.91,2.45,;5.38,1.97,;6.75,2.67,;7.45,1.3,;6.08,.6,;8.91,.82,;10.06,1.85,;9.23,-.69,;10.7,-1.16,;3.44,3.91,;8.83,5.24,;10.37,5.24,;11.14,6.58,;10.37,7.91,;8.83,7.91,;8.06,6.58,;8.06,9.24,;6.52,9.24,;8.83,10.58,;7.29,7.91,)|
CNC(=O)CCCn1c(nc2cccc(C(=O)N[C@@H](C)c3ccc(cc3)C(F)(F)F)c12)-c1cncc2ccccc12
CNC(=O)[C@H]1C[C@@H](C1)n1c(nc2cccc(C(=O)N[C@@H](C)c3ccc4ccccc4c3)c12)-c1cncc2ccccc12 |wU:6.8,wD:4.3,19.20,(10.7,-1.16,;9.23,-.69,;8.91,.82,;10.06,1.85,;7.45,1.3,;6.75,2.67,;5.38,1.97,;6.08,.6,;3.91,2.45,;2.67,1.54,;1.42,2.45,;1.9,3.91,;1.13,5.24,;1.9,6.58,;3.44,6.58,;4.21,5.24,;5.75,5.24,;6.52,6.58,;6.52,3.91,;8.06,3.91,;8.83,2.58,;8.83,5.24,;10.37,5.24,;11.14,6.58,;10.37,7.91,;11.14,9.24,;10.37,10.58,;8.83,10.58,;8.06,9.24,;8.83,7.91,;8.06,6.58,;3.44,3.91,;2.67,,;1.33,-.77,;1.33,-2.31,;2.67,-3.08,;4,-2.31,;5.33,-3.08,;6.67,-2.31,;6.67,-.77,;5.33,,;4,-.77,)|
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCCCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCCCCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCCCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCCCCCCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCOCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCOCCOCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCOCCOCCOCC(=O)Nc5cccc6C(=O)N(Cc56)C5CCC(=O)NC5=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCOCCOCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cn(CCOCCOCCOCC(=O)Nc5cccc6C(=O)N(C7CCC(=O)NC7=O)C(=O)c56)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccccc3)c(Cl)cc2n1
Cc1ccc(Cn2c(=O)n(Cc3cnn[nH]3)c(=O)[nH]\c2=N/c2cc3cn(C)nc3cc2Cl)cc1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(cc3)C(C)(C)C)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(cc3)[N+]([O-])=O)c(Cl)cc2n1
COc1ccc(Cn2c(=O)n(Cc3cnn[nH]3)c(=O)[nH]\c2=N/c2cc3cn(C)nc3cc2Cl)cc1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(OC(F)(F)F)cc3)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(F)cc3)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(Cl)cc3)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(Br)cc3)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(cc3)-c3ccccc3)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3ccc(cc3)C(F)(F)F)c(Cl)cc2n1
Cc1cc(C)cc(Cn2c(=O)n(Cc3cnn[nH]3)c(=O)[nH]\c2=N/c2cc3cn(C)nc3cc2Cl)c1
COc1cc(Cn2c(=O)n(Cc3cnn[nH]3)c(=O)[nH]\c2=N/c2cc3cn(C)nc3cc2Cl)cc(OC)c1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnn[nH]4)c(=O)n3Cc3cc(F)cc(F)c3)c(Cl)cc2n1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnnn4C)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
CCn1nncc1Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)cc2F)c1=O
CCn1nncc1Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2ccc(cc2)C(F)(F)F)c1=O
CCn1nncc1Cn1c(=O)[nH]\c(=N/c2ccc3nn(C)cc3c2)n(Cc2ccc(F)cc2)c1=O
CCn1nncc1Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2ccc(F)cc2)c1=O
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnnn4C4CC4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
CC(C)n1nncc1Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)cc2F)c1=O
CC(C)Cn1nncc1Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)cc2F)c1=O
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4cnnn4C4CCC4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)C(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl |r|
COC(OC)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)c1cc2ccccc2[nH]1 |r|
CC(C)C[C@@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO |r|
CC(C)C[C@H](NC(=O)c1cc2c(C)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)c1cc2c(C)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1cc2c(C)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl |r|
CC(C)C[C@H](NC(=O)c1cc2c(C)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO |r|
CC(C)C[C@H](NC(=O)c1cc2c(C)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)O[Na] |r|
CC(C)C[C@H](CC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C2(C)C |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](NC(=O)C(F)(F)F)C1CC1 |r|
CC(C)C(=O)N[C@@H](C1CC1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](NC(=O)C1CC1)C1CC1 |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](NC(=O)C(F)F)C1CC1 |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)C(=O)[C@@H](NC(=O)C(F)F)C1CC1 |r|
CC1(C)[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@H](C[C@@H]1CCCNC1=O)C#N)C(=O)[C@@H](NC(=O)C(F)F)C1CC1 |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C(C)C)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C(C)C)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C(C)C)C(=O)CCl)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C(C)(C)C)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C(C)(C)C)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C(=O)CCl)C(C)(C)C)C2(C)C |r|
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)C(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C2(C)C |r|
CC(C)C[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)C(C)(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)C(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)C1CC1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(C)(C)C)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
CC(C)C(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(N)=O)C2(C)C)C(C)(C)C |r|
CC(C)(C)[C@H](NC(=O)C1CC1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)C(F)F)[C@@H](C)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
c1ccc(cc1)CN
CCN(CC)S(=O)(=O)c1ccc(N)cc1
Nc1nc(cs1)-c1ccc(Cl)c(Cl)c1
NC(=O)c1c(N)sc2CCCCc12
Nc1ccc(OC(F)F)cc1
CN1C(=O)c2ccc(N)cc2C1=O
Nc1ccc2C(=O)NC(=O)c2c1
CC(C)(C)c1cc(N)n(n1)-c1ccccc1
CC1=CC(=O)Oc2c1ccc(c2)N
NCC(N1CCOCC1)c1cccnc1
CNCc1ccccc1Br
CNCc1ccc(Cl)cc1
[O-][N+](=O)c1ccccc1N1CCNCC1
Cc1sc(N)nc1-c1ccc(Cl)cc1
CN(C1CCNC1)C(=O)OC(C)(C)C
Nc1c(F)cccc1Br
Cc1cc(N)cc(C)c1Br
Nc1ccnc(Br)c1
CC(N)c1ccc(Br)cc1
Nc1cccc2ccc(O)cc12
Nc1c(F)cc(F)cc1[N+]([O-])=O
Cc1cc(Br)c(Cl)cc1N
COc1cc(Cl)nc(N)n1
Nc1ccc(cc1I)C#N
Nc1ccc(Cl)nc1Cl
O=C(C1COc2ccccc2O1)N1CCNCC1
c1c(cncc1Br)N
Nc1cccc(Cl)c1Br
Nc1cc(Cl)ccc1Br
Nc1cc(F)c(Br)c(F)c1
Nc1cc(ccn1)C(F)(F)F
Nc1nnc(Cl)cc1Br
CC(C)Sc1ccccc1N
C[C@H]1CN(CCN1)C(=O)OC(C)(C)C
CCc1ccc(cc1N)[N+]([O-])=O
Nc1cccnc1Br
Nc1c(F)cc(F)cc1Cl
CCc1cc(Br)ccc1N
Oc1ccccc1N1CCNCC1
Nc1ccc(C#N)c(Br)c1
Nc1nnc(s1)-c1ccncc1
Nc1cnc(Cl)c(Br)c1
COc1ccc(cc1)[C@H](C)N
Nc1cc(F)c(F)cc1Br
Nc1cccc(F)c1[N+]([O-])=O
Cc1cc(N)c(F)cc1Br
O=C(OCc1ccccc1)N1CCNCC1
c1cc(ncc1C(F)(F)F)N
Nc1ccc(Oc2ccc(Cl)cc2)cc1
Nc1ncccc1C(F)(F)F
CCN1CCN(CC1)c2ccc(cc2)N
CC(C)(C)OC(=O)NC1CNC1
CN1CCN(CC1)c2ccccc2N
c1ccc2c(c1)c3c([nH]2)CNCC3
COc1cc(Br)ccc1N
Cc1cccc(C)c1NC(=O)CN1CCNCC1
CC12CC3CC(C)(C1)CC(N)(C3)C2 |TLB:7:1:4.5.8:11,10:9:4:2.7.1,0:1:4:8.9.11,THB:7:5:11:2.1.12,12:1:4:8.9.11,12:9:4:2.7.1,6:5:11:2.1.12|
Nc1cc(Cl)c(O)c(Cl)c1
CN(C)C(=O)CN1CCNCC1
Nc1cc(Cl)cc(c1O)[N+]([O-])=O
COc1ccc(N)cc1C(F)(F)F
Nc1cc(Cl)cc(Cl)c1O
Cc1cc(N)cc(Br)c1
NCCCN1CCS(=O)(=O)CC1
Nc1c(Cl)cc(cc1Cl)C#N
c1cc(ccc1C2(CCNCC2)O)Cl
Nc1ncc(Br)cc1O
Nc1ncnc(Cl)c1Cl
COc1ncc(N)cc1Br
Nc1cc(Cl)c(F)cc1F
Cc1nc(Cl)c(N)c(Cl)n1
Nc1ccc(Cl)cc1C#N
Nc1ncc(Br)nc1Cl
Cc1cc(F)cc(Br)c1N
NCC(c1ccccc1)c1ccccc1
Cc1cc(N)cnc1Br
Nc1cc(Cl)c(F)c(Cl)c1
Nc1ccc(Br)c(Cl)c1Cl
Cc1c(Br)cnc(N)c1[N+]([O-])=O
Cc1cc(Br)c(N)c(c1)[N+]([O-])=O
CN1CCNC(C1)c1ccccc1
c1cc(c(cc1CCN)Cl)Cl
Cc1cc(N)ncc1I
Nc1ccc2OC(F)(F)Oc2c1
NCc1ccc(Br)cc1F
CNC(c1ccccc1)c1ccccc1
c1ccc(cc1)C(c2ccccc2)N
c1cc2c(c(c1)Cl)nc(s2)N
Cc1ccc2ccccc2c1N
C[C@H]1CNCCN1C(=O)OC(C)(C)C
NCc1cc(F)c(F)c(F)c1
CC(C)(C)NCc1ccccc1
Nc1ccccc1-c1nc2ccccc2[nH]1
Nc1ccc(OCc2ccccc2)cc1
Nc1ccccc1Oc1ccccc1
Nc1cccc2c1c(=O)[nH][nH]c2=O
Nc1ccc(cc1[N+]([O-])=O)C(F)(F)F
N[C@@H](Cc1ccc(O)cc1)C(N)=O
Cc1c(N)c(=O)n(-c2ccccc2)n1C
Nc1ccc(cc1)-c1ccccc1
Nc1n[nH]cc1Br
CCNCc1ccc(F)cc1
Oc1ccc(cc1)N1CCNCC1
c1cc(ccc1[C@H](CN)O)O
CCCc1nn(C)c(C(N)=O)c1N
C1CCC(CC1)NC1CCCCC1
Nc1cccc(c1F)C(F)(F)F
c1c(c(c(cn1)Cl)N)Cl
Nc1ccc(cc1C(F)(F)F)[N+]([O-])=O
Nc1ccc(OC(F)(F)F)cc1Cl
Nc1cnc(Br)c(Cl)n1
c1cc(c(cc1N)Cl)Cl
CC(=O)Nc1ccc(N)cc1
Cc1ccc(N)cc1I
Cc1cc(I)ccc1N
CC(C)(C)OC(=O)[C@H]1CCCN1
C1CC(=CCN1)c1ccccc1 |c:2|
Nc1cc(ccc1N1CCCC1)C(F)(F)F
COc1cc2CCNCc2cc1OC
Cc1ccc2c(c1)sc(n2)N
CNC(=O)c1ccccc1N
Nc1ccc(cc1Cl)[N+]([O-])=O
Nc1ccc(I)cc1
CC(C)(C)c1ccc(O)c(N)c1
Nc1c(cnn1-c1ccccn1)C#N
Nc1cc(ccc1Cl)C(F)(F)F
c1cc(ccc1CN)I
Nc1c(Cl)cc(Cl)cc1Br
Cc1ccc(Cl)cc1N1CCNCC1
c1cc2c(cc1CN)OCO2
Nc1cccc(Br)c1
Nc1ccccc1I
Nc1ncc(cc1Cl)C(F)(F)F
Nc1cc(Cl)c(Br)cn1
CC(C)c1cccc(C(C)C)c1N
Nc1nc(Cl)nc2nc[nH]c12
c1ccc(cc1)CC2CCNCC2
c1cc(oc1)C(=O)N2CCNCC2
CCn1c2ccccc2c2cc(N)ccc12
NC1CCN(Cc2ccccc2)CC1
Nc1ccccc1Sc1ccccc1
Nc1ccccc1-c1ccccc1
COc1cc(N)cc(OC)c1
Cc1ccc(N)c(Br)c1
c1cc(ccc1C(F)(F)F)N
NCCc1ccc(Cl)cc1Cl
CCOC(=O)C1CCCNC1
Nc1cccc(I)c1
COc1cc2c(cc1N)oc1ccccc21
Nc1ccccc1Cc1ccccc1
Cc1cc(N)c(Cl)cc1F
COc1cc(Cl)c(C)cc1N
Nc1ccc2nccnc2c1Br
Nc1ccc(Br)c(c1)C(F)(F)F
CN(Cc1ccccc1N)C1CCCCC1
Nc1cc(Cl)cnc1Br
Nc1c(F)c(F)cc(F)c1F
COc1ccc(NC(C)=O)cc1N
CC(N)c1cccc2ccccc12
Nc1cccc(c1)-c1ccccc1
COc1ccc(N)c(c1)[N+]([O-])=O
NC12CC3CC(C1)CC(O)(C3)C2 |TLB:4:3:11:5.6.7,4:5:11:2.3.10,THB:7:5:2:11.8.10,7:8:2:4.5.6|
Cc1cnc(N)c(c1)[N+]([O-])=O
Nc1nc2[nH]cnc2c(=O)[nH]1
Nc1cc(F)c(cc1F)C#N
Nc1ccc(cc1)-c1ccccn1
Nc1cc(Cl)ccc1OC(F)(F)F
c1cc2c(cc1Br)c(n[nH]2)N
C[C@H](N)c1ccc(cc1)[N+]([O-])=O
Cc1nccn1-c1ccc(N)cc1
C1CN(CCN1)c1nsc2ccccc12
CN1CCN(CC1)c1ccc(N)cc1F
C(Cc1ccccc1)N1CCNCC1
Nc1cccc(Cl)c1C#N
O=C(NC1CCNCC1)c1ccccc1
c1ccc(cc1)COc2cccnc2N
CC(C)(C)c1csc(N)n1
Cc1n[nH]c(N)c1Br
FC(F)(F)C1CCNCC1
CSc1ncc(C#N)c(N)n1
c1cc(ccc1CN)OC(F)(F)F
CNCc1csc(n1)C(C)C
C1CC(CCN1)c1nc2ccccc2[nH]1
CC(=O)Nc1ccc(N)c(c1)C(F)(F)F
Nc1ccccc1OCC(F)(F)F
NCc1cc(Cl)cc(Cl)c1
Nc1ccc(cc1)-n1cccn1
Nc1ccc(cc1)-n1ccnc1
Nc1cccc(OC(F)(F)F)c1
Nc1nc2cc(Cl)ccc2s1
Cc1ccc(N)cc1Br
Nc1ccc(cc1)N1CCOCC1=O
O=C(C1CC1)N1CCNCC1
Nc1ncnc2n(CCO)cnc12
NC(=O)c1ccc(Cl)c(N)c1
NCc1ccc(Cl)c(c1)C(F)(F)F
Nc1nnc(s1)C(F)(F)F
Nc1c(cnn1-c1ccc(cc1)[N+]([O-])=O)C#N
Nc1ccc2ccccc2c1O
Cc1cc(Br)cc(C)c1N
NCc1c(Cl)cccc1Cl
CCOc1ccc(CN)cc1
COc1ccccc1N1CCNCC1
C1CC(CCN1)Oc1ccccc1
Nc1ccc2OCCOc2c1
C1CN(CCN1)c1ncccn1
COc1ccc(CN)c(OC)c1
NCCc1ccc(cc1)C(F)(F)F
FC(F)(F)c1ccc(CN2CCNCC2)cc1
Cc1cc(C)c(CN)c(=O)[nH]1
c1cc(ccc1CN)Br
COc1cccc(CN)c1OC
COc1cc(CN)cc(OC)c1
NCc1ccccc1Br
Nc1ccc(Oc2ccccc2Cl)cc1
Nc1ccc(F)cc1Br
COc1cc(CN)ccc1O
CNCc1cccc(c1)[N+]([O-])=O
CN1CCN(CC1)C1CCNCC1
Nc1c(Cl)c(F)nc(F)c1Cl
Brc1ccc(nc1)N1CCNCC1
Nc1ccc(F)nc1Br
CNC1CCN(CC1)C(=O)OC(C)(C)C
Nc1ccc(Br)cc1O
Nc1ccc(SC(F)(F)F)cc1
COc1nc(Br)cnc1N
[O-][N+](=O)c1cccc(c1)N1CCNCC1
COc1cccc(CCN)c1
Nc1ccc2scnc2c1
Nc1cccc(Br)n1
Nc1ccc(O)cc1[N+]([O-])=O
Nc1cc(Br)ccc1F
CNCc1cccc2ccccc12
CNC1CCN(Cc2ccccc2)C1
NCc1cc(F)ccc1Br
c1cc(ccc1CN)[N+](=O)[O-]
Nc1cccc(c1)N1CCOCC1
Nc1ccc(Br)c(c1)[N+]([O-])=O
COc1c(N)cccc1Cl
c1cc(ncc1N)Br
NCCc1ccccc1C(F)(F)F
CCC1(CCC(=O)NC1=O)c1ccc(N)cc1
Nc1c(Cl)cccc1[N+]([O-])=O
COc1ccc(Cl)c(N)c1
Cc1cn(cn1)-c1cc(N)cc(c1)C(F)(F)F
N[C@H]1C(O)O[C@H](CO)[C@@H](O)[C@@H]1O
Nc1ccc(OCc2ccccn2)c(Cl)c1
NCc1ccc(Oc2ccccc2)cc1
c1cc(cc(c1)Br)CN
CCS(=O)(=O)N1CCNCC1
Nc1cccc(n1)C(F)(F)F
COc1ncc(Br)cc1N
CCCOc1ccc(N)cc1
c1cc(c(cc1CN)Cl)F
C1[C@@H]([C@H](O[C@H]1N2C=CC(=NC2=O)N)CO)O
NCc1ccc(cc1)-c1ccccc1
Cc1c(c(c(cn1)CO)CN)O
Cc1ccc2c(c1)c(c[nH]2)CCN
COc1cc2nc(Cl)nc(N)c2cc1OC
Cc1c(N)cccc1Br
Cc1ccc2cccc(N)c2n1
Nc1ccc(F)cc1C(F)(F)F
Nc1ccc(Cl)c(Cl)c1F
Nc1ccc(F)c(F)c1Br
CCOc1ccccc1CN
C1Cc2ccccc2C(N1)c1ccccc1
c1ccc(cc1)C[C@H](CO)N
Nc1ccc(I)cn1
COc1cc(N)c(Cl)cc1Cl
COc1ccc(cc1)-c1cc(N)[nH]n1
Nc1ncc(Br)c(n1)C(F)(F)F
CS(=O)(=O)c1ccc(O)c(N)c1
c1cncc(c1N)Br
FC(F)(F)c1nnc2CNCCn12
Nc1c(Br)cncc1[N+]([O-])=O
Nc1c(F)cc(Br)cc1F
Nc1cc(Cl)nc(Cl)n1
Nc1ccc2cc(Br)ccc2c1
Cc1ccc(c(N)c1)[N+]([O-])=O
Cc1nc(Br)ccc1N
COc1cc(N)nc(OC)n1
Nc1ccc(F)c(Br)c1
Nc1ccc(I)cc1F
Nc1ccc(F)cc1I
NCc1cccc(F)c1Cl
Fc1cccc(CN2CCNCC2)c1
Nc1cnc(Br)cn1
Cc1c(ccc(n1)N)Br
Nc1cc(Br)cc(c1)C(F)(F)F
Nc1ccncc1I
Nc1ccc(I)c(F)c1
N[C@@H]([C@@H](O)c1ccccc1)c1ccccc1
COc1cc(N)ccc1Br
Nc1cc(ccc1Cl)C#N
Nc1ncc(F)cc1Br
Nc1ccc(Br)c2ccccc12
Nc1ccc([N+]([O-])=O)c2ccccc12
c1ccc(cc1)N
Clc1cccc(CN2CCN(C2=O)c2nccc3n[nH]cc23)c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
O=C(Cc1[nH]nc2ccccc12)N(Cc1ccccc1)c1ccc(cc1)N1CCCCC1=O
Clc1ccc2OCCC(C(=O)Nc3cccc4c[nH]nc34)c2c1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1[nH]nc2ccccc12)C(=O)c1ccco1
FC(F)c1nc2ccc(cc2[nH]1)C(=O)N1CCC(CC1)C1CCNC1
Cn1cnc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc3c(CCCS3(=O)=O)c2)c2cccnc2)c1
CS(=O)(=O)Cc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C2CCCCCC2)C(=O)c2cnc[nH]2)c2cccnc2)c1
FC(F)CN1C(=O)CCc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc3ncsc3c2)c2cccnc2)c1
CC(C)S(=O)(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
CN1C(=O)CCc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Cn1ccc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
COc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
COc1ccccc1CN(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
CC(C)Oc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(Cc2cccnc2)C(=O)c2cnc[nH]2)c2cccnc2)c1
Cn1ncc2cc(ccc12)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Cc1nc2ccc(cc2o1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc(Cn3cccn3)cc2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2cccc(Oc3cccnn3)c2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(Cc2ccccc2)C(=O)c2cnc[nH]2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCC3OCCC3C2)C(=O)c2cnc[nH]2)c2cccnc2)c1
COc1cc(ccc1S(=O)(=O)N(C)C)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc(cc2)C2COC2)c2cccnc2)c1
CCOc1ccc(cn1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2cnc(nc2)C2CCC2)c2cccnc2)c1
FC(F)Oc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc3CCOCc3c2)c2cccnc2)c1
COCc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cnc[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2cccc(c2)C2COC2)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C2CCC3(CCO3)CC2)C(=O)c2cnc[nH]2)c2cccnc2)c1 |(6.41,-2.5,;7.92,-2.21,;8.42,-.76,;9.93,-.47,;10.94,-1.63,;10.44,-3.08,;11.45,-4.25,;12.96,-3.96,;13.97,-5.12,;15.48,-4.83,;15.98,-3.38,;16.49,-6,;18,-5.7,;19.01,-6.87,;20.52,-6.58,;21.53,-7.74,;21.02,-9.2,;22.56,-9.31,;22.45,-10.84,;20.91,-10.73,;19.51,-9.49,;18.5,-8.32,;18.5,-4.25,;17.5,-3.08,;20.02,-3.96,;20.67,-2.56,;22.2,-2.75,;22.49,-4.27,;21.14,-5.01,;15.98,-7.45,;16.99,-8.61,;16.49,-10.07,;14.98,-10.36,;13.97,-9.2,;14.47,-7.74,;8.93,-3.38,)|
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cc(CO)n[nH]1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cnc[nH]2)c2ccc(Cl)cc2)c2cccnc2)c1
Clc1ccc2N(Cc3nnc[nH]3)CCC(C(=O)Nc3cncc4ccccc34)c2c1
NS(=O)(=O)c1n[nH]cc1C(=O)NC[C@]1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1ccc2OCCC(CC(=O)N3CCCCC3c3nnc[nH]3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CC(=O)N3CCCC3c3nn[nH]n3)(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OCCC(CC(=O)N3CCCCC3c3ccn[nH]3)(C(=O)Nc3cncc4ccccc34)c2c1
NC(=O)C1Cc2nc[nH]c2CN1C(=O)CC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cnc[nH]1)c1cccnc1)C(=O)c1cocn1
Cc1ncc(CN2CC(C(=O)Nc3cncc4ccc(F)cc34)c3cc(Cl)ccc3C2)[nH]1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cc(=O)[nH]c2ccccc12)C(=O)c1cnc[nH]1
Cc1nnc(CN2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)[nH]1
Clc1ccc2CN(Cc3nnc[nH]3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1cccc(CC(=O)N2CC(=O)c3ccccc3C2)c1
CNS(=O)(=O)c1cc(CNC[C@@]2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)ccc1F
CNS(=O)(=O)c1cc(CNC[C@]2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)ccc1F
OC1CN(C(=O)Cc2cccc(Cl)c2)c2ccccc2C1
CC(C(=O)Nc1cncnc1)c1ccccc1
C[C@@H](C(=O)Nc1cncnc1)c1ccccc1
C[C@H](C(=O)Nc1cncnc1)c1ccccc1
OC1CN(Cc2ccccc12)C(=O)Cc1cccc(Cl)c1
Fc1cccc(c1)S(=O)(=O)N1CCN(CC1)C(=O)\C=C\c1ccccc1
Fc1cccc(c1)S(=O)(=O)N1CCCC(=O)CC1
Fc1cccc(c1)S(=O)(=O)N1CCC(=O)CC1
O=C1CCN(CC1)S(=O)(=O)c1cccs1
Fc1cccc(c1)S(=O)(=O)N1CCN(CC1)C(=O)C=C
O=C1CCCN(CC1)S(=O)(=O)c1cccs1
C=CC(=O)N1CCN(CC1)S(=O)(=O)c1cccs1
NS(=O)(=O)c1ccc(CNC[C@]2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1F
NS(=O)(=O)c1ccc(CNC[C@@]2(CCOc3ccc(Cl)cc23)C(=O)Nc2cncc3ccccc23)cc1F
CNS(=O)(=O)c1ccc2c(NC(=O)C3(CCOc4ccc(Cl)cc34)OC)cncc2c1
Clc1cccc(c1)[C@H](NC(=O)[C@H]1CC[C@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)[C@H](NC(=O)[C@@H]1CC[C@@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
Clc1cccc(c1)[C@@H](NC(=O)[C@H]1CC[C@H](O1)C(=O)N1CCCC1)C(=O)Nc1cncc2ccccc12
c1ccc2c(c1)cncc2NC(=O)[C@@H](c3cccc(c3)Cl)NC(=O)[C@@H]4CC[C@@H](O4)C(=O)N5CCCC5
CS(=O)(=O)Nc1ccc2cncc(NC(=O)C3CCS(=O)(=O)c4ccc(Cl)cc34)c2c1
Clc1ccc2c(c1)C(CCS2(=O)=O)C(=O)Nc1cnn2ccccc12
Fc1ccc2c(NC(=O)[C@@H]3CCS(=O)(=O)c4ccc(Cl)cc34)cncc2c1
CC1(CNC(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
Clc1cccc(CC(=O)Nc2cncc3[nH]ccc23)c1
CS(=O)(=O)c1ccc2cncc(NC(=O)C3CNC(=O)c4c(F)cc(F)cc34)c2c1
Clc1cccc(CC(=O)Nc2cnc3CCCCn23)c1
Clc1ccc2OCC[C@@]3(CC(=O)N(C3=O)c3cncc4ccccc34)c2c1
c1ccc2c(c1)cncc2N3C(=O)C[C@@]4(C3=O)CCOc5c4cc(cc5)Cl
Cc1nc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2s1
Clc1cccc(CC(=O)Nc2cncc3oncc23)c1
CNC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CS(=O)(=O)Nc1ccc2cncc(NC(=O)C3CNC(=O)c4ccc(Cl)cc34)c2c1
CN(C)C(=O)c1cc2c(NC(=O)C3CCOc4ccc(Cl)cc34)cncc2s1
Fc1ccc2c(NC(=O)C3CNC(=O)c4ccc(Cl)cc34)cncc2c1
Clc1ccc2C(=O)NCC(C(=O)Nc3cnn4CCCCc34)c2c1
Clc1ccc2C(=O)NCC(C(=O)Nc3cnn4ccccc34)c2c1
COc1cccc2ncc(NC(=O)Cc3cccc(Cl)c3)n12
Cc1cccc2ncc(NC(=O)Cc3cccc(Cl)c3)n12
CCC1(CNC(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CNC1CCc2c1cncc2NC(=O)C1CCOc2ccc(Cl)cc12
COc1ccc(cc1)-c1ccsc1S(=O)(=O)N1CCN(CC1)C(=O)CCl
CCOC(=O)\C=C\N1CCN(CC1)S(=O)(=O)c1ccccc1
C=CC(=O)N1CCN(CC1)S(=O)(=O)c1ccccc1
COc1ccc(cc1)-c1ccccc1S(=O)(=O)N1CCN(CC1)C(=O)CCl
C=CS(=O)(=O)N1CCN(CC1)S(=O)(=O)c1ccccc1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1CC1
Cc1ccn2c(NC(=O)Cc3cccc(Cl)c3)cnc2c1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)NC1CCC1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC#N)CC1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1CS(=O)(=O)C1
Cc1ccc2ncc(NC(=O)Cc3cccc(Cl)c3)n2c1
Cn1ccn2c(CNC(=O)c3ccc4ncsc4c3)nnc2c1=O
CC1CCN(CCN1Cc1ccccc1)c1cc(C)nc2ncnn12
CN(Cc1nnc2ccccn12)C(=O)c1ccnc2ccccc12
Cc1nnc(CNc2ccc3nnc(-c4ccccc4)n3n2)o1
Brc1cnc2sc(cn12)C(=O)Nc1cnc2nccn2c1
CC(CNC(=O)c1cnc2ccccn12)Nc1nc2ccccc2o1
Cn1c2ccc(cc2oc1=O)S(=O)(=O)Nc1ccc2ncccc2c1
CN(Cc1nc2ccccc2s1)C(=O)c1ccc2n(C)nnc2c1
Cc1cn2c(CNC(=O)c3cnn4ccccc34)c(C)nc2s1
O=C(Nc1cccc2cc[nH]c12)c1cccc2[nH]c(=O)oc12
C(N1CCCC(C1)c1nc2ccccc2o1)c1cnc2cnccn12
CC(Nc1ncnc2cccc(C)c12)c1ccc2[nH]c(=O)[nH]c2c1
Cn1cnnc1-c1cccc(NS(=O)(=O)c2c(Cl)nc3sccn23)c1
Cc1noc2ncc(CNc3ccc(cc3)-c3nnnn3C)cc12
CC(Cc1nc2ccccc2s1)Nc1ccc2nnnn2n1
Cc1ccc(cn1)C(=O)Nc1c(nc2ccccn12)-c1cnn(C)c1
CC(NC(=O)c1c(Cl)nc2ccccn12)c1nnc2ccccn12
CC(NC(=O)c1nccc2cccnc12)c1ccc2[nH]c(=O)oc2c1
Cc1cn2ccc(cc2n1)C(=O)Nc1nc(cs1)-c1cnn(C)c1
CC(NC(=O)c1nc(Br)ccc1C)c1nnc2n1cc[nH]c2=O
Cn1c(NC(=O)Cc2csc3nccn23)nc2ccc(F)cc12
Cc1ccn2ncc(C(=O)Nc3ccc4[nH]c(C)cc(=O)c4c3)c2n1
Cc1ccc(NCc2nnc3n(C)c(=O)c4ccccc4n23)cc1C
O=C(Nc1ccc2c(c1)[nH]ccc2=O)c1ccc2ccncc2c1
O=C(N\N=c1/cc[nH]c2ccccc12)c1ccc2ncccc2c1
Cc1nn(C)c2nc(Cl)cc(NNC(=O)c3ccnc4[nH]nnc34)c12
O=C(Nc1nn2cnnc2s1)c1csc(n1)-c1ccccc1
Brc1cnc2c(cnn2c1)C(=O)Nc1cccc(CC#N)n1
Oc1cc(NNC(=O)c2ccc3[nH]ccc3c2)c2cccnc2n1
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2cc(F)ccc12
Clc1cccc(CC(=O)Nc2cncn2-c2ccccc2)c1
Clc1ccccc1NC(=S)Nc1ccc2[nH]c(=O)[nH]c2c1
CCC(C)c1ccc(cc1)C(NCC(=O)Nc1ccc2[nH]c(=O)[nH]c2c1)c1cccs1
O=C(CCc1nc2ccccc2[nH]1)N1CCC(CCc2ccccc2)CC1
Cc1c(C)n2c(nc3n(C)c(=O)n(CCCO)c(=O)c23)n1-c1ccc(C)c(Cl)c1
OC(CN1CCOCC1)Cn1nc(-c2ccc(Br)cc2)c2ccccc2c1=O
Fc1ccc(CNc2nc(cs2)-c2ccc3[nH]c(=O)oc3c2)cc1
Cc1cccc(CN2CCN(CC2)c2nc3ccccc3nc2C)c1
CC(NC(C)c1ccccc1C)C(=O)Nc1ccc2[nH]c(=O)[nH]c2c1
C\C=C\C=C\C(=O)N1CCC(=CC1)c1c[nH]c2ncccc12 |c:10|
C(N1CCC(=CC1)c1c[nH]c2ccccc12)c1ccno1 |c:4|
CCc1n[nH]c(=O)c(-c2nc(cs2)-c2c[nH]c3ncccc23)c1CC
Fc1ccc(c(F)c1)C1(CCC1)C(=O)NCCCc1nc(=O)[nH][nH]1
CC1CCc2c(C1)sc(\N=C\c1c(C)[nH]c3ccccc13)c2C#N
NC(=O)CN1CCCN(CC1)C(=O)CCSc1ccc(F)cc1
Fc1ccc(NC(=O)NCc2ccc3[nH]c(=O)[nH]c3c2)cc1F
O=C(Cn1ccc(=O)[nH]c1=O)OCc1ccc(cc1)-c1ccccc1
OC(=O)c1ccc(CNCc2c[nH]nc2-c2cccs2)cc1
FC(F)(F)c1ccccc1C1CCCCCC1NC(=O)Cn1cn[nH]c1=O
COC(=O)C1CC1C(=O)N1CCC(CC1)c1c[nH]c2ncccc12
Cc1nc(n[nH]1)-c1cccc(NCc2ccccc2C)c1
CC(C)N1CCCC(N2CCN(CC2)c2ccc3nccnc3n2)C1=O
CC1N(CCNC1=O)C(=O)CCCc1c[nH]c2ccccc12
O=C(CNC(=O)C1CCCC1)N1CCCC1c1nc2ccccc2[nH]1
Clc1ccccc1-c1cc2nc([nH]c(=O)c2s1)-c1nnc[nH]1
Cc1sc2ncnc(N3CCc4c(C3)ncn4C3CC3)c2c1C
O=C(NCC(c1c[nH]c2ccccc12)c1ccccc1)c1cnccn1
Oc1cc(C(=O)NCCc2nnc3CCCn23)c2ccccc2n1
CC(C)(CNC(=O)C1CNC(=O)N1)N1CCc2ccccc2C1
Clc1cccc2C(CCOc12)Nc1ncccn1
CCCCn1nnnc1CNC1CCc2nc(nn2C1)C(C)C
CCN1CCCC1C1CCCN1C(=O)CCc1c[nH]c2ccccc12
Clc1scc(CN2CCC(CC2)c2ccn[nH]2)c1Cl
CCC(N(C)C(=O)Cc1c[nH]c2ncccc12)c1ccncc1
O=C(Nc1cccnc1)N1CCC(CN2CCc3ccccc23)CC1
Oc1ccc2CN(CCOc2c1)C(=O)c1cc(F)cc(F)c1
CC(C(=O)N1CCCCC1c1cccc(C)c1C)c1cncnc1
CCC(N1CCCC(C1)NC(=O)c1ccc2ccccc2c1)C(O)=O
Cc1ccc(cc1)-c1ccc(C(=O)N2CC[C@H](N)C2)c(F)c1
Cc1cc(C)n(n1)C1CCCN(C1)C(=O)c1c[nH]c2ncccc12
Cc1c(Cl)cccc1S(=O)(=O)N(Cc1ccc(F)cc1)c1ccc2[nH]c(=O)[nH]c2c1
O=C(N1CCCC(C1)c1ccn[nH]1)c1ccc(nc1)N1CCCC1
Cc1nnc([nH]1)C1CCN(CC1)C(=O)c1ccc(Br)cc1
O=CNc1ccc(cc1)C(=O)NC(C1CCOCC1)c1ccccc1
O=C(COC(=O)c1cc(=O)[nH]c(=O)[nH]1)N1CCC(Cc2ccccc2)CC1
Oc1ccccc1N1CCN(CC1)C(=O)Cn1ccc(=O)[nH]c1=O
Fc1cccc(C(=O)Nc2ccc(cc2)-c2nnc[nH]2)c1F
CC(NCc1c[nH]c2nccnc12)c1cc(F)ccc1N1CCC(O)CC1
CSc1ccc(cc1)C1N(Cc2cccnc2)C(=O)c2[nH]nc(c12)-c1ccccc1O
Cc1cc(C)c(c(C)c1)S(=O)(=O)N1CCCC1C(=O)Nc1ccc2[nH]c(=O)sc2c1
COc1ccc(cc1COC(=O)c1cnc2ccccc2n1)[N+]([O-])=O
NC(=O)C1Cc2ccccc2CN1CC(=O)N1CCN(CC1)c1ncccn1
Cc1[nH]c2ccccc2c1C(=O)CSc1nc2cc(Cl)cnc2[nH]1
O=C(COC(=O)C1(CCC1)c1ccccc1)c1c[nH]c2ccccc12
Clc1ccc(cc1)-c1n[nH]cc1C(=O)OC1CCN(CC1)C=O
Cc1c(Cl)cc(cc1[N+]([O-])=O)S(=O)(=O)N1CCC(=CC1)c1c[nH]c2ncccc12 |c:18|
COC1CCC2OCCN(C2C1)C(=O)c1ccc2nc[nH]c2c1
Cc1csc2ncc(C(=O)Nc3cccc4ncccc34)c(=O)n12
Cn1c(NC(=O)c2cccnc2-n2cccn2)nc2cc(F)ccc12
Clc1ccc2c(CC(=O)Nc3cccc4[nH]c(=O)[nH]c34)c[nH]c2c1
Cc1cc(nn1-c1ccc(F)cc1)C(=O)Nc1cnc2nccn2c1
Oc1cc(C(=O)NNc2nc3ccccc3[nH]2)c2ccccc2n1
CN(Cc1c(C)nc2sccn12)C(=O)c1cn2ccccc2n1
Fc1cc(F)c2C(=O)NCC(C(=O)Nc3cncc4ccccc34)c2c1
CCC1(CNC(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(cc12)S(C)(=O)=O
Cn1ccc2cncc(NC(=O)Cc3cccc(Cl)c3)c12
Clc1ccc2CN(CC(=O)NC3CC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2CN(CC(=O)NCC#N)CC(C(=O)Nc3cncc4ccccc34)c2c1
Cc1cccn2ncc(NC(=O)C3CNC(=O)c4ccc(Cl)cc34)c12
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCOCC1)C#N
FC1(F)CC1CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CN(C1CC1)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
COc1cc2cncc(NC(=O)Cc3cccc(Cl)c3)c2cc1F
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC#N
COC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CC1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCS(=O)(=O)CC1)C#N
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1CCOCC1
CC(C)(CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1)C#N
CN(CCC#N)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CCN(C)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CC(C)CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
COCCN(C)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Cc1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CN(CC#N)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
COc1cc2c(cc1F)cncc2NC(=O)Cc3cccc(c3)Cl
CC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CS(=O)(=O)C1
FC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CC1
CC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CC1
CNC(=O)CN1Cc2ccc(cc2[C@@H](C1)C(=O)Nc3cncc4c3cccc4)Cl
CNC(=O)CN1C[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2C(=O)N(CC3CC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
CNC(=O)C(C)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2C(=O)NC[C@H](C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2C(=O)NC[C@@H](C(=O)Nc3cncc4ccccc34)c2c1
Cn1ncc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)c12
CNC(=O)CN1CC(C(=O)Nc2cncc3ccc(NS(C)(=O)=O)cc23)c2cc(Cl)ccc2C1=O
Clc1ccc2OCCC(C(=O)Nc3cncn3-c3cccnc3)c2c1
Fc1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
COCCN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
COC(C)(C)CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CC(C)NS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
COc1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
Clc1ccc2CN(CC(C(=O)Nc3cncc4cc(Cl)ccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
COc1ccn2c(NC(=O)Cc3cccc(Cl)c3)cnc2c1
CS(=O)(=O)NCc1ccc(cc1CC(=O)Nc2cncc3c2cccc3)Cl
Clc1ccc(CNS(=O)(=O)N2CC(C2)C#N)c(CC(=O)Nc2cncc3ccccc23)c1
COc1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CNC(=O)CN1C[C@H](c2cc(ccc2C1=O)Cl)C(=O)Nc3cncc4c3cccc4
CNC(=O)CN1C[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CS(=O)(=O)CCN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
NC1CCc2c1cncc2NC(=O)C1CCOc2ccc(Cl)cc12
Clc1ccc2OCCC3(CCN(C3)c3cncc4ccccc34)c2c1
CC1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CN(CCO)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CS(=O)(=O)Nc1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)c2c1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCCC1)C#N
CNC(=O)CN1CC(C(=O)Nc2cncc3ccc(NS(C)(=O)=O)cc23)c2cc(Cl)ccc2C1
FC(F)c1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CC(C)(c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl)O
CCS(=O)(=O)Nc1ccc2cncc(NC(=O)Cc3cccc(Cl)c3)c2c1
COc1ccc2ncc(NC(=O)Cc3cccc(Cl)c3)n2c1
Clc1cccc(CC(=O)Nc2cncc3cccc(Cl)c23)c1
Clc1ccc2c(c1)C(CNS2(=O)=O)C(=O)Nc1cncc2ccccc12
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(Cl)ccc23)c2cc(Cl)ccc2C1
Clc1ccc2OCCC3(CN(C(=O)C3)c3cncc4ccccc34)c2c1
Clc1cccc(CC(=O)Nc2cncc3cc(ccc23)C#N)c1
Clc1cccc(CNC(=O)c2cncc3ccccc23)c1
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)NC1CC1
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1
COc1cc2cncc(NC(=O)Cc3cccc(Cl)c3)c2cc1OC
Cc1nn2c(CNc3ccc(Cn4cncn4)cc3)c(C)nc2s1
Cc1nc2cc(ccc2o1)C(=O)NNc1nc2ccncc2s1
CC(NC(=O)c1ccc2oc(=S)[nH]c2c1)c1nnc2ccccn12
CN(C)CCOc1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
Clc1cccc(CC(=O)Nc2cncc3ccc(OCCN4CCCC4)cc23)c1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CC(=O)N(C2=O)c2cncc3ccccc23)C1
CCNS(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
Clc1ccc2CN(CC3(CC(=O)N(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
ClCC(=O)N1CCN([C@H](C1)C(=O)NC(c1ccccc1)c1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)Nc1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)N1CCOCC1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)NCc1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@H](C1)C(=O)Nc1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)NC(c1ccccc1)c1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)NCC1CCCCC1)S(=O)(=O)c1ccsc1
CCOC(=O)c1cccc(NC(=O)[C@@H]2CN(CCN2S(=O)(=O)c2ccsc2)C(=O)CCl)c1
ClCC(=O)N1CCN([C@@H](C1)C(=O)Nc1ccc2ccccc2c1)S(=O)(=O)c1ccsc1
Cc1cccc(C)c1NC(=O)[C@@H]1CN(CCN1S(=O)(=O)c1ccsc1)C(=O)CCl
COc1ccc(NC(=O)[C@@H]2CN(CCN2S(=O)(=O)c2ccsc2)C(=O)CCl)cc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)Nc1cccc(c1)C#N)S(=O)(=O)c1ccsc1
Cc1ccc(cc1)S(=O)(=O)N1CCN(C[C@H]1C(=O)NCc1ccccc1)C(=O)CCl
Cc1ccc(cc1)S(=O)(=O)N1CCN(C[C@H]1C(=O)NCCc1ccccc1)C(=O)CCl
Fc1ccc(NC(=O)[C@@H]2CN(CCN2S(=O)(=O)c2ccsc2)C(=O)CCl)cc1
Cc1ccc(cc1)S(=O)(=O)N1CCN(C[C@H]1C(=O)NC1CCCCC1)C(=O)CCl
ClCC(=O)N1CCN([C@H](C1)C(=O)NCc1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)N1CCN(CC1)c1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)NC1CCCCC1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@H](C1)C(=O)NCCc1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)NCCc1ccccc1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@H](C1)C(=O)Nc1ccccn1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@H](C1)C(=O)NCc1ccccn1)S(=O)(=O)c1ccsc1
ClCC(=O)N1CCN([C@@H](C1)C(=O)NCc1ccccn1)S(=O)(=O)c1ccsc1
FC(F)(F)COc1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CN(C)C(=O)c1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
Clc1ccc2OCCC3(CCN(C3)c3cncc4cccc(Cl)c34)c2c1
CN(C)c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl
NC(=O)c1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
Cc1cccc2cncc(N3CCC4(C3)CCOc3ccc(Cl)cc43)c12
CN(C)CCOc1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl
Clc1ccc2CN(CC(C(=O)Nc3cncc4c[nH]nc34)c2c1)S(=O)(=O)CC1(CC1)C#N
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1=O
FC(F)(F)COc1ccc2cncc(NC(=O)Cc3cccc(Cl)c3)c2c1
CS(=O)(=O)Oc1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
CS(=O)(=O)Nc1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
CC1NC(=O)c2ccc(Cl)cc2C1C(=O)Nc1cncc2ccc(cc12)S(C)(=O)=O
CN(C)C(=O)c1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cc(cc3)C(=O)N
CC(=O)Nc1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2ccc(c3)C(=O)O
CNC(=O)CN1CC(C(=O)Nc2cncc3cccc(C)c23)c2cc(Cl)ccc2C1=O
Clc1ccc2OCCC3(CCN(C3=O)c3cncc4ccccc34)c2c1
CC(C)N(C)S(=O)(=O)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1
CS(=O)(=O)N1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
CNC(=O)CN1CC(C(=O)Nc2cncc3ccc(F)cc23)c2cc(Cl)ccc2C1=O
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2cc(cc3)C(=O)O
CN(C)c1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
CNC(=O)c1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl
CN(c1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl)S(=O)(=O)C
CNC(=O)c1ccc2cncc(c2c1)NC(=O)Cc3cccc(c3)Cl
c1cc(cc(c1)Cl)CC(=O)Nc2cncc3c2ccc(c3)OCCN4CCCC4
Clc1ccc2CN(CC(C(=O)Nc3cncc4ccccc34)c2c1)C1CCNC1=O
Fc1ccc2c(NC(=O)C3CN(CC(=O)NC4COC4)C(=O)c4ccc(Cl)cc34)cncc2c1
CCCNC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2C(=O)N(CC(=O)NC3COC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2C(=O)N(CC(=O)NCC3CCC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2CCN(C(C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)C1CC1
CN(C)S(=O)(=O)N1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
CCCNC(=O)CN1CC(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1=O
c1cc2c(cc1F)cncc2NC(=O)C34CC(C3)Oc5c4cc(cc5)Cl
COCc1ccc2cncc(NC(=O)Cc3cccc(Cl)c3)c2c1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
CC(C)NC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Fc1ccc2c(NC(=O)C3CN(CC(=O)NCC(F)(F)F)C(=O)c4ccc(Cl)cc34)cncc2c1
FC(F)(F)CNC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2OC3CC(C3)(C(=O)Nc3cncc4ccccc34)c2c1 |THB:3:4:7:9,24:23:7:9,(4.03,2.02,;3.77,.5,;4.95,-.49,;4.69,-2,;3.25,-2.54,;2.99,-1.02,;1.26,-1.04,;.33,-3.04,;.48,-1.74,;.22,-.23,;-1.06,-1.78,;-1.79,-3.14,;-1.87,-.47,;-3.41,-.51,;-4.14,-1.87,;-5.68,-1.91,;-6.48,-.6,;-5.75,.76,;-6.56,2.07,;-5.82,3.42,;-4.28,3.47,;-3.48,2.15,;-4.21,.8,;2.07,-1.55,;2.33,-.04,)|
CC(C)(C)NC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CNS(=O)(=O)N1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
CC(=O)Nc1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
Cc1cc(F)cc2cncc(NC(=O)Cc3cccc(Cl)c3)c12
CS(=O)(=O)Oc1ccc2c(c1)cncc2NC(=O)Cc3cccc(c3)Cl
CC(C)NC(=O)CN1CC(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1=O
Fc1ccc2c(NC(=O)C3CN(CC(=O)NCC4CC4)C(=O)c4ccc(Cl)cc34)cncc2c1
Clc1ccc2C(=O)N(CC(=O)NCC3CC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
CNC(=O)CN1CC(C(=O)Nc2cncc3cccc(Cl)c23)c2cc(Cl)ccc2C1=O
Clc1ccc2C(=O)N(CC(=O)NC3CCC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Fc1ccc2c(NC(=O)C3CN(CC(=O)NC4CCC4)C(=O)c4ccc(Cl)cc34)cncc2c1
Clc1ccc2C(=O)N(CC(=O)NC3CC3)CC(C(=O)Nc3cncc4ccccc34)c2c1
Clc1ccc2OC3CC(C3)(C(=O)Nc3cncc4cc(Cl)ccc34)c2c1 |TLB:25:24:7:9,(6.81,.41,;5.62,-.57,;5.88,-2.09,;4.69,-3.07,;3.25,-2.54,;2.29,-1.74,;.48,-1.74,;.22,-.23,;1.26,-1.04,;.33,-3.04,;1.76,.41,;.74,1.57,;3.27,.72,;3.76,2.18,;2.74,3.33,;3.23,4.79,;4.74,5.1,;5.76,3.94,;7.27,4.24,;8.29,3.09,;9.8,3.39,;7.8,1.63,;6.29,1.32,;5.27,2.48,;2.99,-1.02,;4.18,-.04,)|
C[C@@]1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
C[C@]1(CNS(=O)(=O)c2c1cc(cc2)Cl)C(=O)Nc3cncc4c3cccc4
COC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2=O)CC1
Clc1ccc2CN(C[C@@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCOCC1)C#N
Clc1ccc2CN(C[C@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCOCC1)C#N
Clc1ccc2CN(C[C@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCS(=O)(=O)CC1)C#N
Clc1ccc2CN(C[C@@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCS(=O)(=O)CC1)C#N
COC1(CC1)CS(=O)(=O)N2Cc3ccc(cc3[C@@H](C2)C(=O)Nc4cncc5c4cccc5)Cl
COC1(CS(=O)(=O)N2C[C@H](C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CC1
CC1(CS(=O)(=O)N2C[C@H](C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CS(=O)(=O)C1
CC1(CS(=O)(=O)C1)CS(=O)(=O)N2Cc3ccc(cc3[C@@H](C2)C(=O)Nc4cncc5c4cccc5)Cl
CC(C)(CS(=O)(=O)N1C[C@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1)C#N
CC(C)(CS(=O)(=O)N1C[C@@H](C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1)C#N
Clc1ccc2CN(C[C@@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1CS(=O)(=O)C1
Clc1ccc2CN(C[C@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1CS(=O)(=O)C1
Fc1cc(Cl)c2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CNC(=O)CN1CC(C)(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CNC(=O)CN1CC(C)(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2S1(=O)=O
CNC(=O)CN1CC2(CC(=O)N(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CN(C)C(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CCNC(=O)CN1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Fc1ccc2c(NC(=O)C3CN(CC(=O)NC4CC4)C(=O)c4ccc(Cl)cc34)cncc2c1
CS(=O)(=O)c1ccc2c(NC(=O)C3CN(CC(=O)NC4COC4)C(=O)c4ccc(Cl)cc34)cncc2c1
CS(=O)(=O)c1ccc2c(NC(=O)C3CN(CC(=O)NCC4CC4)C(=O)c4ccc(Cl)cc34)cncc2c1
CCCNC(=O)CN1CC(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CS(=O)(=O)c1ccc2c(NC(=O)C3CN(CC(=O)NCC(F)(F)F)C(=O)c4ccc(Cl)cc34)cncc2c1
CC(C)NC(=O)CN1CC(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CC1(CS(=O)(=O)N2C[C@H](C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CC1
CC1(CS(=O)(=O)N2C[C@@H](C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)CC1
CNC(=O)CN1CC(C)(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2S1(=O)=O
CNC(=O)CN1CC(C)(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2S1(=O)=O
CNC(=O)CN1CC(C)(C(=O)Nc2cncc3cc(Cl)ccc23)c2cc(Cl)ccc2S1(=O)=O
C[C@@H]1NC(=O)c2ccc(Cl)cc2[C@@H]1C(=O)Nc1cncc2ccccc12
c1ccc2c(c1)cncc2NC(=O)[C@@H]3CN(Cc4c3cc(cc4)Cl)[C@@H]5CCNC5=O
CS(=O)(=O)c1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
CNC(=O)N1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
Clc1ccc2CN(C[C@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CNC1)C#N
Clc1ccc2CN(C[C@@H](C(=O)Nc3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CNC1)C#N
CS(=O)(=O)c1ccc2c(NC(=O)C34CC(C3)Oc3ccc(Cl)cc43)cncc2c1 |TLB:22:23:13:15,(-1.33,7.96,;-.31,6.8,;-1.47,5.78,;.84,7.82,;.71,5.65,;.21,4.19,;1.23,3.03,;2.74,3.33,;3.76,2.18,;3.27,.72,;1.76,.41,;.74,1.57,;1.26,-1.04,;.22,-.23,;.48,-1.74,;.33,-3.04,;2.29,-1.74,;3.25,-2.54,;4.69,-3.07,;5.88,-2.09,;5.62,-.57,;6.81,.41,;4.18,-.04,;2.99,-1.02,;5.27,2.48,;5.76,3.94,;4.74,5.1,;3.23,4.79,;2.21,5.95,)|
Clc1ccc2OC3CC(C3)(C(=O)Nc3cncc4cccc(Cl)c34)c2c1 |THB:3:4:7:9,25:24:7:9,(4.03,2.02,;3.77,.5,;4.95,-.49,;4.69,-2,;3.25,-2.54,;2.99,-1.02,;1.26,-1.04,;.33,-3.04,;.48,-1.74,;.22,-.23,;-1.06,-1.78,;-1.79,-3.14,;-1.87,-.47,;-3.41,-.51,;-4.14,-1.87,;-5.68,-1.91,;-6.48,-.6,;-5.75,.76,;-6.56,2.07,;-5.82,3.42,;-4.28,3.47,;-3.48,2.15,;-1.94,2.2,;-4.21,.8,;2.07,-1.55,;2.33,-.04,)|
CC(C)(C)NC(=O)CN1CC(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CC(C)(C)NC(=O)CN1CC(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1=O
COC1(CCOc2ccc(Cl)cc12)C(=O)Nc1cncc2cc(ccc12)S(=O)(=O)N(C)C
CS(=O)(=O)c1ccc2c(NC(=O)C3CN(CC(=O)NC4CC4)C(=O)c4ccc(Cl)cc34)cncc2c1
CCNC(=O)CN1CC(C(=O)Nc2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1=O
CS(=O)(=O)c1ccc2c(NC(=O)C3CN(CC(=O)NC4CCC4)C(=O)c4ccc(Cl)cc34)cncc2c1
CCNC(=O)CN1CC(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CNC(=O)CN1C[C@H](C(=O)Nc2cncc3ccc(F)cc23)c2cc(Cl)ccc2C1=O
CNC(=O)C1(CC1)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2C(=O)N(CC(C(=O)Nc3cncc4ccccc34)c2c1)C1CNC(=O)C1
CNC(=O)CN1C[C@H](c2cc(ccc2C1=O)Cl)C(=O)Nc3cncc4c3cc(cc4)F
CC1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2cc(ccc12)S(C)(=O)=O
CC1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccc(F)cc12
CCC1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(COC)ccc23)c2cc(Cl)ccc2C1
Clc1ccc2C(=O)N(CC(C(=O)Nc3cncc4ccccc34)c2c1)C1CCNC1=O
CNC(=O)CN1Cc2ccc(Cl)cc2[C@]2(CCN(C2=O)c2cncc3ccccc23)C1
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4cccc5)Cl
CNC(=O)CN1CC(C)(C(=O)Nc2cncc3cccc(Cl)c23)c2cc(Cl)ccc2S1(=O)=O
CC(=O)N1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
CN(c1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1)S(C)(=O)=O
Clc1ccc2c(c1)C(CNS2(=O)=O)C(=O)Nc1cncc2CCCCc12
CN(c1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1)S(C)(=O)=O
CC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4cc(ccc34)S(C)(=O)=O)c3cc(Cl)ccc3C2)CS(=O)(=O)C1
COC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4cc(ccc34)S(C)(=O)=O)c3cc(Cl)ccc3C2=O)CC1
CC1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2CCCCc12
CC(C)(O)c1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)c2c1
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(NS(C)(=O)=O)ccc23)c2cc(Cl)ccc2C1=O
CN1C[C@@H](c2cccc(c2)S(=O)(=O)NCCOCCOCCNC(=O)NCCCCNC(=O)NCCOCCOCCNS(=O)(=O)c2cccc(c2)[C@@H]2CN(C)Cc3c(Cl)cc(Cl)cc23)c2cc(Cl)cc(Cl)c2C1 |r|
CC(C)C1NC(=O)C(CCCCN)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(CSSCC(NC1=O)C(=O)NC(C(C)O)C(N)=O)NC(=O)C(N)Cc1ccc2ccccc2c1
NCCCCC(NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CSSC[C@H](N)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(N)=O)C(=O)N1)C(=O)NCC(N)=O
C[C@@H](NC(=O)[C@@H](CCCNC(N)=N)NC(=O)[C@@H](CCCNC(N)=N)NC(=O)[C@@H](CCCNC(N)=N)NC(=O)[C@@H](C)NC(=O)[C@@H](CSSC[C@H](N)C(O)=O)NC(C)=O)C(=O)N[C@H](CCCNC(N)=N)C(N)=O
[H][C@@]12CC[C@]3(C)[C@]([H])(CC=C4[C@]5([H])[C@@H](C)[C@H](C)CC[C@@]5(CC[C@@]34C)C(=O)O[C@@H]3O[C@H](CO[C@@H]4O[C@H](CO)[C@@H](O[C@@H]5O[C@@H](C)[C@H](O)[C@@H](O)[C@H]5O)[C@H](O)[C@H]4O)[C@@H](O)[C@H](O)[C@H]3O)[C@@]1(C)C[C@@H](O)[C@H](O)[C@@]2(C)CO |t:9|
C[C@H](C(O)=O)C(=O)SCCNC(=O)CCNC(=O)[C@H](O)C(C)(C)COP(O)(=O)OP(O)(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1OP(O)(O)=O)n1cnc2c(N)ncnc12
CC(C)(COP(O)(=O)OP(O)(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1OP(O)(O)=O)n1cnc2c(N)ncnc12)[C@@H](O)C(=O)NCCC(=O)NCCSC(=O)CCC(O)=O
CCCCCC(=O)SCCNC(=O)CCNC(=O)[C@H](O)C(C)(C)COP(O)(=O)OP(O)(=O)OC[C@H]1O[C@H]([C@H](O)[C@@H]1OP(O)(O)=O)n1cnc2c(N)ncnc12
CC[C@H](C)[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](C)NC(=O)[C@@H](N)CC(N)=O)C(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(O)=O
COC(=O)N[C@@H](C(C)C)C(=O)N1CCC[C@H]1c1ncc([nH]1)-c1ccc(cc1)-c1ccc(cc1)-c1cnc([nH]1)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)OC)C(C)C
CC(C)C[C@@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H](N)Cc1ccccc1)C(=O)N[C@H](CCCCN)C(=O)N1CCC(N)(CC1)C(O)=O |r|
[#6]-[#6](-[#6])-[#6](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#8])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6]-[#6]-[#7])-[#7]-[#6](=O)-[#6@@H](-[#7])-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccc(-[#8])cc1)-[#6](-[#8])=O
Cc1cc(O)cc(C)c1C[C@H](NC(=O)[C@H](N)CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
C[C@H](N)C(=O)N[C@@H](CCC(N)=O)C(O)=O
Cn1ncc2cc(cnc12)C(=O)NNc1nc2cccnc2s1
Cc1cc(C)n2ncc(C(=O)Nc3ccc4ncsc4c3)c2n1
CC(NCc1cnc2n(C)ncc2c1)c1nc2ccccc2s1
O=C(NCc1nnc2n1cc[nH]c2=O)c1ccnc2ccnn12
Cc1ccc2ncnc(NCc3ccc4nonc4c3)c2c1
Cc1cc2ncc(C(=O)Nc3ccc4oc(C)nc4c3)c(C)n2n1
Cc1cccc2nc(NC3CCN(C3)c3ccc4nncn4n3)sc12
O=C(NNc1nc2cccnc2s1)c1ccc2ccncc2c1
Cc1nc2cc(NC(=O)Cn3cnc4n(C)ncc4c3=O)ccc2o1
Oc1cc(NNC(=O)c2ccnc3ccccc23)c2cccnc2n1
CC(C(=O)Nc1cccc2nccnc12)n1cnc2c(N)ncnc12
O=C(Nc1ccc2nccnc2c1)c1csc2cncn12
Cc1nc2ccc(NCc3cnc4ccccn34)cn2n1
O=C(N1CCn2c(C1)cc1ccccc21)c1ccc2nnnn2c1
Cn1c(NCc2cn3ccnc3s2)nc2ccccc12
CC1NCCn2c1ccc2-c1nc(no1)-c1cnc2cnccn12
Cn1ncc2c1nc(NNC(=O)c1cccn3nccc13)[nH]c2=O
Cc1nc2cc(ccc2o1)C(=O)NNc1ccnc2cccnc12
Cc1nc2ccc(Nc3cc(C)nc4ncnn34)cc2s1
Cc1ccc2nnc(CNc3ccc4nnc(n4n3)C(F)(F)F)n2c1
Cn1ncc2c(NCc3ccc4cccnc4c3)ncnc12
CC(CNc1ccc2nnnn2n1)c1nc2ccccc2s1
Cn1ccn2c(CNc3nc4ccccc4s3)nnc2c1=O
CC(NCc1cnc2ccccn12)c1nnc2ccccn12
Cc1cc2c(nccn2n1)N1CCc2[nH]c3ccccc3c2C1
O=C(Nc1ccc2nncn2c1)c1ccc2scnc2c1
Cc1nc2ccc(NC(=O)Cn3ncn4nccc4c3=O)cc2s1
CC(NC(=O)Nc1ccn2ccnc2c1)c1ccc2[nH]c(=O)oc2c1
CNC(=O)CN1C[C@@H](C(=O)Nc2cncc3cccc(Cl)c23)c2cc(Cl)ccc2C1=O
CNC(=O)CN1C[C@@]2(CC(=O)N(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2OCC[C@@]3(CCCN(C3=O)c3cncc4ccccc34)c2c1
CC1(CN(CC(=O)NC2CC2)S(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2cc(ccc12)S(C)(=O)=O
Clc1cccc(CC(=O)Nc2cncn3cnnc23)c1
CNC(=O)CN1C[C@]2(CC(=O)N(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2CCN(C(C(=O)Nc3cncc4ccccc34)c2c1)C(=O)CC#N
Cc1nc2ccc(NS(=O)(=O)c3cccc4nonc34)cc2o1
Cc1cn2nc(NCc3ccc4ncccc4c3)sc2n1
CN(Cc1c(C)nc2sccn12)C(=O)c1cnc2sccn2c1=O
Cc1nc2ccc(NC(=O)NCc3ccc4[nH]c(=O)[nH]c4c3)cc2o1
CCS(=O)(=O)Nc1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
CC1(CN(CC2CC2)S(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2cc(ccc12)S(C)(=O)=O
CN(C)C(=O)CN1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
CNC(=O)c1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)c2c1
CNC(=O)CN1CC2(CCN(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CC1(CN(CC2CC2)S(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2ccccc12
c1ccc2c(c1)cncc2N3CCC[C@@]4(C3=O)CCOc5c4cc(cc5)Cl
CN(C)CCOc1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)c2c1
CNC(=O)CN1C[C@](C)(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2S1(=O)=O
CC1(CNS(=O)(=O)c2ccc(Cl)cc12)C(=O)Nc1cncc2cccc(Cl)c12
Clc1ccc2CN(CC(C(=O)Nc3cncc4cccc(Cl)c34)c2c1)S(=O)(=O)CC1(CC1)C#N
C[C@]1(CN(S(=O)(=O)c2c1cc(cc2)Cl)CC(=O)NC)C(=O)Nc3cncc4c3cccc4
CNC(=O)CN1C[C@H](C(=O)Nc2cncc3cccc(Cl)c23)c2cc(Cl)ccc2C1=O
CNC(=O)CN1CC(C(=O)Nc2cncc3ccc(cc23)C(C)(C)O)c2cc(Cl)ccc2C1=O
COC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccc(cc34)C(C)(C)O)c3cc(Cl)ccc3C2)CC1
CNC(=O)CN1CC(C(=O)Nc2cncc3CCCCc23)c2cc(Cl)ccc2C1=O
CNC(=O)CN1CC(C(=O)Nc2cncc3ccc(cc23)C(C)(C)O)c2cc(Cl)ccc2C1
Cn1ncc2c(NC(=O)Cc3cccc(Cl)c3)cncc12
Fc1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)c2c1
CNC(=O)CN1C[C@@H](C(=O)Nc2cncc3cc(Cl)ccc23)c2cc(Cl)ccc2C1=O
CNC(=O)CN1C[C@H](C(=O)Nc2cncc3cc(Cl)ccc23)c2cc(Cl)ccc2C1=O
Cc1ncc(CN2CC(C(=O)Nc3cncc4cc(ccc34)S(C)(=O)=O)c3cc(Cl)ccc3C2=O)[nH]1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccc(F)cc23)C1
CC(C)S(=O)(=O)Nc1ccc2c(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
CS(=O)(=O)Nc1ccc2c(NC(=O)[C@H]3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(CC3)C#N)cncc2c1
CS(=O)(=O)Nc1ccc2c(c1)cncc2NC(=O)[C@@H]3CN(Cc4c3cc(cc4)Cl)S(=O)(=O)CC5(CC5)C#N
CC1(CN(Cc2ccc(Cl)cc12)S(=O)(=O)CC1(CC1)C#N)C(=O)Nc1cncc2ccccc12
CC(C)CS(=O)(=O)N1CC(C(=O)Nc2cncc3ccc(cc23)C(C)(C)O)c2cc(Cl)ccc2C1
CNC(=O)c1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(C)CS(=O)(=O)C3)c2c1
CC1(CS(=O)(=O)N2CC(C(=O)Nc3cncc4cccc(Cl)c34)c3cc(Cl)ccc3C2)CS(=O)(=O)C1
CNC(=O)CN1CC(C(=O)Nc2cncc3cc(NS(C)(=O)=O)ccc23)c2cc(Cl)ccc2C1
CN(C)CCOc1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(C)CS(=O)(=O)C3)c2c1
COCCN1CCc2ccc(Cl)cc2C1C(=O)Nc1cncc2ccccc12
CC(C)(O)c1ccc2cncc(NC(=O)C3CN(Cc4ccc(Cl)cc34)S(=O)(=O)CC3(C)CS(=O)(=O)C3)c2c1
Clc1ccc2CN(CC(C(=O)Nc3cncc4cc(NS(=O)(=O)C5CC5)ccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc(CNS(=O)(=O)CC2(CC2)C#N)c(CC(=O)Nc2cncc3ccccc23)c1
CS(=O)(=O)Nc1ccc2c(NC(=O)Cc3cccc(Cl)c3)cncc2c1
CNC(=O)CN1C(C)C(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CN1CC(C)(C(=O)Nc2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2S1(=O)=O
CC(C)CN1CC(C)(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2S1(=O)=O
Clc1ccc2CN(C[C@]3(CC(=O)N(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc2CN(C[C@@]3(CC(=O)N(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc2CN(C[C@@]3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
c1ccc2c(c1)cncc2N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N
[H][C@@]1([#6]-[#6][C@]2([#6])[C@]1([H])[#6@H](-[#8])-[#6][C@]1([H])[C@@]3([#6])[#6]-[#6]-[#6@H](-[#8][C@]4([H])[#8]-[#6@H](-[#6]-[#8])-[#6@@H](-[#8])-[#6@H](-[#8])-[#6@H]4-[#8])C([#6])([#6])[C@]3([H])[#6]-[#6][C@@]21[#6])[C@]([#6])([#8])[#6]-[#6]\[#6]=[#6](\[#6])-[#6] |r|
COc1c(O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)cc2oc(cc(=O)c2c1O)-c1ccc(O)cc1 |r|
C[C@@H]1[C@@]2(CC[C@@H](C)CO2)O[C@H]2C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@]12O |t:16|
COC(C)(C)\C=C\C[C@@H](C)[C@H]1CC[C@@]2(C)[C@@H]3[C@@H](O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)C=C4[C@@H](CC[C@H](O)C4(C)C)[C@@]3(CC[C@]12C)C=O |c:30|
C[C@H](C\C=C\C(C)(C)O)[C@H]1CC[C@@]2(C)[C@@H]3C=C[C@]45OC(O)[C@@]3(CC[C@]12C)[C@@H]4CC[C@H](O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)C5(C)C |c:15,TLB:20:19:14.15.16:26|
CC(CCC(OC1OC(COC2OC(CO)C(O)C(O)C2O)C(O)C(O)C1O)C(C)(C)O)C1CCC2(C)C3CC=C4C(CCC(O)C4(C)C)C3(C)C(O)CC12C |c:41|
CC1=C[C@H]([C@H]([C@@H](C1)c1ccc(O)cc1O)C(=O)c1ccc(O)cc1O)c1c(O)cc(cc1O)-c1cc2ccc(O)cc2o1 |t:1|
C[C@H](C\C=C\C(C)(C)O)[C@H]1CC[C@@]2(C)[C@@H]3C=C[C@@]45OC[C@]3(CC[C@]12C)[C@@H]4CC[C@H](O)C5(C)C |c:15|
[#6]\[#6](-[#6])=[#6]\[#6]-[#6]\[#6](-[#6])=[#6]\[#6]-[#6]\[#6](-[#6])=[#6]\[#6]-[#6]\[#6](-[#6])=[#6]\[#6]-c1cc(-[#8])cc2\[#6](=[#6](/[#6])-[#6])-[#6](=O)-[#8]-c12
[#6]-[#8]-c1cc(-[#8])c(-[#6]\[#6]=[#6](/[#6])-[#6])c(-[#8])c1-[#6](=O)\[#6]=[#6]\c1ccc(-[#8])cc1
CC(C)(O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CNC(=O)Nc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CC1(OCCO1)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
OCCNC(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CCNC(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)-n2ccnc2)c2cccnc2)c1
OC1(COC1)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
OCCCNC(=O)c1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(cc2)C#N)c2cccnc2)c1
Fc1cccc(CCNC(=O)C(N(C(=O)c2cocn2)c2ccc(NC(=O)NC3CC3)cc2)c2cccnc2)c1
COCOc1ccc(cc1)N(C(C(=O)NCCc1cccc(F)c1)c1cccnc1)C(=O)c1cocn1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3CCCCc23)C1
c1cc2c(cc1Cl)[C@@H](CNS2(=O)=O)C(=O)Nc3cncc4c3CCCC4
Clc1ccc2c(c1)[C@H](CNS2(=O)=O)C(=O)Nc1cncc2CCCCc12
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4CCCCc34)c2c1)S(=O)(=O)CC1(CC1)C#N
CNC(=O)C(C)(C)N1CC(C(=O)Nc2cncc3ccccc23)c2cc(Cl)ccc2C1=O
C[C@]1(CNS(=O)(=O)c2c1cc(cc2)Cl)C(=O)Nc3cncc4c3CCCC4
C[C@@]1(CNS(=O)(=O)c2c1cc(cc2)Cl)C(=O)Nc3cncc4c3CCCC4
COC1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4cc(ccc34)S(C)(=O)=O)C2)CC1
Fc1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCOCC1)C#N
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCC1)C#N
COC1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccccc34)C2)CC1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1CS(=O)(=O)C1
CC1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccccc34)C2)CC1
CNC(=O)C1(CC1)N1CC2(CCN(C2=O)c2cncc3cc(ccc23)S(C)(=O)=O)c2cc(Cl)ccc2C1=O
CNC(=O)CN1CC2(CCN(C2=O)c2cncc3ccc(Cl)cc23)c2cc(Cl)ccc2C1=O
CNC(=O)CN1CC2(CCN(C2=O)c2cncc3cccc(Cl)c23)c2cc(Cl)ccc2C1=O
CN(C)CCOc1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
CNC(=O)CN1CC2(CCN(C2=O)c2cncc3cc(F)ccc23)c2cc(Cl)ccc2C1=O
CC(C)(CS(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1)C#N
CNC(=O)CN1CC2(CCN(C2=O)c2cncc3cc(Cl)ccc23)c2cc(Cl)ccc2C1=O
COC1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccc(OCCN(C)C)cc34)C2)CC1
CCN(C)S(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CNC(=O)C1(CC1)N1CC2(CCN(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4cccc(Cl)c34)c2c1)S(=O)(=O)CC1(CC1)C#N
Cc1cc(C(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccccc34)C2)n(C)n1
Cc1cnn(C)c1C(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)N1CCC1
CCn1nccc1C(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CS(=O)(=O)c1ccc2c(cncc2c1)N1CCC2(CN(Cc3ccc(Cl)cc23)S(=O)(=O)CC2(CC2)C#N)C1=O
CC1(CC1)NC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
Clc1ccc2CN(CC(=O)NCC#N)CC3(CCN(C3=O)c3cncc4ccccc34)c2c1
CN1CC(CS(=O)(=O)N2CC(C(=O)Nc3cncc4ccccc34)c3cc(Cl)ccc3C2)(C1)C#N
COCCN(C)S(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CC1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccccc34)C2)CS(=O)(=O)C1
CC1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4cc(ccc34)S(C)(=O)=O)C2)CC1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCS(=O)(=O)CC1)C#N
COC1CN(C1)S(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CNC(=O)CN1CC2(CCN(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2S1(=O)=O
CN(CCC#N)S(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)N1CC(C1)C#N
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC#N)CC1
Clc1ccc2CN(CC(=O)NCC3CC3)CC3(CCN(C3=O)c3cncc4ccccc34)c2c1
CNC(=O)C1(CC1)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
Clc1ccc2CN(CC(C(=O)Nc3nncn3C3CC3)c2c1)S(=O)(=O)CC1(CC1)C#N
Fc1cc(Cl)c2c(cncc2c1)N1CCC2(CN(Cc3ccc(Cl)cc23)S(=O)(=O)CC2(CC2)C#N)C1=O
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)C(=O)c1ccnn1C1CC1
CC(C)n1nccc1C(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CNC(=O)CN1Cc2ccc(Cl)cc2[C@]2(CCN(C2=O)c2cncc3CCCCc23)C1
CNC(=O)CN1Cc2ccc(cc2[C@]3(C1)CCN(C3=O)c4cncc5c4CCCC5)Cl
CNC(=O)CN1C[C@]2(CCN(C2=O)c3cncc4c3cccc4)c5cc(ccc5C1=O)Cl
CNC(=O)CN1C[C@@]2(CCN(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CCCC1)C#N
CN(CC#N)S(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccc(OCCN(C)C)cc23)C1
FC(F)(F)C1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccccc34)C2)CC1
FC(F)C1(CS(=O)(=O)N2Cc3ccc(Cl)cc3C3(CCN(C3=O)c3cncc4ccccc34)C2)CC1
CNC(=O)C1(CC1)N1C[C@@]2(CCN(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2C1=O
CNC(=O)C1(CC1)N2C[C@]3(CCN(C3=O)c4cncc5c4cccc5)c6cc(ccc6C2=O)Cl
CN(CCO)S(=O)(=O)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccccc23)C1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3cccc(Cl)c23)C1
CNC(=O)CN1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccc(OC)cc23)C1
Clc1ccc2c(c1)C1(CCN(C1=O)c1cncc3ccccc13)CN(CC(=O)NCC1CC1)S2(=O)=O
CC1CN(C(=O)C11CN(Cc2ccc(Cl)cc12)S(=O)(=O)CC1(CC1)C#N)c1cncc2ccccc12
CCNC(=O)CN1CC2(CCN(C2=O)c2cncc3ccccc23)c2cc(Cl)ccc2S1(=O)=O
CCC1CN(C(=O)C11CN(Cc2ccc(Cl)cc12)S(=O)(=O)CC1(CC1)C#N)c1cncc2ccccc12
COc1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
FC(F)c1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
CNC(=O)C1(CC1)N1Cc2ccc(Cl)cc2C2(CCN(C2=O)c2cncc3ccc(OCCN(C)C)cc23)C1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccc(OCCN5CCOCC5)cc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccc(OCCCN5CCCC5)cc34)c2c1)S(=O)(=O)CC1(CC1)C#N
CN(C)CCCOc1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
CN(C)CCOc1ccc2cncc(N3CC[C@@]4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
CN(C)CCOc1ccc2cncc(c2c1)N3CC[C@@]4(C3=O)CN(Cc5c4cc(cc5)Cl)S(=O)(=O)CC6(CC6)C#N
Clc1ccc2CN(CC3(CCCN(C3=O)c3cncc4ccccc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccc(OCCN5CCCC5)cc34)c2c1)S(=O)(=O)CC1(CC1)C#N
CCN(C)CCOc1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
CCN(CC)CCOc1ccc2cncc(N3CCC4(CN(Cc5ccc(Cl)cc45)S(=O)(=O)CC4(CC4)C#N)C3=O)c2c1
Clc1ccc2CN(CC3(CCN(C3=O)c3cncc4ccc(Cl)cc34)c2c1)S(=O)(=O)CC1(CC1)C#N
Clc1ccc2CN(Cc3nncs3)CC3(CCN(C3=O)c3cncc4ccccc34)c2c1
CC(=O)Nc1nc2c(s1)cccc2S(=O)(=O)NCCc3ccccc3
CC(=O)NCCc1c[nH]c2c1cccc2CN3CCN(CC3)C(=O)C
CC(=O)N1CC2CC1CN2Cc1cccc(Cl)c1 |THB:1:3:6:8.9,10:9:3.4:6|
c1cc(c2cc[nH]c2c1)C=O
CSC1=C(C#N)C2(CCCCC2)C(C#N)=C(NC(C)=O)N1 |c:2,t:15|
Cc1cc(c(n1NC(=O)C2=NNC(=O)c3c2cccc3)C)C(=O)C
OCC(=O)[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cc(F)cc(F)c2[nH]1 |r|
OCC(=O)[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cccc(Cl)c2[nH]1 |r|
OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cc(F)cc(F)c2[nH]1 |r|
OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cccc(Cl)c2[nH]1 |r|
OCC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cccc(F)c2[nH]1 |r|
OCC(=O)[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cccc(F)c2[nH]1 |r|
CC(C)[C@H](N)C(=O)OCC(=O)[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2cc(F)cc(F)c2[nH]1 |r|
COc1cc2c3CC4CCCN4Cc3c3cc(OC)c(OC)cc3c2cc1OC
CCN1CC(O)c2c(C1)c1cc(OC)c(OC)cc1c1cc(OC)ccc21
CCN1Cc2c(C(O)C1C)c1ccc(OC)cc1c1cc(OC)c(OC)cc21
COc1cc2c3CC4CCCCN4Cc3c3cc(OC)c(OC)cc3c2cc1OC
CCN1CCc2c(C1)c1cc(OC)c(OC)cc1c1cc(OC)ccc21
COc1cc2c3CC4CCC[N+]4([O-])Cc3c3cc(OC)c(OC)cc3c2cc1OC
Oc1nn2ccccc2c1C(=O)Nc1c(F)c(F)c(-c2ccccc2)c(F)c1F
Cc1c(nc2ccc(F)cc2c1C(O)=O)-c1ccc(cc1)-c1ccccc1F
CCCO[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CCCO[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CCCO[C@@H]1C[C@H](N(C1)C(=O)C(NC(=O)NC(C)(C)C)C(C)C)C(=O)N[C@@H](CC1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CCCN(CCC)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CCCC(=O)N[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CC1([C@@H]2[C@H]1[C@H](N(C2)C(=O)[C@H](C(C)(C)C)NC(=O)NC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)c4nc5ccccc5s4)C
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(=O)NCc3ccccc3)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc(cs1)-c1ccccc1)C2(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(N)=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
CCCO[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc(cs1)-c1ccccc1 |r|
CCCN(CCC)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CCCC(=O)N[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1 |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)N1CCCC1)C(C)(C)C |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)N1CCOCC1)C(C)(C)C |r|
CCCN(CCC)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)c1nc(cs1)-c1ccccc1 |r|
CC(C)(C)[C@H](NC(=O)NCc1ccncc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc(cs1)-c1ccccc1)C2(C)C |r|
CN(C)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc(cs1)-c1ccccc1 |r|
CCN(CC)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc(cs1)-c1ccccc1 |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc(co1)-c1ccccc1)C2(C)C)C(C)(C)C |r|
CC(=O)OC(C#N)[C@H](CC1CCCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)C(NC(=O)NC(C)(C)C)C(C)(C)C)C2(C)C |r,w:4.3|
CCCN(CCC)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(F)=O)C(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C#N |r|
CCCN(CCC)[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C#N |r|
CCCO[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)NC(C[C@@H]1CCNC1=O)C#N |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)NC(C[C@@H]1CCNC1=O)C#N)C2(C)C)C(C)(C)C |r|
CC(C)(C)[C@H](NC(=O)c1ccccc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C |r|
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc2NC(=O)CCc2c1
CN1C(=O)CCc2cc(ccc12)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc2NC(=O)OCc2c1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc2NC(=O)CCCc2c1
CC(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CCC(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CCCC(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1)C1CC1
O=C(Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1)C1CCC1
FC(F)(F)C(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CCOC(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
NC(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1)N1CCOCC1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCNC1=O
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCNC1=O
CN1CCN(C1=O)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CC(C)N1CCN(C1=O)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCOC1=O
CN(C(C)=O)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCC1=O
CC1(C)CN(C1=O)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCCC1=O
FC1(F)CCC(=O)N(C1)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
OC1CCC(=O)N(C1)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCCCC1=O
Fc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
COc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
Oc1ccc(cc1)C(=O)Nc1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CC(=O)Nc1ccc(cc1F)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CC(=O)Nc1ccc(cc1O)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CC(=O)Nc1ccc(nn1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCN(CC1=O)C1CCC1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCN(CC2CCC2)CC1=O
Cc1nc2ccc(cc2o1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CC2(CCC2)C1=O
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCC2(CCC2)C1=O
O=C(NC1CC1)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(NC1CCC1)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(NC1CCCC1)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)-c1ccn[nH]1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)-c1nnco1
CN(C)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
COC(=O)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
CC(C)(C)OC(=O)c1ccc(cc1)C(=O)Nc1cccc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)C1(CC1)C#N
COc1cc(NC(=O)c2ccc3NC(=O)CCc3c2)cc(c1)C#Cc1ccccn1
Cc1cc(NC(=O)c2ccc3NC(=O)CCc3c2)nc(c1)C#Cc1ccccn1
COc1cc(NC(=O)c2ccc(cc2)N2CCCCC2=O)cc(c1)C#Cc1ccccn1
CC(=O)Nc1ccc(cc1)-c1nc2ccc(cc2[nH]1)C#Cc1ccccn1
FC(F)(F)Oc1cc(NC(=O)c2ccc(cc2)N2CCCCC2=O)cc(c1)C#Cc1ccccn1
COc1cc(NC(=O)c2ccc3NC(=O)CCCc3c2)cc(c1)C#Cc1ccccn1
Nc1cc(NC(=O)c2ccc(cc2)N2CCCCC2=O)cc(c1)C#Cc1ccccn1
O=C(Nc1cc(OCC2CC2)cc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCCC1=O
O=C(Nc1ccc2NC(=O)CCc2c1)c1cccc(c1)C#Cc1ccccn1
CC(=O)Nc1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
CCN(C(C)=O)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
O=C(Nc1ccc(cc1)N1CCC1=O)c1cccc(c1)C#Cc1ccccn1
CC1(C)CN(C1=O)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
O=C(Nc1ccc(cc1)N1CCCCC1=O)c1cccc(c1)C#Cc1ccccn1
O=C(Nc1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1)N1CCC1
CC1(CC1)NC(=O)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
O=C(NC1CCCC1)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
COC(=O)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
COC(=O)c1cccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)c1
CC(C)OC(=O)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
O=C(Nc1ccc(cc1)C(=O)OCC1CC1)c1cccc(c1)C#Cc1ccccn1
CC(C)(C)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
OC(c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1)(C(F)(F)F)C(F)(F)F
CC(C)n1nccc1-c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
O=C(Nc1ccc(cc1)N1CCCCS1(=O)=O)c1cccc(c1)C#Cc1ccccn1
CC(=O)Nc1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cn1
COc1cc(cc(c1)C(=O)Nc1ccc(cc1)N1CCCCC1=O)C#Cc1ccccn1
CCOP(=O)(OCC)c1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
O=C(Nc1ccc(cc1)N1CCCS1(=O)=O)c1cccc(c1)C#Cc1ccccn1
COc1cc(cc(c1)C(=O)Nc1ccc(cc1)N1CCCCS1(=O)=O)C#Cc1ccccn1
COc1cc(NC(=O)c2ccc(cc2)N2CCCCS2(=O)=O)cc(c1)C#Cc1ccccn1
O=C(Nc1cccc(c1)C#Cc1ccccn1)c1ccc(cc1)N1CCCCS1(=O)=O
O=C(Nc1cc(cc(c1)C#Cc1ccccn1)C#N)c1ccc(cc1)N1CCCCC1=O
COc1cc(cc(c1)C(=O)Nc1ccc(CC2CC(=O)NC2=O)cc1)C#Cc1ccccn1
NS(=O)(=O)Cc1ccc(NC(=O)c2cccc(c2)C#Cc2ccccn2)cc1
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1ccc(F)cc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(CC(C)C)C(=O)Nc1cc(F)cc(F)c1)C(=O)N1C[C@]2(C[C@H]1C(N)=O)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)[C@@H](CC(C)C)C(=O)Nc1cc(F)cc(F)c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)OC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)c1cc2c(F)cc(F)cc2[nH]1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(C)(C)C(O)=O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(C)(C)C(=O)Nc1cc(F)ccc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)C(C)(C)C(=O)Nc1c(C)cccc1C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1c(C)cccc1C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)(C)C[C@H](NC(=O)C(C)(C)C(=O)Nc1cc(F)ccc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
Cc1cccc(C)c1NC(=O)C(C)(C)C(=O)N[C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CS(=O)(=O)Nc1c(C)cccc1C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)S(=O)(=O)CC(=O)Nc1c(C)cccc1C |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)NCC(C)(C)O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)NCc1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H](C)c1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1cccc2ccccc12)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H](C)c1ccccc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1ccccn1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1cccnc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1ccncc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1ccccc1F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1cccc(F)c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1ccc(F)cc1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)Nc1cn[nH]c1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CN([C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21)C(=O)C1(CCC1)C(=O)Nc1c(C)cccc1C |r|
Cc1cccc(C)c1NC(=O)C1(CC1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](NC(=O)C1(CCCC1)C(=O)Nc1c(C)cccc1C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)NC[C@H](C)O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)NC[C@@H](C)O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H](C)CO)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H](C)CO)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)NCC(F)F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H]1CCN(C1)C(=O)OC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H]1CCN(C1)C(=O)OC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](NC(=O)C1(CCOCC1)C(=O)Nc1c(C)cccc1C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](NC(=O)C1(CCC1)C(=O)NCC(C)(C)O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
Cc1cccc(C)c1NC(=O)C1(CCOCC1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H]1CCC[C@@H]1O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H]1CCC[C@@H]1O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H]1CCC[C@H]1O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H]1CCC[C@H]1O)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H]1CC[C@H](O)C1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H]1CC[C@H](O)C1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@@H]1CC[C@@H](O)C1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)N[C@H]1CC[C@@H](O)C1)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
CC(C)C[C@H](N(C)C(=O)CC(=O)NC(C)C(F)(F)F)C(=O)N1C[C@]2(C[C@H]1C#N)C(=O)Nc1ccccc21 |r|
Nc1nc(N)c2c3ccn(Cc4ccccc4C(F)(F)F)c3ccc2n1
Cc1ccccc1Cn1ccc2c1ccc1nc(N)nc(N)c21
Cc1cc2c(ccc3nc(N)nc(N)c23)n1Cc1ccc(cc1)C#N
Nc1nc(N)c2c3ccn(CC=C)c3ccc2n1
O=C(N1C[C@@H]2CNC[C@@H]2C1)c1sc(nc1-c1ccccc1)-c1ccccc1 |r|
Clc1ccc(cc1)-c1nc(sc1C(=O)N1C[C@@H]2CNC[C@@H]2C1)-c1ccccc1 |r|
Clc1ccc(cc1)-c1nc(c(s1)C(=O)N1C[C@@H]2CNC[C@@H]2C1)-c1ccccc1 |r|
c1ccc(c(c1)Cn2ccc3c2ccc4c3c(nc(n4)N)N)F
Nc1nc(N)c2c3ccn(Cc4cccnc4)c3ccc2n1
Nc1nc(N)c2c3ccn(Cc4ccncc4)c3ccc2n1
Nc1nc(N)c2c3ccn(Cc4ccccn4)c3ccc2n1
Nc1nc(N)c2c3ccn(CC4CCCCC4)c3ccc2n1
CC(C)CCCC(C)(C)[C@H]1CC[C@@]2(C)\C(CCC[C@]12C)=C\C=C1\C[C@@H](C)CC[C@H]1C |r|
CC(CCCC(C)(C)O)[C@H]1CC[C@H]2C3=CC=C4C[C@@H](O)CC[C@@]4(C)[C@@H]3CC[C@]12C |r,t:13,15|
C[C@H](CCCC(C)(C)C)[C@H]1CC[C@H]2\C(CCC[C@]12C)=C\C=C1\C[C@@H](C)C[C@H](C)[C@H]1C |r|
CC(C)CCC[C@](C)(O)[C@H]1CC[C@H]2C3=CC=C4C[C@@H](O)CC[C@@]4(C)[C@@H]3CC[C@]12C |r,t:13,15|
CC(C)[C@@H](O)CCC(C)[C@H]1CC[C@H]2C3=CC=C4C[C@@H](O)CCC4(C)[C@@H]3CC[C@]12C |r,t:13,15|
CC(C)CCCC(C)(C)[C@@]1(C)CC[C@H]2C3=CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C |r,t:14,16|
O=C[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
COc1ccccc1C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C=O
OC1Oc2ccccc2CC1NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
COc1ccc2OC(O)C(Cc2c1)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
Cc1ccc2OC(O)C(Cc2c1)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
COC(=O)c1ccc2OC(O)C(Cc2c1)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
CN1CCN(CC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)NC1Cc2ccccc2OC1O
CN1CCN(CC1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1ccc[nH]c1=O)C=O
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc[nH]c1=O)C=O)c1ccccc1
CC(C)[C@H](NC(C)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1ccc[nH]c1=O)C=O)c1ccccc1
CC(C)C[C@H](NC(=O)C(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](Cc1ccc[nH]c1=O)C=O
O=C[C@H](Cc1ccc[nH]c1=O)NC(=O)[C@@H](NC(=O)C(=O)c1cc2ccccc2[nH]1)C1CCCCC1
[O-][N+](=O)c1ccc(cc1)[C@H](NC(=O)C(=O)c1cc2ccccc2[nH]1)C(=O)N[C@@H](Cc1ccc[nH]c1=O)C=O
CC(C)[C@H](NC(C)=O)C(=O)N1CCC[C@H]1C(=O)C(=O)N[C@@H](Cc1ccc[nH]c1=O)C=O
CC(C)[C@H](NC(C)=O)C(=O)N1CCC[C@H]1C(=O)C(=O)N[C@@H](Cc1ccc[nH]c1=O)C#N
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1 |r|
Cc1cc(C(=O)N[C@@H]2CCN(C2)c2c(cc(Br)cc2C(F)(F)F)C(=O)N2CCOCC2)c(F)c(=O)[nH]1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1 |r|
Fc1cccc2c(C(=O)N[C@@H]3CCN(C3)c3c(cc(cc3C(F)(F)F)C#N)C(=O)N3CCOCC3)c(F)c(=O)[nH]c12 |r|
Fc1c(C(=O)N[C@@H]2CCN(C2)c2c(cc(cc2C(F)(F)F)C#N)C(=O)N2CCOCC2)c2ccccc2[nH]c1=O |r|
Fc1cc(F)c2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(cc3C(F)(F)F)C#N)C(=O)N3CCOCC3)c2c1 |r|
Fc1ccc2c(cc(=O)[nH]c2c1F)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(cc3C(F)(F)F)C#N)C(=O)N3CCOCC3)c12 |r|
Cc1cc(C(=O)N[C@@H]2CCN(C2)c2c(cc(cc2C(F)(F)F)C#N)C(=O)N2CCOCC2)c(F)c(=O)[nH]1 |r|
Cc1[nH]c(=O)c(F)c(C(=O)N[C@@H]2CCN(C2)c2c(cc(cc2C(F)(F)F)C#N)C(=O)N2CCOCC2)c1Cl |r|
Cc1cc(C(=O)N[C@@H]2CCN(C2)c2c(cc(cc2C(=O)N2CCOCC2)C#N)C(F)F)c(F)c(=O)[nH]1 |r|
Cc4cc(C(=O)N[C@@H]3CCN(c2c(C(=O)N1CCOCC1)cc(C#N)cc2C(F)(F)F)C3)c(F)c(=O)[nH]4
CN1CCN(CC1)C(=O)c1cc(cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCCCC1 |r|
C[C@@]12COC[C@@H]1CN(C2)C(=O)c1cc(cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CC2CC(C1)O2 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1C[C@@H]2COC[C@@H]2C1 |r|
COCCN1CCN(CC1)C(=O)c1cc(cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCCC1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCC(F)(F)C1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CC(F)(F)C1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCN2CCOCC2C1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCN(CC2CCCO2)CC1 |r|
CCS(=O)(=O)N1CCN(CC1)C(=O)c1cc(cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCC(CC1)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCNC(=O)C1 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(cc3C(F)(F)F)C#N)C(=O)NC(C)C)c12 |r|
CC(C)CNC(=O)c1cc(cc(c1N1CC[C@H](C1)NC(=O)c1cc(C)[nH]c(=O)c1)C(F)(F)F)C#N |r|
C[C@@H]1C[C@H](CN1c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12 |r|
C[C@@H]1C[C@H](CN1c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1)NC(=O)c1cc(=O)[nH]c2c(F)c(F)ccc12 |r|
CO[C@H]1CN(C[C@@H]1NC(=O)c1cc(=O)[nH]c2c(F)cccc12)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1 |r|
Fc1cc(F)c2[nH]c(=O)cc(C(=O)N[C@H]3CN(C(=O)C3)c3c(cc(cc3C(F)(F)F)C#N)C(=O)N3CCOCC3)c2c1 |r|
Fc1ccc2c(cc(=O)[nH]c2c1F)C(=O)N[C@H]1CN(C(=O)C1)c1c(cc(cc1C(F)(F)F)C#N)C(=O)N1CCOCC1 |r|
NC(=O)c1cc(C(=O)N2CCOCC2)c(N2CC[C@H](C2)NC(=O)c2cc(=O)[nH]c3c(F)cccc23)c(c1)C(F)(F)F |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Cl)cc1C(F)(F)F)C(=O)N1CCOCC1 |r|
CN1CCN(CC1)C(=O)c1cc(Cl)cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F |r|
Fc1cc(C(=O)N2CCOCC2)c(N2CC[C@H](C2)NC(=O)c2cc(=O)[nH]c3c(F)cc(F)cc23)c(c1)C(F)(F)F |r|
FC(F)c1cc(cc(C(=O)N2CCOCC2)c1N1CC[C@H](C1)NC(=O)c1c(F)c(=O)[nH]c2c(F)cccc12)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(cc1C(=O)N1CCOCC1)C#N)C1CC1 |r|
CN1CCN(CC1)C(=O)c1cc(cc(C2CC2)c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C#N |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(OC(F)(F)F)cc(Br)cc1C(=O)N1CCOCC1 |r|
FC(F)Oc1cc(Cl)cc(C(=O)N2CCOCC2)c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(OC(F)(F)F)cc(Cl)cc1C(=O)N1CCOCC1 |r|
Cc1cc(C2CC2)c(N2CC[C@H](C2)NC(=O)c2cc(=O)[nH]c3c(F)cccc23)c(c1)C(=O)N1CCOCC1 |r|
Fc1cc(C2CC2)c(N2CC[C@H](C2)NC(=O)c2cc(=O)[nH]c3c(F)cccc23)c(c1)C(=O)N1CCOCC1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1cccc2c(C(=O)N[C@@H]3CCN(C3)c3c(cc(Br)cc3C(F)(F)F)C(=O)N3CCOCC3)c(F)c(=O)[nH]c12 |r|
Fc1cc(F)c2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(Br)cc3C(F)(F)F)C(=O)N3CCOCC3)c2c1 |r|
Fc1ccc2c(C(=O)N[C@@H]3CCN(C3)c3c(cc(Br)cc3C(F)(F)F)C(=O)N3CCOCC3)c(F)c(=O)[nH]c2c1F |r|
Fc1ccc2c(cc(=O)[nH]c2c1F)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1ccc(F)c2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCOCC1 |r|
Fc1c(C(=O)N[C@@H]2CCN(C2)c2c(cc(Br)cc2C(F)(F)F)C(=O)N2CCOCC2)c2ccccc2[nH]c1=O |r|
FC(F)c1cc(Br)cc(C(=O)N2CCOCC2)c1N1CC[C@H](C1)NC(=O)c1c(F)c(=O)[nH]c2c(F)cccc12 |r|
Fc1cccc2c(C(=O)N[C@@H]3CCN(C3)c3c(cc(Cl)cc3C(F)(F)F)C(=O)N3CCOCC3)c(F)c(=O)[nH]c12 |r|
FC(F)(F)c1cc(Br)cc(C(=O)N2CCOCC2)c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2ccccc12 |r|
COc1cc(F)cc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(Br)cc3C(F)(F)F)C(=O)N3CCOCC3)c12 |r|
FC(F)(F)c1cc(Br)cc(C(=O)N2CCOCC2)c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(Cl)cccc12 |r|
Cc1[nH]c(=O)cc(C(=O)N[C@@H]2CCN(C2)c2c(cc(Br)cc2C(F)(F)F)C(=O)N2CCOCC2)c1F |r|
Cc1cc(C2CC2)c(N2CC[C@H](C2)NC(=O)c2cc(C)[nH]c(=O)c2F)c(c1)C(=O)N1CCOCC1 |r|
FC(F)c1cc(cc(=O)[nH]1)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCOCC1 |r|
Cc1cc(C(=O)N[C@@H]2CCN(C2)c2c(cc(Br)cc2C(=O)N2CCOCC2)C(F)F)c(F)c(=O)[nH]1 |r|
CN1CCN(CC1)C(=O)c1cc(Br)cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCCCC1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CC2CC(C1)O2 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CC2COCC2C1 |r|
COCCN1CCN(CC1)C(=O)c1cc(Br)cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCCC1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCC(F)(F)C1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CC(F)(F)C1 |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CCN2CCOCC2C1 |r|
COCCN(C)C(=O)c1cc(Br)cc(c1N1CC[C@H](C1)NC(=O)c1cc(=O)[nH]c2c(F)cccc12)C(F)(F)F |r|
Fc1cccc2c(cc(=O)[nH]c12)C(=O)N[C@@H]1CCN(C1)c1c(cc(Br)cc1C(F)(F)F)C(=O)N1CC2(COC2)C1 |r|
Cc1cc(C2CC2)c(N2C[C@@H](CC2=O)NC(=O)c2cc(=O)[nH]c3c(F)cc(F)cc23)c(c1)C(=O)N1CCOCC1 |r|
Cc1cc(C2CC2)c(N2C[C@@H](CC2=O)NC(=O)c2cc(=O)[nH]c3c(F)c(F)ccc23)c(c1)C(=O)N1CCOCC1 |r|
Cc1cc(C2CC2)c(N2C[C@@H](CC2=O)NC(=O)c2cc(=O)[nH]c3c(F)cccc23)c(c1)C(=O)N1CCOCC1 |r|
Fc1ccc2c(C(=O)N[C@H]3CN(C(=O)C3)c3c(cc(Br)cc3C(F)(F)F)C(=O)N3CCOCC3)c(F)c(=O)[nH]c2c1F |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(ccc(F)c3C(=O)N3CCOCC3)C3CC3)c12 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(F)cc3C(=O)N3CCOCC3)C3CC3)c12 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(ccc(C)c3C(=O)N3CCOCC3)C3CC3)c12 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(cc(C)cc3C(=O)N3CCOCC3)C3CC3)c12 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(nc(Cl)cc3C(=O)N3CCOCC3)C3CC3)c12 |r|
C[C@@H]1C[C@H](CN1c1c(cc(C)cc1C(=O)N1CCOCC1)C1CC1)NC(=O)c1cc(=O)[nH]c2c(F)c(F)ccc12 |r|
CO[C@H]1CN(C[C@@H]1NC(=O)c1cc(=O)[nH]c2cccc(OC)c12)c1c(cc(C)cc1C(=O)N1CCOCC1)C1CC1 |r|
COc1cccc2[nH]c(=O)cc(C(=O)N[C@@H]3CCN(C3)c3c(Cl)cc(C)cc3C(=O)N3CCOCC3)c12 |r|
O=C1NC2(CC(C2)C2CCC2)C(=O)N1c1cncc2ccccc12 |(.99,4.33,;.99,2.79,;2.24,1.89,;1.76,.42,;1.52,-1.1,;3.04,-1.34,;3.28,.18,;3.95,-2.58,;3.71,-4.11,;5.23,-4.35,;5.47,-2.83,;.22,.42,;-.68,-.82,;-.25,1.89,;-1.72,2.36,;-2.04,3.87,;-3.5,4.35,;-4.65,3.32,;-4.33,1.81,;-5.47,.78,;-5.15,-.73,;-3.69,-1.2,;-2.54,-.17,;-2.86,1.33,)|
O=C1NC2(CC(C2)c2ccccc2)C(=O)N1c1cncc2ccccc12 |(.54,4.78,;.54,3.24,;1.78,2.33,;1.31,.87,;1.07,-.65,;2.59,-.89,;2.83,.63,;3.49,-2.14,;2.86,-3.55,;3.77,-4.79,;5.3,-4.63,;5.93,-3.22,;5.02,-1.98,;-.23,.87,;-1.14,-.38,;-.71,2.33,;-2.17,2.81,;-2.49,4.32,;-3.96,4.79,;-5.1,3.76,;-4.78,2.25,;-5.93,1.22,;-5.61,-.28,;-4.14,-.76,;-3,.27,;-3.32,1.78,)|
Cc1c(Br)cncc1N1C(=O)NC2(CC(C2)C(C)(C)C)C1=O |(-1.31,3.97,;-2.45,2.94,;-3.92,3.42,;-4.24,4.92,;-5.06,2.39,;-4.74,.88,;-3.28,.4,;-2.13,1.43,;-.67,.96,;.58,1.86,;.58,3.4,;1.82,.96,;1.35,-.51,;1.11,-2.03,;2.63,-2.27,;2.87,-.75,;3.53,-3.52,;2.91,-4.92,;5.06,-3.35,;4.44,-4.76,;-.19,-.51,;-1.1,-1.75,)|
Cc1c(Br)cncc1N1C(=O)NC2(CC(C2)C2CCC2)C1=O |(-1.3,4.15,;-2.45,3.12,;-3.91,3.59,;-4.23,5.1,;-5.06,2.56,;-4.74,1.06,;-3.27,.58,;-2.13,1.61,;-.66,1.13,;.58,2.04,;.58,3.58,;1.83,1.13,;1.35,-.33,;1.11,-1.85,;2.63,-2.09,;2.87,-.57,;3.54,-3.34,;3.3,-4.86,;4.82,-5.1,;5.06,-3.58,;-.19,-.33,;-1.09,-1.58,)|
Cc1c(Br)cncc1N1C(=O)NC2(CC(C2)c2ccccc2)C1=O |(-1.76,4.59,;-2.91,3.56,;-4.37,4.04,;-4.69,5.54,;-5.52,3.01,;-5.2,1.5,;-3.73,1.03,;-2.59,2.06,;-1.12,1.58,;.12,2.49,;.12,4.03,;1.37,1.58,;.89,.12,;.65,-1.41,;2.17,-1.65,;2.41,-.13,;3.08,-2.89,;2.45,-4.3,;3.36,-5.54,;4.89,-5.38,;5.52,-3.98,;4.61,-2.73,;-.65,.12,;-1.55,-1.13,)|
Cc1ccncc1N1C(=O)NC2(CC(C2)C(C)(C)C)C1=O |(-2.96,-.35,;-3.28,1.16,;-4.74,1.63,;-5.06,3.14,;-3.92,4.17,;-2.45,3.69,;-2.13,2.19,;-.67,1.71,;.58,2.62,;.58,4.16,;1.82,1.71,;1.35,.25,;1.11,-1.28,;2.63,-1.52,;2.87,.01,;3.53,-2.76,;2.91,-4.17,;5.06,-2.6,;4.44,-4.01,;-.19,.25,;-1.1,-1,)|
Cc1cccnc1CN1C(=O)NC2(CC(C2)C(C)(C)C)C1=O |(-5.7,.24,;-4.93,1.58,;-5.7,2.91,;-4.93,4.24,;-3.39,4.24,;-2.62,2.91,;-3.39,1.58,;-2.62,.24,;-1.08,.24,;-.18,1.49,;-.65,2.95,;1.29,1.01,;1.29,-.53,;1.53,-2.05,;3.05,-1.81,;2.81,-.29,;4.3,-2.71,;5.7,-2.09,;4.13,-4.24,;5.54,-3.62,;-.18,-1,;-.65,-2.47,)|
Cc1ccncc1N1C(=O)NC2(CC(C2)C2CCC2)C1=O |(-2.95,-.17,;-3.27,1.33,;-4.74,1.81,;-5.06,3.32,;-3.91,4.35,;-2.45,3.87,;-2.13,2.36,;-.66,1.89,;.58,2.79,;.58,4.33,;1.83,1.89,;1.35,.42,;1.11,-1.1,;2.63,-1.34,;2.87,.18,;3.54,-2.58,;3.3,-4.11,;4.82,-4.35,;5.06,-2.83,;-.19,.42,;-1.09,-.82,)|
Cc1ccncc1N1C(=O)NC2(CC(C2)c2ccccc2)C1=O |(-3.41,.27,;-3.73,1.78,;-5.2,2.25,;-5.52,3.76,;-4.37,4.79,;-2.91,4.32,;-2.59,2.81,;-1.12,2.33,;.12,3.24,;.12,4.78,;1.37,2.33,;.89,.87,;.65,-.65,;2.17,-.89,;2.41,.63,;3.08,-2.14,;2.45,-3.55,;3.36,-4.79,;4.89,-4.63,;5.52,-3.22,;4.61,-1.98,;-.65,.87,;-1.55,-.38,)|
CC(C)(C)C1CC2(C1)NC(=O)N(C2=O)c1cncc(F)c1 |(3.32,-4.17,;3.94,-2.76,;5.48,-2.6,;4.85,-4.01,;3.04,-1.52,;1.52,-1.28,;1.76,.25,;3.28,.01,;2.23,1.71,;.99,2.62,;.99,4.16,;-.26,1.71,;.22,.25,;-.69,-1,;-1.72,2.19,;-2.04,3.69,;-3.51,4.17,;-4.65,3.14,;-4.33,1.63,;-5.48,.6,;-2.87,1.16,)|
Fc1cncc(c1)N1C(=O)NC2(CC(C2)C2CCC2)C1=O |(-5.47,.78,;-4.33,1.81,;-4.65,3.32,;-3.5,4.35,;-2.04,3.87,;-1.72,2.36,;-2.86,1.33,;-.25,1.89,;.99,2.79,;.99,4.33,;2.24,1.89,;1.76,.42,;1.52,-1.1,;3.04,-1.34,;3.28,.18,;3.95,-2.58,;3.71,-4.11,;5.23,-4.35,;5.47,-2.83,;.22,.42,;-.68,-.82,)|
Brc1cncc(c1)N1C(=O)NC2(CC(C2)C2CCC2)C1=O |(-5.47,.78,;-4.33,1.81,;-4.65,3.32,;-3.5,4.35,;-2.04,3.87,;-1.72,2.36,;-2.86,1.33,;-.25,1.89,;.99,2.79,;.99,4.33,;2.24,1.89,;1.76,.42,;1.52,-1.1,;3.04,-1.34,;3.28,.18,;3.95,-2.58,;3.71,-4.11,;5.23,-4.35,;5.47,-2.83,;.22,.42,;-.68,-.82,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(5.65,-.57,;5.02,-1.98,;5.93,-3.22,;5.3,-4.63,;3.77,-4.79,;2.86,-3.55,;3.49,-2.14,;2.59,-.89,;1.07,-.65,;1.31,.87,;2.83,.63,;1.78,2.33,;.54,3.24,;.54,4.78,;-.71,2.33,;-.23,.87,;-1.14,-.38,;-2.17,2.81,;-2.49,4.32,;-3.96,4.79,;-5.1,3.76,;-4.78,2.25,;-5.93,1.22,;-5.61,-.28,;-4.14,-.76,;-3,.27,;-3.32,1.78,)|
Brc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Fc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
COc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(3.54,-.81,;4.44,-2.05,;3.81,-3.46,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Clc1cccc(Cl)c1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(.1,-5.24,;1.63,-5.08,;2.54,-6.33,;4.07,-6.16,;4.7,-4.76,;3.79,-3.51,;4.42,-2.1,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Fc1cccc(C2CC3(C2)NC(=O)N(C3=O)c2cncc3ccccc23)c1Cl |(5.46,-4.6,;3.93,-4.76,;3.3,-6.16,;1.77,-6.33,;.87,-5.08,;1.49,-3.67,;.59,-2.43,;-.93,-2.19,;-.69,-.66,;.83,-.91,;-2.23,-.66,;-2.71,.8,;-4.17,1.28,;-1.46,1.71,;-.22,.8,;1.25,1.28,;-1.46,3.25,;-.13,4.02,;-.13,5.56,;-1.46,6.33,;-2.79,5.56,;-4.13,6.33,;-5.46,5.56,;-5.46,4.02,;-4.13,3.25,;-2.79,4.02,;3.03,-3.51,;3.65,-2.1,)|
Fc1ccc(C2CC3(C2)NC(=O)N(C3=O)c2cncc3ccccc23)c(Cl)c1
Fc1ccc(C2CC3(C2)NC(=O)N(C3=O)c2cncc3ccccc23)c(Cl)c1
Fc1ccc(Cl)c(c1)C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(1.91,-7.03,;2.54,-5.62,;4.07,-5.46,;4.7,-4.05,;3.79,-2.81,;4.42,-1.4,;2.26,-2.97,;1.63,-4.38,;1.35,-1.72,;-.17,-1.48,;.07,.04,;1.6,-.2,;-1.47,.04,;-1.94,1.5,;-3.41,1.98,;-.7,2.41,;.55,1.5,;2.02,1.98,;-.7,3.95,;.64,4.72,;.64,6.26,;-.7,7.03,;-2.03,6.26,;-3.36,7.03,;-4.7,6.26,;-4.7,4.72,;-3.36,3.95,;-2.03,4.72,)|
Fc1cccc(Cl)c1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(.1,-5.24,;1.63,-5.08,;2.54,-6.33,;4.07,-6.16,;4.7,-4.76,;3.79,-3.51,;4.42,-2.1,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
CC1(CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12)c1ccccc1 |(.27,-3.52,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,;2.26,-3.67,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,)|
Clc1sccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(4.63,-2.48,;3.86,-3.81,;4.34,-5.28,;3.09,-6.18,;1.85,-5.28,;2.32,-3.81,;1.42,-2.57,;-.1,-2.33,;.14,-.81,;1.66,-1.05,;-1.4,-.81,;-1.88,.66,;-3.34,1.13,;-.63,1.56,;.61,.66,;2.08,1.13,;-.63,3.1,;.7,3.87,;.7,5.41,;-.63,6.18,;-1.97,5.41,;-3.3,6.18,;-4.63,5.41,;-4.63,3.87,;-3.3,3.1,;-1.97,3.87,)|
Clc1ccsc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(.51,-5.68,;1.99,-5.28,;3.24,-6.18,;4.49,-5.28,;4.01,-3.81,;2.47,-3.81,;1.57,-2.57,;.04,-2.33,;.28,-.81,;1.81,-1.05,;-1.26,-.81,;-1.73,.66,;-3.2,1.13,;-.49,1.56,;.76,.66,;2.23,1.13,;-.49,3.1,;.85,3.87,;.85,5.41,;-.49,6.18,;-1.82,5.41,;-3.15,6.18,;-4.49,5.41,;-4.49,3.87,;-3.15,3.1,;-1.82,3.87,)|
Brc1ccsc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(.51,-5.68,;1.99,-5.28,;3.24,-6.18,;4.49,-5.28,;4.01,-3.81,;2.47,-3.81,;1.57,-2.57,;.04,-2.33,;.28,-.81,;1.81,-1.05,;-1.26,-.81,;-1.73,.66,;-3.2,1.13,;-.49,1.56,;.76,.66,;2.23,1.13,;-.49,3.1,;.85,3.87,;.85,5.41,;-.49,6.18,;-1.82,5.41,;-3.15,6.18,;-4.49,5.41,;-4.49,3.87,;-3.15,3.1,;-1.82,3.87,)|
O=C1NC2(CC(C2)c2cn(Cc3ccccc3)nn2)C(=O)N1c1cncc2ccccc12 |(-3.2,3.44,;-1.73,2.97,;-1.26,1.5,;.28,1.5,;.04,-.02,;1.57,-.26,;1.81,1.26,;2.47,-1.5,;1.99,-2.97,;3.24,-3.91,;3.24,-5.45,;1.91,-6.22,;1.91,-7.76,;.57,-8.53,;-.76,-7.76,;-.76,-6.22,;.57,-5.45,;4.49,-2.97,;4.01,-1.5,;.76,2.97,;2.23,3.44,;-.49,3.87,;-.49,5.41,;.85,6.18,;.85,7.72,;-.49,8.49,;-1.82,7.72,;-3.15,8.49,;-4.49,7.72,;-4.49,6.18,;-3.15,5.41,;-1.82,6.18,)|
O=C1NC2(CC(C2)OCc2ccccc2)C(=O)N1c1cncc2ccccc12 |(-4.62,1.82,;-3.16,1.34,;-2.68,-.12,;-1.14,-.12,;-1.38,-1.64,;.14,-1.88,;.38,-.36,;1.04,-3.13,;2.57,-2.97,;3.48,-4.21,;5.01,-4.05,;5.92,-5.3,;5.29,-6.71,;3.76,-6.87,;2.85,-5.62,;-.67,1.34,;.8,1.82,;-1.91,2.25,;-1.91,3.79,;-.58,4.56,;-.58,6.1,;-1.91,6.87,;-3.25,6.1,;-4.58,6.87,;-5.91,6.1,;-5.91,4.56,;-4.58,3.79,;-3.25,4.56,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Fc1ccc2cncc(N3C(=O)NC4(CC(C4)c4ccccc4Cl)C3=O)c2c1 |(-5.36,3.25,;-4.03,4.02,;-4.03,5.56,;-2.7,6.33,;-1.36,5.56,;-.03,6.33,;1.3,5.56,;1.3,4.02,;-.03,3.25,;-.03,1.71,;-1.27,.8,;-2.74,1.28,;-.8,-.66,;.74,-.66,;.5,-2.19,;2.02,-2.43,;2.26,-.91,;2.93,-3.67,;2.3,-5.08,;3.21,-6.33,;4.74,-6.16,;5.36,-4.76,;4.46,-3.51,;5.08,-2.1,;1.22,.8,;2.68,1.28,;-1.36,4.02,;-2.7,3.25,)|
Fc1ccc2c(cncc2c1)N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(-5.36,6.33,;-4.03,5.56,;-4.03,4.02,;-2.7,3.25,;-1.36,4.02,;-.03,3.25,;1.3,4.02,;1.3,5.56,;-.03,6.33,;-1.36,5.56,;-2.7,6.33,;-.03,1.71,;-1.27,.8,;-2.74,1.28,;-.8,-.66,;.74,-.66,;.5,-2.19,;2.02,-2.43,;2.26,-.91,;2.93,-3.67,;2.3,-5.08,;3.21,-6.33,;4.74,-6.16,;5.36,-4.76,;4.46,-3.51,;5.08,-2.1,;1.22,.8,;2.68,1.28,)|
COc1ccc2cncc(N3C(=O)NC4(CC(C4)C4CCC4)C3=O)c2c1 |(-5.57,3.57,;-4.24,2.8,;-2.91,3.57,;-2.91,5.11,;-1.57,5.88,;-.24,5.11,;1.1,5.88,;2.43,5.11,;2.43,3.57,;1.1,2.8,;1.1,1.26,;-.15,.35,;-1.61,.83,;.33,-1.11,;1.87,-1.11,;1.63,-2.63,;3.15,-2.87,;3.39,-1.35,;4.05,-4.12,;3.81,-5.64,;5.33,-5.88,;5.57,-4.36,;2.34,.35,;3.81,.83,;-.24,3.57,;-1.57,2.8,)|
Cc1ccc2cncc(N3C(=O)NC4(CC(C4)C4CCC4)C3=O)c2c1 |(-4.91,2.8,;-3.57,3.57,;-3.57,5.11,;-2.24,5.88,;-.9,5.11,;.43,5.88,;1.76,5.11,;1.76,3.57,;.43,2.8,;.43,1.26,;-.82,.35,;-2.28,.83,;-.34,-1.11,;1.2,-1.11,;.96,-2.63,;2.48,-2.87,;2.72,-1.35,;3.38,-4.12,;3.14,-5.64,;4.66,-5.88,;4.91,-4.36,;1.68,.35,;3.14,.83,;-.9,3.57,;-2.24,2.8,)|
CN1C(=O)N(C(=O)C11CC(C1)c1ccccc1Cl)c1cncc2ccccc12 |(-2.37,-1.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;.07,-.66,;-.17,-2.19,;1.35,-2.43,;1.6,-.91,;2.26,-3.67,;1.63,-5.08,;2.54,-6.33,;4.07,-6.16,;4.7,-4.76,;3.79,-3.51,;4.42,-2.1,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
CN1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12 |(-1.91,-2.36,;-1.01,-1.11,;-1.48,.35,;-2.95,.83,;-.24,1.26,;1.01,.35,;2.47,.83,;.53,-1.11,;.29,-2.63,;1.81,-2.87,;2.05,-1.35,;2.72,-4.12,;2.48,-5.64,;4,-5.88,;4.24,-4.36,;-.24,2.8,;1.1,3.57,;1.1,5.11,;-.24,5.88,;-1.57,5.11,;-2.91,5.88,;-4.24,5.11,;-4.24,3.57,;-2.91,2.8,;-1.57,3.57,)|
NC(=O)CN1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12 |(-2.19,-5.01,;-1.29,-3.76,;.25,-3.92,;-1.91,-2.36,;-1.01,-1.11,;-1.48,.35,;-2.95,.83,;-.24,1.26,;1.01,.35,;2.47,.83,;.53,-1.11,;.29,-2.63,;1.81,-2.87,;2.05,-1.35,;2.72,-4.12,;2.48,-5.64,;4,-5.88,;4.24,-4.36,;-.24,2.8,;1.1,3.57,;1.1,5.11,;-.24,5.88,;-1.57,5.11,;-2.91,5.88,;-4.24,5.11,;-4.24,3.57,;-2.91,2.8,;-1.57,3.57,)|
Clc1cc(CN2C(=O)N(C(=O)C22CC(C2)C2CCC2)c2cncc3ccccc23)cc(Cl)n1 |(-5.32,.22,;-4.55,-1.11,;-3.01,-1.11,;-2.24,-2.44,;-.7,-2.44,;.07,-1.11,;-.4,.35,;-1.87,.83,;.84,1.26,;2.09,.35,;3.55,.83,;1.61,-1.11,;1.37,-2.63,;2.89,-2.87,;3.13,-1.35,;3.8,-4.12,;3.56,-5.64,;5.08,-5.88,;5.32,-4.36,;.84,2.8,;2.18,3.57,;2.18,5.11,;.84,5.88,;-.49,5.11,;-1.83,5.88,;-3.16,5.11,;-3.16,3.57,;-1.83,2.8,;-.49,3.57,;-3.01,-3.78,;-4.55,-3.78,;-5.32,-5.11,;-5.32,-2.44,)|
O=C1N(CC#N)C2(CC(C2)C2CCC2)C(=O)N1c1cncc2ccccc12 |(-2.58,.83,;-1.11,.35,;-.64,-1.11,;-1.54,-2.36,;-3.08,-2.2,;-4.61,-2.03,;.9,-1.11,;.66,-2.63,;2.18,-2.87,;2.42,-1.35,;3.09,-4.12,;2.85,-5.64,;4.37,-5.88,;4.61,-4.36,;1.38,.35,;2.84,.83,;.13,1.26,;.13,2.8,;1.46,3.57,;1.46,5.11,;.13,5.88,;-1.2,5.11,;-2.54,5.88,;-3.87,5.11,;-3.87,3.57,;-2.54,2.8,;-1.2,3.57,)|
O=C(CN1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12)c1ccccn1 |(-2.8,-.68,;-2.17,-2.09,;-.64,-2.25,;.27,-1,;-.21,.46,;-1.67,.94,;1.04,1.37,;2.28,.46,;3.75,.94,;1.81,-1,;1.57,-2.52,;3.09,-2.77,;3.33,-1.24,;3.99,-4.01,;3.75,-5.53,;5.27,-5.77,;5.51,-4.25,;1.04,2.91,;2.37,3.68,;2.37,5.22,;1.04,5.99,;-.3,5.22,;-1.63,5.99,;-2.96,5.22,;-2.96,3.68,;-1.63,2.91,;-.3,3.68,;-3.08,-3.33,;-2.45,-4.74,;-3.35,-5.99,;-4.89,-5.83,;-5.51,-4.42,;-4.61,-3.17,)|
C=CCN1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12 |(-2.19,-5.01,;-1.29,-3.76,;-1.91,-2.36,;-1.01,-1.11,;-1.48,.35,;-2.95,.83,;-.24,1.26,;1.01,.35,;2.47,.83,;.53,-1.11,;.29,-2.63,;1.81,-2.87,;2.05,-1.35,;2.72,-4.12,;2.48,-5.64,;4,-5.88,;4.24,-4.36,;-.24,2.8,;1.1,3.57,;1.1,5.11,;-.24,5.88,;-1.57,5.11,;-2.91,5.88,;-4.24,5.11,;-4.24,3.57,;-2.91,2.8,;-1.57,3.57,)|
CCN1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12 |(-3.45,-2.36,;-1.91,-2.36,;-1.01,-1.11,;-1.48,.35,;-2.95,.83,;-.24,1.26,;1.01,.35,;2.47,.83,;.53,-1.11,;.29,-2.63,;1.81,-2.87,;2.05,-1.35,;2.72,-4.12,;2.48,-5.64,;4,-5.88,;4.24,-4.36,;-.24,2.8,;1.1,3.57,;1.1,5.11,;-.24,5.88,;-1.57,5.11,;-2.91,5.88,;-4.24,5.11,;-4.24,3.57,;-2.91,2.8,;-1.57,3.57,)|
O=C1N(Cc2ccccn2)C2(CC(C2)C2CCC2)C(=O)N1c1cncc2ccccc12 |(-1.8,.83,;-.34,.35,;.14,-1.11,;-.77,-2.36,;-2.31,-2.36,;-3.08,-3.69,;-4.62,-3.69,;-5.39,-2.36,;-4.62,-1.02,;-3.08,-1.02,;1.68,-1.11,;1.44,-2.63,;2.96,-2.87,;3.2,-1.35,;3.86,-4.12,;3.62,-5.64,;5.14,-5.88,;5.39,-4.36,;2.16,.35,;3.62,.83,;.91,1.26,;.91,2.8,;2.24,3.57,;2.24,5.11,;.91,5.88,;-.42,5.11,;-1.76,5.88,;-3.09,5.11,;-3.09,3.57,;-1.76,2.8,;-.42,3.57,)|
O=C1N(Cc2ncc[nH]2)C2(CC(C2)C2CCC2)C(=O)N1c1cncc2ccccc12 |(-2.16,.83,;-.69,.35,;-.22,-1.11,;-1.12,-2.36,;-2.66,-2.36,;-3.57,-3.6,;-5.03,-3.13,;-5.03,-1.59,;-3.57,-1.11,;1.32,-1.11,;1.08,-2.63,;2.6,-2.87,;2.85,-1.35,;3.51,-4.12,;3.27,-5.64,;4.79,-5.88,;5.03,-4.36,;1.8,.35,;3.26,.83,;.55,1.26,;.55,2.8,;1.89,3.57,;1.89,5.11,;.55,5.88,;-.78,5.11,;-2.11,5.88,;-3.45,5.11,;-3.45,3.57,;-2.11,2.8,;-.78,3.57,)|
O=C1CCCN1CN1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12 |(-3.09,-5.07,;-3.57,-3.6,;-5.03,-3.13,;-5.03,-1.59,;-3.57,-1.11,;-2.66,-2.36,;-1.12,-2.36,;-.22,-1.11,;-.69,.35,;-2.16,.83,;.55,1.26,;1.8,.35,;3.26,.83,;1.32,-1.11,;1.08,-2.63,;2.6,-2.87,;2.85,-1.35,;3.51,-4.12,;3.27,-5.64,;4.79,-5.88,;5.03,-4.36,;.55,2.8,;1.89,3.57,;1.89,5.11,;.55,5.88,;-.78,5.11,;-2.11,5.88,;-3.45,5.11,;-3.45,3.57,;-2.11,2.8,;-.78,3.57,)|
CC(=O)N1C(=O)N(C(=O)C11CC(C1)C1CCC1)c1cncc2ccccc12 |(-3.45,-2.36,;-1.91,-2.36,;-1.21,-3.73,;-1.01,-1.11,;-1.48,.35,;-2.95,.83,;-.24,1.26,;1.01,.35,;2.47,.83,;.53,-1.11,;.29,-2.63,;1.81,-2.87,;2.05,-1.35,;2.72,-4.12,;2.48,-5.64,;4,-5.88,;4.24,-4.36,;-.24,2.8,;1.1,3.57,;1.1,5.11,;-.24,5.88,;-1.57,5.11,;-2.91,5.88,;-4.24,5.11,;-4.24,3.57,;-2.91,2.8,;-1.57,3.57,)|
O=C1N(Cc2ccn[nH]2)C2(CC(C2)C2CCC2)C(=O)N1c1cncc2ccccc12 |(-2.16,.83,;-.69,.35,;-.22,-1.11,;-1.12,-2.36,;-2.66,-2.36,;-3.57,-1.11,;-5.03,-1.59,;-5.03,-3.13,;-3.57,-3.6,;1.32,-1.11,;1.08,-2.63,;2.6,-2.87,;2.85,-1.35,;3.51,-4.12,;3.27,-5.64,;4.79,-5.88,;5.03,-4.36,;1.8,.35,;3.26,.83,;.55,1.26,;.55,2.8,;1.89,3.57,;1.89,5.11,;.55,5.88,;-.78,5.11,;-2.11,5.88,;-3.45,5.11,;-3.45,3.57,;-2.11,2.8,;-.78,3.57,)|
FC(F)(F)c1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(4.5,-.65,;3.88,-2.05,;2.47,-1.43,;5.28,-2.68,;3.25,-3.46,;4.13,-4.76,;3.51,-6.16,;1.97,-6.33,;1.07,-5.08,;1.7,-3.67,;.79,-2.43,;-.73,-2.19,;-.49,-.66,;1.03,-.91,;-2.03,-.66,;-2.51,.8,;-3.97,1.28,;-1.26,1.71,;-.01,.8,;1.45,1.28,;-1.26,3.25,;.07,4.02,;.07,5.56,;-1.26,6.33,;-2.59,5.56,;-3.93,6.33,;-5.26,5.56,;-5.26,4.02,;-3.93,3.25,;-2.59,4.02,)|
Cc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
O=C1NC2(CC(C2)c2ccccc2C#N)C(=O)N1c1cncc2ccccc12 |(-3.58,1.28,;-2.12,.8,;-1.64,-.66,;-.1,-.66,;-.34,-2.19,;1.18,-2.43,;1.42,-.91,;2.09,-3.67,;1.46,-5.08,;2.36,-6.33,;3.9,-6.16,;4.52,-4.76,;3.64,-3.46,;4.27,-2.05,;4.89,-.65,;.38,.8,;1.84,1.28,;-.87,1.71,;-.87,3.25,;.46,4.02,;.46,5.56,;-.87,6.33,;-2.2,5.56,;-3.54,6.33,;-4.87,5.56,;-4.87,4.02,;-3.54,3.25,;-2.2,4.02,)|
Clc1cccc(c1)C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12 |(5.46,-4.6,;3.93,-4.76,;3.3,-6.16,;1.77,-6.33,;.87,-5.08,;1.49,-3.67,;3.03,-3.51,;.59,-2.43,;-.93,-2.19,;-.69,-.66,;.83,-.91,;-2.23,-.66,;-2.71,.8,;-4.17,1.28,;-1.46,1.71,;-.22,.8,;1.25,1.28,;-1.46,3.25,;-.13,4.02,;-.13,5.56,;-1.46,6.33,;-2.79,5.56,;-4.13,6.33,;-5.46,5.56,;-5.46,4.02,;-4.13,3.25,;-2.79,4.02,)|
Clc1ccc(cc1)C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12
Fc1ccc(cc1)C1CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2cccnc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2cnccc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2nccnc12 |(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Fc1cccc2cncc(N3C(=O)NC4(CC(C4)c4ccccc4Cl)C3=O)c12 |(-3.36,1.89,;-3.36,3.25,;-4.7,4.02,;-4.7,5.56,;-3.36,6.33,;-2.03,5.56,;-.7,6.33,;.64,5.56,;.64,4.02,;-.7,3.25,;-.7,1.71,;-1.94,.8,;-3.41,1.28,;-1.47,-.66,;.07,-.66,;-.17,-2.19,;1.35,-2.43,;1.6,-.91,;2.26,-3.67,;1.63,-5.08,;2.54,-6.33,;4.07,-6.16,;4.7,-4.76,;3.79,-3.51,;4.42,-2.1,;.55,.8,;2.02,1.28,;-2.03,4.02,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)C1=CN=CC2CCCCC12 |c:22,t:20,(4.42,-2.1,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,;2.26,-3.67,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,)|
Fc1cc2c(cncc2c(F)c1F)N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(-5.36,2.48,;-4.03,3.25,;-2.7,2.48,;-1.36,3.25,;-.03,2.48,;1.3,3.25,;1.3,4.79,;-.03,5.56,;-1.36,4.79,;-2.7,5.56,;-2.7,7.1,;-4.03,4.79,;-5.36,5.56,;-.03,.94,;-1.27,.03,;-2.74,.51,;-.8,-1.43,;.74,-1.43,;.5,-2.96,;2.02,-3.2,;2.26,-1.68,;2.93,-4.44,;2.3,-5.85,;3.21,-7.1,;4.74,-6.93,;5.36,-5.53,;4.46,-4.28,;5.08,-2.87,;1.22,.03,;2.68,.51,)|
Fc1ncccc1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(1.33,3.25,;-.01,4.02,;-.01,5.56,;-1.34,6.33,;-2.67,5.56,;-2.67,4.02,;-1.34,3.25,;-1.34,1.71,;-2.59,.8,;-4.05,1.28,;-2.11,-.66,;-.57,-.66,;-.81,-2.19,;.71,-2.43,;.95,-.91,;1.61,-3.67,;.99,-5.08,;1.89,-6.33,;3.42,-6.16,;4.05,-4.76,;3.15,-3.51,;3.77,-2.1,;-.09,.8,;1.37,1.28,)|
Clc1ccccc1C1CC2(C1)NC(=O)C(C2=O)c1cccnn1
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cnccc1Oc1ccccc1
CC1(CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12)c1ccc(F)cc1Cl |(.27,4.38,;.43,2.84,;.19,1.32,;1.71,1.08,;1.95,2.6,;3.25,1.08,;3.73,-.38,;5.19,-.86,;2.48,-1.29,;1.24,-.38,;-.23,-.86,;2.48,-2.83,;3.81,-3.6,;3.81,-5.14,;2.48,-5.91,;1.15,-5.14,;-.19,-5.91,;-1.52,-5.14,;-1.52,-3.6,;-.19,-2.83,;1.15,-3.6,;-.98,3.47,;-2.23,2.57,;-3.63,3.2,;-3.78,4.73,;-5.19,5.36,;-2.54,5.63,;-1.14,5,;.11,5.91,)|
Fc1ncc(Br)cc1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(-1.93,2.93,;-3.27,2.16,;-4.6,2.93,;-5.93,2.16,;-5.93,.62,;-7.27,-.15,;-4.6,-.15,;-3.27,.62,;-1.93,-.15,;-1.77,-1.68,;-2.92,-2.71,;-.26,-2,;.51,-.67,;1.7,-1.64,;2.67,-.44,;1.47,.53,;4.2,-.28,;4.83,1.13,;6.36,1.29,;7.27,.04,;6.64,-1.36,;5.11,-1.52,;4.48,-2.93,;-.52,.48,;-.2,1.98,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1c(Cl)ncc2ccccc12
Fc1cc(Cl)c(cc1F)C1CC2(C1)NC(=O)N(C2=O)c1c(Cl)ncc2ccccc12
Fc1cccc2cnc(Cl)c(N3C(=O)NC4(CC(C4)c4ccccc4Cl)C3=O)c12
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2cccnc12
Cc1ccnc(F)c1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O
COc1ccnc(F)c1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O
FC(F)(F)c1ccncc1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O
CN(C)c1ccncc1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cnnc2ccccc12
CC1(CC2(C1)NC(=O)N(C2=O)c1cncc2cccc(F)c12)c1ccccc1Cl |(-.67,4.33,;-.27,2.84,;-.51,1.32,;1.01,1.09,;1.26,2.61,;2.55,1.09,;3.03,-.38,;4.5,-.85,;1.78,-1.28,;.54,-.38,;-.93,-.85,;1.78,-2.82,;3.12,-3.59,;3.12,-5.13,;1.78,-5.9,;.45,-5.13,;-.88,-5.9,;-2.22,-5.13,;-2.22,-3.59,;-.88,-2.82,;-.88,-1.59,;.45,-3.59,;-1.68,3.47,;-2.93,2.56,;-4.33,3.19,;-4.5,4.72,;-3.25,5.63,;-1.84,5,;-.6,5.9,)|
CC1(CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12)c1ccccc1Cl |(-.67,4.33,;-.27,2.84,;-.51,1.32,;1.01,1.09,;1.26,2.61,;2.55,1.09,;3.03,-.38,;4.5,-.85,;1.78,-1.28,;.54,-.38,;-.93,-.85,;1.78,-2.82,;3.12,-3.59,;3.12,-5.13,;1.78,-5.9,;.45,-5.13,;-.88,-5.9,;-2.22,-5.13,;-2.22,-3.59,;-.88,-2.82,;.45,-3.59,;-1.68,3.47,;-2.93,2.56,;-4.33,3.19,;-4.5,4.72,;-3.25,5.63,;-1.84,5,;-.6,5.9,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2cc[nH]c12 |(.04,5.24,;-1.49,5.08,;-2.39,6.32,;-3.93,6.16,;-4.55,4.75,;-3.65,3.51,;-2.12,3.67,;-1.21,2.42,;-1.44,.9,;.08,.67,;.32,2.19,;1.62,.67,;2.09,-.8,;3.56,-1.27,;.85,-1.7,;-.4,-.8,;-1.86,-1.27,;.85,-3.24,;-.48,-4.01,;-.48,-5.55,;.85,-6.32,;2.18,-5.55,;3.65,-6.03,;4.55,-4.78,;3.65,-3.54,;2.18,-4.01,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2[nH]c(=O)[nH]c12 |(-.73,5.24,;-2.26,5.08,;-3.16,6.32,;-4.7,6.16,;-5.32,4.75,;-4.42,3.51,;-2.89,3.67,;-1.98,2.42,;-2.21,.9,;-.69,.67,;-.45,2.19,;.85,.67,;1.32,-.8,;2.79,-1.27,;.08,-1.7,;-1.17,-.8,;-2.63,-1.27,;.08,-3.24,;-1.25,-4.01,;-1.25,-5.55,;.08,-6.32,;1.41,-5.55,;2.88,-6.03,;3.78,-4.78,;5.32,-4.78,;2.88,-3.54,;1.41,-4.01,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncc2nccn12 |(-.54,-5.24,;.99,-5.08,;1.89,-6.33,;3.42,-6.16,;4.05,-4.76,;3.15,-3.51,;1.61,-3.67,;.71,-2.43,;-.81,-2.19,;-.57,-.66,;.95,-.91,;-2.11,-.66,;-2.59,.8,;-4.05,1.28,;-1.34,1.71,;-.09,.8,;1.37,1.28,;-1.34,3.25,;-2.67,4.02,;-2.67,5.56,;-1.34,6.33,;-.01,5.56,;1.46,6.03,;2.36,4.79,;1.46,3.54,;-.01,4.02,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cccnc1
O=C1NC2(CC(C2)n2cccn2)C(=O)N1c1cncc2ccccc12 |(-3.2,1.13,;-1.73,.66,;-1.26,-.81,;.28,-.81,;.04,-2.33,;1.57,-2.57,;1.81,-1.05,;2.47,-3.81,;1.99,-5.28,;3.24,-6.18,;4.49,-5.28,;4.01,-3.81,;.76,.66,;2.23,1.13,;-.49,1.56,;-.49,3.1,;.85,3.87,;.85,5.41,;-.49,6.18,;-1.82,5.41,;-3.15,6.18,;-4.49,5.41,;-4.49,3.87,;-3.15,3.1,;-1.82,3.87,)|
CN(C)c1cc2c(cncc2c(F)c1F)N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(-6.03,3.25,;-4.7,2.48,;-4.7,.94,;-3.36,3.25,;-2.03,2.48,;-.7,3.25,;.64,2.48,;1.97,3.25,;1.97,4.79,;.64,5.56,;-.7,4.79,;-2.03,5.56,;-2.03,7.1,;-3.36,4.79,;-4.7,5.56,;.64,.94,;-.61,.03,;-2.07,.51,;-.13,-1.43,;1.41,-1.43,;1.17,-2.96,;2.69,-3.2,;2.93,-1.68,;3.59,-4.44,;2.97,-5.85,;3.87,-7.1,;5.4,-6.93,;6.03,-5.53,;5.13,-4.28,;5.75,-2.87,;1.88,.03,;3.35,.51,)|
CC(C)c1ccncc1N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(-4.65,4.71,;-3.56,3.62,;-3.96,2.13,;-2.07,4.02,;-2.07,5.56,;-.74,6.33,;.59,5.56,;.59,4.02,;-.74,3.25,;-.74,1.71,;-1.99,.8,;-3.45,1.28,;-1.51,-.66,;.03,-.66,;-.21,-2.19,;1.31,-2.43,;1.55,-.91,;2.21,-3.67,;1.59,-5.08,;2.49,-6.33,;4.02,-6.16,;4.65,-4.76,;3.75,-3.51,;4.37,-2.1,;.5,.8,;1.97,1.28,)|
CN(C)c1cncc(c1)N1C(=O)NC2(CC(C2)c2ccccc2Cl)C1=O |(-4.7,4.79,;-3.36,5.56,;-3.35,7.1,;-2.03,4.79,;-.7,5.56,;.64,4.79,;.64,3.25,;-.7,2.48,;-2.03,3.25,;-.7,.94,;-1.94,.03,;-3.41,.51,;-1.47,-1.43,;.07,-1.43,;-.17,-2.96,;1.35,-3.2,;1.6,-1.68,;2.26,-4.44,;1.63,-5.85,;2.54,-7.1,;4.07,-6.93,;4.7,-5.53,;3.79,-4.28,;4.42,-2.87,;.55,.03,;2.02,.51,)|
Clc1ccccc1C1CC2(C1)NC(=O)N(C2=O)c1cncnc1 |(3.77,-2.1,;3.15,-3.51,;4.05,-4.76,;3.42,-6.16,;1.89,-6.33,;.99,-5.08,;1.61,-3.67,;.71,-2.43,;-.81,-2.19,;-.57,-.66,;.95,-.91,;-2.11,-.66,;-2.59,.8,;-4.05,1.28,;-1.34,1.71,;-.09,.8,;1.37,1.28,;-1.34,3.25,;-2.67,4.02,;-2.67,5.56,;-1.34,6.33,;-.01,5.56,;-.01,4.02,)|
Clc1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)cc1Cl
O=C(Cn1nnc2ccccc12)N(CC1CCCC1)c1ccc(cc1)-c1ccc[nH]c1=O
Cc1[nH]ncc1-c1ccc(cc1)N(Cc1cccc(Cl)c1)C(=O)Cn1nnc2ccccc12
O=C(Cn1nnc2ccccc12)N(CC1COC1)c1ccc(cc1)-c1cccnc1
Cc1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2cccnc2)cc1Cl
Fc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
C[C@@H](N(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1)c1cc(F)cc(Cl)c1 |r|
Cc1[nH]cnc1-c1ccc(cc1)N(Cc1cc(F)cc(Cl)c1)C(=O)Cn1nnc2ccccc12
Fc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cn2)-c2c[nH]cn2)c1
FC(F)(F)c1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
O=C(Cn1nnc2ccccc12)N(Cc1cccc(c1)C#N)c1ccc(cc1)-c1c[nH]cn1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
O=C(Cn1nnc2ccccc12)N(CC1CCC1)c1ccc(cc1)-c1c[nH]cn1
Fc1ccc(F)c(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1F
Fc1cccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1ccc(Cl)cc1CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
Fc1c(Cl)cccc1CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
Clc1cncc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
COc1ccc(Cl)cc1CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
COc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
CC(N(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1)c1cc(F)cc(F)c1
CC(C)CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2CCNCC2)c1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2=CCNC2)c1 |t:30|
COC(=O)Cc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
OC(=O)Cc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
NC(=O)Cc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
FC(F)(F)c1cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)ccn1
FC(F)(F)c1cncc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cncc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cccc(F)c1CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
OCCc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2ncc[nH]2)c1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)N2CCNCC2=O)c1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C#N)c1
Fc1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)nc1
Cc1nc(c[nH]1)-c1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]nn2)c1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2nnc[nH]2)c1
NCCc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2CCNC2)c1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2=CC(=O)NC2)c1 |t:30|
COc1ccc(F)cc1CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
COc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cn2ccnn2)c2ccc(cc2)-c2c[nH]cn2)c1
Clc1cccc(CN(C(=O)Cn2ccnn2)c2ccc(cc2)-c2cn[nH]c2)c1
CC(C)(C)CN(C(=O)Cn1nnc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2CNC(=O)C2)c1
Fc1cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)ccc1Cl
COc1ccc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)cc1F
Fc1cc(F)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2CNC2)c1
Fc1cncc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2CNC2)c1
Fc1cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)cc(OC(F)(F)F)c1
Fc1cc(Cl)cc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2CNC2)c1
Fc1cncc(CN(C(=O)Cn2nnc3ccccc23)c2ccc(cc2)C2=CCNC2)c1 |t:29|
CC(=O)NCc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
NCc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cn1nnc2ccccc12
Clc1cccc(CN(C(=O)Cc2nnc3ccccn23)c2ccc(cc2)-c2cn[nH]c2)c1
Clc1cccc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2cn[nH]c2)c1
Fc1ccc2nnc(CC(=O)N(Cc3cccc(Cl)c3)c3ccc(cc3)-c3cn[nH]c3)n2c1
Clc1cccc(CN(C(=O)Cc2cnc3ccccn23)c2ccc(cc2)-c2cn[nH]c2)c1
Clc1cccc(CN(C(=O)Cc2cnccn2)c2ccc(cc2)-c2cn[nH]c2)c1
Clc1cccc(CN(C(=O)Cc2cccnn2)c2ccc(cc2)-c2cn[nH]c2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2nnc3ccccn23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1ccc2nnc(CC(=O)N(Cc3cc(F)cc(Cl)c3)c3ccc(cc3)-c3c[nH]cn3)n2c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cnc3ccccn23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
C[C@@H](N(C(=O)Cc1nnc2ccccn12)c1ccc(cc1)-c1c[nH]cn1)c1cc(F)cc(Cl)c1 |r|
C[C@@H](N(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1)c1cc(F)cc(Cl)c1 |r|
Fc1ccc(Cl)cc1CN(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
Fc1c(Cl)cccc1CN(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
Clc1cncc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
COc1ccc(Cl)cc1CN(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
COc1cc(Cl)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1ccc(F)c(CN(C(=O)Cc2nnc3ccccn23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1ccc(F)c(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cccc(CN(C(=O)Cc2nnc3ccccn23)c2ccc(cc2)-c2c[nH]cn2)c1F
Fc1cccc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1F
Fc1cccc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(F)cc(CN(C(=O)Cc2nnc3ccccn23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cn2)-c2c[nH]cn2)c1
CC(N(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1)c1cc(F)cc(F)c1
Fc1cc(F)cc(CN(C(=O)Cc2cccnn2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)N2CCNCC2=O)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)N2CCNC(=O)C2)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C#N)c1
FC(F)(F)c1cncc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cncc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Cc1ccc2nnc(CC(=O)N(Cc3cc(F)cc(F)c3)c3ccc(cc3)-c3c[nH]cn3)n2n1
Cc1ccc2nnc(CC(=O)N(Cc3cc(F)cc(Cl)c3)c3ccc(cc3)-c3c[nH]cn3)n2n1
Fc1cc(Cl)cc(CN(C(=O)Cc2cccnc2)c2ccc(cc2)-c2c[nH]cn2)c1
Clc1cccc(CN(C(=O)Cc2cccnc2)c2ccc(cc2)-c2c[nH]cn2)c1
CC(C)(C)CN(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
CC(C)CN(C(=O)Cc1nnc2ccccn12)c1ccc(cc1)-c1c[nH]cn1
Fc1cccc(CN(C(=O)Cc2nnc3ccccn23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cncnc2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2noc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)CC2NC(=O)c3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
NC(=O)c1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cc1cncc2ccccc12
Fc1cc(Cl)cc(CN(C(=O)Cc2cccnn2)c2ccc(cc2)-c2c[nH]cn2)c1
COc1ccc(F)cc1CN(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1
COc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cnccn2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C2=CCNC2)c1 |t:31|
Fc1cc(Cl)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C2=CCNC2)c1 |t:31|
Fc1cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)ccc1Cl
Fc1cc(Cl)cc(CN(C(=O)CC2C(=O)Nc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cncc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C2CNC2)c1
Fc1cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)cc(OC(F)(F)F)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C2CNC2)c1
CC(C)(C)NC(=O)C(N(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)C1=CCNC1)c1cc(F)cc(F)c1 |t:31|
CC(C)(C)NC(=O)C(N(C(=O)Cc1cncc2ccccc12)c1ccc(cc1)-c1c[nH]cn1)c1cc(F)cc(F)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc(Br)c2)c2ccc(cc2)-c2c[nH]cn2)c1
Cc1cncc(CC(=O)N(Cc2cc(F)cc(F)c2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(F)cc(CN(C(=O)Cc2cncc(c2)C2CC2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cncc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C2=CCNC2)c1 |t:30|
Fc1cncc(CC(=O)N(Cc2cc(F)cc(Cl)c2)c2ccc(cc2)-c2c[nH]cn2)c1
Cc1cncc(CC(=O)N(Cc2cc(F)cc(Cl)c2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cncc(c2)C2CC2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cncc3ccccc23)c2ccc(cc2)C2CNC2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2nncc3ccccc23)c2ccc(cc2)-c2c[nH]cn2)c1
NCc1ccc(cc1)N(Cc1cc(F)cc(F)c1)C(=O)Cc1cncc2ccccc12
Fc1cc(Cl)cc(CN(C(=O)Cc2cnccc2C(F)(F)F)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2cnccc2Cl)c2ccc(cc2)-c2c[nH]cn2)c1
Cc1ccncc1CC(=O)N(Cc1cc(F)cc(Cl)c1)c1ccc(cc1)-c1c[nH]cn1
COc1ccncc1CC(=O)N(Cc1cc(F)cc(Cl)c1)c1ccc(cc1)-c1c[nH]cn1
Fc1cc(Cl)cc(CN(C(=O)Cc2cncc(c2)C2CC2)c2ccc(cc2)C2CNC2)c1
Cc1cncc(CC(=O)N(Cc2cc(F)cc(Cl)c2)c2ccc(cc2)C2CNC2)c1
Fc1cncc(CN(C(=O)Cc2cncc(F)c2)c2ccc(cc2)-c2c[nH]cn2)c1
Fc1cc(Cl)cc(CN(C(=O)Cc2nncc3ccccc23)c2ccc(cc2)C2CNC2)c1
Fc1cncc(CN(C(=O)Cc2cncc(F)c2)c2ccc(cc2)C2CNC2)c1
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)NC(=O)OCc2ccccc2
[2H]c1c([2H])c([2H])c(C([2H])([2H])OC(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C=O)C[C@@H]2CCNC2=O)c([2H])c1[2H]
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)c1ccccc1
[2H]c1c([2H])c([2H])c(C([2H])([2H])OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(O)S(=O)(=O)[O-])c([2H])c1[2H]
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-])c1ccccc1
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(OC(C)=O)S(=O)(=O)[O-])c1ccccc1
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(OC(=O)CCCCC)S(=O)(=O)[O-])c1ccccc1
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CC(F)(F)C2)cc(Br)cc1[N+](=O)[O-])c1cncc2ccccc12
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCCCC2)cc(Br)cc1[N+](=O)[O-])c1cncc2ccccc12
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCCC2)cc(Br)cc1[N+](=O)[O-])c1cncc2ccccc12
O=C(c1cccnc1)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(Br)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CCC(F)(F)CC1
CC1(C)C2CN(C(=O)c3cc(Br)cc([N+](=O)[O-])c3N[C@@H]3CCCN(C(=O)c4cncc5ccccc45)C3)CC21
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3cc(Cl)ccc23)C1)N1CCCCC1
O=C(N[C@H]1CCCC[C@H]1Nc3c(C(=O)N2CCCCC2)cc(Br)cc3C(F)(F)F)c4cncc5ccccc45
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CCNCC1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cnnc3ccccc23)C1)N1CCCCC1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCN(C(=O)c2cncc3ccccc23)C1)N1CCCCC1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CCCCC1
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCCCC2)cc(Br)cc1[N+](=O)[O-])c1cncc(Br)c1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CC2CC2C1
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCC(F)(F)CC2)cc(Br)cc1[N+](=O)[O-])c1cc(=O)[nH]c2ccccc12
C[C@@H]1CN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCN(C(=O)c3cncc4[nH]ccc34)C2)C[C@H](C)O1
C[C@@H]1CN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCN(C(=O)C3CCNC(=O)C3)C2)C[C@H](C)O1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCC(N5CCOCC5)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)N[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCN(CC(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCN(C(=O)C(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
O=C(c1cc[nH]c(=O)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCC(F)(F)CC3)cc(Br)cc2[N+](=O)[O-])C1
O=C1CN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCC[C@@H]2NC(=O)c2cncc3cc(Cl)ccc23)CCN1
Cc1cc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCOCC4)cc(Br)cc3[N+](=O)[O-])C2)cc(=O)[nH]1
Cc1cc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C2)cc(=O)[nH]1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3[nH]ccc23)C1)N1CCC(F)(F)CC1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCN(C)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
Cc1cc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCN(C(=O)C(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C2)cc(=O)[nH]1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CC(Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)c1
C[C@H]1CCCN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCN(C(=O)[C@H]3CC(=O)N[C@@H](C)C3)C2)C1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCO[C@H](C)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCCC(F)(F)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCO[C@H](CF)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CCOCC1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CCCC1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCN(C(=O)c2cncc3ccccc23)C1)N1CCCC1
N#Cc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C2)c1
Nc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C2)c1
Cc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C2)c1
O=C(c1cncc(Br)c1)N1CCC[C@@H](Nc2c(C(=O)N3CC4CC4C3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(C2CC2)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
Cc1c(Br)cncc1C(=O)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(Br)c1)N4CC[C@@H](Nc3c(C(=O)N2CCCCC2)cc(Br)cc3C(F)(F)F)C4
O=C(c1cc(Br)cc(C(F)(F)F)c1N[C@@H]4CCN(C(=O)c2cncc3ccccc23)C4)N5CCCCC5
O=C(c1cncc(Br)c1)N4CCC[C@@H](Nc3c(C(=O)N2CCC(F)(F)CC2)cc(Br)cc3C(F)(F)F)C4
O=C(c1cncc(O)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCC(F)(F)CC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCN(C(=O)c2cncc3cc(Cl)ccc23)C1)N1CC2CC2C1
O=C(N[C@H]1CCCC[C@H]1Nc3c(C(=O)N2CCOCC2)cc(Br)cc3C(F)(F)F)c4cncc5cc(Cl)ccc45
O=C(c1cc(=O)[nH]c(=O)[nH]1)N1CCC[C@@H](Nc2c(C(=O)N3CCC(F)(F)CC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cc(=O)[nH]c3ccccc23)C1)N1CCC(F)(F)CC1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCO[C@H](C(F)F)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cnnc3ccccc23)C1)N1CCCCC1
O=C(c1cc(O[N+](=O)[O-])cc(Cl)c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1)N1CCCCC1
N#Cc1cc(Cl)cc(C(=O)N2CCCCC2)c1N[C@@H]1CCCN(C(=O)c2cncc3ccccc23)C1
O=C(c1cncnc1)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(OC(F)F)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
COc1ncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C2)cn1
O=C(c1cnc(Cl)nc1)N1CCC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(Br)c1)N1CC[C@@H](Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(Br)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCCC3)cc(Br)cc2[N+](=O)[O-])C1
O=C(c1cncc(Br)c1)N4CCC[C@@H](Nc3c(C(=O)N2CCCCC2)cc(Br)cc3C(F)(F)F)C4
O=C(c1cc(Br)cc(C(F)(F)F)c1N[C@@H]4CCCN(C(=O)c2cncc3ccccc23)C4)N5CCCCC5
O=C(c1cncc(Br)c1)N4CC[C@@H](Nc3c(C(=O)N2CCCCC2)cc(Br)cc3C(F)(F)F)C4
O=C(c1cncc(Br)c1)N4CC[C@@H](Nc3c(C(=O)N2CCC(F)(F)CC2)cc(Br)cc3C(F)(F)F)C4
O=C(c1cncc(C(F)(F)F)c1)N4CCC[C@@H](Nc3c(C(=O)N2CCC(F)(F)CC2)cc(Br)cc3[N+](=O)[O-])C4
Nc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCC(F)(F)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
C[C@@H]1C[C@H](C)CN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCN(C(=O)c3cncc(Br)c3)C2)C1
C[C@@H]1CN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCN(C(=O)c3cncc(Br)c3)C2)C[C@H](C)N1
Cc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCC(F)(F)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
O=C(c1cncc(I)c1)N1CCC[C@@H](Nc2c(C(=O)N3CCC(F)(F)CC3)cc(Br)cc2[N+](=O)[O-])C1
C[C@@H]1CN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCN(C(=O)c3cncc(Br)c3)C2)C[C@H](C)O1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCN(C(=O)C(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CCN(C)CC4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4C[C@@H](C)N(C)[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CC[C@@H](NC(=O)C(F)(F)F)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4CC5C(C4)C5(C)C)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCN(CC(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCN(CC(F)(F)F)C(=O)C4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@H](C)C[C@H](C)C4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCC(C)(C)CC4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)c1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4CC5C(C4)C5(C)C)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)NCC(F)(F)F)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCN(CC(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCN(CC(F)(F)F)C(=O)C4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@H](C)C[C@H](C)C4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCC(C)(C)CC4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCC5(CC4)CC5)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
Cc1cc(C(=O)N2C[C@H](Nc3c(C(=O)N4CCC5(CCC5)CC4)cc(Br)cc3[N+](=O)[O-])C3(CC3)C2)cc(=O)[nH]1
CNc1cncc(C(=O)N2CCC[C@@H](Nc3c(C(=O)N4CC(=O)NC(C)C4)cc(Br)cc3[N+](=O)[O-])C2)c1
CNc1cncc(C(=O)N2CC(Nc3c(C(=O)C4CC5C(C4)C5(C)C)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)c1
CNc1cncc(C(=O)N2CC(Nc3c(C(=O)N4CCN(CC(F)(F)F)CC4)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)c1
CNc1cncc(C(=O)N2CC(Nc3c(C(=O)N4CCN(CC(F)(F)F)C(=O)C4)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)c1
CNc1cncc(C(=O)N2CC(Nc3c(C(=O)N4C[C@H](C)C[C@H](C)C4)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)c1
Cc1cc(C(=O)N2CC(Nc3c(C(=O)N4CCCCC4)cc(Br)cc3[N+](=O)[O-])C(F)(F)C2)cc(=O)[nH]1
CC1(Nc2c(C(=O)N3CCCCC3)cc(Br)cc2[N+](=O)[O-])CCCN(C(=O)c2cncc3ccccc23)C1
O=C(c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCN(C(=O)c2cncc3cc(F)ccc23)C1)N1CCCCC1
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CNc5cncc(C(=O)N3C[C@H](Nc2c(C(=O)N1C[C@H](C)O[C@H](C)C1)cc(Br)cc2[N+](=O)[O-])C[C@H]3C(=O)Nc4cc(C(F)(F)F)ncn4)c5
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)N[C@H]2CC(=O)N(C)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)Nc2nn(C3C[C@@H](C)O[C@@H](C)C3)cc2Br)c1
CO[C@H]1CN(C(=O)c2cncc3[nH]nc(C)c23)C[C@@H]1Nc1c(C(=O)N2C[C@@H](C)O[C@@H](C)C2)cc(Br)cc1[N+](=O)[O-]
CNc1cncc(C(=O)N2C[C@H](Nc3c(-c4nnn(C)n4)cc(Br)cc3[N+](=O)[O-])[C@@H](OC)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)Nc2cc(Cl)ncn2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)Nc2ccnc(Cl)n2)c1
[2H]C([2H])([2H])Nc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OC)C2)c1
CO[C@H]1CN(C(=O)c2cncc3[nH]nc(Cl)c23)C[C@@H]1Nc1c(C(=O)N2C[C@@H](C)O[C@@H](C)C2)cc(Br)cc1[N+](=O)[O-]
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)Nc2ncc(Br)cn2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@@H](OCCOC)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2COC)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@@H](O[C@@H]3CCOC3)C2)c1
CO[C@H]1CN(C(=O)c2cncc3[nH]c(C)nc23)C[C@@H]1Nc1c(C(=O)N2C[C@@H](C)O[C@@H](C)C2)cc(Br)cc1[N+](=O)[O-]
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)NCc2ccnc(C(F)(F)F)n2)c1
[2H]C([2H])([2H])Nc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OC([2H])([2H])[2H])C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@@H](O[C@H]3CCOC3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])C[C@H]2C(=O)NC2CCN(CCOC)CC2(F)F)c1
CO[C@H]1CN(C(=O)c2cncc3[nH]nnc23)C[C@@H]1Nc1c(C(=O)N2C[C@@H](C)O[C@@H](C)C2)cc(Br)cc1[N+](=O)[O-]
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3ccccc3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3ccc(OC)nc3)C2)c1
CNc5cncc(C(=O)N4C[C@H](Nc2c(C(=O)N1C[C@H](C)O[C@H](C)C1)cc(Br)cc2[N+](=O)[O-])[C@@H](OCc3ccc(C(F)(F)F)nc3)C4)c5
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3ccccn3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3ccc(F)cn3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3ncco3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3nccs3)C2)c1
CNc1cncc(C(=O)N2C[C@H](Nc3c(C(=O)N4C[C@@H](C)O[C@@H](C)C4)cc(Br)cc3[N+](=O)[O-])[C@@H](OCc3cncn3C)C2)c1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)Cc1ccc2c(c1)OCO2)C1CCN(C(C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)Cc1ccc2c(c1)OCO2)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)Cc1cccc(F)c1)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)Cc1ccccc1)C1CCN(C(C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C1CC1)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C1CCC1)C1CCN(C(C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C1CCC1)C1CCN([C@H](C)c2cccc3ccccc23)CC1
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NC/C=C/C(N)=O)C(=O)C2CCC2)CC1
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NC/C=C/S(C)(=O)=O)C(=O)C2CCC2)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C1CCCC1)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C1CCCCC1)C1CCN([C@H](C)c2cccc3ccccc23)CC1
C#CCNC(=O)CNC(=O)CNC1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(C)=O)C1CCN(C(C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C(F)(F)F)C1CCN([C@H](C)c2cccc3ccccc23)CC1
CCC(=O)N(CC(=O)NCC(=O)NC/C=C/C(=O)OC)C1CCN(C(C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)CC(F)(F)F)C1CCN(C(C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)C(C)C)C1CCN([C@H](C)c2cccc3ccccc23)CC1
CCCC(=O)N(CC(=O)NCC(=O)NC/C=C/C(=O)OC)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C(=O)CC(C)C)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(N)(=O)=O
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)NC(=O)OC(C)(C)C
COC(=O)/C=C/CNC(=O)CNC(=O)CNC1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(C)C1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)[C@H](CN)NC1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)[C@H](CNC(=O)OC(C)(C)C)NC3CCN([C@H](C)c1cccc2ccccc12)CC3
COC(=O)/C=C/CNC(=O)CNC(=O)[C@@H](C)NC1CCN([C@H](C)c2cccc3ccccc23)CC1
COC(=O)/C=C/CNC(=O)CNC(=O)C[C@H](NCc1ccc2c(c1)OCO2)C1CCN(C(C)c2cccc3ccccc23)CC1
C#CCNC(=O)CCNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C[C@H](c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NC/C=C/S(C)(=O)=O)S(C)(=O)=O)CC1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)C1CC1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)c1ccccc1
C[C@H](c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NCC=O)S(C)(=O)=O)CC1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)N1CCCC1
COC(=O)/C=C/CNC(=O)CNC(=O)CN(/C=C/C(=O)C(F)(F)F)C3CCN([C@H](C)c1cccc2ccccc12)CC3
C#CCNC(=O)CNC(=O)CN(CCC(C)=O)C1CCN([C@H](C)c2cccc3ccccc23)CC1
C#CCNC(=O)CNC(=O)CN(C3CCN([C@H](C)c1cccc2ccccc12)CC3)S(=O)(=O)C(F)(F)F
C#CCNC(=O)CCC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3cccnc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2c(F)ccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccc(Cl)cc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccnc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN([C@@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN([C@@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)C1CC1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)N1CCCC1
C#CCNC(=O)CNC(=O)[C@@H]1CNS(=O)(=O)N1C1CCN([C@H](C)c2cccc3ccccc23)CC1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1F)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(Cl)c2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccc(OC)c3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(=O)(=O)N1CCCC1
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(C)c2C)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C3CCN(C(c1cccc2ccccc12)C(F)(F)F)CC3)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccccc2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccccc2C(F)(F)F)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(CC)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C2(c3cccc4ccccc34)CC2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccc(F)c3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(Br)c2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccc3ccccc3c2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2nccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(-c3ccccc3)c2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccccc2-c2ccccc2)CC1)S(C)(=O)=O
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NCC#N)S(C)(=O)=O)CC1
CCOC(=O)CN1CCN(S(=O)(=O)N(CC(=O)NCC(=O)NCC#N)C2CCN(C(C)c3cccc4ccccc34)CC2)CC1
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NCC#N)S(=O)(=O)N2CCN(CC(=O)O)CC2)CC1
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NCC#N)C(=O)CCC(=O)O)CC1
C#CCNC(=O)CNC(=O)CN(C1CCN(c2nc3ccccc3s2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccc(Cl)cc2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccc(OC)c(Cl)c2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(OC)c2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2c(Cl)cccc2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(c2nc3cc(Cl)ccc3s2)CC1)S(C)(=O)=O
C#CCCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CC(C)NC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccccc2F)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccccc2OC)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(=O)(=O)CCC(=O)OC
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NCC(=O)CF)S(C)(=O)=O)CC1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)CCC(N)=O
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)N1CCC(C(=O)OC)C1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)CCCO
COC(=O)/C=C/CNC(=O)c1nnc(CNC(=O)CN(C2CCN(C(C)c3cccc4ccccc34)CC2)S(C)(=O)=O)o1
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(=O)(=O)N1CCC(C(N)=O)C1
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2ccc(OC)cc2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cc(Cl)ccc2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(-c3cccs3)c2)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc(C)c2Cl)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(CO)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(CF)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(N)(=O)=O
C#CC(=O)NNC(=O)CN(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=O)CNC(=O)CN(C1CCN(C(c2cccc3ccccc23)C(F)F)CC1)S(C)(=O)=O
[2H]C([2H])([2H])C(c1cccc2ccccc12)N3CCC(N(CC(=O)NCC(=O)NCC#C)S(C)(=O)=O)CC3
C#CCNC(=O)CNC(=O)[C@@H](C)N(C1CCN([C@H](C)c2cccc3ccccc23)CC1)S(C)(=O)=O
[2H]C([2H])(C#C)NC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
COC(CNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O)OC
C#CC(C)(C)CNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCCNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
CC(c1cccc2ccccc12)N1CCC(N(CC(=O)NCC(=O)NC/C=C/C(N)=O)S(C)(=O)=O)CC1
COC(=O)/C(C#N)=C/CNC(=O)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#CCNC(=S)CNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C=CC(=O)NNC(=O)CN(C1CCN(C(C)c2cccc3ccccc23)CC1)S(C)(=O)=O
C#Cc1nnc(NC(=O)CN(C2CCN(C(C)c3cccc4ccccc34)CC2)S(C)(=O)=O)o1
Cc1cncc(-c2nnc3n2CCN(C(c2ccccc2)c2ccccc2)C3)c1
Cc1cncc(C(=O)N2CCC(=C3c4ccccc4CS(=O)c4ccccc43)CC2)c1
Cc1cncc(C(=O)N2CCC(=C3c4ccccc4CS(=N)(=O)c4ccccc43)CC2)c1
O=C(c1cncc2cc[nH]c12)N1CCC(=C2c3ccccc3CSc3ccccc32)CC1
O=C(c1cncc2cc[nH]c12)N1CCC(=C2c3ccccc3CS(=O)c3ccccc32)CC1
N=S1(=O)Cc2ccccc2C(=C2CCN(C(=O)c3cncc4cc[nH]c34)CC2)c2ccccc21
Cc1cncc(C(=O)N2CCN(C3c4ccccc4CS(=O)(=O)c4ccc(F)cc43)CC2)c1
O=C(c1cncc2cc[nH]c12)N1CCN(C2c3ccccc3CS(=O)(=O)c3ccc(F)cc32)CC1
Cc1cncc(C(=O)N2CCN(C3c4cc(F)ccc4CS(=O)(=O)c4ccccc43)CC2)c1
O=C(c1cncc2cc[nH]c12)N1CCN(C2c3cc(F)ccc3CS(=O)(=O)c3ccccc32)CC1
Cc1cncc(C(=O)N2CCC(=C3c4ccccc4CC(=O)c4sccc43)CC2)c1
O=C1Cc2ccccc2C(=C2CCN(C(=O)c3cncc4cc[nH]c34)CC2)c2ccsc21
O=C(c1cncc2cc[nH]c12)N1CCC(=C2c3ccccc3C3OC3c3ccccc32)CC1
O=C1Cc2ccccc2C(=C2CCN(C(=O)c3cncc4cc[nH]c34)CC2)c2ccccc21
Cc1cncc(-n2c(=O)c(Oc3ccccc3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)c1
N#CCn1c(N2Cc3cn[nH]c3C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cc[nH]c(=O)c2)c1=O
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C)c(C)c3)n(C(C)C#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C)c(C)c3)n(CC#N)c2=O)c1
CC(C)(O)C1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cncc(N2C(=O)N(CC#N)CC3(CCOc4ccc(Cl)cc43)C2=O)c1
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2Cc3ccccc3C2)c(C(=O)c2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2Cc3ccccc3C2)c(Sc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2cccc(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCc1c(N2Cc3ccccc3C2)n(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
COc1ccc(Oc2c(Cc3cc(F)c(F)c(F)c3)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)cc1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
N#CCn1c(N2CC(O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(Cl)cnn2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(c3ncc(F)cn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(CO)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(O)(c2ccccc2)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)(F)F)c2)c1=O
Cc1cncc(N2C(=O)N(CC#N)CC3(COc4ccc(Cl)cc43)C2=O)c1
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(CCC(N)=O)c1=O
Cn1cnc(Cn2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4cn[nH]c4C3)n(CC#N)c2=O)n1
CN1C[C@@H]2CN(c3c(Cc4cc(F)c(F)c(F)c4)c(=O)n(Cc4ncn(C)n4)c(=O)n3CC#N)C[C@@H]2C1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(OC(C(F)(F)F)C(F)(F)F)n(CC#N)c2=O)c1
Cn1cnc(Cn2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3cc4ccccc4s3)n(CC#N)c2=O)n1
Cn1cnc(Cn2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCc4ccccc4C3)n(CC#N)c2=O)n1
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncnc2)c1=O
Cn1cnc(Cn2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)n1
COc1ccc(Oc2c(-c3cccc4ccccc34)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)cc1
Cc1cncc(-n2c(=O)c(Oc3cc(F)c(F)c(F)c3)c(Oc3cc(F)c(F)c(F)c3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(C(=O)c3cc(F)c(F)c(F)c3)c(-c3cc4ccccc4s3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3cccc(C#N)c3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(Cl)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(Cl)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3cccc4ccccc34)c(N3Cc4cn[nH]c4C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3cnc4ccccc4c3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Oc3cc(F)c(F)c(F)c3)c(-c3cc4ccccc4s3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3cc4ccccc4s3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3cc4ccccc4s3)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(CCCO3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3cnc(C)nc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3Cc4ccccc4C3=O)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C(=O)O)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N(C)Cc3ccccc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3cc4ccccc4[nH]3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C(=O)OC(C)(C)C)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(Oc3cccc4[nH]ccc34)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(Oc3cccc4ccccc34)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(Oc3ccc(F)cc3Cl)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C(F)(F)F)c(Cl)c3)n(CC#N)c2=O)c1
Cc1cc(-n2c(=O)c(-c3cc(F)c(F)c(Cl)c3)c(N3CC4(CCOCC4)C3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3cc(F)c(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3cc(F)c(F)c(Cl)c3)c(N3CCC(C(F)(F)F)CC3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cnnc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3C[C@H]4C[C@@H](C3)O4)n(CC#N)c2=O)c1
Cc1cnnc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3ccccn23)c1=O
N#CCn1c(N2CC3CCC(CC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3ccccn23)c1=O
Cc1cnnc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)c1
N#CCn1c(N2Cc3ccccc3C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3ccccn23)c1=O
CCCOc1cc(Cl)cc(-c2c(N3Cc4ccccc4C3)n(CC#N)c(=O)n(-c3cncc(C)c3)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3cccc(Cl)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3ccccn23)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC4(CCNC4=O)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(Cl)n(C(C)C#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(/C=C/CO)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C)c(C)c3)n(C(F)C#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C)c(C)c3)n(C3(C#N)CC3)c2=O)c1
CC(C)(C)OC(=O)C(C#N)n1c(N2CCC(C(F)(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC3(CNC(=O)C3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(CCCO)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(CCOC4)C3)n(C(C)C#N)c2=O)c1
N#CCn1c(Cl)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C)c(C)c3)n(C(C#N)C(=O)O)c2=O)c1
Cc1ccc(-c2c(Cc3cc(F)c(F)c(F)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)cc1C
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC3(CCC(=O)N3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3CNC(=O)C3C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC3(CNC(=O)C3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2Cc3cn[nH]c3C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(-c3ccc(C)c(C)c3)n(C(C)(C)C#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C(F)(F)F)c(Cl)c3)n(CC#N)c2=O)c1
N#CCn1c(N2CCC3(CC2)CNC(=O)O3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CN1CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)CC1=O
N#CCn1c(N2CCC(C(F)(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC4(CCOC4)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C4CC4)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3Cc4cn[nH]c4C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3Cc4cccnc4C3)n(CC#N)c2=O)c1
N#CCn1c(N2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(c3nccs3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(n3cccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCN(c3ccccc3)C(=O)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2C[C@@H]3[C@@H](O)[C@@H]3C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(c3ccccc3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC(C)OC1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1
N#CCn1c(N2CC(N3CCOCC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(O)(C(F)(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cn1cnc(Cn2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC(F)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C#N)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(CCOCC4)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC4(CCC(=O)N4)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC4(C3)NC(=O)NC4=O)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC[C@@H](C(N)=O)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCCC(C(F)(F)F)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCN(C)C(=O)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C(N)=O)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)c1
COC1CCN(c2c(Cc3cc(F)c(F)c(F)c3)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)C1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4CC(F)(F)C4C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(CO)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
COC1CCN(c2c(Cc3cc(F)c(F)c(F)c3)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)CC1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C(F)F)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(S(N)(=O)=O)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C)(O)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC4(CCC(O)C4)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC4(CCOCC4)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C(N)=O)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C(F)(F)F)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC4(CC3)CNC(=O)O4)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C)(F)C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(O)(C(F)(F)F)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3C[C@H]4CN(C)C[C@H]4C3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C(F)F)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCC(C(F)(F)F)CC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3nc4ccccc4s3)n(CC#N)c2=O)c1
N#CCn1c(N2Cc3ccccc3C2)c(-c2cccc(Cl)c2)c(=O)n(C2CCn3cnnc32)c1=O
Cn1cnc(Cn2c(=O)c(-c3cccc(Cl)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)n1
Cc1cc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)cc(=O)[nH]1
N#CCn1c(N2Cc3ccccc3C2)c(-c2cccc(Cl)c2)c(=O)n(Cc2ccc[nH]c2=O)c1=O
N#CCn1c(Cl)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3ccc(F)cn23)c1=O
N#CCn1c(Cl)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3cnccn23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnn3ccccc23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3ccc(F)cn23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3ccc(F)cn23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3nc4ccccc4o3)n(CC#N)c2=O)c1
CC(C)(O)C1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cnc4cc(Cl)ccn34)c(=O)n2CC#N)C1
N#CCn1c(N2CC3(CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
CC1(O)CC2(CN(c3c(-c4ccc(F)c(Cl)c4)c(=O)n(-c4cnc5cc(F)ccn45)c(=O)n3CC#N)C2)C1
CC1(O)CC2(CN(c3c(-c4ccc(F)c(Cl)c4)c(=O)n(-c4cnc5cc(Cl)ccn45)c(=O)n3CC#N)C2)C1
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
N#CCn1c(N2CCC(O)(C(F)(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(Cl)ccn23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2nsc3ccccc23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3cccnn23)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2C[C@H]3C[C@@H]2CN3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2CCC(F)(F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2CCC(O)(C(F)(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2CC3(CCCO3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2CCC(C(F)(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
CC1(C)CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cnc4cc(F)ccn34)c(=O)n2CC#N)C1
N#CCn1c(N2Cc3ccccc3C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(C2CCNC(=O)C2)c1=O
N#CCn1c(N2Cc3ccccc3C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2nnc3ccccn23)c1=O
Cn1c(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)cc(=O)n1C
N#CCn1c(N2Cc3ccccc3C2)c(Cc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(=O)[nH]2)c1=O
Cc1cc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4ccccc4C3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cnnc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)c1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(CCOCC4)C3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC(C(F)(F)F)CC3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)cc(=O)[nH]1
Cc1[nH]ncc1-n1c(=O)c(Cc2cc(F)c(F)c(F)c2)c(N2Cc3ccccc3C2)n(CC#N)c1=O
CC1(C)CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cc4n(c(=O)c3)CCC4)c(=O)n2CC#N)CC1
N#CCn1c(-c2cc3ccccc3s2)c(Sc2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2cccc(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC(C)(C)CC3)n(CC#N)c2=O)cc(=O)[nH]1
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccccc2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3C[C@H]4CCCC[C@H]4C3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3cc4ccccc4s3)n(CC#N)c2=O)cc(=O)[nH]1
N#CCn1c(N2CCC(F)(F)CC2)c(-c2cccc(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC1(C)CN(c2c(-c3cccc(C#N)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1
CC1(C)CCN(c2c(-c3cccc(C#N)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)CC1
N#CCn1c(N2CC3(CCOC3)C2)c(-c2cccc(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC1(C)[C@@H]2CN(c3c(-c4cccc(Cl)c4)c(=O)n(-c4cncc(Cl)c4)c(=O)n3CC#N)C[C@@H]21
N#CCn1c(N2CC3(CCOC3)C2)c(-c2cc(Cl)cc(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2cc(F)cc(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C4CC4)cc3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(C#CC3CC3)n(CC#N)c2=O)cc(=O)[nH]1
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(C(F)(F)F)[nH]c(=O)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(Cl)[nH]c(=O)c2)c1=O
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)cnn1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3nc4ccccc4s3)n(CC#N)c2=O)cc(=O)[nH]1
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)(F)F)n2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)n2)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(CCOC4)C3)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC(C(F)F)CC3)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(CCCO4)C3)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC(C)(C)C3)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC(F)(F)CC3)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)n1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CCC(C(F)(F)F)CC3)n(CC#N)c2=O)n1
Cc1cc(-n2c(=O)c(-c3cc(Cl)cc(C(F)(F)F)c3)c(N3CCC(C(F)(F)F)CC3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3cc(Cl)cc(C(F)(F)F)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3CCCC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(Cc3cc(F)c(F)c(F)c3)c(N3Cc4cn[nH]c4C3)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)n2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)(F)F)n2)c1=O
N#CCc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)n1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(CC#N)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(C3=CCOCC3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(/C=C/c3ccc(C(F)(F)F)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3cc(F)c(F)c(F)c3)c(CCC(C)(C)O)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(Cl)cnn2)c1=O
COc1cnnc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(C#N)cnn2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(OCC(F)F)cnn2)c1=O
CNc1cnnc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
CN(C)c1cnnc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C(F)F)cc3)n(CC#N)c2=O)cc(=O)[nH]1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)[nH]c(=O)c1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(=O)cc(Br)[nH]2)c1=O
CC(C)N1CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)CC1=O
CCN1CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)CC1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3C[C@@H]4C[C@H]3CO4)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3C[C@H]4C[C@@H]3CO4)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(CCOC3)C2)c(C2=CCCCCC2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cnnc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(C(F)(F)F)cnn2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(F)c2)c1=O
N#CCn1c(N2CC(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@H](C(=O)N3CC(F)(F)C3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@@H](C(=O)C3CC(F)(F)C3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(c3cnccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@@](O)(c3ccccc3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@](O)(c3ccccc3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCCO2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCOC2=O)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CN1CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1=O
N#CCn1c(OC2CC(F)(F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(Oc2cncc(Cl)c2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(C#CC3CC3)n(CC#N)c2=O)c1
N#CCn1c(N2CCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC1(c2ccc(F)c(Cl)c2)CN(CC#N)C(=O)N(c2cncc(Cl)c2)C1=O
N#CCn1c(N2CCCCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cnc(F)c(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c1
N#CCn1c(N2CC(O)(c3nccs3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2cncc(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
COc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)n1
C[C@@H](C#N)n1c(N2CC3(CCOC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC(=O)Nc1cccc(-c2c(N3CCC(F)(F)CC3)n(CC#N)c(=O)n(-c3cncc(Cl)c3)c2=O)c1
N#CCn1c(N2CC3(CCOC3)C2)c(C2=CCCCC2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(-c2ccc(C3CC3)cc2)c(N2CCCCC2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(C2CCC(F)(F)CC2)c(-c2ccnc(C(F)(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2C[C@@H]3CC[C@H]2C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
C[C@H](C#N)n1c(N2CC(C(C)(C)O)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC(C)(O)C1(F)CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1
Cc1ccc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)cc1
COc1ccc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C)c3)c(=O)n2CC#N)cc1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(F)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(C(N)=O)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(N(C)C)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3ccc(S(N)(=O)=O)cc3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(NS(=O)(=O)c3ccccc3)n(CC#N)c2=O)c1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(Cl)n(CC#N)c2=O)c[n+]([O-])c1
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)c[n+]([O-])c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(-c3cn[nH]c3)n(CC#N)c2=O)c1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(Oc3ccccc3)n(CC#N)c2=O)c1
N#CCn1cc(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CCCCc1c(N2CC3(CCOC3)C2)n(CC#N)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(C2CCCCC2)c(=O)n(-c2cncc(Cl)c2)c1=O
CCCCc1c(-c2ccc(F)cc2)n(CC#N)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(F)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(F)(F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cncc(-n2c(=O)c(-c3cc(F)c(F)c(F)c3)c(/C=C/C(C)(C)O)n(CC#N)c2=O)c1
N#CCn1c(N2CC3(CCOCC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CN1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C=N1
C[C@@]1(O)CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(F)c2)c1=O
CC1(O)CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)C1
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(C3=CC4(CCOCC4)C3)n(CC#N)c2=O)c1
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
N#CCn1c(N2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(F)c2)c1=O
CC(C)=Cc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
Cn1ccc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)n1
Cn1ccc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)cc1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2onc3cc(F)ccc23)c1=O
N#CCn1c(N2CCC(F)(C#N)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC(C)(O)CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
CC(C)(F)Cc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
CC(C)(O)Cc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
N#CCn1c(N2CC(F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CC(OC(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CC(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
CC(C)(O)[C@@H]1CCN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C#N)c3)c(=O)n2CC#N)C1
Cc1cc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)on1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)(F)F)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2C[C@@H]3C[C@H]2CO3)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)c(F)cn23)c1=O
N#CCn1c(CCC(F)(F)F)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2cc(F)c(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2cc(F)c(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cc(-c2c(N3CCC(F)(F)CC3)n(CC#N)c(=O)n(-c3cncc(Cl)c3)c2=O)cs1
N#CCn1c(N2CCC(F)(F)CC2)c(-c2csc3ccccc23)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2cc(Cl)cc(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2cc(O)cc(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OC(F)F)n2)c1=O
N#CCn1c(N2CC(O)(C(F)F)C2)c(-c2cc(F)c(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)(F)F)n2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)(F)F)n2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
Cc1cncc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC(O)(c4ncccn4)C3)n(CC#N)c2=O)n1
N#CCn1c(N2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2C[C@@H]3C[C@H]2CO3)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1cc(-n2c(=O)c(-c3ccc(F)c(Cl)c3)c(N3CC4(C3)CC(F)(F)C4)n(CC#N)c2=O)cc(=O)o1
N#CCn1c(N2CC(O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)c2)c1=O
N#CCn1c(N2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)c2)c1=O
N#CCn1c(C2(O)CCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(C2=CCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(CCC(F)F)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cnc3cc(F)ccn23)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
CC1(O)CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(OC(F)F)n3)c(=O)n2CC#N)C1
CC1(O)CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(OCF)n3)c(=O)n2CC#N)C1
N#CCn1c(N2CC[C@@](O)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
CC(C)(F)CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
N#CCn1c(-c2nnc(C3CC3)s2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1coc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)n1
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Br)c2)c1=O
N#CCn1c(N2CC3(C=C(F)C3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(I)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(CC2CC(F)(F)C2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(CCOC3)C2)c(CCCC(F)(F)F)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2cc(F)c(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2cc(F)c(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2cc(F)c(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2cc(F)c(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2C[C@@H]3C[C@H]2CO3)c(-c2cc(F)c(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(C2CC(O)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2C[C@@H]3C[C@H]2CO3)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OC(F)F)n2)c1=O
COc1ccc(-c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(Cl)c3)c(=O)n2CC#N)cn1
N#CCn1c(-c2ccc(CO)nc2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
CC1(O)CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C(F)F)n3)c(=O)n2CC#N)C1
N#CCn1c(N2CC(O)(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
N#CCn1c(-c2ccc(C#N)nc2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(-c2ccc(F)nc2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
C[C@@H](C#N)n1c(N2CCC(F)(F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(-c2ccc(C(F)F)nc2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(C2CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
COCC1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C(F)F)n3)c(=O)n2CC#N)C1
N#CCn1c(C2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C(F)F)n2)c1=O
N#CCn1c(CCC2CC(F)(F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
C[C@](O)(CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N)C(F)F
C[C@@](O)(CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N)C(F)F
N#CCn1c(C2CC(F)(F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(C2CCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
COC1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C(F)F)n3)c(=O)n2CC#N)C1
N#CCn1c(N2CCC(C(F)F)CC2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(C(F)F)CC2)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CC[C@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(C(F)(F)F)CC2)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CCC(C(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
CCCNC(=O)c1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
CC(C)NC(=O)c1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
N#CCn1c(CC2(O)CCC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CC(CO)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CC(F)(C3CC3)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CC(O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CCC(C(F)F)CC2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CCC(C(F)F)CC2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
CC(C)(O)CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c(=O)n1CC#N
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CC(O)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(N2CCC(F)(F)CC2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
CCOC1CN(c2c(-c3ccc(F)c(Cl)c3)c(=O)n(-c3cncc(C(F)F)n3)c(=O)n2CC#N)C1
C[C@@H](C#N)n1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CC(C(F)(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
N#CCn1c(N2CCC(C(F)F)CC2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(OCF)n2)c1=O
C[C@H](C#N)n1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(CCC2(O)CCC2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
N#CCn1c(CCC2(O)CCC2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC3(C2)CC(F)(F)C3)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cc(Cl)c[n+]([O-])c2)c1=O
C[C@@H](C#N)n1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(C#N)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
C[C@@H](C#N)n1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
C[C@](O)(CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c(=O)n1CC#N)C(F)F
C[C@@](O)(CCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c(=O)n1CC#N)C(F)F
C[C@@H](C#N)n1c(N2CC[C@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
C[C@@H](C#N)n1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
C[C@@H](C#N)n1c(N2CC[C@@](O)(C(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
C[C@@H](C#N)n1c(N2CC[C@](O)(C(F)F)C2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
COCc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC#N
N#CCn1c(CCC2(O)CCC2)c(-c2ccc(F)c(F)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(OC(F)F)C2)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
C#CCn1c(C)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
N#CCn1c(N2CC(O)(c3ncccn3)C2)c(-c2ccc(F)c(C(F)F)c2)c(=O)n(-c2cncc(C#N)c2)c1=O
C#CCn1c(CC(C)(C)F)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC(N)=O
CC(=O)Cn1c(C)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c(=O)n1CC(=O)CO
CC(=O)OCC(=O)Cn1c(C)c(-c2ccc(F)c(Cl)c2)c(=O)n(-c2cncc(Cl)c2)c1=O
Cc1nc2cc(C)c(Nc3nc(=O)n(Cc4c[nH]cn4)c(=O)n3Cc3cc(F)c(F)c(F)c3)cc2s1
Cc1cncc(-n2c(=O)nc(Nc3cc4cn(C)nc4cc3F)n(Cc3cc(F)c(F)c(F)c3)c2=O)c1
Cc1cncc(c1)-n1c(=O)nc(Nc2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)c(F)c2)c1=O
Cc1cncc(-n2c(=O)nc(Nc3cc4cn(C)nc4cc3C)n(Cc3cc(F)c(F)c(F)c3)c2=O)c1
Cn1cc2cc(c(cc2n1)Cl)NC3=NC(=O)N(C(=O)N3Cc4cc(c(cc4F)F)F)Cc5ncn(n5)C
O=c1nc(Nc2cc3cn(CCO)nc3cc2Cl)n(Cc2cc(F)c(F)c(F)c2)c(=O)n1-c1cncc2ccccc12
CC(=O)N1CC(n2cc3cc(Nc4nc(=O)n(-c5cncc6ccccc56)c(=O)n4Cc4cc(F)c(F)c(F)c4)c(Cl)cc3n2)C1
Cn1cc2cc(Nc3nc(=O)n(-c4cncc(CO)c4)c(=O)n3Cc3cc(F)c(F)c(F)c3)ccc2n1
N#Cc1cc(Cn2c(Nc3ccc4nn(CC(F)F)cc4c3)nc(=O)n(-c3cncc4ccccc34)c2=O)ccc1F
Cn1cc2cc(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3ccc(F)c(C#N)c3)ccc2n1
Cc1cncc(-n2c(=O)nc(Nc3ccc4nn(CC(F)F)cc4c3)n(Cc3ccc(F)c(C#N)c3)c2=O)c1
Cc1cncc(c1)-n1c(=O)nc(Nc2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)cc2F)c1=O
Cc1cc2nn(C)cc2cc1Nc1nc(=O)n(-c2cncc3ccccc23)c(=O)n1Cc1cc(F)c(F)c(F)c1
Cn1cc2cc(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
Cn1cc2cc(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3ccc(F)c(C#N)c3)c(Cl)cc2n1
Cn1cc2cc(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3cc(F)c(F)c(F)c3)ccc2n1
Cc1cncc(-n2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3ccc(F)c(C#N)c3)c2=O)c1
Cc1cncc(-n2c(=O)nc(Nc3cc4cn(C)nc4cc3F)n(Cc3ccc(F)c(C#N)c3)c2=O)c1
Cc1cncc(-n2c(=O)nc(Nc3cc4cn(C)nc4cc3C)n(Cc3ccc(F)c(C#N)c3)c2=O)c1
O=c1nc(Nc2cc3cn(CCN4CCOCC4)nc3cc2Cl)n(Cc2cc(F)c(F)c(F)c2)c(=O)n1-c1cncc2ccccc12
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)n1
Cc1nc2cc(Cl)c(Nc3nc(=O)n(Cc4ncn(C)n4)c(=O)n3Cc3cc(F)c(F)c(F)c3)cc2n1C
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)c1
N#Cc1cc(Cn2c(Nc3cc4cn(C(F)F)nc4cc3Cl)nc(=O)n(-c3cncc4ccccc34)c2=O)ccc1F
Cn1cc2cc(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3ccc(F)c(C#N)c3)c(F)cc2n1
Cc1cncc(-n2c(=O)nc(Nc3cc4cn(C(F)F)nc4cc3Cl)n(Cc3ccc(F)c(C#N)c3)c2=O)c1
Cc1cc2nn(C)cc2cc1Nc1nc(=O)n(-c2cncc3ccccc23)c(=O)n1Cc1ccc(F)c(C#N)c1
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(CCO)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)n1
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(CC(F)F)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)n1
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C(F)F)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)n1
N#Cc1cc(Cn2c(Nc3ccc4nn(CCO)cc4c3)nc(=O)n(-c3cncc4ccccc34)c2=O)ccc1F
Cc1nc2cc(Cl)c(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3cc(F)c(F)c(F)c3)cc2n1C
CC(=O)NCCn1cc2cc(Nc3nc(=O)n(-c4cncc5ccccc45)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
O=c1nc(Nc2ccc3nn(CC(F)F)cc3c2)n(Cc2cc(F)c(F)c(F)c2)c(=O)n1-c1cncc2ccccc12
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3F)c2=O)n1
CC(C)NC[C@H]1CN(c2cncc3ccccc23)C(=O)[C@@]12CN(Cc1cn(C)nn1)C(=O)c1ccc(Cl)cc12
CCNC[C@H]1CN(c2cncc3ccccc23)C(=O)[C@@]12CN(Cc1cc(C)no1)C(=O)c1ccc(Cl)cc12
CCNC[C@H]1CN(c2cncc3ccccc23)C(=O)[C@@]12CN(CC1CCOCC1)C(=O)c1ccc(Cl)cc12
CCNC[C@H]1CN(c2cncc3ccccc23)C(=O)[C@@]12CN(Cc1cc(C)ncn1)C(=O)c1ccc(Cl)cc12
CC(C)NC[C@H]1CN(c2cncc3ccccc23)C(=O)[C@@]12CN(CC1CCOCC1)C(=O)c1ccc(Cl)cc12
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)CC1C(=C=O)Nc3ccccc31)C2(C)C
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=C=O)N(C(=O)[C@@H](NC(=O)C(F)(F)F)C34CC5CC(CC(C5)C3)C4)C[C@@H]21
CC5(C)[C@H]4CN(C(=O)C(NC(=O)C(F)(F)F)C2CC1(CCC1)C2)[C@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)[C@H]45
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)N(C(=O)[C@H](Cc3ccc4ccccc4c3)NC(=O)C(F)(F)F)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)CC3C(=O)Nc4ccccc43)N(C(=O)[C@@H](NC(=O)C(F)(F)F)C34CC5CC(CC(O)(C5)C3)C4)C[C@@H]21
CN(C)C1CCC([C@H](NC(=O)C(F)(F)F)C(=O)N2C[C@H]3[C@@H]([C@H]2C(=O)N[C@H](C#N)C[C@@H]2CCNC2=O)C3(C)C)CC1
CN(C)CCCC[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]4[C@@H]([C@H]1C(=O)N[C@H](C#N)CC3C(=O)Nc2ncccc23)C4(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)Cl)C(=O)N1C[C@H]4[C@@H]([C@H]1C(=O)N[C@H](C#N)CC3C(=O)Nc2ccccc23)C4(C)C
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)CC3CCNC3=O)N(C(=O)[C@@H](NC(=O)C(F)(F)Cl)C34CC5CC(CC(O)(C5)C3)C4)C[C@@H]21
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
[2H]C([2H])(c1ncn(C)n1)n1c(=O)nc(Nc2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)cc2F)c1=O
[2H]C([2H])(c1cc(F)c(F)cc1F)n1c(Nc2cc3cn(C)nc3cc2Cl)nc(=O)n(Cc2ncn(C)n2)c1=O
[2H]C([2H])([2H])n1cc2cc(Nc3nc(=O)n(Cc4ncn(C)n4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(Nc3cc4cn(C([2H])([2H])[2H])nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
[2H]C([2H])([2H])n1cc2cc(Nc3nc(=O)n(Cc4ncn(C)n4)c(=O)n3Cc3cc(F)ccc3F)c(Cl)cc2n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)ccc3F)c2=O)n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)cc(F)c3F)c2=O)n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3ccc(F)c(F)c3F)c2=O)n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3c(F)cc(F)cc3F)c2=O)n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)nc(NC3=CC4OC(F)(F)OC4C=C3Cl)n(Cc3c(F)cc(F)cc3F)c2=O)n1
[2H]C([2H])([2H])n1cnc(Cn2c(=O)[nH]/c(=Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
CC1[C@H]2CN([C@@H]([C@@H]12)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
c1ccc2c(c1)CC(=O)N(C2=O)O
Oc1c(Cc2c(O)c3ccccc3oc2=O)c(=O)oc2ccccc12
c1cc(c(cc1Cc2ccc(c(c2)C(=O)O)O)C(=O)O)O
O=C(NCc1ncc[nH]1)c1c(O)cnc2ccccc12
c1cc(ccc1CCC(=O)c2c(cc(cc2O)O)O)O
O=C(O)c1cccc(Cc2cccc(C(=O)O)c2O)c1O
O=C(O)c1cc2cc(-c3ccccc3)ccc2[nH]c1=O
Oc1ccc(CC2NCCc3cc(O)c(O)cc23)cc1O
CC(C)=CCc1cc(C(=O)/C=C/c2ccc(O)cc2)c(O)cc1O
COc1cc(O)c(CC=C(C)C)c(O)c1C(=O)/C=C/c1ccc(O)cc1
OC(=O)c1c(O)c(Cc2ccc(Cl)cc2)nc2c3CCCCc3ccc12
Cc1c(S(=O)(=O)[O-]->[Na+])oc2c1C(=O)C(=O)c1c-2ccc2c1CCCC2(C)C
CC(C)c1cc(Cc2cc(C(C)C)cc(C(=O)O)c2O)c(O)c(C(=O)O)c1
CC(C)=CCOc1ccc(/C=C/C(=O)c2ccc(OCC=C(C)C)cc2OCC(=O)O)cc1
CC(C)=CCc1c2c(c3occ(-c4ccc(O)c(O)c4)c(=O)c3c1O)C=CC(C)(C)O2
CC(C)=CCc1c(O)cc(O)c(C(=O)/C=C/c2ccc(O)cc2)c1O
CC(C)=CCc1c(O)ccc(C(=O)/C=C/c2ccc(O)c(O)c2)c1O
CC1(C)CCc2c(O)ccc(C(=O)/C=C/c3ccc(O)cc3)c2O1
CC(C)=CCc1c(O)ccc(C(=O)/C=C/c2ccc(O)cc2)c1O
OC(=O)c1ccc2ccc(\C=C\c3ccc(O)c(O)c3)nc2c1O
OC(=O)c1ccc2ccc(nc2c1O)C(=O)NCc1ccc(O)c(O)c1
COc1cc(\C=C\c2ccc3ccc(C(O)=O)c(O)c3n2)cc(O)c1O
OC(=O)c1ccc2ccc(nc2c1O)C(=O)NCc1cccc(O)c1O
OC(=O)c1ccc2ccc(nc2c1O)C(=O)NCc1cc(O)cc(O)c1
OC(=O)c1ccc2ccc(\C=C\c3cc(Br)c(O)c(Br)c3)nc2c1O
OC(=O)c1ccc2ccc(\C=C\c3ccc(F)c(F)c3)nc2c1O
OC(=O)c1ccc2ccc(\C=C\c3ccc(O)c(c3)C(O)=O)nc2c1O
Oc1ccc(\C=C\c2ccc3cccc(O)c3n2)cc1O
Oc1ccc(\C=C\c2ccc3ccc(C(=O)c4ccc(F)c(F)c4)c(O)c3n2)cc1O
OC(=O)c1ccc2ccc(CCc3ccc(O)c(O)c3)nc2c1O
O=C(c1ccccc1)c1ccc2ccc(/C=C/c3ccc(O)c(O)c3)nc2c1O
O=C(O)c1ccc2nc(/C=C/c3ccc(O)c(O)c3)ccc2c1O
O=P(O)(O)c1ccc2ccc(CCc3ccc(O)c(O)c3)nc2c1O
Oc1ccc(\C=C\c2ccc3ccc(C(=O)c4ccc(cc4)[N+]([O-])=O)c(O)c3n2)cc1O
O=C(c1ccccn1)c1ccc2ccc(/C=C/c3ccc(O)c(O)c3)nc2c1O
Oc1ccc(\C=C\c2ccc3ccc(C(=O)c4ccncc4)c(O)c3n2)cc1O
COC(=O)c1ccc(Cn2nc3n(c(=O)c2=O)CCN3c2ccc(F)cc2)o1
O=c1c2c(ncn1CCc1ccc(F)cc1)C1C=CC=CC1N2
CC1(C)C=C2C(=O)C(=O)C(C(=O)N3CCOCC3)=CC2=C2C=CN3C=CCC3=C21
Oc1ccc2C3c4cc(O)c(O)cc4CC3(O)COc2c1O
COc1ccc2[nH]c(=O)c(cc2c1)-c1noc(n1)-c1ccc(F)cc1
COc1ccc2[nH]c(=O)c(cc2c1)-c1noc(n1)-c1ccccc1
ON1C(=O)C(C(=O)NCc2ccc(F)cc2)c2ccc(F)cc2C1=O
ON1C(=O)C(C(=O)NCc2ccc(F)cc2)c2ccc(cc2C1=O)C(F)(F)F
ON1C(=O)C(C(=O)NCc2ccc(F)cc2)c2ccc(Br)cc2C1=O
ON1C(=O)C(C(=O)NC2CCCCC2)c2ccccc2C1=O
ON1C(=O)C(Cc2ccccc2)c2ccccc2C1=O
ON1C(=O)C(C(=O)Nc2ccccc2)c2ccccc2C1=O
Oc1ccc(\C=C\c2ccc3ccc(C(=O)c4cccnc4)c(O)c3n2)cc1O
c1ccc(cc1)[C@@H]2CCN(C[C@H]2NC(=O)c3ccc[nH]3)C(=O)c4cccn5c4cnc5
CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2ccccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1ccn[nH]1
O=C(NC1CN(C(=O)c2cccn3cncc23)CCC1c1cccc(Cl)c1)c1ncc[nH]1
O=C(NC1CN(C(=O)c2cccn3cncc23)CCC1c1cccc(Cl)c1)c1cnc[nH]1
O=C(NC1CN(C(=O)c2cccn3cncc23)CCC1c1ccc(Cl)cc1)c1cnc[nH]1
O=C(NC1CN(C(=O)c2cccn3cncc23)CCC1c1ccc(Cl)cc1)c1ncc[nH]1
O=C(c1cccn2cncc12)N1CCC(c2ccccc2)C(NC(=O)C2(O)CCCCC2)C1
CCc1ncc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)[nH]1
CS(=O)(=O)NCC(=O)NC1CN(C(=O)c2cccn3cncc23)CCC1c1ccccc1
CS(=O)(=O)NCC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
CC(C)(C)[C@H](NS(C)(=O)=O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
CC(=O)NCC(=O)NC1CN(C(=O)c2cccn3cncc23)CCC1c1ccccc1
CC(=O)N[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)C(C)(C)C
O=C(c1cccn2cncc12)N1CC[C@@H](c2ccccc2)[C@H](N2CCNC2=O)C1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
CC(C)[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@H]1NC(=O)[C@@H](NS(C)(=O)=O)C(C)(C)C
CC(C)[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@@H]1NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C
N[C@H]1CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)C1=O
NC1CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)C1=O
O=C(c1cccn2cncc12)N1CC[C@@H](c2ccccc2)[C@H](N2CCCNC2=O)C1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2ccc(CO)cc2[nH]1
N#Cc1cccc2cc(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)[nH]c12
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2cccc(F)c2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2c(F)cccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2ncccc2[nH]1
O=C(c1cccn2cncc12)N1CC[C@@H](c2ccccc2)[C@H](NC(=O)C2(c3ccccc3)CC2)C1
COc1cccc2[nH]c(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)cc12
NS(=O)(=O)c1cccc2[nH]c(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)cc12
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1nc2ccccc2[nH]1
O=C(N[C@@H]1CN(C(=O)C2=CC=CN3C=NCC23)CC[C@H]1c1ccccc1)c1cc2sccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2cnccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1cc2c([nH]1)CCOC2
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nc2ccccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nc2ccccc2[nH]1
CCc1cnc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cccc(Cl)c2)[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nccs1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1cncs1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nc2ccccc2s1
CC1=CNC(C(=O)N[C@@H]2CN(C(=O)C3CC=CN4C=NCC34)CC[C@H]2C2=CC(Cl)CC=C2)N1
Cc1nc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cccc(Cl)c2)[nH]c1C
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1ncc[nH]1
C[C@@H](NS(C)(=O)=O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
CCS(=O)(=O)NCC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
O=C(Cc1ccn[nH]1)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
CN(C(=O)c1cc2ccccc2[nH]1)[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1
CN(C(=O)c1ncc[nH]1)[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nnc[nH]1
CC(C)(C)C[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@H]1NC(=O)c1ncc[nH]1
CC(C)C[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@H]1NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C
CC(C)(C)C[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@H]1NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C
CC(C)(C)[C@H](NS(C)(=O)=O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(F)c1)c1cc2ccccc2[nH]1
N#Cc1cc(Cl)c2[nH]c(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)cc2c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1cc2cccc(F)c2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nc2cccc(F)c2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)c1nc2c(F)ccc(F)c2[nH]1
COc1cccc2nc(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3cccc(Cl)c3)[nH]c12
O=C(CNC(=O)C(F)(F)F)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)c1nc2ccccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)c1cc2ncccc2[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)c1ncc[nH]1
CC(C)c1nc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)cs1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1ncc(C(F)(F)F)[nH]1
CC(C)c1cnc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)[nH]1
CC(C)CC[C@@H](N)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1
CC(C)[C@H](NS(C)(=O)=O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1
Cc1nc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cccc(Cl)c2)sc1C
O=C1Cc2c(cccc2C(=O)N2CC[C@@H](c3cccc(Cl)c3)[C@H](NC(=O)c3nc4ccccc4[nH]3)C2)N1
Cc1cnc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cccc(Cl)c2)s1
Cc1csc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cccc(Cl)c2)n1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccccc1)c1nc2cccc(F)c2[nH]1
COc1cccc2[nH]c(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)nc12
COc1ccc(F)c2[nH]c(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)cc12
Cc1cccc([C@@H]2CCN(C(=O)c3cccn4cncc34)C[C@H]2NC(=O)c2ncc[nH]2)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)C(F)F
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(F)c1)c1cncs1
CC(C)COC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(F)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CN1CCCC[C@]1(C)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1C1CCOCC1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3sncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CC(F)(F)C1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCCC1
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cncc3sncc23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CC(F)(F)C1
O=C(N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)[C@H](O)C1CCOCC1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3sncc23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCCC[C@]1(C)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
Cc1csc([C@@H]2CCN(C(=O)c3cncc4cccnc34)C[C@H]2NC(=O)[C@@H](C)N2CCCC2)c1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2c(F)ccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCC(C)(C)[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3nn(C)cc23)CC[C@H]1c1cc(F)cc(Cl)c1
CN1CCC(F)(F)C[C@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
C[C@H](C(=O)NC1CN(C(=O)c2nccn3cncc23)CC[C@H]1C1CC(F)(F)C1)N1CCCC1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCCC1
CN1CCC(F)(F)C[C@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CCC(F)(F)F
CN1CCC(C)(C)[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)C[C@@H]1CCN(C(=O)c2cncc3cccnc23)C[C@H]1NC(=O)[C@H](NC(=O)C(F)(F)F)C(C)C
CN1CCC(C)(C)[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCC(C)(C)[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
O=C(N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)[C@@H](NCC(F)F)C1CCOCC1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cn(C)nc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)S(=O)(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)C(O)(C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)C(F)(F)F
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CC(F)(F)C1)N1CCCC1
CC(C)[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1)N1CCC1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)[C@@H](NCC(F)F)C1CCOCC1
O=C(N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)C(N1CCCC1)C(F)(F)F
CN1CCCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)CS(=O)(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CCC(F)(F)F)N1CCCC1
CN1CCC(C)(C)[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccnc2)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CN1CCC(C)(C)[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)S(=O)(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)C[C@H]1c1cc(F)cc(Cl)c1
CC(C)S(=O)(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1
O=C(CN1CCCC12CC2)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)c(F)cc1F
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CCC(F)(F)F)N1CCCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(Cl)c1
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1
Cc1ncn2cccc(C(=O)N3CC[C@@H](c4cc(F)cc(F)c4)[C@H](NC(=O)[C@H](NC(=O)C(F)(F)F)C(C)C)C3)c12
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
CC(C)C[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
O=C(N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(F)c1)[C@H](O)C1CCCC1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CCC(F)(F)F
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc(F)c2)CC[C@H]1c1cc(F)cc(F)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CCC(F)(F)F)c1ncc[nH]1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CC(C)(C)C1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)ccc1F
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)[C@@]1(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(F)c2)CCCN1
CC(C)[C@H](NC(=O)C(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@]1(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(F)c2)CCCN1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccnc2)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)C[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCOCC1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)C[C@H]1c1cc(F)cc(Cl)c1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)C(O)C1(C(F)F)CCCC1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCOCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(Cl)ccc1F
CC(C)[C@@H](NC(=O)C(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)ccc1F)N1CCCC1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CC1CC1(F)F)c1ncc[nH]1
CC1(C)COCCN1CC(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
O=C(CN1CCCC12CC2)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)c(F)c(F)c1
CC1(C)COCCN1CC(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC1(C)COCCN1CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CC(C)C[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@H]1NC(=O)[C@@H](C(C)C)N1CCCC1
CN1CCOC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
C[C@]1(NC(=O)C(F)(F)F)CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1=O
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CC1(C)COCCN1CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1F
CN1CCOC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
C[C@]1(NC(=O)C(F)(F)F)CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1=O
O=C(CN1CCCC12CC2)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1F
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccc(F)c(F)c1)N1CCCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(C(F)(F)F)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(C(F)F)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1)N1CCCC1
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1F
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CCC(F)(F)CC1
C[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CCC(F)(F)CC1
CC(C)C[C@@H]1CCN(C(=O)c2cccn3cncc23)C[C@H]1NC(=O)[C@H](NC(=O)C(F)(F)F)C(C)C
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)(C)C[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1F)N1CCCC1
CC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1CC(C)C)N1CCCC1
Cc1cc(C(=O)N2CC[C@@H](c3cc(F)cc(Cl)c3)[C@H](NC(=O)[C@@H](C)NC(=O)C(F)(F)F)C2)c2cncn2c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1F
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](NCC(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)c(F)c(Cl)c1
N[C@H](CCC(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@@]1(O)CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1=O
CC1(O)CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1=O
C[C@@]1(O)CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1=O
CC[C@@]1(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(F)c2)CCCN1
CC[C@@]1(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(F)c2)CCCN1
CC(C)(C)[C@H](O)C(=O)NC1CN(C(=O)c2cncc3cccnc23)CCC1c1cc(F)cc(Cl)c1
CC(C)c1cnc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(F)c2)[nH]1
Cc1nc(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(F)c2)[nH]c1C
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](NC(=O)C2(NCC(F)F)CCOCC2)C1
C[C@@]1(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)CCCN1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
O=C(CN1CCCCC1)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](NC(=O)C(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(=O)N[C@@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)C(C)C
CN1CCC[C@@H]1C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CCC(F)(F)CC1
CC(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC1(C[C@@H]2CCN(C(=O)c3cccn4cncc34)C[C@H]2NC(=O)c2ncc[nH]2)CC1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)[C@H](O)CC1CCCC1
CC(C)(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
Cc1ccc(C(=O)N2CC[C@@H](c3cc(F)cc(Cl)c3)[C@H](NC(=O)[C@@H](C)NC(=O)C(F)(F)F)C2)c2cncn12
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)[C@H](O)C1CCCC1
CC(C)(C)[C@H](NC(=O)C(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)C[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)ccc1F)N1CCCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CCCCC1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCOCC1
O=C(CN1CCCC12CC2)N[C@@H]1CN(C(=O)c2cccn3cncc23)C[C@H]1c1ccccc1
Cc1cncc(C(=O)N2CC[C@@H](c3cc(F)cc(Cl)c3)[C@H](NC(=O)[C@@H](C)NC(=O)C(F)(F)F)C2)c1C
CC(C)(C)[C@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@@H](O)C(=O)NC1CN(C(=O)c2cncc3cccnc23)CCC1c1cc(F)cc(Cl)c1
CC(C)(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](N2CC[C@]3(CCCN3)C2=O)C1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](N2CC[C@]3(CCCN3)C2=O)C1
O=C(CN1CCOCC1)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)ccc1F
C[C@@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCOCC1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)C[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@]1(C(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)CCCN1
O=C(CN1CCCCC1)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(Cl)cc(F)c1F
Cc1ccc(C(=O)N2CC[C@@H](c3cc(F)cc(Cl)c3)[C@H](NC(=O)[C@H](C)NC(=O)C(F)(F)F)C2)c2cncn12
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@H]1CN(C(=O)c2cncc3cccnc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@H](C(=O)N[C@@H]1CN(CC[C@H]1c2cc(cc(c2)Cl)F)C(=O)c3cncc4c3nccc4)NC(=O)C(F)(F)F
CC(C)(C)CC[C@@H]1CCN(C(=O)c2cccn3cncc23)CC1NC(=O)c1ncc[nH]1
C[C@@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
CC(C)[C@H](NC(=O)C(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)N1CCCC1
C[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(CN1CCCC12CC2)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)[C@@H]1CC(F)(F)C(=O)N1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)[C@@H]1CC(F)(F)C(=O)N1
C[C@]1(C#N)CCN(CC(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1
C[C@]1(C#N)CCN(CC(=O)N[C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2cc(F)cc(Cl)c2)C1
CC(C)[C@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cccc(F)c1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cccc(F)c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)[C@H](NC(=O)C(F)(F)F)C1CCC1
CC1(C)CCCN1CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](NC(=O)C2(NCC(F)(F)F)CCOCC2)C1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1ccc(F)c(Cl)c1
CC(C)(C)[C@H](O)C(=O)N[C@@H]1CN(C(=O)c2cncc3cncn23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@H](O)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
COC[C@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)C(C)C
C[C@H](NCC(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@@H]1CCCN1CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
C[C@H]1CCCN1CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccnc2)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)NC1CN(C(=O)c2cncc3cncn23)CCC1c1cccc(F)c1
CC(C)(CC(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2nccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](N2CCC(NC(=O)C(F)(F)F)C2=O)C1
C[C@@H](OCC(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccc3c2CC(=O)N3)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)[C@H](O)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(Cl)cc(C#N)c1
C[C@H](OCC(F)(F)F)C(=O)N[C@@H]1CN(C(=O)C2CC=CN3C=NCC23)CC[C@H]1C1=CC(Cl)CC(F)=C1
Cn1cc([C@@H]2CCN(C(=O)c3cccn4cncc34)C[C@H]2NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)cn1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)C[C@H]1c1cccc(Cl)c1
CC(NCC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)C(F)(F)F
C[C@@H](NCC(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)C(F)(F)F
CC(F)(F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(CN1CCC(F)(F)C1)N[C@@H]1CN(C(=O)C2CC=CN3C=NCC23)CC[C@H]1C1=CC(Cl)CC(F)=C1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](NC(=O)C2(NC(=O)C(F)(F)F)CCCCC2)C1
Cc1cc([C@@H]2CCN(C(=O)c3cccn4cncc34)C[C@H]2NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)nn1C
CC(C)(CC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1)C(F)(F)F
O=C(CN1CCCC1)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(C)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(CNCC(F)(F)F)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cncc(Cl)c1)c1ncc[nH]1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)c1nc2c([nH]1)CCCC2
C[C@](O)(C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(F)c1)C(F)(F)F
Cn1ccc([C@@H]2CCN(C(=O)c3cccn4cncc34)C[C@H]2NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)n1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)NC1CN(C(=O)c2cccn3cncc23)CCC1C1CC(F)(F)C1
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1C1CC(F)(F)C1
CC(CC#N)OC(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(F)c1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](NC(=O)C2(NC(=O)C(F)(F)F)CCOCC2)C1
Cc1nc([C@@H]2CCN(C(=O)c3cccn4cncc34)C[C@H]2NC(=O)[C@H](NC(=O)C(F)(F)F)C(C)C)cs1
O=C(N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cncc(F)c1)c1ncc[nH]1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](NC(=O)C2(NC(=O)C(F)(F)F)CCCC2)C1
CS(=O)(=O)N[C@@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)C(F)(F)F
CS(=O)(=O)N[C@@H](C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cccc(Cl)c1)C(F)(F)F
CS(=O)(=O)N[C@H]1CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)C1=O
C[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CS(=O)(=O)N[C@H]1CCN([C@@H]2CN(C(=O)c3cccn4cncc34)CC[C@H]2c2ccccc2)C1=O
C[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC(C)(NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC[C@@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
CC[C@H](NC(=O)C(F)(F)F)C(=O)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
O=C(c1cccn2cncc12)N1CC[C@@H](c2cc(F)cc(Cl)c2)[C@H](NC(=O)C2(NC(=O)C(F)(F)F)CCC2)C1
CNS(=O)(=O)c1cccc2[nH]c(C(=O)N[C@@H]3CN(C(=O)c4cccn5cncc45)CC[C@H]3c3ccccc3)cc12
O=C(CCC(F)(F)F)N[C@@H]1CN(C(=O)c2cccn3cncc23)CC[C@H]1c1cc(F)cc(Cl)c1
Cc1ccc(N2CC3CCC(C2)N3)cc1C(=O)NC1(c2cccc3cc(F)ccc23)CC1
Cc1ccc(N2CCNCC2)cc1C(=O)NC1(c2ccc(F)c3ccccc23)CC1
Cc1ccc(N2CC3CCC(C2)N3)cc1C(=O)NC1(c2ccc(F)c3ccccc23)CC1
Cc1ccc(N2CC3CCC(C2)N3C)cc1C(=O)NC1(c2cccc(-c3cccs3)c2)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3cc(F)ccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3cc(F)c(F)cc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(Cl)c3ccccc23)CC1
COc1ccc(C2(NC(=O)c3cc(N4CC(N(C)C)C4)ccc3C)CC2)c2ccccc12
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(Br)c3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(C)c3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(F)c3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3c(Cl)cccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3c(F)cccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2csc3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3c2CCCC3)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3occc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(F)c3ncccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cccc3ncccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccnc3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccnc3c(Cl)cccc23)CC1
COc1cccc2c(C3(NC(=O)c4cc(N5CC(N(C)C)C5)ccc4C)CC3)ccnc12
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(OC(F)(F)F)c3ncccc23)CC1
COc1ccc2c(C3(NC(=O)c4cc(N5CC(N(C)C)C5)ccc4C)CC3)ccc(F)c2n1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccnc3c(F)cccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(OC(F)F)c3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(OC(F)F)c3ncccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(C#N)c3ccccc23)CC1
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2cnc(O)c3ccccc23)CC1
COc1ncc(C2(NC(=O)c3cc(N4CC(N(C)C)C4)ccc3C)CC2)c2ccccc12
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(C)c3ncccc23)CC1
COc1ccc(C2(NC(=O)c3cc(N4CC(N(C)C)C4)ccc3C)CC2)c2cccnc12
Cc1ccc(N2CC(N(C)C)C2)cc1C(=O)NC1(c2ccc(N(C)C)c3ccccc23)CC1
Cc1ccc2c(C3(NC(=O)c4cc(N5CC(N(C)C)C5)ccc4C)CC3)ccc(F)c2n1
[2H]C1([2H])C(N(C)C)C([2H])([2H])N1c1ccc(C)c(C(=O)NC2(c3ccc(F)c4ncccc34)CC2)c1
CC(C)C[C@H](NC(=O)OC1CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OC1CCN(CC1)S(C)(=O)=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1(Cc2ccccc2)CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OC1(Cc2ccccc2)CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1(Cc2ccccc2)CCN(CC1)S(C)(=O)=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CCC1(CCN(CC1)C(=O)OC(C)(C)C)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CCC1(CCN(CC1)C(=O)OC(C)(C)C)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1CCN(CC1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1CCN(CC1)S(C)(=O)=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CCOC(=O)N1CCC(CC1)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CCOC(=O)N1CCC(CC1)OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OC1(Cc2ccccc2)CCN(CC1)S(C)(=O)=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)c2cc(C)on2)C(C)C)\C=C\C(=O)OCC)CCNC1=O
[H][C@@]1([#6]-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]\[#6]=[#6](\[#6])-[#6])-[#6]-[#6](=O)-[#6@@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#8])-[#7]-[#6](=O)-[#8]C([#6])([#6])[#6])-[#6](-[#6])-[#6])\[#6]=[#6]\[#6](=O)-[#8]-[#6]-[#6])[#6]-[#6]-[#7]-[#6]1=O
CCN1C(Sc2ccc(cc12)-c1nc2ccccc2s1)=C/C=C/c1sc2ccc(cc2[n+]1CC)-c1nc2ccccc2s1
CCN1\C(Sc2ccccc12)=C/C=C/C1=C/C(/CC(C)C1)=C/c1sc2ccccc2[n+]1CC |t:16|
CCN1\C(Sc2ccccc12)=C/C=c1\s\c(=C/c2sc3ccccc3[n+]2CC)n(CC)c1=O
CCN1C(SC(=C1c1ccccc1)c1ccccc1)=C/C=C/c1sc2c(ccc3ccccc23)[n+]1CC
CCN1\C(Sc2cc(C)c(C)cc12)=C/C(/CC)=C/c1sc2c(ccc3ccccc23)[n+]1CC
CCN1C(Sc2cc(C=Cc3ccccc3)ccc12)=C/C(/CC)=C/c1sc2cc(C)c(C)cc2[n+]1CC
CCN1\C(Sc2ccc(OC)cc12)=C/C(/OC)=C\c1sc2ccccc2[n+]1CCCS([O-])(=O)=O
C1CC(\C=C2\CC[n+]3c2sc2ccccc32)=C2Sc3ccccc3N12 |t:18|
CC(C)(C)OC(=O)Nc1ccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NCc2ccccc2)c(=O)c1 |r|
CC(C)C=CC(=O)c1cc(O)c2c(O)ccc(O)c2c1O |w:4.4|
Cn1nc(nc2c1cc(=O)n(C)c2=O)-c1ccc(cc1)C(F)(F)F
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)N[C@@H](CCC(=O)N(C)Cc1ccccc1)C(=O)C(F)(F)F |r|
CCN(CC)C(=O)CC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)C)C(=O)c1nccs1 |r|
C[C@@H]1C[C@@H]2[C@@](C)(CC[C@]3(C)C4=CC=c5c(cc(O)c(O)c5=C)[C@]4(C)CC[C@@]23C)CC1=O |r,c:12,t:10|
COc1cc(C=CC(=O)CC(=O)C=Cc2ccc(O)c(OC)c2)ccc1O |w:12.11,5.4|
C[C@]12CC[C@](C)(C[C@H]1[C@]1(C)CC[C@]3(C)C(=CC=c4c3cc(O)c(O)c4=C)[C@@]1(C)CC2)C(O)=O |r,c:15,17|
[H][C@@]12CCC(=C)[C@H](CC\C(C)=C/CO)[C@@]1(C)CCC[C@@]2(C)CO |r|
COc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)c(-c3cc(ccc3OC)-c3cc(O)c4c(cc(OC)cc4=O)o3)c2o1 |(10.61,-33.01,;9.27,-32.25,;7.94,-33.02,;7.94,-34.56,;6.61,-35.34,;5.28,-34.57,;5.27,-33.03,;6.6,-32.26,;3.95,-35.34,;3.95,-36.87,;2.63,-37.63,;2.63,-39.17,;1.31,-36.87,;-.03,-37.66,;-.03,-39.2,;-1.36,-36.89,;-1.36,-35.35,;-2.69,-34.58,;-.02,-34.58,;-.02,-33.04,;-1.36,-32.27,;-1.35,-30.73,;-.03,-29.96,;1.31,-30.73,;1.31,-32.27,;2.65,-33.04,;3.98,-32.27,;-2.68,-29.97,;-2.68,-28.42,;-4.03,-27.64,;-4.03,-26.1,;-5.36,-28.42,;-5.36,-29.97,;-6.7,-30.74,;-8.03,-29.97,;-9.37,-30.74,;-10.7,-29.97,;-8.03,-28.42,;-6.7,-27.64,;-6.7,-26.1,;-4.02,-30.74,;1.3,-35.35,;2.62,-34.57,)|
Oc1ccc(cc1)-c1cc(=O)c2c(O)cc(O)c(-c3cc(ccc3O)-c3cc(O)c4c(cc(O)cc4=O)o3)c2o1 |(13.25,-26.01,;14.59,-25.24,;14.59,-23.7,;15.92,-22.93,;17.26,-23.7,;17.26,-25.24,;15.93,-26.01,;18.58,-22.93,;19.91,-23.69,;21.23,-22.92,;22.57,-23.69,;21.22,-21.4,;22.56,-20.64,;23.88,-21.41,;22.55,-19.1,;21.22,-18.33,;21.22,-16.79,;19.9,-19.11,;18.57,-18.34,;17.23,-19.1,;15.9,-18.33,;15.9,-16.79,;17.23,-16.02,;18.57,-16.79,;19.91,-16.02,;14.57,-19.09,;14.56,-20.65,;13.21,-21.42,;13.21,-22.96,;11.87,-20.64,;11.88,-19.08,;10.54,-18.32,;9.21,-19.09,;7.87,-18.32,;9.21,-20.64,;10.54,-21.41,;10.54,-22.95,;13.22,-18.3,;19.9,-20.64,;18.58,-21.4,)|
COc1cc2oc(cc(O)c2c(=O)c1)-c1ccc(OC)c(c1)-c1c(O)cc(O)c2c1oc(cc2=O)-c1ccc(O)cc1 |(-8.64,-2.46,;-8.63,-4,;-7.29,-4.77,;-5.96,-3.99,;-4.63,-4.75,;-3.3,-3.96,;-1.95,-4.73,;-1.94,-6.28,;-3.28,-7.06,;-3.27,-8.6,;-4.61,-6.3,;-5.94,-7.06,;-5.93,-8.6,;-7.27,-6.31,;-.63,-3.95,;-.64,-2.41,;.68,-1.63,;2.03,-2.39,;3.35,-1.62,;3.34,-.08,;2.04,-3.94,;.71,-4.71,;3.37,-4.69,;3.38,-6.24,;2.05,-7.01,;4.72,-7,;6.05,-6.22,;7.39,-6.98,;6.04,-4.68,;4.7,-3.92,;4.68,-2.38,;6.02,-1.6,;7.36,-2.36,;7.36,-3.9,;8.7,-4.67,;6.02,-.06,;7.35,.72,;7.34,2.26,;6,3.02,;5.99,4.56,;4.67,2.23,;4.68,.7,)|
COc1ccc(cc1-c1c(O)cc(O)c2c1oc(cc2=O)-c1ccc(O)cc1)-c1cc(O)c2c(cc(O)cc2=O)o1 |(3.27,-31.58,;3.27,-33.11,;1.94,-33.89,;.61,-33.11,;-.73,-33.89,;-.73,-35.42,;.61,-36.2,;1.94,-35.42,;3.27,-36.2,;4.6,-35.42,;4.6,-33.89,;5.93,-36.2,;5.93,-37.73,;7.27,-38.51,;4.6,-38.51,;3.27,-37.73,;1.94,-38.51,;1.94,-40.04,;3.27,-40.81,;4.6,-40.04,;5.93,-40.81,;.61,-40.81,;.61,-42.35,;-.73,-43.12,;-2.06,-42.35,;-3.39,-43.12,;-2.06,-40.81,;-.73,-40.04,;-2.06,-36.2,;-2.06,-37.73,;-3.39,-38.51,;-3.39,-40.04,;-4.73,-37.73,;-4.73,-36.2,;-6.06,-35.42,;-7.39,-36.2,;-8.72,-35.42,;-7.39,-37.73,;-6.06,-38.51,;-6.06,-40.04,;-3.39,-35.42,)|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(Cl)cc2)cc1 |c:12|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(OC(F)(F)F)cc2)cc1 |c:12|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2cccc(Cl)c2)cc1 |c:12|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(F)cc2)cc1 |c:12|
COc1ccc(cc1)N1N=C(\C(=C\c2ccc(cc2)C(O)=O)C1=O)c1ccccc1 |c:10|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccccc2)cc1 |c:12|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2cccc(c2)[N+]([O-])=O)cc1 |c:12|
OC(=O)c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(Cl)c(Cl)c2)cc1 |c:12|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)c1cc(C)on1)C(C)C)C(=O)N[C@@H](CCC(N)=O)C#N |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCC(N)=O)C#N |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](CCC(N)=O)C#N |r|
Oc1cc(O)cc(Oc2c(O)cc(O)c3Oc4c(Oc23)c(O)cc2oc3c(Oc5cc(O)cc(O)c5)c(O)cc(O)c3c42)c1
Oc1cc(O)c(Oc2cc(O)c3Oc4cc(O)cc(O)c4Oc3c2Oc2cc(O)cc(O)c2)c(O)c1
c1c(cc(cc1O)O)O
Oc1cc(O)cc(Oc2c(O)cc(Oc3c(O)cc(O)cc3O)cc2O)c1
Oc1cc(O)c2oc3c(oc2c1)c(O)cc1oc2c(O)cc(O)cc2oc31
OCc1cc(O)c2C(=O)c3c(O)cccc3C(=O)c2c1
Oc1cc(O)c(Oc2cc(O)c3Oc4c(Oc5cc(O)cc(O)c5)c(O)cc(O)c4Oc3c2)c(O)c1
COc1ccc(cc1O)[C@@H]2CC(=O)c3c(cc(cc3O2)O)O
Oc1cc(O)c(Oc2cc(O)cc(O)c2Oc2cc(O)cc(O)c2-c2c(O)cc(O)cc2O)c(O)c1 |(18.25,-3.55,;19.59,-2.79,;20.91,-3.56,;22.25,-2.8,;23.58,-3.59,;22.27,-1.25,;23.6,-.49,;23.61,1.05,;22.28,1.82,;22.29,3.35,;20.95,4.13,;23.63,4.13,;24.96,3.35,;26.3,4.11,;24.95,1.81,;26.28,1.03,;27.62,1.79,;27.61,3.33,;28.94,4.11,;28.93,5.65,;30.28,3.36,;30.3,1.82,;31.64,1.07,;28.96,1.03,;28.98,-.51,;27.65,-1.29,;26.31,-.53,;27.66,-2.83,;29,-3.59,;29.02,-5.13,;30.33,-2.8,;30.32,-1.26,;31.64,-.48,;20.93,-.48,;20.93,1.06,;19.59,-1.24,)|
Oc1cc(O)cc(Oc2c(O)cc(O)c3Oc4cc(Oc5c(O)cc(Oc6c(O)cc(O)c7Oc8cc(O)cc(O)c8Oc67)cc5O)cc(O)c4Oc23)c1
Oc1cc(O)cc(Oc2c(O)cc(O)c3Oc4cc(O)cc(O)c4Oc23)c1
c1cc(ccc1C2=COc3cc(ccc3C2=O)O)O
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)OCc2ccccc2)C(=O)C(=O)NC(C)C)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)OCc2ccccc2)C=O)CCNC1=O |r|
Fc1ccc(cc1)N1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1
FC(F)(F)c1cccc(c1)N1CCN(CC1)S(=O)(=O)c1ccc2NC(=O)C(=O)c2c1
COc1ccc(cc1)C(=O)Cn1c(NCCO)nc2ccccc12
COc1ccc(cc1)N(CC(=O)NCc1ccco1)S(C)(=O)=O
Brc1cncc(c1)C(=O)N1CCN(Cc2ccsc2)CC1
Clc1cc(CSC(=S)NCc2cccnc2)c(Cl)s1
Nc1ccc(F)c(c1)S(=O)(=O)Nc1cccc(c1)C(F)(F)F
CCOc1ccc(cc1C)S(=O)(=O)NCc1ccc2OCOc2c1
OCCCc1nc2ccccc2n1CCOc1ccccc1
COCCOCCn1c(CCCO)nc2ccccc12
C(\C=C\c1ccccc1)[N+]1(C\C=C\c2ccccc2)CCN(CC1)C(c1ccccc1)c1ccccc1
CN(CC(=O)NC1CCCC1)S(=O)(=O)c1cccc(Cl)c1
COc1ccccc1CNC(=O)[C@H](C)NS(=O)(=O)c1ccccc1 |r|
CCCCC(CC)CNC(=N)NC(=N)NCCCCCCNC(=N)NC(=N)NCC(CC)CCCC
[#6]-n1c(-[#7]\[#7]=[#6]-2/[#6](=O)-[#7]-[#6](=O)-[#7]-[#6]-2=O)nc2n(-[#6])c(=O)n(-[#6])c(=O)c12
Cc1cc(C)n(c(=O)n1)S(=O)(=O)c1ccc(N)cc1
O=C(NC1=CC=CC2C1OC(=CC2=O)c1nn[nH]n1)c1ccc(OCCCCc2ccccc2)cc1 |c:5,11,t:3|
Nc1ccc(cn1)[N+]([O-])=O
c1cc(c2c(c1[N+](=O)[O-])non2)Cl
c1cc(c(cc1[N+](=O)[O-])O)O
c1ccnc(c1)NS(=O)(=O)c2ccc(cc2)/N=N/c3ccc(c(c3)C(=O)O)O
COCC(=O)\C=C1/Sc2ccccc2N1C
c1cc(c(cc1C=O)O)O
OC(=O)c1cc(\C=C\c2ccc(cc2)N2CCOCC2)nc2ccccc12
[O-][N+](=O)c1ccc(cc1)N1CCNCC1
Cc1ccc(C)c(CSc2nc(C3CCCCC3)c(C#N)c(=O)[nH]2)c1
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2)C(C)C)C(C)C |r,c:19|
CC(C)C[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2 |r,c:27|
CC[C@@H]1NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC3CC3)NC(=O)[C@@H](NC1=O)C(C)(C)C)C(N)=O)ccn2 |r,c:9|
C[C@@H](O)[C@@H]1NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC3CC3)NC(=O)[C@@H](NC1=O)[C@@H](C)O)C(N)=O)ccn2 |r,c:10|
CC(C)C[C@@H]1NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)C(C)C)C(C)C)C(N)=O)ccn2 |r,c:20|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2)C(C)C |r,c:15|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2)C(C)C |r,c:25|
CC[C@@H]1NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC3CC3)NC(=O)[C@@H](NC1=O)C(C)(C)C)C(N)=O)ccn2 |r,c:14|
CC[C@@H]1NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC3CC3)NC(=O)[C@@H](NC1=O)C(C)(C)C)C(N)=O)ccn2 |r,c:9|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2)C(C)C |r,c:25|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2)C(C)C |r,c:25|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCC(O)=O)NC1=O)C(N)=O)ccn2)C(C)C)C(C)C |r,c:19|
CC(C)C[C@@H]1NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCC(O)=O)NC1=O)C(N)=O)ccn2 |r,c:27|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC1=O)C(N)=O)ccn2)C(C)C |r,c:25|
NCCCC[C@@H]1NC(=O)[C@H](CO)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC1=O)C(N)=O)ccn2 |r,c:39|
CC(C)C[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]2CSC(=N2)c2cc(C[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](Cc3ccccc3)NC(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CCC(N)=O)NC1=O)C(N)=O)ccn2)[C@@H](C)O)C(C)C |r,c:30|
CC[C@@H]1NC(=O)[C@@H](N)CCNC(=O)[C@@H]2CSC(=N2)c2cccc(n2)C2=N[C@@H](CS2)C(=O)NCCCC[C@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC1=O)C(C)(C)C)C(N)=O |r,c:16,t:26|
CC[C@H](N)C(=O)N[C@H](C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccnc(c1)C#N)C(N)=O)C(C)(C)C |r|
CC[C@H](NC(C)=O)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(N)=O)C(C)(C)C |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@@H]1CSCN1)C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccnc(c1)C#N)C(N)=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(C)=O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CO)C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccccc1)C(N)=O |r|
Oc1ccccc1\C=N\NC(=N)c1nonc1NCNc1nonc1C(=N)N\N=C\c1ccccc1O
COc1cc(ccc1O)C(NC1=NC(=O)C(CC(=O)Nc2ccc(cc2)C(O)=O)S1)c1c(O)[nH]c(=O)[nH]c1=O |t:12|
Cn1cc(SCC(=O)NCc2ccccc2)c2ccccc12
Cn1cc(SCC(=O)N(Cc2ccccc2)Cc2ccccc2)c2ccccc12
CN(C)CCOc1ccc(CNC(=O)CSc2cn(C)c3ccccc23)cc1
COc1ccccc1CNC(=O)CSc1cn(C)c2ccccc12
Cn1cc(SCC(=O)NCc2ccc(Cl)c(Cl)c2)c2ccccc12
O=C(CSc1c[nH]c2ccccc12)NCc1ccccc1
FC(F)(F)c1ccc(CNC(=O)CSc2c[nH]c3ccccc23)cc1
CN(C)CCOc1ccc(CNC(=O)CSc2c[nH]c3ccccc23)cc1
COc1ccccc1CN(C)C(=O)CSc1c[nH]c2ccccc12
C[C@@H](NC(=O)CSc1c[nH]c2ccccc12)c1ccccc1 |r|
COc1ccccc1CNC(=O)CSc1c[nH]c2cccc(Br)c12
Clc1ccc(CNC(=O)CSc2c[nH]c3cccc(Br)c23)cc1Cl
COc1ccccc1CNC(=O)CSc1c[nH]c2ccc(Br)cc12
Clc1ccc(CNC(=O)CSc2c[nH]c3ccc(Br)cc23)cc1Cl
COc1ccccc1CNC(=O)CSc1c[nH]c2cc(Br)ccc12
Clc1ccc(CNC(=O)CSc2c[nH]c3cc(Br)ccc23)cc1Cl
COc1ccccc1CNC(=O)CSc1c[nH]c2c(Br)cccc12
Clc1ccc(CNC(=O)CSc2c[nH]c3c(Br)cccc23)cc1Cl
CN(Cc1ccccc1)C(=O)CSc1c[nH]c2cccc(Br)c12
CN(Cc1ccccc1)C(=O)CSc1c[nH]c2c(Br)cccc12
Brc1cccc2c(SCC(=O)N(Cc3ccccc3)Cc3ccccc3)c[nH]c12
O=C(CSc1c[nH]c2ccccc12)N(Cc1ccccc1)Cc1ccccc1
CN(Cc1ccccc1)C(=O)CSc1c[nH]c2ccccc12
COc1ccccc1CNC(=O)CSc1c[nH]c2c(cccc12)-c1ccccc1
Brc1cccc2[nH]cc(SCC(=O)N(Cc3ccccc3)Cc3ccccc3)c12
CCOc1ccccc1CN(OC)C(=O)CSc1c[nH]c2cccc(Br)c12
[H][C@@]1(C[C@@H](NC(=O)[C@@H](CC2CCCCC2)n2cccc(NC(=O)OC(C)(C)C)c2=O)C(=O)C(=O)NC2CC2)CCNC1=O |r|
[H][C@@]1(C[C@@H](NC(=O)[C@@H](CC2CCCCC2)NC(=O)\C=C\c2ccccc2)C(=O)C(=O)NCc2ccccc2)CCNC1=O |r|
[H][C@@]1(C[C@@H](NC(=O)[C@@H](CC2CC2)n2cccc(NC(=O)OC(C)(C)C)c2=O)C(=O)C(=O)NCc2ccccc2)CCNC1=O |r|
CSCC[C@@H](NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(C)=O)C=O |r|
CCC[C@@H](NC(=O)[C@@H](CC(C)C)NC(=O)OCc1ccccc1)C(=O)C(=O)NCc1ccccn1 |r|
[H][C@@]1(C[C@@H](NC(=O)[C@@H](CC2CCCCC2)NC(=O)c2cc3ccccc3[nH]2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@@H](NC(=O)[C@@H](Cc2cccc(F)c2)NC(=O)c2cc3ccccc3[nH]2)C=O)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](CCCC)C(=O)C(=O)NC3CC3)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC1(CS(=O)(=O)C(C)(C)C)CCCCC1)C(C)(C)C |r|
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NS(=O)(=O)c1ccc(F)cc1)C(C)C)C=O |r|
[#6]-[#7](-[#6])-[#6](=O)-[#6]-[#8]-[#6](=O)-[#6]-c1ccc(-[#8]-[#6](=O)-c2ccc(cc2)\[#7]=[#6](\[#7])-[#7])cc1
CC(C)[C@H](NC(=O)N(C)Cc1csc(n1)C(C)C)C(=O)N[C@H](C[C@H](O)[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 |r|
C[C@H](NC(=O)c1cc(N)ccc1C)c1cccc2ccccc12 |r|
C[C@H](NC(=O)c1cc(NC(C)=O)ccc1C)c1cccc2ccccc12 |r|
COc1ccc(cc1)-c1cc(=O)c2c(O)c(OC)c(O[C@@H]3O[C@H](CO[C@@H]4O[C@@H](C)[C@H](O)[C@@H](O)[C@H]4O)[C@@H](O)[C@H](O)[C@H]3O)cc2o1 |r|
C[C@@H]1O[C@@H](O[C@H]2[C@H](Oc3cc(O)c4c(c3)oc(cc4=O)-c3ccc(O)cc3)O[C@H](CO)[C@@H](O)[C@@H]2O)[C@H](O)[C@H](O)[C@H]1O |r|
c1cc(ccc1C2=C(C(=O)c3c(cc(c(c3O2)O)O)O)O)O
Oc1ccc(CC\C=C\C(=O)CCc2ccc(O)c(O)c2)cc1O
[H][C@]12CCC(=C)[C@@H](C\C=C3/[C@H](O)COC3=O)[C@]1(C)CC[C@@H](O)[C@@]2(C)CO |r|
O=C(NCc1ccco1)C1CN(CCN1)C(=O)c1cc(=O)[nH]c(=O)[nH]1
c1cc(cnc1)C(=O)N2CCN([C@@H](C2)C(=O)NCc3cccs3)c4ccc(c(c4)Cl)Cl
c1cc(c(cc1N2CCN(CC2)C(=O)C3=CC(=O)NC(=O)N3)Cl)Cl
Clc1ccc(CN2CCN(C[C@H]2C(=O)NCc2cccs2)C(=O)c2cc(=O)[nH]c(=O)[nH]2)c(Cl)c1 |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1cccs1)C(=O)c1cncc2ccccc12 |r|
Clc1ccc(cc1Cl)N1CCN(CC1C(=O)NCc1ccco1)C(=O)c1cc(=O)[nH]c(=O)[nH]1
c1cc(sc1)CNC(=O)[C@@H]2CN(CCN2c3ccc(c(c3)Cl)Cl)C(=O)C4=CC(=O)NC(=O)N4
Clc1ccc(cc1Cl)N1CCN(C[C@@H]1C(=O)NCc1ccco1)C(=O)c1cc(=O)[nH]c(=O)[nH]1 |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1ccco1)C(=O)c1cc(=O)[nH]c(=O)[nH]1 |r|
c1cc(sc1)CNC(=O)[C@@H]2CN(CCN2c3ccc(c(c3)Cl)Cl)C(=O)C4=CC(=O)NC(=O)N4
Clc1ccc(CN2CCN(CC2C(=O)NCc2ccco2)C(=O)c2cc(=O)[nH]c(=O)[nH]2)c(Cl)c1
Clc1ccc(CN2CCN(C[C@H]2C(=O)NCc2ccco2)C(=O)c2cc(=O)[nH]c(=O)[nH]2)c(Cl)c1 |r|
c1ccc(c(c1)COc2cc(cc(c2)Cl)C3=CC(=CN(C3=O)c4cccnc4)C5=CNC(=O)NC5=O)Cl
C[C@H](NC(=O)[C@H](N(C(=O)CCl)c1ccc(cc1)-n1cccc1)c1cccnc1)c1ccccc1 |r|
CCS(=O)(=O)N1CCC(CC1)[C@@H](C)n1c(C)c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c2ccccc12 |r|
C[C@@H](NC(=O)c1cc(NC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC[C@H]2CCCO2)s1 |r|
CCCCC(=O)Nc1ccc(C)c(c1)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
Cc1ccc(cc1C(=O)N[C@H](C)c2cccc3c2cccc3)NC(=O)C=C
Cc1ccc(cc1C(=O)N[C@H](C)c2cccc3c2cccc3)NC(=O)NC(=O)N
C[C@@H](NC(=O)c1cc(NC(=O)Oc2ccc(cc2)[N+]([O-])=O)ccc1C)c1cccc2ccccc12 |r|
CCCCNC(=O)Nc1ccc(C)c(c1)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
Nc1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc2ccccc12
C[C@@H](NC(=O)c1ccc(N)cc1C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1cc(ccc1C)N(C)C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1ccc(NS(C)(=O)=O)cc1C)c1cccc2ccccc12 |r|
C[C@@H](N1Cc2ccccc2C1)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1ccccc1Cl)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1sccc1C)c1cccc2ccccc12 |r|
CC(N(C)Cc1cc(O)ccc1Cl)c1ccccc1Cl
C[C@@H](N(C)Cc1cc(O)ccc1Cl)c1ccccc1C |r|
C[C@@H](N(C)Cc1cccc2[nH]ccc12)c1cccc2ccccc12 |r|
C[C@@H](N(C)Cc1ccc2[nH]ncc2c1)c1cccc2ccccc12 |r|
C[C@H](c1cccc2c1cccc2)N(C)Cc3c[nH]c4c3cccc4
C[C@@H](N(C)Cc1cc(O)ccc1C)c1cccc2ccccc12 |r|
C[C@@H](N(C)Cc1ccc(O)cc1C)c1cccc2ccccc12 |r|
C[C@@H](N(C)Cc1ccc(O)cc1Cl)c1cccc2ccccc12 |r|
COc1cc(O)ccc1CN(C)[C@H](C)c1cccc2ccccc12 |r|
C[C@@H](N(C)Cc1cc(N)ccc1C)c1cccc2ccccc12 |r|
C[C@H](c1cccc2c1cccc2)N(C)Cc3ccc(cc3)O
C[C@H](N(C)Cc1ccc(O)cc1)c1cccc2ccccc12 |r|
C[C@H](c1cccc2c1cccc2)N3CCC(CC3)C(=O)NCc4cccc(c4)F
C[C@H](c1cccc2c1cccc2)N3CCC(CC3)C(=O)NCc4cccc(c4)NC(=O)C
COc1cc(CNC(=O)C2CCN(CC2)[C@H](C)c2cccc3ccccc23)ccn1 |r|
C[C@@H](N1CCC(CC1)C(=O)NCc1cc(F)cc(NC(C)=O)c1)c1cccc2ccccc12 |r|
C[C@@H](N1CCC(CC1)C(=O)NCC1CCN(C)CC1)c1cccc2ccccc12 |r|
C[C@@H](N1CCC(CC1)C(=O)NCc1cccc(NC(=O)CN(C)C)c1)c1cccc2ccccc12 |r|
C[C@@H](N1CCC(CC1)C(=O)NCc1cccc(NC(=O)N2CCN(C)CC2)c1)c1cccc2ccccc12 |r|
C[C@@H](N1CCC(CC1)C(=O)NCc1cc(F)cc(NC(=O)CN(C)C)c1)c1cccc2ccccc12 |r|
C[C@@H](N1CCC(CC1)C(=O)NCc1cc(F)cc(NC(=O)N2CCN(C)CC2)c1)c1cccc2ccccc12 |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H](CC2CC2)n2cccc(NC(=O)OC(C)(C)C)c2=O)C(=O)C(=O)NCc2ccccc2)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C(CC2CC2)n2cccc(NC(=O)OC(C)(C)C)c2=O)C(=O)C(=O)NCc2ccccc2)CCNC1=O |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)[C@H](F)Cl |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)[C@H](F)Cl |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)[C@@H](F)Cl |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)NN(C[C@H]1CCNC1=O)C(=O)[C@H](F)Cl |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)NN(C[C@H]1CCNC1=O)C(=O)[C@H](F)Cl |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)NN(C[C@H]1CCNC1=O)C(=O)[C@@H](F)Cl |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)NN(C[C@@H]1CCNC1=O)C(C)=O |r|
Clc1ccc2n(Cc3ccccc3)c(SCC(=O)N3CCNC3=O)nc2c1
Clc1ccc2n(Cc3ccccc3)c(SCC(=O)N3CCOC3=O)nc2c1
CC(C)(C)c1ccc2n(Cc3ccccc3)c(SCC(=O)N3CCOC3=O)nc2c1
Clc1ccc2n(Cc3ccccc3)c(SC(Cc3ccccc3)C(=O)N3CCNC3=O)nc2c1
Cc1ccc2n(Cc3ccccc3)c(SC(Cc3ccccc3)C(=O)N3CCNC3=O)nc2c1
Clc1ccc2n(Cc3ccccc3)c(SC(Cc3ccccc3)C(=O)N3CCOC3=O)nc2c1
Cc1ccc2n(Cc3ccccc3)c(SC(Cc3ccccc3)C(=O)N3CCOC3=O)nc2c1
CC(C)(C)c1ccc2n(Cc3ccccc3)c(SC(Cc3ccccc3)C(=O)N3CCOC3=O)nc2c1
Clc1ccc2n(Cc3ccccc3)c(SC(Cc3ccco3)C(=O)N3CCOC3=O)nc2c1
Clc1ccc2nc(SC(Cc3ccco3)C(=O)N3CCOC3=O)n(Cc3ccccc3)c2c1
COc1ccc2nc(SC(Cc3ccco3)C(=O)N3CCOC3=O)n(Cc3ccccc3)c2c1
Oc1ccc2nc(SC(Cc3ccco3)C(=O)N3CCOC3=O)n(Cc3ccccc3)c2c1
Clc1cc2nc(SCC(=O)N3CCOC3=O)n(Cc3ccccc3)c2cc1Cl
COc1cc2n(Cc3ccccc3)c(SCC(=O)N3CCOC3=O)nc2cc1Cl
Oc1cc2n(Cc3ccccc3)c(SCC(=O)N3CCOC3=O)nc2cc1Cl
Clc1cc2nc(SC(Cc3ccco3)C(=O)N3CCOC3=O)n(Cc3ccccc3)c2cc1Cl
COc1cc2n(Cc3ccccc3)c(SC(Cc3ccco3)C(=O)N3CCOC3=O)nc2cc1Cl
Oc1cc2n(Cc3ccccc3)c(SC(Cc3ccco3)C(=O)N3CCOC3=O)nc2cc1Cl
COCCn1c(nc2ccccc2c1=O)C(=O)NCC(O)c1ccccc1
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(C)=C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccco1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1ccccc1)C1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@](C)(NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)C[C@H](NC(=O)C(C)(C)NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)C1(CC1)NC(=O)OCc1ccccc1 |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)[C@@H](NC(=O)OCc1ccccc1)C1CC1 |r|
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cccc(Cl)c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OCc1cccc(Cl)c1)[C@@H](C)OC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OCc1cccc(Cl)c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)NC(=O)[C@H](C(C)C)NC(=O)c2cc3ccccc3[nH]2
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
CC1([C@@H]2[C@H]1[C@H](N(C2)C(=O)[C@H](C(C)(C)C)NC(=O)NC(C)(C)C)C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)C
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(=O)NC3CC3)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(=O)NCC3CC3)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(=O)NCC)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(=O)NCCCC)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(=O)NCCCCCC)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(C)(C)C |r|
CC(C)(C)C[C@H](NC(=O)[C@@H](NC(=O)NC(C)(C)C)C(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)(C)NC(=O)N[C@H](C(=O)N[C@@H](CC1CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)CC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)C(N)=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)CC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)CC(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)OCc1ccccc1)C(C)(C)C |r|
C[C@@H](OC(C)(C)C)[C@H](NC(=O)NC(C)(C)C)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)OC(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)CC(C)(C)C)C(C)(C)C |r|
NC(=N)Nc1ccc2COB(O)c2c1
NC(=N)Nc1ccc(cc1)C(=O)Nc1ccc2COB(O)c2c1
OB1OCc2ccc(NC(=O)c3cccc(OCc4ccccc4)c3)cc12
OB1OCc2ccc(NC(=O)c3cccc(NCc4ccccc4)c3)cc12
OB1OCc2ccc(NC(=O)c3cccc(NC(=O)c4ccccc4)c3)cc12
OB1OCc2ccc(NC(=O)c3cccc(OCc4ccccc4)n3)cc12
Cc1cccc(COc2cccc(c2)C(=O)Nc2ccc3COB(O)c3c2)c1
[#6]\[#6](-[#6])=[#6]\[#6]-c1cc(\[#6]=[#6]-2/[#8]-[#6](=O)-[#6](=[#6]-2-[#8])-c2cc3-[#6]-[#6]C([#6])([#6])[#8]-c3cc2-[#8])ccc1-[#8] |c:13|
CC(C)(O)C1Cc2cc(\C=C3/OC(=O)C(=C3O)c3cc4CC(O)C(C)(C)Oc4cc3O)ccc2O1 |c:14|
[#6]\[#6](-[#6])=[#6]\[#6]-c1cc(\[#6]=[#6]-2/[#8]-[#6](=O)-[#6](=[#6]-2-[#8])-c2cc(-[#6]-[#6]C([#6])([#6])[#8])c(-[#8])cc2-[#8])ccc1-[#8] |c:13|
[#6]\[#6](-[#6])=[#6]\[#6]-[#6]\[#6](-[#6])=[#6]\[#6]-[#6][C@@]1([#6])[#8]-c2c(-[#8])c(-[#6])c(-[#8])c(-[#6]=O)c2-[#6]=[#6]1 |r,c:26|
Cn1cnc(Cn2c(=O)nc(Nc3cc4c(F)n(C)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
CCn1cc2cc(Nc3nc(=O)n(Cc4ncn(C)n4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(CC(F)F)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(Cl)c(F)cc3F)c2=O)n1
Cn1cnc(Cn2c(=O)nc(NC3=CC4CCOC4C=C3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)n1 |c:20,t:12|
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(Cl)c(F)c(Cl)c3)c2=O)n1
Cn1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cccc4ccccc34)c2=O)n1
Cn1cc2cc(Nc3nc(=O)n(Cc4cc5ccsc5[nH]c4=O)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
Cc1cncc(c1)-n1c(=O)nc(Nc2cc3cn(C)nc3cc2Cl)n(Cc2cc(C#N)c(F)cc2C)c1=O
Cn1cc2cc(Nc3nc(=O)n(-c4cncc5COCc45)c(=O)n3Cc3cc(Cl)c(F)cc3F)c(Cl)cc2n1 |(-6.65,4.87,;-5.88,3.54,;-4.34,3.37,;-4.02,1.87,;-2.69,1.1,;-2.69,-.44,;-1.36,-1.21,;-.02,-.44,;-.02,1.1,;1.31,1.87,;1.31,3.41,;2.64,1.1,;3.98,1.87,;5.32,1.1,;6.65,1.87,;6.64,3.4,;5.31,4.18,;4.99,5.68,;3.46,5.84,;2.84,4.44,;3.98,3.41,;2.64,-.44,;3.98,-1.21,;1.31,-1.21,;1.31,-2.75,;2.64,-3.52,;3.98,-2.75,;5.31,-3.52,;6.64,-2.75,;5.31,-5.06,;6.64,-5.83,;3.98,-5.83,;2.64,-5.07,;1.31,-5.84,;-4.02,-1.21,;-4.02,-2.75,;-5.36,-.44,;-5.36,1.1,;-6.5,2.13,)|
Cn1cc2cc(Nc3nc(=O)n(-c4cncc(c4)C(F)(F)F)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
Cn1cc2cc(Nc3nc(=O)n(Cc4cc(Cl)ccn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
CCNC(=O)Cn1c(=O)nc(Nc2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)c(F)c2)c1=O
Cc1cnc(Cn2c(=O)nc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)nc1
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1cc2c3OCCc3ccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
CC(C)C[C@H](NC(=O)c1cc2c(OC(F)(F)F)cccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
CCOc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cc(Cl)cc2[nH]c(cc12)C(=O)N[C@@H](CC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COc1cc(Cl)cc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C#N |r|
COC1C[Se]c2ccc3cc(ccc3[n+]12)C#C
[O-][N+](=O)c1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1
Brc1ccc2[nH]c-3c(CC(=O)Nc4ccccc-34)c2c1
[H][C@]12CCC(=C)[C@@H](C\C=C(/C)[C@@H]3CCc4c(O)c(CC5C(O)C(C)(C)C(O)=C(C(C)=O)C5=O)c(O)c(C(=O)CCC)c4O3)[C@]1(C)CCC[C@]2(C)C(O)=O |r,t:26|
[H][C@]12CCC(=C)[C@@H](C\C=C(/C)[C@H]3CCc4c(O)c(CC5C(O)C(C)(C)C(O)=C(C(C)=O)C5=O)c(O)c(C(=O)CCC)c4O3)[C@]1(C)CCC[C@]2(C)C(O)=O |r,t:26|
CCCOc1ccc(cc1)-c1cc(OCCN2CCN(Cc3ccccc3)CC2)c2c(OC)cc(OC)cc2n1
CCCOc1ccc(cc1)-c1cc(OCCN2CCc3cc(OC)c(OC)cc3C2)c2c(OC)cc(OC)cc2n1
CCCOc1ccc(cc1)-c1cc(OCCN2CCCCC2)c2c(OC)ccc(OC)c2n1
CCCOc1ccc(cc1)-c1cc(OCCN2CCCC2)c2cc(OC)cc(OC)c2n1
[O-][N+](=O)c1ccccc1SCc1nnc(S)n1CC=C
CC(C)C[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)NN(CCC(N)=O)C(=O)CCl |r|
O=C(Sc1nncs1)c1cc2ccccc2[nH]1
Cc1nnc(SC(=O)c2cc3ccccc3[nH]2)s1
Cc1nnc(SC(=O)c2cccc3[nH]ccc23)s1
Cc1nnc(SC(=O)c2ccc3[nH]ccc3c2)s1
Cc1nnc(SC(=O)c2ccc3cc[nH]c3c2)s1
Cc1nnc(SC(=O)c2cccc3cc[nH]c23)s1
Cc1nnc(SC(=O)c2cc3ccccc3n2C)s1
CSc1nnc(SC(=O)c2cc3ccccc3[nH]2)s1
COc1nnc(SC(=O)c2cc3ccccc3[nH]2)s1
Cc1nnc(SC(=O)c2cc3ccccc3[nH]2)o1
Cc1nnc(SC(=O)c2cc3ccccc3[nH]2)n1C(=O)c1cc2ccccc2[nH]1
Cc1nnc(SC(=O)c2cc3ccccc3o2)s1
Cc1nnc(SC(=O)c2ccc(Br)o2)s1
Cc1nnc(SC(=O)c2ccc(o2)-c2ccccc2)s1
Cc1nnc(SC(=O)c2ccc(o2)C#Cc2ccccc2)s1
Cc1nnc(SC(=O)c2ccc([nH]2)-c2ccccc2)s1
Cc1nnc(SC(=O)c2ccc3ccccc3c2)s1
O=C(Sc1ncccn1)c1cc2ccccc2[nH]1
Cc1ccnc(SC(=O)c2cc3ccccc3[nH]2)n1
Cc1cc(C)nc(SC(=O)c2cc3ccccc3[nH]2)n1
O=C(Sc1ncccn1)c1ccc(o1)-c1ccccc1
Cc1cc(C)nc(SC(=O)c2ccc(o2)C#Cc2ccccc2)n1
O=C(Sc1ncccn1)c1cc2ccccc2s1
O=C(Sc1ncccn1)c1ccc(s1)-c1ccccc1
Brc1ccc(cc1)-c1ccc(s1)C(=O)Sc1ncccn1
O=C(Sc1ncccn1)c1ccc2ccccc2n1
COc1ccc2cc(ccc2c1)[C@H](C)C(=O)Sc1ncccn1 |r|
O=C(Sc1nc2ccccc2s1)c1cc2ccccc2[nH]1
O=C(Sc1nc2ccccc2s1)c1ccc(o1)-c1ccccc1
Brc1ccc(cc1)-c1ccc(o1)C(=O)Sc1nc2ccccc2s1
O=C(Sc1nc2ccccc2s1)c1cc2ccccc2s1
O=C(Sc1nc2ccccc2s1)c1ccc(s1)-c1ccccc1
O=C(Sc1nc2ccccc2s1)c1ccc2ccccc2n1
Oc1ccc2ccccc2c1SSc1c(O)ccc2ccccc12
O=C(NCCN1C(=O)C=CC1=O)c1cc2ccccc2[nH]1 |c:8|
S=C(SSC(=S)N1CCOCC1)N1CCOCC1
Nc1cccn([C@@H](CC2CC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NCc2ccccc2)c1=O |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)c1cc2ccccc2[nH]1 |r|
CC(=O)N[C@@H](CCc1nc2ccccc2s1)C(=O)N[C@@H](CN)C(=O)NCC(=O)NC\C=C\C(O)=O |r|
CC(=O)N[C@@H](CCc1ccc(O)cc1)C(=O)N[C@@H](CN)C(=O)NCC(=O)NC\C=C\C(O)=O |r|
O=C1c2ccccc2-c2nc3nnnn3nc12
Cc1cc2nc3c(nc(=O)[nH]c3=O)n(C)c2cc1C=O
Cc1nc2c(s1)C(=O)C=C(Nc1ccc(C)cc1)C2=O |t:9|
C[C@@H](N(C)Cc1cc(O)ccc1Cl)c1ccccc1Cl |r|
COc1cc(CNC(=O)C2CCN(CC2)C(C)c2cccc3ccccc23)ccn1
COC(=O)c1ccc(c(c1)O)O
c1cc(ccc1CCO)O
c1cc(ccc1C=O)O
Nc1nc2nc[nH]c2c(=S)[nH]1
O=C1c2nc(oc2C(=O)c2ccccc12)-c1ccccc1
COCC[n+]1c(C)n(Cc2cnccn2)c2c1C(=O)c1ccccc1C2=O
Cc1c2c(oc1S([O-])(=O)=O)-c1ccc3c(CCCC3(C)C)c1C(=O)C2=O
Oc1c(Cl)cc(Cl)c2cccnc12
CC1(C)OC2=C(C1n1cc(nn1)-c1ccccc1)C(=O)C(=O)c1ccccc21 |c:4|
CN(Cc1cn(nn1)C1C2=C(OC1(C)C)c1ccccc1C(=O)C2=O)C1=CC(=O)c2ccccc2C1=O |c:10,t:29|
CN(Cc1cn(nn1)C1C2=C(OC1(C)C)c1ccccc1C(=O)C2=O)C1=C(Br)C(=O)c2ccccc2C1=O |c:10,29|
[H][C@]1(O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@@]1([H])c2cccc(O)c2C(=O)c2c(O)cc(CO)cc12
[H][C@]1(O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@]1([H])c2cccc(O)c2C(=O)c2c(O)cc(CO)cc12 |r|
COC(=O)\C=C\C(=O)NNC(=O)CCc1ccccc1C(=O)N[C@H](C)c1cccc2ccccc12 |r|
COC(=O)\C=C\C(=O)NNC(=O)CCc1ccc(NC(C)=O)cc1C(=O)N[C@H](C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1ccccc1CCC(=O)NNC(=O)C#C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1ccccc1CCC(=O)NNC(=O)CCl)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1ccccc1CCC(=O)NNC(=O)CC#N)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)c1ccccc1CCC(=O)NNC(=O)C(=C\C1CC1)\C#N)c1cccc2ccccc12 |r|
Brc1ccccc1-n1[se]c2ccccc2c1=O
Oc1cccnc1-n1[se]c2ccccc2c1=O
[O-][N+](=O)c1ccc(cc1)-n1[se]c2ccccc2c1=O
COc1ccc(c(OC)c1)-n1[se]c2ccccc2c1=O
Fc1ccc(Cl)cc1-n1[se]c2ccccc2c1=O
Cc1ccc(Cl)cc1-n1[se]c2ccccc2c1=O
Cc1c(Cl)cccc1-n1[se]c2ccccc2c1=O
C#CC[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)NC(=O)/C=C/c2ccccc2
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)NC(=O)/C=C/c2ccccc2
CCCC[C@@H](C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)NC(=O)/C=C/c2ccccc2
CCCC[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)/C=C/c2ccccc2
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)[C@H](C(C)C)NC(=O)c2ccc3ccccc3c2
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)[C@H](C(C)C)NC(=O)c2ccc(cc2)[N+](=O)[O-]
O=C[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@H](CC1CC1)NC(=O)\C=C\c1ccccc1 |r|
CC(C)C[C@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
C[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c2ccccc2)C(C)C)C=O)CCCNC1=O |r|
CC(C)(C)[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
O=C[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@@H](NC(=O)\C=C\c1ccccc1)c1ccccc1 |r|
C=CC[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
O=C[C@H](C[C@@H]1CCCNC1=O)NC(=O)[C@H](CC#C)NC(=O)\C=C\c1ccccc1 |r|
CCC[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC[C@H](C)[C@H](NC(=O)\C=C\c1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccc(C)cc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccc(cc1)C(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccc(cc1)-c1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)[C@H](C(C)C)NC(=O)/C=C/c2ccc(cc2)OC
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccc(cc1)N(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccc(F)cc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1ccccc1F)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)\C=C\c1cccc(F)c1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1cc2ccccc2[nH]1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc2cc[nH]c2c1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)CCc1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc(cc1)-c1ccccc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)[C@H](C(C)C)NC(=O)C2CCCCC2
CC(C)C[C@@H](C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O)NC(=O)[C@H](C(C)C)NC(=O)c2ccco2
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccoc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc[nH]1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccncc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1cccnc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccccn1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc(F)cc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc(Cl)cc1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc(cc1)C(F)(F)F)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)C1CCOCC1)C(C)C)C(=O)N[C@@H](C[C@@H]1CCCNC1=O)C=O |r|
Nc1nonc1-c1nc2ccccc2n1CC(=O)N\N=C\c1ccc(o1)-c1cccc(c1)C(O)=O
Cc1cc(c(cc1Cl)-c1ccc(\C=N\NC(=O)c2nonc2N)o1)[N+]([O-])=O
Cc1cc(-c2ccc(\C=N\NC(=O)Cn3nnnc3N)o2)c(cc1C)[N+]([O-])=O
Cc1c(NC(=S)N\N=C\c2ccc(o2)-c2ccc(cc2)[N+]([O-])=O)c(=O)n(-c2ccccc2)n1C
NC(=S)N\N=C\c1ccc(o1)-c1cccc(c1)[N+]([O-])=O
NC(=S)N\N=C\c1ccc(o1)-c1ccc(cc1)[N+]([O-])=O
NC(=S)N\N=C\c1ccc(o1)-c1cccc(c1)C(O)=O
NC(=S)N\N=C\c1ccc(o1)-c1ccc(cc1)C(O)=O
NC(=S)N\N=C\c1ccc(o1)-c1ccc(O)c(c1)C(O)=O
NC(=S)N\N=C\c1ccc(o1)-c1ccc(O)c(c1)C#N
COc1ccc(cc1OC)-c1ccc(\C=N\NC(N)=S)o1
NC(=S)N\N=C\c1ccc(o1)-c1ccncc1
NC(=S)N\N=C\c1ccc(o1)-c1ccc(F)nc1
NC(=S)N\N=C\c1ccc(o1)-c1ccc2cccnc2c1
NC(=S)N\N=C\c1ccc(o1)-c1cnc2ccccc2c1
NC(=S)N\N=C\c1ccc(Cc2ccccc2)o1
NC(=S)N\N=C\c1ccc(o1)-c1ccc(cc1)C(N)=O
NC(=S)N\N=C\c1ccc(o1)-c1ccc(cc1)S(N)(=O)=O
NC(=S)N\N=C\c1ccc(o1)-c1ccccc1
NC(=S)N\N=C\c1ccc(o1)-c1ccc(cc1F)C(O)=O
Cc1cc(ccc1-c1ccc(\C=N\NC(N)=S)o1)C(O)=O
NC(=S)N\N=C\c1ccc(o1)-c1ccc(C(O)=O)c(O)c1
NC(=S)N\N=C\c1ccc(o1)-c1ccc(C(O)=O)c(Cl)c1
NC(=S)N\N=C\c1ccc(o1)-c1cccc(C(O)=O)c1Cl
NC(=S)N\N=C\c1ccc(o1)-c1ccc(Cl)c(c1)C(O)=O
NC(=S)N\N=C\c1ccc(o1)-c1cc(ccc1Cl)C(O)=O
NC(=S)N\N=C\c1cc(co1)-c1ccc(cc1)C(O)=O
NC(=S)N\N=C\c1ccc(s1)-c1ccc(cc1)C(O)=O
NC(=S)N\N=C\c1cccc(c1)-c1ccc(cc1)C(O)=O
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CC2)NC(=O)n2cccc(NC(=O)OC(C)(C)C)c2=O)C(=O)C(=O)NCc2ccccc2)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@]3([H])CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)COc1ccc(OC(F)(F)F)cc1 |r|
Cc1ccc(cc1Nc2nc(cs2)c3cccnc3)NC(=O)c4ccc(cc4)CN5CCN(CC5)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)NCCC1CCNC1=O)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](CO)C[C@@H]1CCNC1=O)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(N)=O)C2(C)C |r|
COC(=O)[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C2(C)C |r|
CCOC(=O)C=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1)C2(C)C |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COCc1ccccc1)C2(C)C |r|
[H][C@@]12C[C@@]3([H])[C@]4([H])CC[C@]([H])([C@H](C)[C@@]5([H])CC(C)=C(CO)C(=O)O5)[C@@]4(C)CC[C@]3([H])[C@@]3(C)C(=O)C=C[C@H](O)[C@@]13O2 |r,c:37,t:17|
[H][C@@]12O[C@]1([H])[C@@]1(O)CC=CC(=O)[C@]1(C)[C@@]1([H])CC[C@@]3(C)[C@@]([H])(CC[C@]3(O)[C@H](C)[C@@]3([H])CC(C)=C(C)C(=O)O3)[C@]21[H] |r,c:9,t:35|
Fc1ccc2c(c1)sn(CC(=O)Nc1cc(Cl)cc(Cl)c1)c2=O
Fc1ccc2c(c1)sn(CC(=O)Nc1ccccc1)c2=O
Fc1ccc2c(c1)sn(CC(=O)NC1CCCCC1)c2=O
Fc1ccc2c(c1)sn(CC(=O)NC1CCCC1)c2=O
CCNC(=O)Cn1sc2cc(F)ccc2c1=O
Fc1ccc2c(c1)sn(CC(=O)Nc1ccccc1Cl)c2=O
Fc1ccc2c(c1)sn(CC(=O)Nc1cccc(Cl)c1)c2=O
Fc1ccc2c(c1)sn(CC(=O)Nc1ccc(Cl)cc1)c2=O
COc1ccccc1NC(=O)Cn1sc2cc(F)ccc2c1=O
COc1cccc(NC(=O)Cn2sc3cc(F)ccc3c2=O)c1
COc1ccc(NC(=O)Cn2sc3cc(F)ccc3c2=O)cc1
COc1cc(NC(=O)Cn2sc3cc(F)ccc3c2=O)cc(OC)c1
CC(C)(C)c1ccc(NC(=O)Cn2sc3cc(F)ccc3c2=O)cc1
Fc1ccc2c(c1)sn(CC(=O)Nc1ccccc1C(F)(F)F)c2=O
Fc1ccc2c(c1)sn(CC(=O)Nc1cccc(c1)C(F)(F)F)c2=O
Fc1ccc2c(c1)sn(CC(=O)Nc1ccc(cc1)C(F)(F)F)c2=O
c1cc2c(cc1F)SNC2=O
CC(C)(C)OC(=O)Cn1sc2cc(F)ccc2c1=O
OC(=O)Cn1sc2cc(F)ccc2c1=O
Fc1ccc2c(c1)sn(CC(=O)NCc1ccccc1)c2=O
Fc1ccc2c(c1)sn(CC(=O)NCCc1ccccc1)c2=O
Fc1ccc2c(c1)sn(C(=O)Nc1ccccc1)c2=O
CC(=O)NCn1sc2cc(F)ccc2c1=O
Fc1ccc2c(c1)sn(CCCc1ccccc1)c2=O
O=C(Cn1sc2ccccc2c1=O)Nc1ccccc1
Fc1cccc2sn(CC(=O)Nc3ccccc3)c(=O)c12
Fc1ccc2sn(CC(=O)Nc3ccccc3)c(=O)c2c1
Fc1cccc2c1sn(CC(=O)Nc1ccccc1)c2=O
COc1cccc2sn(CC(=O)Nc3ccccc3)c(=O)c12
COc1ccc2sn(CC(=O)Nc3ccccc3)c(=O)c2c1
COc1ccc2c(c1)sn(CC(=O)Nc1ccccc1)c2=O
FC(F)(F)c1cccc2sn(CC(=O)Nc3ccccc3)c(=O)c12
FC(F)(F)c1ccc2sn(CC(=O)Nc3ccccc3)c(=O)c2c1
FC(F)(F)c1ccc2c(c1)sn(CC(=O)Nc1ccccc1)c2=O
Nc1cccc2sn(CC(=O)Nc3ccccc3)c(=O)c12
Nc1ccc2sn(CC(=O)Nc3ccccc3)c(=O)c2c1
Nc1ccc2c(c1)sn(CC(=O)Nc1ccccc1)c2=O
Nc1cccc2c1sn(CC(=O)Nc1ccccc1)c2=O
Clc1c2C(=O)CC(=O)c2c(Cl)c(Cl)c1Cl
[H][C@]1(O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)c1c(O)cc(C)c2c1oc(CC(C)=O)cc2=O |r|
COc1cc(C)c2c(oc(C[C@@H](C)O)cc2=O)c1[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1OC(=O)\C=C\c1ccc(O)cc1 |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNCc2ccc3ccccc3c2)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNC(=O)c2ccc3ccccc3c2)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc3ccccc3c2)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc3cccnc3c2)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc3nc(Cl)ccc3c2)[C@@H](O)[C@H]1O |r|
CC(=O)Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc3ccccc3c2)[C@@H](O)[C@H]1O |r|
Nc1ncnn2c(ccc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc3ccccc3c2)[C@@H](O)[C@H]1O |r|
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CCl
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(=O)c1c(Cl)cccc1Cl
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CCCCC1
COc1cccc2[nH]c(cc12)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@]3([H])CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)c1cc2c(OC(F)F)cccc2[nH]1 |r|
FC(F)Oc1cccc2[nH]c(cc12)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
CC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(C)(C)C
CCC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(C)(C)C
CC(C)C(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C)C(C)(C)C
CC(C)(C)[C@H](NC(=O)C1CCCCC1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
CC(C)(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C2(C)C
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CCCCC2)n2cccc(NC(=O)OC(C)(C)C)c2=O)C(=O)C(=O)NCc2ccccc2)CCNC1=O |r|
FC(F)(C(=O)N1CCN([C@@H](C1)C(=O)NCc1cccs1)c1ccc(Cl)c(Cl)c1)S(F)(=O)=O |r|
c1cc(sc1)CNC(=O)[C@@H]2CN(CCN2c3ccc(c(c3)Cl)Cl)C(=O)CCl
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1cccs1)C(=O)CBr |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1cccs1)C(=O)C#C |r|
[2H][C@](N(C(=O)C(C)=O)c1ccc2c(c1)oc1ccccc21)(C(=O)N[C@@H](C)c1ccc(F)cc1)c1cccnc1 |r|
O=C1C=C(Nc2ccccc2N2CCNCC2)C2=NS(=O)(=O)c3cccc1c23
O=C(N[C@@H](CC1CCCCC1)C(=O)N[C@@H](CC1CCNC1=O)C(=O)C(=O)NCc1ccccc1)\C=C\c1ccccc1 |r|
CC1=NC2C(S1)C(=O)C=C(Nc1ccc(C)cc1)C2=O |t:1,9|
COC(=O)\C=C\C(=O)NNC(=O)\C=C\c1ccccc1C(=O)N[C@H](C)c1cccc2ccccc12 |r|
C[C@H](NC(=O)[C@H](N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cnccn1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C1CCCCC1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1cccs1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)-c1ccccc1)c1cnccn1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccno1)c1ccc(cc1)C1CCCCC1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-n1cccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
O=C(NCCCc1ccccc1)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1
O=C(NCC(c1ccccc1)c1ccccc1)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccn1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)[Si](C)(C)C)c1cccnc1)c1ccccc1 |r|
CC(C)(C)CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cccnc1)C(=O)c1ccco1
C[C@H](NC(=O)C(N(C(=O)c1ccno1)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCC1)c1cccnc1)C(=O)c1ccco1
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccco1)c1cccnc1)c1ccccc1 |r|
O=C(NC1CCCCC1)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CC1)c1cccnc1)C(=O)c1ccco1
O=C(NC1CCCC1)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(N(C(=O)c1cnco1)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
CC(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)N1CCCCC1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1)c1ccccc1 |r|
O=C(NC1CCCCC1)C(N(C(=O)c1c[nH]cn1)c1ccc(cc1)-c1ccccc1)c1cccnc1
O=C(NC1CCCC1)C(N(C(=O)c1cnc[nH]1)c1ccc(cc1)-c1ccccc1)c1cccnc1
COc1ccc(NC(=O)C(N(C(=O)c2ccco2)c2ccc(cc2)C(C)(C)C)c2cccnc2)cc1
CC(C)(C)c1ccc(cc1)N(C(C(=O)Nc1ccc(F)cc1)c1cccnc1)C(=O)c1ccco1
CC(C)(C)c1ccc(cc1)N(C(C(=O)NCn1nnc2ccccc12)c1cccnc1)C(=O)c1ccco1
O=C(NC1CC1)C(N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1
CC(C)(C)CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
Cc1cccc(C)c1NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
Cc1ccc(cc1)S(=O)(=O)CNC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cccnc1
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1c[nH]cn1
CC(C)(C)NC(=O)C(N(C(=O)c1ccco1)c1ccc(cc1)C(C)(C)C)c1cncnc1
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(OC(C)(C)C)cc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)C(N(C(=O)c1ccco1)c1ccc(Cc2ccccc2)cc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC(=O)[C@@H](N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ccccn1
CCc1ccc(O)c2-c3cccc(-c4ccccn4)c3CC(COC(C)=O)c12
CC(C)c1ccc(O)c2-c3cccc(-c4ccccn4)c3CC(COC(C)=O)c12
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C3CCCCC3)c12)-c1ccccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(cc3)C#N)c12)-c1ccccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(Cc3ccccc3)c12)-c1ccccn1
CC(=O)OCC1Cc2c(ccc(C)c2-c2c(O)ccc(C)c12)-c1ccccn1
COc1ccc(-c2ccccn2)c2CC(COC(C)=O)c3c(C)ccc(O)c3-c12
CC(=O)OCC1Cc2c(ccc(F)c2-c2c(O)ccc(C)c12)-c1ccccn1
CC(=O)OCC1Cc2c(ccc(Cl)c2-c2c(O)ccc(C)c12)-c1ccccn1
CC(=O)OCC1Cc2c(ccc(Br)c2-c2c(O)ccc(C)c12)-c1ccccn1
CC(=O)OCC1Cc2c(cc(C)cc2-c2c(O)ccc(C)c12)-c1ccccn1
CC(=O)OCC1Cc2c(ccc(C)c2-c2ccccn2)-c2c(O)ccc(C)c12
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ncccc1C
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1cc(C)ccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1cc(ccn1)-c1ccccc1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ccc(F)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ccc(Cl)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ccc(Br)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1nccc2ccccc12
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1cc2ccccc2cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ccc2ccccc2n1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ncccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C)c12)-c1ccncn1
CC(=O)OCC1Cc2c(cccc2-n2cccn2)-c2c(O)ccc(C)c12
CC(=O)OCC1Cc2c(cccc2-c2ncnc3n(CC4CC4)cnc23)-c2c(O)ccc(C)c12
CC(=O)OCC1Cc2c(cccc2-c2ncnc3n(CC=C)cnc23)-c2c(O)ccc(C)c12
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(C3CCCCC3)c12)-c1cc(ccn1)-c1ccccc1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(ccn1)-c1ccccc1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(C)ccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(Cl)ccn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(ccn1)C#N
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(C=O)ccn1
CCNc1ccnc(c1)-c1cccc-2c1CC(COC(C)=O)c1c(ccc(O)c-21)-c1ccc(Br)cc1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(ccn1)N1CCCC1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(ccn1)N1CCOCC1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(C)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(F)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(Cl)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(Br)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(cn1)C#N
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(C=O)cn1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(cn1)S(C)(=O)=O
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(cn1)C(C)=O
CN(C)c1ccc(nc1)-c1cccc-2c1CC(COC(C)=O)c1c(ccc(O)c-21)-c1ccc(Br)cc1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(cn1)-c1ccccc1
CC(=O)OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(NCc2ccccc2)cn1
OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(ccn1)-c1ccccc1
OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1cc(C=O)ccn1
Cc1ccc(nc1)-c1cccc-2c1CC(CO)c1c(ccc(O)c-21)-c1ccc(Br)cc1
OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(F)cn1
OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(Cl)cn1
OCC1Cc2c(cccc2-c2c(O)ccc(-c3ccc(Br)cc3)c12)-c1ccc(cn1)C#N
CCNc1ccc(nc1)-c1cccc-2c1CC(CO)c1c(ccc(O)c-21)-c1ccc(Br)cc1
CC1=C(C#N)C(=O)N(CCCO)C(=O)\C1=N/Nc1ccc(Br)cc1C(O)=O |c:1|
NC(=O)CN1C(=O)C(O)(CC(=O)\C=C/c2ccc3OCOc3c2)c2ccccc12
ClCC(=O)N1CCNC(=O)C1CC(=O)Nc1cccc(Cl)c1
[H][C@]12SC(C)(C)[C@@H](N1C(=O)[C@H]2NC(=O)COc1ccccc1)C(=O)OCc1ccccc1 |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12C[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1F)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1cccc(F)c1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc(F)cc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1cc(F)cc(F)c1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc(F)cc1F)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1c(F)cc(F)cc1F)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1cccc(c1)[N+]([O-])=O)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc(OC)cc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc(o1)C(F)(F)F)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1cc(C)no1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OC)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCC)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCC#C)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCC#N)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCOc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)CCc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3c(F)c(F)c(F)c(F)c3F)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccc(OC)cc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COCc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COC3CCCCC3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3cccc4ccccc34)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12N([C@@H](C(=O)OCc3ccccc3)C(C)(C)S1(=O)=O)C(=O)C2(Br)Br |r|
[H][C@@]12[C@@H](Br)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12N([C@@H](C(O)=O)C(C)(C)S1(=O)=O)C(=O)C2(Br)Br |r|
[H][C@@]12N([C@@H](C(=O)OCc3ccc(cc3)[N+]([O-])=O)C(C)(C)S1(=O)=O)C(=O)C2(Br)Br |r|
[H][C@@]12N([C@@H](C(=O)OCc3ccc(cc3)[N+]([O-])=O)C(C)(C)[S+]1[O-])C(=O)C2(Br)Br |r|
CC1([C@@H](N2[C@H](S1)[C@@H](C2=O)NC(=O)COc3ccccc3)C(=O)O)C
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)[S@@+]2[O-] |r|
[H][C@@]12[C@@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)[S@@+]2[O-] |r|
[H][C@@]12[C@@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1cc(F)c(F)c(F)c1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc(cc1)[N+]([O-])=O)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)COc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc3ccccc3c1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)Cc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)OCc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)c3c(C)onc3-c3c(Cl)cccc3Cl)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r,wU:2.2,wD:23.26,1.0,(2.97,4.57,;3,3.02,;1.46,3.02,;.36,4.12,;-.99,3.37,;-1.02,1.83,;-2.3,4.19,;-2.41,5.73,;-1.32,6.82,;-3.9,6.1,;-4.72,4.79,;-3.73,3.61,;-4.12,2.13,;-3.04,1.04,;-1.55,1.44,;-3.43,-.45,;-4.92,-.84,;-6.01,.24,;-5.62,1.73,;-6.71,2.82,;1.46,1.48,;.36,.4,;3,1.49,;4.47,1.02,;4.96,-.44,;6.47,-.76,;3.93,-1.6,;4.41,-3.06,;3.39,-4.21,;3.87,-5.67,;2.85,-6.82,;1.34,-6.5,;.86,-5.05,;1.87,-3.89,;5.37,2.26,;6.71,1.49,;6.45,3.36,;4.44,3.51,;4.84,5,;5.96,3.8,)|
[H][C@@]12[C@H](NC(=O)CNC(=O)c3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)CNC(=O)OCc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)[C@H](NC(=O)NC3CCN(CC)C(=O)C3=O)c3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)C(C)Oc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@@]12[C@H](NC(=O)C(C)Oc3ccccc3)C(=O)N1[C@@H](C(=O)OCc1ccc(F)cc1)C(C)(C)S2(=O)=O |r|
[H][C@]12SC(C)(C)[C@@H](N1C(=O)C2(Br)Br)C(=O)OCc1ccccc1 |r|
[H][C@]12SC(C)(C)[C@@H](N1C(=O)C2(Br)Br)C(=O)OCc1ccc(cc1)[N+]([O-])=O |r|
CC1([C@@H](N2[C@H](S1(=O)=O)CC2=O)C(=O)O)C
[H][C@@]12CC(=O)N1[C@@H](C(=O)OCc1ccccc1)C(C)(C)S2(=O)=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)C(=O)OC(C)(C)C)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)C(=O)OC(C)(C)C)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)C(=O)C(C)C)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)C(=O)C(C)C)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)C(=O)Cc2ccccc2)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)C(=O)Cc2ccccc2)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)S(C)(=O)=O)C=O)CCNC1=O |r|
CC(C)C[C@H](NC(=O)OC1C[C@@]2(C1)CCN(C2)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r,wU:4.3,11.13,wD:27.29,29.31,(3.44,4.42,;3.44,2.88,;4.78,2.11,;2.11,2.11,;2.11,.57,;.78,-.2,;-.56,.57,;-.56,2.11,;-1.89,-.2,;-3.22,.57,;-3.62,2.06,;-5.14,1.65,;-4.74,.16,;-5.32,3.11,;-6.8,3.5,;-7.57,2.17,;-6.54,1.03,;-9.11,2.17,;-9.88,3.5,;-9.88,.84,;-9.11,-.5,;-9.88,-1.83,;-7.57,-.5,;-8.34,-1.83,;3.44,-.2,;3.44,-1.74,;4.78,.57,;6.11,-.2,;6.11,-1.8,;7.45,-2.57,;7.61,-4.1,;9.11,-4.42,;9.88,-3.09,;8.85,-1.94,;9.25,-.45,;7.45,.57,;7.45,2.11,)|
CC(C)C[C@H](NC(=O)OC1C[C@@]2(C1)CCN(C2)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CN(C3)S(C)(=O)=O)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CCC3(CN(C3)C(=O)OC(C)(C)C)C2)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CCC3(CN(C3)C(=O)OC(C)(C)C)C2)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C(=O)OC(C)(C)C)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C(=O)OC(C)(C)C)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C(=O)C(C)C)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C(=O)C(C)C)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C(=O)Cc2ccccc2)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C(=O)Cc2ccccc2)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)S(C)(=O)=O)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)S(C)(=O)=O)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C#N)C=O)CCNC1=O |r|
[H][C@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OC2CC3(C2)CCN(CC3)C#N)C(=O)C(O)S([O-])(=O)=O)CCNC1=O |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1CN(C1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OC1CN(C1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OC1(C)CN(C1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OC1(C)CN(C1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC1CN(C1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC1CN(C1)C(=O)OC(C)(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC1CN(C1)C(=O)Cc1ccccc1)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC1CN(C1)C(=O)Cc1ccccc1)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC1CN(C1)C(=O)C1CC2CCC1C2)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r,TLB:14:16:22:19.20|
CC(C)C[C@H](NC(=O)OCC1CN(C1)C(=O)C1CC2CCC1C2)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r,TLB:14:16:22:19.20|
CC(C)C[C@H](NC(=O)OCC1CN(C1)S(C)(=O)=O)C(=O)N[C@@H](C[C@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC1CN(C1)S(C)(=O)=O)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O |r|
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@H]1CCNC1=O)C(=O)C(O)S([O-])(=O)=O)C1CN(C1)C(=O)OC(C)(C)C |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1 |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)C(=O)C(=O)NC2CC2)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc2cccc(c2)C(F)(F)F)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@]3([H])CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)COc1ccc(OC)cc1 |r|
c1c(cc(cc1F)F)CCC(=O)N2C[C@@H]3CCC[C@@H]3[C@H]2C(=O)N[C@@H](C[C@@H]4CCNC4=O)C=O
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)COc2ccc(Cl)cc2Cl)C=O)CCNC1=O |r|
c1cc(c2c(c1O)C(=O)C=CC2=O)O
C[C@H](NC[C@H](N(C(=O)C(Cl)Cl)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
C[C@H](NC[C@H](N(C(=O)C(Br)(Br)Br)c1ccc(cc1)-c1ccccc1)c1cccnc1)c1ccccc1 |r|
F[C@H](Cl)C(=O)N([C@@H](C(=O)NCCc1cccc(F)c1)c1cncnc1)c1ccc(cc1)S(F)(F)(F)(F)F |r|
c1ccc(cc1)C2=NN([C@H](C2)c3cccc4c3nccn4)C(=O)CCl
Fc1ccc(Cl)cc1C1=NN(C(C1c1ccccc1)c1ccc2nccnc2c1)C(=O)CCl |t:9|
CSc1ccc2C(=O)C(F)(F)C(=O)Nc2c1
CCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1)C(=O)C(=O)NCc1ccccn1 |r|
CSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(C)=O)C=O |r|
CCOC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)OC(C)(C)C |r|
CC(=O)\C=C\[C@H](CCc1ccccc1)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1ccc(F)cc1 |r|
CC(C)C[C@H](NC(=O)OCc1ccc(cc1)[N+]([O-])=O)C(=O)N[C@@H](CCc1ccccc1)\C=C\C(C)=O |r|
[O-]S(=O)(=O)C(F)(F)F.[H][C@]12OCc3c(NC(C)(C)C)n4c(c(sc4[n+]3[C@@]1([H])CC(=O)C=C2)-c1ccc(OC)cc1)-c1ccc(OC)cc1 |r,c:32|
COc1cc(c2c(c1)OC(=C(C2=O)O)c3cc(c(c(c3)O)O)O)O
COc1cc(O)c2C(=O)[C@H](O)[C@H](Oc2c1)c1cc(O)c(O)c(O)c1 |r|
COc1ccc2cc(ccc2c1)[C@@H](C)C(=O)Oc1cncc(Cl)c1 |r|
Cc1cccc(C(=O)Oc2c(C)cccc2C(=O)Oc2cncc(Cl)c2)c1O
COc1cccc(Cn2[se]c3ccccc3c2=O)c1
O=C(N1CCOCC1)c1cccc(Cn2[se]c3ccccc3c2=O)c1
COc1cncc(Cn2[se]c3ccccc3c2=O)c1
Clc1ccc(Cn2[se]c3ccccc3c2=O)cc1
CC(C)CCn1sc2ccccc2c1=O
O=c1n(CC2CCCCC2)sc2ccccc12
CCCCCn1sc2ccccc2c1=O
Brc1ccc2sn(-c3ccccc3)c(=O)c2c1
CC(C)CCn1sc2ccc(Br)cc2c1=O
Cc1c(oc2cc(O)cc(O)c2c1=O)-c1ccc(O)c(O)c1
CCCc1c(oc2cc(O)cc(O)c2c1=O)-c1ccc(O)c(O)c1
CCCCc1c(oc2cc(O)cc(O)c2c1=O)-c1ccc(O)c(O)c1
CCCCOc1c(oc2cc(O)cc(O)c2c1=O)-c1ccc(O)c(O)c1
OCCOc1c(oc2cc(O)cc(O)c2c1=O)-c1ccc(O)c(O)c1
OCCCOc1c(oc2cc(O)cc(O)c2c1=O)-c1ccc(O)c(O)c1
Oc1ccc(Cc2cc(=O)c3c(O)cccc3o2)cc1O
CC(c1ccc(O)c(O)c1)c1cc(=O)c2c(O)cccc2o1
CCCCC(c1ccc(O)c(O)c1)c1cc(=O)c2c(O)cccc2o1
Oc1ccc(CCc2cc(=O)c3c(O)cccc3o2)cc1O
Oc1ccc(\C=C\c2cc(=O)c3c(O)cccc3o2)cc1O
Oc1ccc(NC(=O)c2cc(=O)c3c(O)cccc3o2)cc1O
Oc1ccc(OC(=O)c2cc(=O)c3c(O)cccc3o2)cc1O
Oc1ccc(CCOC(=O)c2cc(=O)c3c(O)cccc3o2)cc1O
Oc1ccc(cc1O)C(=O)NCCNC(=O)c1cc(=O)c2c(O)cccc2o1
Oc1ccc(NC(=S)NCCNC(=O)c2cc(=O)c3c(O)cccc3o2)cc1O
Cc1ccc(cc1NC(=O)c2cccc(c2)NC(=O)Nc3cccc(c3)C(=O)Nc4cc(ccc4C)C(=O)Nc5ccc(c6c5c(cc(c6)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O)C(=O)Nc7ccc(c8c7c(cc(c8)S(=O)(=O)O)S(=O)(=O)O)S(=O)(=O)O
c1ccc(cc1)C2=CC(=C3N(C2=O)c4cc(ccc4S3)OC5CCCCC5)C(=O)N[C@@H](Cc6ccc(cc6)O)C(=O)O
Cc1ccccc1Cn1c(=O)sn(-c2cccc3ccccc23)c1=O
CN(C(=O)c1ccccc1C)c1ccccc1
CC(C)(C)OC(=O)Nc1cccn([C@@H](CC2CCCCC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)C(=O)NC2CC2)c1=O
[#6]\[#6](-[#6])=[#6]/[#6][C@]12[#8]-c3cc(-[#8])c(-[#6@H]-4-[#6]=[#6](-[#6])-[#6]-[#6@@H](-[#6@H]-4-[#6](=O)-c4ccc(-[#8])cc4-[#8])-c4ccc(-[#8])cc4-[#8])c(-[#8])c3-[#6](=O)[C@@]1([#8])[#8]-c1cc(-[#8])ccc21 |r,t:13|
[#6]\[#6](-[#6])=[#6]/[#6][C@@]12[#8]-c3cc(-[#8])c(-[#6@H]-4-[#6]=[#6](-[#6])-[#6]-[#6@@H](-[#6@H]-4-[#6](=O)-c4ccc(-[#8])cc4-[#8])-c4ccc(-[#8])cc4-[#8])c(-[#8])c3-[#6](=O)[C@]1([#8])[#8]-c1cc(-[#8])ccc21 |r,t:13|
[#6]\[#6](-[#6])=[#6]\[#6]C12[#8]-c3cc(-[#8])c(-[#6]-4-[#6]=[#6](-[#6])-[#6]-[#6](-[#6]-4-[#6](=O)-c4ccc(-[#8])cc4-[#8])-c4ccc(-[#8])cc4-[#8])c(-[#8])c3-[#6](=O)C1([#8])[#8]-c1cc(-[#8])ccc21 |t:13|
[#6]\[#6](-[#6])=[#6]\[#6]-[#6]-[#6]-1=[#6]-[#6@@H](-[#6@H](-[#6@@H](-[#6]-1)-c1ccc(-[#8])cc1-[#8])-[#6](=O)-c1ccc(-[#8])cc1-[#8])-c1c(-[#8])cc2-[#8]-[#6@@H](-[#6]-[#6](=O)-c2c1-[#8])-c1ccc(-[#8])cc1-[#8] |r,t:6|
CC1=C[C@@H]([C@H]([C@@H](C1)c1ccc(O)cc1O)C(=O)c1ccc(O)cc1O)c1c(O)ccc([C@@H]2CC(=O)c3c(O)cc(O)cc3O2)c1O |t:1|
[#6]\[#6](-[#6])=[#6]\[#6]-c1c(-[#8])c2c(cc(-[#8])cc2=O)oc1-c1ccc(-[#8])c2-[#6]=[#6]C([#6])([#6])[#8]-c12 |c:26|
[#6]\[#6](-[#6])=[#6]\[#6]-c1c(oc2c3-[#6]=[#6]C([#6])([#6])[#8]-c3cc(-[#8])c2c1=O)-c1ccc(-[#8])cc1-[#8] |c:10|
[#6]\[#6](-[#6])=[#6]\[#6]=[#6](-[#8]-[#6](-[#6])=O)-c1cc(-[#8])c2c(-[#8])ccc(-[#8])c2c1-[#8] |w:4.3|
CCC(CC)OC(=O)[C@H](C)N[P@@](=O)(CC[C@H]1O[C@](C#N)([C@H](O)[C@@H]1O)c1ccc2c(N)ncnn12)Oc1ccccc1 |r|
CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2CN1)C=O |r|
CC(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CC(=O)NCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
O=C[C@H](Cc1c[nH]cn1)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1Cc2ccccc2CN1 |r|
CC(=O)NCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1ccc(O)cc1)C=O |r|
CC(=O)NCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CC(C)(C)O[C@H]1CN[C@@H](C1)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CC(C)(C)OC(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CCCCCCCC(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]cn1)C=O |r|
CNC(=O)c1cc(Br)cc(c1N[C@@H]1CCCC[C@@H]1NC(=O)c1cccc2ccccc12)[N+]([O-])=O |r|
C[C@H](NC(=O)[C@H](N(C(=O)c1ccco1)c1ccc(cc1)-c1ccccc1)c1ccccc1)c1ccccc1 |r|
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)\C=C\c2ccccc2)n1
C\C=C\C(=O)NCc1nc(no1)-c1ccc(cc1)C(F)(F)F
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)\C=C\c2ccccn2)n1
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)\C=C\c2ccco2)n1
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)\C=C\c2cccs2)n1
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)c2ccccc2)n1
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)CCc2ccccc2)n1
FC(F)(F)c1ccc(cc1)-c1noc(CNC(=O)C#Cc2ccccc2)n1
CC1=C(C1C(=O)NCc1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1cccc(c1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1ccccc1C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1ccccc1)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1cccc(C)c1)c1ccccc1 |t:1|
COc1cccc(c1)-c1noc(CNC(=O)C2C(C)=C2c2ccccc2)n1 |c:19|
CC1=C(C1C(=O)NCc1nc(no1)-c1cccc(F)c1)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1cccc(Cl)c1)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1cccc(c1)[N+]([O-])=O)c1ccccc1 |t:1|
CC1=C(C1C(=O)NCc1nc(no1)-c1cccc(OC(F)(F)F)c1)c1ccccc1 |t:1|
CC(NC(=O)C1C(C)=C1c1ccccc1)c1nc(no1)-c1ccc(cc1)C(F)(F)F |c:7|
CC1=C(C1C(=O)NC(CC1CC1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(CC1CCCCC1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(Cc1ccccc1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(Cc1ccc2ccccc2c1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(Cc1cc2ccccc2[nH]1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(Cc1ccccc1F)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(Cc1cccc(F)c1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
CC1=C(C1C(=O)NC(Cc1ccc(F)cc1)c1nc(no1)-c1ccc(cc1)C(F)(F)F)c1ccccc1 |t:1|
[H][C@@]12CN(Cc3cc(OC)cc(OC)c3)C[C@]3(CN([C@@]4(CC[C@H](OCCCN(C)C)[C@@]1([H])[C@]34[H])C(C)C)S(=O)(=O)c1ccc(C)cc1)O2 |r|
N[C@@H](CCSC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12)C(O)=O
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)[C@@H](NS(=O)(=O)C1CC1)C(C)(C)C |r|
[H][C@]12CCC[C@@]1([H])N([C@@H](C2)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)[C@@H](NS(=O)(=O)C(F)(F)F)C(C)(C)C |r|
Cn1cnc2n(C)c(=O)n(CC(=O)Nc3ccc(cc3)S(=O)(=O)Nc3ncccn3)c(=O)c12
Clc1cccc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)COc1ccc(OC(F)(F)F)cc1 |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#C)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](CCSC)C#C)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](CCSC)C#N)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#C)[C@@]1([H])C2(C)C)C(=O)COc1ccc(OC(F)(F)F)cc1 |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)COc1ccc(cc1)C(F)(F)F |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#C)[C@@]1([H])C2(C)C)C(=O)COc1ccc(cc1)C(F)(F)F |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#Cc3ccccc3)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#Cc3ccc(cc3)[N+]([O-])=O)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#CC(F)(F)F)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
c1ccc(cc1)C[C@@H](C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)NC(=O)c3cc4ccccc4[nH]3
[#8]-[#6](=O)-[#6]-1=[#6]\[#6](-[#6]=[#6]-[#6]-1=O)=[#6](\c1ccc(-[#8])c(c1)-[#6](-[#8])=O)-c1ccc(-[#8])c(c1)-[#6](-[#8])=O |c:6,t:3|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)c2cnoc2)C2CCCCC2)C#N)CCNC1=O |r|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)[C@@H](NC(=O)C(F)(F)F)C1CCCCC1)C(=O)N[C@@H](Cc1n[nH]c2ccccc12)C#N |r|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(C)=O)C2CCCCC2)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)c2ccc(F)cc2)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)C2CCCCC2)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2C[C@@]3([H])CCCC[C@@]3([H])N2C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C#N)CCNC1=O |r|
[H][C@@]12C[C@]1([H])[C@H](N(C2)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C(=O)N[C@@H](C[C@]1([H])CCNC1=O)C#N |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)C2CCCCC2)C(=O)C(=O)NC(C)(C)C)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)C2CCC2)C(=O)C(=O)NC(C)(C)C)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)C2CCCC2)C(=O)C(=O)NC(C)(C)C)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)C2CC3(CCC3)C2)C(=O)C(=O)NC(C)(C)C)CCNC1=O |r|
O=C(CSC#N)N1c2ccccc2CCc2ccccc12
O=C(CSC#N)N1c2ccccc2Sc2ccccc12
Clc1ccc2CCc3ccccc3N(C(=O)CSC#N)c2c1
FC(F)(F)c1ccc2Sc3ccccc3N(C(=O)CSC#N)c2c1
COc1ccc2Sc3ccccc3N(C(=O)CSC#N)c2c1
CC(=O)c1ccc2Sc3ccccc3N(C(=O)CSC#N)c2c1
CCC(=O)c1ccc2Sc3ccccc3N(C(=O)CSC#N)c2c1
O=C(CSC#N)N1c2ccccc2Sc2ccc(cc12)C#N
CCSc1ccc2Sc3ccccc3N(C(=O)CSC#N)c2c1
Clc1ccc2Sc3ccccc3N(C(=O)CSC#N)c2c1
O=C(CSC#N)N1c2ccccc2Oc2ccccc12
COC(=O)CC1COc2c3CCCN4CCCc(cc2-c2c(NC(C)(C)C)n5c(c(C)sc5[n+]12)-c1ccc(F)cc1)c34
[H][C@]12COc3ccc4ccccc4c3[C@@]1([H])N=C1SC(C)=C(N1C2(C)C)c1cccc2OCOc12 |r,c:23,t:19|
[H][C@]12COc3ccc4ccccc4c3[C@@]1([H])N=C1SC=C(N1C2(C)C)c1ccc(cc1)S(=O)(=O)N1CCOCC1 |r,c:22,t:19|
COC(=O)[C@H](Cc1ccc(OC)c(OC)c1)N1CC(=N[C@@H](Cc2ccc(OC)c(OC)c2)C1=O)c1cc(C)ccc1O |r,c:19|
[H][C@@]12CC(=O)C=C[C@@]1(CCC1N2[C@@H](CC11C(=O)Nc2ccccc12)C(=O)OC)OC |r,c:5|
COc1ccc2[nH]cc(CCN3[C@@H](C(=O)NC(C)(C)C)c4ccccc4OC[C@@H](CC(O)=O)[C@@H](c4nnc(o4)-c4cccc(c4)C(F)(F)F)C3=O)c2c1 |r|
[H][C@@]12CC[C@]3(Cc4c(C[C@@]3([H])N1CCc1c2[nH]c2ccccc12)[nH]c1ccc(OC)cc41)OC |r|
[H][C@@]12CC(=O)C=C[C@]1(C)OCC1N2CCc2cccc3[nH]cc1c23 |r,c:5|
[H][C@@]12CC[C@@]3(CC\C(C=C3)=N/Nc3ccc(OC(F)(F)F)cc3)c3[nH]c4cccc(CCN1)c4c23 |r,c:8|
[H][C@@]12CC[C@]3(Cc4c(C[C@@]3([H])N1CCc1cccc3[nH]cc2c13)[nH]c1ccc(OC)cc41)OC |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)C(=O)NC1CC1 |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)(C(=O)NC1CC1)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#N |r|
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O)C(C)(C)Sc1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)[S+]([O-])c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)[S+]([O-])c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)S(=O)(=O)c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)S(=O)(=O)c1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1cccc(F)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1cccc(F)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccc(F)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1ccc(F)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCCSc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCCSc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1nc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Sc1nc2ccccc2[nH]1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1ccc(Cl)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1ccc(Cl)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O)C(C)(C)Oc1ccc(Cl)cc1 |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
[2H]C([2H])(OC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O)C(C)(C)Oc1cccc(Cl)c1 |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1ccc(F)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1ccc(F)cc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1cccc(F)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(C)Oc1cccc(F)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(O)c1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)C[C@H](NC(=O)OCC(C)(O)c1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O |r|
NC(=O)c1ccc2N(Cc3cn(Cc4cccc(Cl)c4)nn3)C(=O)C(=O)c2c1
NC(=O)c1ccc2N(Cc3cn(Cc4ccc(cc4)S(N)(=O)=O)nn3)C(=O)C(=O)c2c1
NC(=O)c1ccc2N(Cc3cn(Cc4ccc(cc4F)C(F)(F)F)nn3)C(=O)C(=O)c2c1
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C#N)[C@@]1([H])C2(C)C)C(=O)[C@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
O=c1n(Cc2ccccc2)[se]c2ccccc12
O=c1n(Cc2ccncc2)[se]c2ccccc12
O=c1n(Cc2cccnc2)[se]c2ccccc12
O=c1n([se]c2ccccc12)-c1ccc(NS(=O)(=O)C2CC2)cc1
CN(C)S(=O)(=O)Nc1ccc(cc1)-n1[se]c2ccccc2c1=O
O=C(Nc1ccc(cc1)-n1[se]c2ccccc2c1=O)C1CC1
Nc1ccc2c(c1)[se]n(-c1ccccc1)c2=O
CC(C)(C)OC(=O)N1CCC(CC1)n1[se]c2ccccc2c1=O
O=c1n([se]c2ccccc12)C1CCN(CC1)S(=O)(=O)C1CC1
O=c1n([se]c2ccccc12)C1CCN(CC1)S(=O)(=O)c1cccnc1
NS(=O)(=O)c1ccc(cc1)C(=O)N1CCC(CC1)n1[se]c2ccccc2c1=O
C1CCC(CC1)[C@@H](C(=O)N2C[C@@H]3CCC[C@@H]3[C@H]2C(=O)N[C@@H](C[C@@H]4CCNC4=O)[C@H](C(=O)NC5CCCC5)O)NC(=O)C(F)(F)F
CNC(=O)c1cc(cc(c1N[C@@H]2CCCC[C@@H]2NC(=O)c3cncc4c3cccc4)N(=O)=O)Br
[H][C@@]1(C[C@H](NC(=O)[C@H](CCC)NC(=O)OCc2ccccc2)\C=C\C(C)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)\C=C\C(C)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CCCC)NC(=O)OCc2ccccc2)\C=C\C(C)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CC2)NC(=O)OCc2ccccc2)\C=C\C(C)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)(C)C)NC(=O)OCc2ccccc2)\C=C\C(C)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CCCCC2)NC(=O)OCc2ccccc2)\C=C\C(C)=O)CCNC1=O |r|
Cc1cccc2nc(CSC(=S)NCc3cccnc3)cn12
S=C(NCc1cccnc1)SCc1ccccc1
CCSC(=S)NCc1cccnc1
Cc1cccc2nc(CNC(=S)NCc3cccnc3)cn12
[S-]C(=S)NCc1cccnc1
S=C(NCc1cccnc1)OCc1ccccc1
[H][C@]12Cc3ccc(Oc4cc5cc(Oc6ccc(cc6Cl)[C@@H](O[C@@H]6O[C@H](CO)[C@@H](O)[C@H](O)[C@H]6NC(C)=O)[C@]6([H])NC(=O)[C@]([H])(NC(=O)[C@]5([H])NC(=O)[C@@]([H])(NC1=O)c1cc(O)cc(Oc5cc(ccc5O)[C@@H](N)C(=O)N2)c1)c1ccc(O)c(c1)-c1c(O[C@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]2O)cc(O)cc1[C@H](NC6=O)C(O)=O)c4O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1NC(=O)CCCCCCCCC)c(Cl)c3
COC(=O)CCC(CC(=O)[C@H](CC(=O)OC)NC(=O)OCc1ccccc1)C(=O)NC(C(C)C)C(=O)NC(CC(=O)OC)C(=O)CF |r|
C[C@@H](c1ccc2cc(ccc2c1)OC)C(=O)O
O=c1[nH]cnc2[nH]ncc12
CN(Cc1ccc(cc1)C(C)(C)C)Cc1cccc2ccccc12
Oc1ccc(cc1)-c1sc2cc(O)ccc2c1C(=O)c1ccc(OCCN2CCCCC2)cc1
c1ccc(cc1)[C@@H]2C[C@H]2N
CC(C)(C)NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2CN1C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NC(=O)c1ccc2ccccc2n1 |@:16|
CC(C)(C)OC(=O)CC[C@H](NC(=O)CNC(=O)OC(C)(C)C)C(=O)CCl |r|
CC(C)(C)OC(=O)CC[C@H](NC(=O)CNC(=O)OC(C)(C)C)C(=O)COC(=O)c1c(Cl)cccc1Cl |r|
CCOC(=O)[C@@H]1O[C@H]1C(=O)N(CCC(N)=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1 |r|
C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)NN(CC(N)=O)C(=O)\C=C\C(=O)c1ccccc1 |r|
O[C@H]1C(Oc2cc(O)cc(O)c2C1=O)c1cc(O)c(O)c(O)c1 |r|
c1cc(c(cc1C2=C(C(=O)c3c(cc(c(c3O)O)O)O2)O)O)O
C[n+]1c2cc(N)ccc2cc2ccc(N)cc12
FC(F)(F)c1cccc(c1)-n1[se]c2ccccc2c1=O
COc1cccc(c1)-n1[se]c2ccccc2c1=O
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CC2)NC(=O)OCCc2cccc(Cl)c2)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@@]1(C[C@@H](NC(=O)[C@@H](CC(C)C)NC(=O)OC([2H])([2H])c2ccccc2)C(O)S([O-])(=O)=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CC2)NC(=O)OCc2cccc(F)c2)C(O)S([O-])(=O)=O)CCNC1=O |r|
CC(C)C[C@H](NC(=O)c1cc2c(F)cccc2[nH]1)C(=O)NN(C[C@@H]1CCNC1=O)C(=O)C(F)Cl |r|
CCN(C[C@]1(C)CN(CCC1=O)C(=O)c1nn(C)c-2c1CCc1ccccc-21)C(=O)c1nn(C)c-2c1CCc1ccccc-21 |r|
[H][C@@]12C([C@@H](C(=O)OCc3ccccc3)C(C)(C)S1(=O)=O)C(=O)C2(Br)Br |r|
[H][C@@]12C([C@@H](C(=O)OCc3ccc(cc3)[N+]([O-])=O)C(C)(C)S1(=O)=O)C(=O)C2(Br)Br |r|
[H][C@@]12C([C@@H](C(=O)OCc3ccc(cc3)[N+]([O-])=O)C(C)(C)[S+]1[O-])C(=O)C2(Br)Br |r|
CC(C)(C)c1ccc(cc1)N(C(C(=O)NC1CCCCC1)c1cccnc1)S(=O)(=O)C=C
c1c(cc(c(c1Cl)Cl)Cl)N2CCN(CC2)C(=O)C3=CC(=O)NC(=O)N3
Cc1c(cc(cc1Cl)N2CCN(CC2)C(=O)C3=CC(=O)NC(=O)N3)Cl
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1F
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(F)c1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc(F)cc1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1Cl
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(Cl)c1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc(Cl)cc1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1Br
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(Br)c1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc(Br)cc1
Cc1ccccc1-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
Cc1cccc(c1)-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
Cc1ccc(cc1)-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1C(F)(F)F
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(c1)C(F)(F)F
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1OC(F)(F)F
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(OC(F)(F)F)c1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1[N+]([O-])=O
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(c1)[N+]([O-])=O
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc(cc1)[N+]([O-])=O
CC(C)c1cccc(c1)-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)(C)c1cccc(c1)-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)(C)c1ccc(cc1)-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1O
Oc1ccc(cc1)-c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccc(F)c1F
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc(F)cc1F
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc(F)c(F)c1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccc1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1cccs1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccccn1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccncc1
Cc1cc(-c2nc3cc(O)c(O)c(O)c3c(=O)[nH]2)n(C)n1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)-c1ccc2ccccc2c1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)C1CC1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)C1CCCC1
Oc1cc2nc([nH]c(=O)c2c(O)c1O)C1CCCCC1
CC(C)c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)(C)c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)Cc1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)(C)Cc1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
Oc1cc2nc(\C=C\c3ccccc3)[nH]c(=O)c2c(O)c1O
Oc1cc2nc(Cc3ccccc3)[nH]c(=O)c2c(O)c1O
CC(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CCC(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)C(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)[nH]1
CC(C)Cn1c(nc2cc(O)c(O)c(O)c2c1=O)-c1ccccc1
OCCn1c(nc2cc(O)c(O)c(O)c2c1=O)-c1ccccc1
CC(C)(C)NC(=O)Cn1c(nc2cc(O)c(O)c(O)c2c1=O)-c1ccccc1
Oc1cc2nc(-c3ccccc3)n(C3CC3)c(=O)c2c(O)c1O
Oc1cc2nc(-c3ccccc3)n(C3CCCC3)c(=O)c2c(O)c1O
Oc1cc2nc(-c3ccccc3)n(C3CCCCC3)c(=O)c2c(O)c1O
Oc1cc2nc(-c3ccccc3)n(-c3ccccc3)c(=O)c2c(O)c1O
Oc1cc2nc(-c3ccccc3)n(-c3ccccc3F)c(=O)c2c(O)c1O |(-5.19,-1.09,;-3.91,-.34,;-2.64,-1.09,;-1.37,-.34,;-.1,-1.09,;1.25,-.34,;2.52,-1.09,;2.52,-2.63,;3.85,-3.4,;5.19,-2.63,;5.19,-1.09,;3.85,-.32,;1.25,1.15,;2.57,1.94,;3.91,1.17,;5.24,1.94,;5.24,3.48,;3.91,4.25,;2.57,3.48,;1.24,4.25,;-.1,1.9,;-.1,3.4,;-1.37,1.15,;-2.64,1.9,;-2.64,3.4,;-3.91,1.15,;-5.19,1.9,)|
Oc1cc2nc(-c3ccccc3)n(-c3cccc(F)c3)c(=O)c2c(O)c1O
Oc1ccc(cc1)-n1c(nc2cc(O)c(O)c(O)c2c1=O)-c1ccccc1
Oc1cc2nc(-c3ccccc3)n(-c3ccc(Br)cc3F)c(=O)c2c(O)c1O |(-5.21,-1.51,;-3.94,-.76,;-2.67,-1.51,;-1.4,-.76,;-.13,-1.51,;1.22,-.76,;2.49,-1.51,;2.49,-3.05,;3.83,-3.82,;5.16,-3.05,;5.16,-1.51,;3.83,-.74,;1.22,.73,;2.55,1.51,;3.88,.74,;5.21,1.51,;5.21,3.05,;6.55,3.82,;3.88,3.82,;2.55,3.05,;1.21,3.82,;-.13,1.48,;-.13,2.98,;-1.4,.73,;-2.67,1.48,;-2.67,2.98,;-3.94,.73,;-5.21,1.48,)|
Cc1cc(ccc1F)-n1c(nc2cc(O)c(O)c(O)c2c1=O)-c1ccccc1
Oc1cc2nc(-c3ccccc3)n(-c3ccc(cc3)-c3ccccc3)c(=O)c2c(O)c1O
Oc1cc2nc(-c3ccccc3)n(-c3cccnc3)c(=O)c2c(O)c1O
Oc1cc2nc(-c3ccccc3)n(-c3cn[nH]c3)c(=O)c2c(O)c1O
CC(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccccc1
CC(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccc(F)c(C)c1
CC(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccccc1F |(3.82,.41,;2.49,-.36,;2.49,-1.9,;1.16,-2.67,;1.16,-4.21,;2.49,-4.98,;3.82,-4.21,;3.82,-2.67,;1.22,.39,;-.13,-.36,;-1.4,.39,;-2.67,-.36,;-3.94,.39,;-5.21,-.36,;-3.94,1.89,;-5.21,2.63,;-2.67,2.63,;-2.67,4.13,;-1.4,1.89,;-.13,2.63,;-.13,4.13,;1.22,1.89,;2.55,2.67,;3.88,1.9,;5.21,2.67,;5.21,4.21,;3.88,4.98,;2.55,4.21,;1.21,4.98,)|
CC(c1ccccc1)c1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccc(Br)cc1F |(3.82,.41,;2.49,-.36,;2.49,-1.9,;1.16,-2.67,;1.16,-4.21,;2.49,-4.98,;3.82,-4.21,;3.82,-2.67,;1.22,.39,;-.13,-.36,;-1.4,.39,;-2.67,-.36,;-3.94,.39,;-5.21,-.36,;-3.94,1.89,;-5.21,2.63,;-2.67,2.63,;-2.67,4.13,;-1.4,1.89,;-.13,2.63,;-.13,4.13,;1.22,1.89,;2.55,2.67,;3.88,1.9,;5.21,2.67,;5.21,4.21,;6.55,4.98,;3.88,4.98,;2.55,4.21,;1.21,4.98,)|
CC(C)Cn1c(nc2cc(O)c(O)c(O)c2c1=O)C(C)c1ccccc1
CC(C)Cc1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccccc1
CC(C)Cc1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccccc1F |(1.16,-3.82,;2.49,-3.05,;3.83,-3.82,;2.49,-1.51,;1.22,-.76,;-.13,-1.51,;-1.4,-.76,;-2.67,-1.51,;-3.94,-.76,;-5.21,-1.51,;-3.94,.73,;-5.21,1.48,;-2.67,1.48,;-2.67,2.98,;-1.4,.73,;-.13,1.48,;-.13,2.98,;1.22,.73,;2.55,1.51,;2.55,3.05,;3.88,3.82,;5.21,3.05,;5.21,1.51,;3.88,.74,;3.88,-.8,)|
Cc1cc(ccc1F)N2C(=Nc3cc(c(c(c3C2=O)O)O)O)CC(C)C
CC(C)Cc1nc2cc(O)c(O)c(O)c2c(=O)n1-c1ccc(Br)cc1F |(1.16,-3.82,;2.49,-3.05,;3.83,-3.82,;2.49,-1.51,;1.22,-.76,;-.13,-1.51,;-1.4,-.76,;-2.67,-1.51,;-3.94,-.76,;-5.21,-1.51,;-3.94,.73,;-5.21,1.48,;-2.67,1.48,;-2.67,2.98,;-1.4,.73,;-.13,1.48,;-.13,2.98,;1.22,.73,;2.55,1.51,;3.88,.74,;5.21,1.51,;5.21,3.05,;6.55,3.82,;3.88,3.82,;2.55,3.05,;1.21,3.82,)|
Oc1cc2nc(Cc3ccccc3)n(-c3ccccc3)c(=O)c2c(O)c1O
Cc1cc(ccc1F)-n1c(Cc2ccccc2)nc2cc(O)c(O)c(O)c2c1=O
CC(C)Cn1c(Cc2ccccc2)nc2cc(O)c(O)c(O)c2c1=O
CC(C)C[C@H](NC(=O)C(=O)Nc1ccccc1F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COc1c(F)c(F)cc(F)c1F |r|
CC(C)C[C@H](NC(=O)C(=O)Nc1ccccc1F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
Fc1ccccc1NC(=O)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C(=O)COC(F)(F)F)[C@@]1([H])C2(C)C)C(=O)C(=O)NC(C)(C)C |r|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)C(=O)NC(C)(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)CC(=O)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)\C=C\C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC1(C)CC(O)(C1)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)C[C@H](NC(=O)C(=O)NCC(F)(F)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)C[C@H](NC(=O)C(=O)NC12CC(F)(C1)C2)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)C[C@H](NC(=O)c1cc(on1)C(C)(C)F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)C[C@H](NC(=O)[C@H]1CCCO1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
CC(C)C[C@H](NC(=O)C(=O)Nc1ccccc1F)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)CO |r|
CC(C)C[C@@H](O)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F)C(F)(F)F |r|
CC(C)C[C@@H](O)C(=O)N1CC2(CC2)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)COC(F)(F)F |r|
Cc1cc2nc3s\c(=C\c4ccc(o4)-c4cccc(c4)C(O)=O)c(=O)n3c2cc1C
Cn1c2cc(cnc2[nH]c1=O)-c1cccc(c1)C(=O)Nc1cccc(c1)C#N
Cc1c(C(=O)\C=C\c2ccc(O)c(c2)[N+]([O-])=O)c(C#N)c2CCCn12
Brc1ccc2nc(COC(=O)c3cc([nH]n3)-c3ccco3)cn2c1
Cn1c2cc(cnc2[nH]c1=O)-c1cccc(c1)C(=O)Nc1ccc(Cl)c(CO)c1
COc1cc(F)cc(NC(=O)c2cccc(c2)-c2cnc3[nH]c(=O)n(C)c3c2)c1
Oc1ccc(CNC(=O)c2[nH]c3ccccc3c2C#N)cc1[N+]([O-])=O
CCc1c(oc2ccccc12)C(=O)\C=C\c1ccc(O)c(c1)[N+]([O-])=O
Cn1c(C(=O)NCc2ccc(O)c(c2)[N+]([O-])=O)c(Br)c2ccccc12
Brc1ccc(NC(=O)COC(=O)c2cc(n[nH]2)-c2ccoc2)cc1
Oc1ccccc1-c1ncnc2[nH]ccc12
ClC(=C)COC(=O)c1cnc2[nH]ccc2c1
CC(C)SCn1cnc2cnn(C)c2c1=O
Brc1c[nH]c(CNc2cncc(n2)C#N)c1
Cn1ncc(N)c1-c1cc2ccccc2[nH]1
O=C(NC1CSC1)c1ncnn2cccc12
Nc1cn2cc(ncc2n1)-c1cscc1Cl
Cc1nc2ncc(cc2[nH]1)-c1c[nH]nn1
CN(Cc1ccncc1)c1cc(Br)ncn1
Cc1cc(sc1C=O)C(=O)Nc1cccc(N2CCNC2=O)c1C
Oc1ccc2c(ccc(NC(=O)c3cc(C=O)n4CCCCc34)c2c1)C#N
CN(C)c1cncc(NC(=O)c2ccc(C=O)cc2O)c1
Fc1cc(C(=O)Nc2cc(Cl)c3OCCOc3c2)c(F)cc1C=O
O=[#6]-c1nc2ccccn2c1\[#6]=[#6]-1\[#6]-[#8]-[#6]-1
CN(C(=O)C=C)c1ccc(cc1)C(=O)Nc1ccc(cc1)-c1cn2ccsc2n1
Clc1ccc2C(C3CCN(CC3)C(=O)CCNC(=O)C=C)C(=O)Nc2c1
Clc1ccc2C(C3CCN(CC3)C(=O)C(=O)CNC(=O)C=C)C(=O)Nc2c1
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CSCCNS(=O)(=O)c2ccccc2)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CSCCNS(=O)(=O)c2ccc(cc2)[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CSCCNS(=O)(=O)c2ccc(cc2)C#N)[C@@H](O)[C@H]1O |r|
Cc1ccc(cc1)S(=O)(=O)NCCSC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CSCCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CSCCNS(=O)(=O)c2ccccc2[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
COc1ccc(c(c1)[N+]([O-])=O)S(=O)(=O)NCCSC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CSCCNS(=O)(=O)c2ccc(Cl)cc2[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CS(=O)(=O)CCNS(=O)(=O)c2ccccc2)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CS(=O)(=O)CCNS(=O)(=O)c2ccc(cc2)[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CS(=O)(=O)CCNS(=O)(=O)c2ccc(cc2)C#N)[C@@H](O)[C@H]1O |r|
Cc1ccc(cc1)S(=O)(=O)NCCS(=O)(=O)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(N)ncnc12 |r|
Nc1ncnc2n(cnc12)[C@@H]1O[C@H](CS(=O)(=O)CCNS(=O)(=O)c2ccc(cc2)C(F)(F)F)[C@@H](O)[C@H]1O |r|
CNC(=O)c1ccc(N)cc1
NCCc1ccc(cc1)C(F)F
NCCc1cccc(Cl)c1
c1cc(cc(c1)F)CN
NCc1ccc(CCO)cc1
Cc1ccc(CCN)cc1
C\N=c1/nc(-c2ccccc2)n(s1)-c1ccccc1
CN=C(S)N=C(Nc1ccccc1)c1ccccc1
C1CC1\N=c1/nc(-c2ccccc2)n(s1)-c1ccccc1
FC1(F)CC(C1)\N=c1/nc(-c2ccccc2)n(s1)-c1ccccc1
C\N=c1/nc(-c2ccccc2)n(s1)-c1ccc(F)cc1
C\N=c1/nc(-c2ccc(Cl)cc2)n(s1)-c1ccccc1
COc1ccc(cc1)-c1n\c(=N/C)sn1-c1ccccc1
C\N=c1/nc(-c2ccc(F)cc2)n(s1)-c1ccccc1
COc1ccc(cc1)-c1n\c(=N/C)sn1-c1ccc(F)cc1
COc1ccc(cc1)-c1n\c(=N/C)sn1-c1cc(F)c(F)c(F)c1
CCOc1ccc(cc1)-c1n\c(=N/C)sn1-c1ccc(F)cc1
COc1ccc(cc1OC)-c1n\c(=N/C)sn1-c1ccc(F)cc1
COc1cc(C)cc2c(ccc(O)c12)-c1c(O)cc(O)c2[C@@H](C)N[C@H](C)Cc12 |r,wU:24.26,wD:21.23,(-6.69,-15.33,;-5.35,-16.09,;-5.34,-17.63,;-6.67,-18.4,;-6.67,-19.95,;-8,-20.72,;-5.33,-20.71,;-4,-19.94,;-2.66,-20.71,;-1.33,-19.93,;-1.34,-18.38,;-2.68,-17.62,;-2.68,-16.08,;-4,-18.4,;-2.66,-22.25,;-3.99,-23.02,;-5.33,-22.25,;-3.99,-24.55,;-2.65,-25.32,;-2.65,-26.86,;-1.32,-24.54,;.01,-25.29,;.02,-26.83,;1.33,-24.52,;1.32,-22.99,;2.65,-22.21,;-.01,-22.22,;-1.33,-23,)|
Nc1ccccc1-c1noc(n1)-c1ccncc1
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)\C=C\C(=O)OC)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)OCc2ccccc2)\C=C\C(=O)N2CCN(CC3CCN(CC3)c3cc4C(=O)N(C5CCC(=O)NC5=O)C(=O)c4cc3F)CC2)CCNC1=O |r|
COC(=O)\C=C\[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)CCC(=O)N1CCN(CC1)C(=O)C1CCN(CC1)c1cccc2C(=O)N(C3CCC(=O)NC3=O)C(=O)c12)C(C)C |r|
CCC(CC)CC1(CCCCC1)C(=O)Nc1ccccc1S
COc1ccccc1CNC(=O)CSc1c[nH]c2ccccc12
CCOc1cccc(CNC(=O)CSc2cn(C(=O)OC(C)(C)C)c3ccccc23)c1
Clc1ccc(cc1Cl)C(=O)CSc1c[nH]c2ccccc12
Cc1cccc(c1)C(=O)CSc1c[nH]c2ccccc12
Clc1ccc(NC(=O)CSc2[nH]c3ccccc3c2SCC(=O)Nc2ccc(Cl)c(Cl)c2)cc1Cl
c1cc(n2c1c(ncn2)N)[C@]3([C@@H]([C@@H]([C@H](O3)COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O)O)C#N
CC1=CCC(=C\C1=N\C(=O)C1=CC=C\C(C1)=N/C(=O)/N=C1/CC(=CC=C1)C(=O)\N=C1\CC(=CC=C1C)C(=O)\N=C1/CC=C(c2cc(cc(c12)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O)C(=O)\N=C1/CC=C(c2cc(cc(c12)S(O)(=O)=O)S(O)(=O)=O)S(O)(=O)=O |c:4,13,24,26,34,36,45,72,t:1,11|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(O)(=O)=O |r|
CC(C)C[C@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](C)C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CO[C@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CO[C@@H]1C[C@H](N(C1)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)OC(C)(C)C |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1C[C@@H](C[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O)OC(C)(C)C |r|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCCC[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC(OC(C)(C)C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)(C)C)NC(=O)c2cc3ccccc3[nH]2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)(C)C)NC(=O)c2cc3c(OC)cccc3[nH]2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC(C)(C)C)NC(=O)OCc2ccccc2)C=O)CCNC1=O |r|
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)OCc1ccccc1 |r|
Clc1cccc(COC(=O)N[C@@H](CC2CCCCC2)C(=O)N[C@@H](C[C@@H]2CCNC2=O)C=O)c1 |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CCCCC2)NC(=O)OCc2cccc(OC(C)=O)c2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H](NC(=O)OCc2ccccc2)[C@@H](C)OC(C)(C)C)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2C[C@H](CN2C(=O)OCc2ccccc2)OC(C)(C)C)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2C[C@H](CN2C(=O)OCc2ccccc2)C2CCCCC2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2CC3(CC3)CN2C(=O)OCc2ccccc2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2CC3(CCC3)CN2C(=O)OCc2ccccc2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CCCC3)CN2C(=O)OCc2ccccc2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CN2C(=O)OCc2ccccc2)CCCCC3)C=O)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@]3([H])CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)CNc1ccc(Cl)cc1 |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2CC3(CC3)CN2C(=O)COc2ccc(Cl)cc2Cl)C=O)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@]3([H])CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)COC1CCCCC1 |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@]3([H])CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)CCC1CCCCC1 |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CCCC3)CN2C(=O)OCc2ccccc2)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CCCC3)CN2C(=O)OCc2cccc(Cl)c2)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CCCC3)CN2C(=O)c2cc3c(OC)cccc3[nH]2)C=O)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CCCC3)CN2C(=O)c2cc3c(OC)cccc3[nH]2)C#N)CCCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)C2CC3(CN2C(=O)OCc2ccccc2)CCCCC3)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@H](CC2CCCCC2)NC(=O)C(F)(F)F)C#N)CCNC1=O |r|
[H][C@@]1(C[C@H](NC(=O)[C@@H]2CC3(CCC3)CN2C(=O)OC(C)(C)C)C=O)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)N[C@@H](C[C@@H]3CCNC3=O)C=O)[C@@]1([H])C2(C)C)C(=O)COc1ccc(Cl)cc1Cl |r|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)COc1ccc(Cl)c(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C=O |r|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2)C(=O)CCl)[N+]([O-])=O |c:6|
CC1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CC(C)(C)C2)[N+]([O-])=O |c:15|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CC1)C(=O)CCl)[N+]([O-])=O |c:6|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CCC1)C(=O)CCl)[N+]([O-])=O |c:6|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CCCC1)C(=O)CCl)[N+]([O-])=O |c:6|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CCCCC1)C(=O)CCl)[N+]([O-])=O |c:6|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccccc1)C(=O)CCl)[N+]([O-])=O |c:6|
Cc1ccc(cc1)C1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CC(C)(C)C2)[N+]([O-])=O |c:22|
COc1ccc(cc1)C1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CC(C)(C)C2)[N+]([O-])=O |c:23|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(OC(F)(F)F)cc1)C(=O)CCl)[N+]([O-])=O |c:6|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(cc1)C(F)(F)F)C(=O)CCl)[N+]([O-])=O |c:6|
CC1(C)CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(F)cc1F)C(=O)CCl)[N+]([O-])=O |c:6|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CC1)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CCC1)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CCCC1)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2C1CCCCC1)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccccc1)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(C)cc1)C(=O)CCl)[N+]([O-])=O |c:5|
COc1ccc(cc1)C1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CC(C)C2)[N+]([O-])=O |c:23|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(OC(F)(F)F)cc1)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(cc1)C(F)(F)F)C(=O)CCl)[N+]([O-])=O |c:5|
CC1CC(=O)C2=C(C1)Nc1cc(ccc1N(C2c1ccc(F)cc1F)C(=O)CCl)[N+]([O-])=O |c:5|
[O-][N+](=O)c1ccc2N(CC3=C(CCCC3=O)Nc2c1)C(=O)CCl |t:9|
CC1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CCC2)[N+]([O-])=O |c:15|
[O-][N+](=O)c1ccc2N(C(C3CC3)C3=C(CCCC3=O)Nc2c1)C(=O)CCl |t:13|
[O-][N+](=O)c1ccc2N(C(C3CCC3)C3=C(CCCC3=O)Nc2c1)C(=O)CCl |t:14|
[O-][N+](=O)c1ccc2N(C(C3CCCC3)C3=C(CCCC3=O)Nc2c1)C(=O)CCl |t:15|
[O-][N+](=O)c1ccc2N(C(C3CCCCC3)C3=C(CCCC3=O)Nc2c1)C(=O)CCl |t:16|
[O-][N+](=O)c1ccc2N(C(C3=C(CCCC3=O)Nc2c1)c1ccccc1)C(=O)CCl |t:9|
Cc1ccc(cc1)C1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CCC2)[N+]([O-])=O |c:22|
COc1ccc(cc1)C1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CCC2)[N+]([O-])=O |c:23|
[O-][N+](=O)c1ccc2N(C(C3=C(CCCC3=O)Nc2c1)c1ccc(OC(F)(F)F)cc1)C(=O)CCl |t:9|
[O-][N+](=O)c1ccc2N(C(C3=C(CCCC3=O)Nc2c1)c1ccc(cc1)C(F)(F)F)C(=O)CCl |t:9|
[O-][N+](=O)c1ccc2N(C(C3=C(CCCC3=O)Nc2c1)c1ccc(F)cc1F)C(=O)CCl |t:9|
COC(=O)c1ccc2N(C(C3=C(CCCC3=O)Nc2c1)c1ccc(cc1)C(F)(F)F)C(=O)CCl |t:10|
FC(F)(F)c1ccc(cc1)C1N(C(=O)CCl)c2ccc(cc2NC2=C1C(=O)CCC2)C#N |c:25|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C#C |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)C(=O)C(=O)Nc1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)C#C |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C#N |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)C=O |r|
CNS(=O)(=O)\C=C\[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)OCc1ccccc1 |r|
COc1cccc2[nH]c(cc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C#C |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)\C=C\C(=O)OCc1ccccc1 |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)C#N |r|
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CCC(N)=O)\C=C\S(C)(=O)=O |r|
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc3c(F)cccc3s1)C2(C)C
CC1([C@@H]2[C@H]1[C@H](N(C2)C(=O)[C@H](C(C)(C)C)NC(=O)C(F)(F)F)C(=S)N[C@@H](C[C@@H]3CCNC3=O)C(=O)c4nc5c(cccc5s4)F)C
FC(F)(F)CCOc1cc(Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Clc1cc(OCC2CC2)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Clc1cc(Cl)cc(c1)-n1cc(-c2ccc(=O)[nH]c2)c(=O)n(-c2cccnc2)c1=O
Clc1cc(Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Clc1cccc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1ccccc1C#N
FC(F)(F)c1ncsc1COc1cc(Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
FC(F)n1c(COc2cc(Cl)cc(c2)-n2cc(-c3ccc[nH]c3=O)c(=O)n(-c3cccnc3)c2=O)nc2ccccc12
Cc1scnc1COc1cc(Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Cc1nc(C)c(COc2cc(Cl)cc(c2)-n2cc(-c3ccc[nH]c3=O)c(=O)n(-c3cccnc3)c2=O)s1
FC(F)n1ccnc1COc1cc(Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Cn1c(COc2cc(Cl)cc(c2)-n2cc(-c3ccc[nH]c3=O)c(=O)n(-c3cccnc3)c2=O)ncc1[N+]([O-])=O
Clc1cc(OCc2ccccc2Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Cn1cc(COc2cc(Cl)cc(c2)-n2cc(-c3ccc[nH]c3=O)c(=O)n(-c3cccnc3)c2=O)c(n1)C(F)(F)F
FC(F)(F)c1scnc1COc1cc(Cl)cc(c1)-n1cc(-c2ccc[nH]c2=O)c(=O)n(-c2cccnc2)c1=O
Cc1scnc1COc1cc(Cl)cc(c1)-n1cc(-c2ccc(=O)[nH]c2)c(=O)n(-c2cccnc2)c1=O
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c1nc[nH]c2=O)S(=O)(=O)c1ccc(OC)c(c1)C#N |r|
CNc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(Br)c(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
CNc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(C)c(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
CNc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(C)c(Cl)c2)[C@@H](O)[C@H]1O |r|
CNc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(OC)c(c2)[N+]([O-])=O)[C@@H](O)[C@H]1O |r|
CNc1ncnc2n(cnc12)[C@@H]1O[C@H](CNS(=O)(=O)c2ccc(OC)c(c2)C#N)[C@@H](O)[C@H]1O |r|
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC)ncnc12)S(=O)(=O)c1ccc(Br)c(c1)[N+]([O-])=O |r|
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC)ncnc12)S(=O)(=O)c1ccc(C)c(c1)[N+]([O-])=O |r|
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC)ncnc12)S(=O)(=O)c1ccc(C)c(Cl)c1 |r|
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC)ncnc12)S(=O)(=O)c1ccc(OC)c(c1)[N+]([O-])=O |r|
CCN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC)ncnc12)S(=O)(=O)c1ccc(OC)c(c1)C#N |r|
CN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2ccccc2)c2c(N)ncnc12)S(=O)(=O)c1ccc(Br)c(c1)[N+]([O-])=O |r|
CN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2ccccc2)c2c(N)ncnc12)S(=O)(=O)c1ccc(C)c(c1)[N+]([O-])=O |r|
CN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2ccccc2)c2c(N)ncnc12)S(=O)(=O)c1ccc(C)c(Cl)c1 |r|
COc1ccc(cc1[N+]([O-])=O)S(=O)(=O)N(C)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2ccccc2)c2c(N)ncnc12 |r|
COc1ccc(cc1C#N)S(=O)(=O)N(C)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2ccccc2)c2c(N)ncnc12 |r|
CN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2cnc3ccccc3c2)c2c(N)ncnc12)S(=O)(=O)c1ccc(Br)c(c1)[N+]([O-])=O |r|
CN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2cnc3ccccc3c2)c2c(N)ncnc12)S(=O)(=O)c1ccc(C)c(c1)[N+]([O-])=O |r|
CN(C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2cnc3ccccc3c2)c2c(N)ncnc12)S(=O)(=O)c1ccc(C)c(Cl)c1 |r|
COc1ccc(cc1[N+]([O-])=O)S(=O)(=O)N(C)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2cnc3ccccc3c2)c2c(N)ncnc12 |r|
COc1ccc(cc1C#N)S(=O)(=O)N(C)C[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cc(C#Cc2cnc3ccccc3c2)c2c(N)ncnc12 |r|
CCCCCCCCCCCCNC(=O)[C@@H](Cc1ccc(O)c(O)c1)OC(=O)\C=C\c1ccc(O)c(O)c1 |r|
CCc1cccc(NC(=O)[C@@H](Cc2ccc(O)c(O)c2)OC(=O)\C=C\c2ccc(O)c(O)c2)c1 |r|
[H][C@@]1(CN(NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)C(=O)[C@H](F)Cl)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)NN(C[C@]3([H])CCNC3=O)C(=O)CCl)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C |r|
[H][C@@]1(CN(NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C(F)(F)C(F)(F)F)[C@@H](C)CC)C(=O)[C@H](F)Cl)CCNC1=O |r|
[H][C@]12CN([C@H](C(=O)NN(C[C@]3([H])CCNC3=O)C(=O)[C@H](F)Cl)[C@@]1([H])C2(C)C)C(=O)[C@@H](NC(=O)C(F)(F)F)C(CC)CC |r|
[H][C@@]1(CN(NC(=O)[C@H]2N(C[C@]3([H])CCC[C@]23[H])C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)CC)C(=O)[C@H](F)Cl)CCNC1=O |r|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)[C@@H](NC(=O)[C@@H](F)Cl)[C@@H](C)CC)C(=O)NN(C[C@]1([H])CCCNC1=O)C(=O)[C@@H](F)Cl |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1cccs1)C(=O)c1cc(=O)[nH]c2ccccc12 |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1cccs1)C(=O)c1cncc2cc[nH]c12 |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1cccs1)C(=O)c1cnccc1Cl |r|
Fc1cncc(c1)C(=O)N1CCN([C@@H](C1)C(=O)NCc1cccs1)c1ccc(Cl)c(Cl)c1 |r|
COc1ccncc1C(=O)N2CCN([C@@H](C2)C(=O)NCc3cccs3)c4ccc(c(c4)Cl)Cl
Oc1cncc(c1)C(=O)N1CCN([C@@H](C1)C(=O)NCc1cccs1)c1ccc(Cl)c(Cl)c1 |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NS(=O)(=O)c1cccs1)C(=O)c1cccnc1 |r|
CN(Cc1cccs1)C(=O)[C@@H]1CN(CCN1c1ccc(Cl)c(Cl)c1)C(=O)c1cccnc1 |r|
Fc1ccc(CNC(=O)[C@@H]2CN(CCN2c2ccc(Cl)c(Cl)c2)C(=O)c2cccnc2)s1 |r|
Clc1ccc(cc1Cl)N1CCN(C[C@H]1C(=O)NCc1ccc(Br)s1)C(=O)c1cccnc1 |r|
COc1ccc(NC(=O)[C@@H]2CN(CCN2c2ccc(Cl)c(Cl)c2)C(=O)c2cccnc2)cc1 |r|
COc1ccc(NC(=O)[C@@H]2CN(CCN2c2ccc(Cl)c(Cl)c2)C(=O)c2cnccc2OC)cc1 |r|
COc1ccncc1C(=O)N1CCN([C@@H](C1)C(=O)Nc1cc(F)c(OC)c(F)c1)c1ccc(Cl)c(Cl)c1 |r|
COc1cc(OC)c(NC(=O)[C@@H]2CN(CCN2c2ccc(Cl)c(Cl)c2)C(=O)c2cnccc2OC)cc1F |r|
COc1ccncc1C(=O)N1CCN([C@@H](C1)C(=O)NCc1ccc(F)s1)c1ccc(Cl)c(Cl)c1 |r|
COc1ccncc1C(=O)N1CCN([C@@H](C1)C(=O)Nc1ccc(OC(F)F)cc1)c1ccc(Cl)c(Cl)c1 |r|
CC(C)C[C@@H]1NC(=O)[C@@H](Cc2ccc(O)cc2)NC(=O)CSC[C@H](CC(=O)[C@H](CCC(O)=O)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc2c[nH]cn2)NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CCC(N)=O)NC1=O)C(C)C)C(C)=O |r|
COc1ccc2c(O[C@@H]3C[C@@H]4[C@@H](C3)C(=O)N(C)CCCC\C=C/[C@@H]3C[C@]3(NC4=O)C(=O)NS(=O)(=O)C3CC3)cc(nc2c1C)-c1nc(cs1)C(C)C |r,c:22|
CC(C)(O)c1ccccc1CC[C@@H](SCCCC([O-])=O)c1cccc(\C=C\c2ccc3ccc(Cl)cc3n2)c1 |r|
[#6]\[#6](-[#6])=[#6]\[#6]=[#6](-[#8]-[#6](=O)-[#6]C([#6])([#6])[#8])-c1cc(-[#8])c2c(-[#8])ccc(-[#8])c2c1-[#8] |w:4.3|
COc1ccc(cc1)-c1nc(N)n(C)c1SSc1c(nc(N)n1C)-c1ccc(OC)cc1
[H][C@]1(NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CNC(=O)[C@H](CS([O-])(=O)=O)NC(=O)\C=C\c2csc(n2)[C@H](Cc2ccc(O)cc2)NC(=O)C1=O)NC(=O)[C@H](C)N)[C@@H](C)CC |r,t:27|
[H][C@]1(NC(=O)[C@H](CCC)NC(=O)[C@H](CNC(=O)[C@H](CS([O-])(=O)=O)NC(=O)\C=C\c2csc(n2)[C@H](Cc2ccc(O)cc2)NC(=O)C1=O)NC(=O)[C@H](C)N)[C@@H](C)CC |r,t:26|
CC(C)C[C@@H]1NC(=O)[C@@H](CCCCNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3cc(Cl)c(O)cc23)N(C)C(=O)[C@H](CC(C)C)NC1=O)NC(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H]1NC(=O)[C@@H](CCCCNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3cc(Cl)ccc23)N(C)C(=O)[C@H](CC(C)C)NC1=O)NC(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
COc1ccc(CNC(=O)C2CCN(CC2)[C@H](C)c2cccc3ccccc23)cc1 |r|
COc1cccc(CNC(=O)C2CCN(CC2)[C@H](C)c2ccc3ccccc3c2)c1 |r|
C[C@@H](NC(=O)c1cc(CN)ccc1C)c1cccc2ccccc12 |r|
CNCc1ccc(C)c(c1)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
COc1ccc([C@@H](C)NC(=O)c2cc(N)ccc2C)c2ccccc12 |r|
COc1ccc(cc1N)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
C[C@@H](NS(=O)(=O)c1cccc(c1)[N+]([O-])=O)c1cccc2ccccc12 |r|
C[C@@H](NS(=O)(=O)c1ccc(cc1)[N+]([O-])=O)c1cccc2ccccc12 |r|
C[C@@H](NS(=O)(=O)c1cccc(N)c1)c1cccc2ccccc12 |r|
C[C@@H](NS(=O)(=O)c1ccc(N)cc1)c1cccc2ccccc12 |r|
CC(C)NC(=O)c1ccc(C)c(c1)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
CCCN(CCC)C(=O)c1ccc(C)c(c1)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
CCCN(CCC)C(=O)c1cccc(c1)C(=O)N[C@H](C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccccc1)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccccc1)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)OC(C)(C)C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)[C@H](N)Cc1ccccc1)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C)c1cccc2ccccc12 |r|
C[C@@H](NC(=O)[C@H](N)Cc1c[nH]c2ccccc12)c1cccc2ccccc12 |r|
N[C@H]1CN2CC(C(=O)N(Cc3ccccc3)Cc3ccccc3)=C(N2C1=O)C(O)=O |r,c:24|
OC(=O)C1=C(CN2C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C(=O)N12)C(=O)N(Cc1ccccc1)Cc1ccccc1 |r,t:3|
OC(=O)C1=C(CN2C[C@H](NC(=O)[C@H](C[C@@H]3CCNC3=O)NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C(=O)N12)C(=O)N(Cc1ccccc1)Cc1ccccc1 |r,t:3|
C[C@H]1[C@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)c2cc3ccccc3[nH]2)C(=O)N1S(O)(=O)=O |r|
[H][C@]12SCC(Cl)=C(N1C(=O)[C@H]2NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc2ccccc2[nH]1)C(O)=O |r,c:5|
O=C(N[C@@H]1CONC1=O)[C@H](Cc1ccccc1)NC(=O)c1cc2ccccc2[nH]1 |r|
[H][C@]12SC(C)(C)[C@@H](N1C(=O)[C@H]2NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc2ccccc2[nH]1)C(O)=O |r|
OC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc2ccccc2[nH]1 |r|
OC(=O)C1=C(CN2C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C(=O)N12)C(=O)NCc1ccccc1 |r,t:3|
OC(=O)C1=C(CN2C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C(=O)N12)C(=O)NCc1ccncc1 |r,t:3|
CN(Cc1ccccc1)C(=O)C1=C(N2N(C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C2=O)C1)C(O)=O |r,t:12|
CCN(CC)C(=O)C1=C(N2N(C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C2=O)C1)C(O)=O |r,t:7|
OC(=O)C1=C(CN2C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C(=O)N12)C(=O)N1CCCC1 |r,t:3|
OC(=O)C1=C(CN2C[C@H](NC(=O)[C@H](Cc3ccccc3)NC(=O)c3cc4ccccc4[nH]3)C(=O)N12)C(=O)OCC=C |r,t:3|
COC(=O)N[C@H](C(=O)N1CCC2(CC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(N)=O)C(C)(C)C |r|
CNC(=O)C(=O)[C@H](CCC(C)(F)F)NC(=O)[C@@H]1CC2(CC2)CCN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C |r|
COC(=O)N[C@H](C(=O)N1CCC2(CC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C |r|
COC(=O)N[C@H](C(=O)N1CCC2(CCCC2)CC1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C |r|
[H][C@@]12CCC[C@]1([H])[C@H](N(C2)C(=O)[C@H](CC(F)(F)F)NC(=O)OC)C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC |r|
CNC(=O)C(=O)[C@H](CCC(C)(F)F)NC(=O)C1C2CC(C)(C)C2CN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C |r|
CC(C)[C@]1(O)C(OC(=O)c2ccc[nH]2)[C@@]2(O)[C@@]3(C)C[C@]4(O)O[C@@]5([C@H](O)[C@@H](C)CC[C@]35O)[C@@]2(O)[C@@]14C |r,THB:20:19:29:31.14,33:19:29:31.14|
[H][C@]12CC[C@]3([H])[C@@]([C@@H]1O)(C(=O)C2=C)[C@@]1(O)OC[C@]32[C@@H](O)CCC(C)(C)[C@@]2([H])[C@@H]1O |r,THB:12:11:4.3.2:7,10:9:4.3.2:7|
Cc1ccc(N)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NCC(C)(C)C)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NC2CCCCC2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NC2CCC(C#N)CC2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
COC1CCC(Nc2ccc(C)c(-c3noc(C(C)c4cccc5ccccc45)n3)c2)CC1
Cc1ccc(NC2CCC(C(=O)O)CC2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NC2CCCC(C(=O)O)C2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(Nc2ccc(C(=O)O)cc2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
COC(=O)c1ccc(Nc2ccc(C)c(-c3noc(C(C)c4cccc5ccccc45)n3)c2)cc1
Cc1ccc(NCc2ccc(C(=O)O)cc2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
COC(=O)c1ccc(CNc2ccc(C)c(-c3noc(C(C)c4cccc5ccccc45)n3)c2)cc1
Cc1ccc(NCc2cccc(C(=O)O)c2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NCc2ccc(C#N)cc2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NCc2ccc(O)cc2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NCc2ccc(S(C)(=O)=O)cc2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NCc2ccc(C(=O)O)o2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
Cc1ccc(NCc2ccc(C(=O)O)s2)cc1-c1noc(C(C)c2cccc3ccccc23)n1
CC(c1nc(-c2cccc(NCc3ccc(C(=O)O)cc3)c2)no1)c1cccc2ccccc12
CC(c1nc(-c2cccc(NCc3ccc(C(=O)O)s3)c2)no1)c1cccc2ccccc12
CC(c1nc(-c2cccc(NCc3ccc(C(=O)O)o3)c2)no1)c1cccc2ccccc12
CC(c1nc(-c2cc(NCc3ccc(C(=O)O)cc3)ccc2Br)no1)c1cccc2ccccc12
CC(c1nc(-c2cc(NCc3ccc(C(=O)O)cc3)cc(C(F)(F)F)c2)no1)c1cccc2ccccc12
Cc1ccc(-c2noc(C(C)c3cccc4ccccc34)n2)cc1NCc1ccc(C(=O)O)cc1
CC(c1nc(-c2cc(NCc3ccc(C(=O)O)s3)cc(C(F)(F)F)c2)no1)c1cccc2ccccc12
Cc1ccc(-c2noc(C(C)c3cccc4ccccc34)n2)cc1NCc1ccc(C(=O)O)s1
COc1ccc(-c2noc(C(C)c3cccc4ccccc34)n2)cc1NCc1ccc(C(=O)O)s1
CC(c1nc(-c2ccc(NCc3ccc(C(=O)O)cc3)cc2)no1)c1cccc2ccccc12
CC(c1nc(-c2ccc(NCc3ccc(C(=O)O)s3)cc2)no1)c1cccc2ccccc12
CC(c1nc(-c2ccc(N(C)Cc3ccc(C(=O)O)s3)cc2)no1)c1cccc2ccccc12
CC(c1nc(-c2ccc(Nc3ccc(C(=O)O)cc3)cc2)no1)c1cccc2ccccc12
CC(c1nc(-c2ccc(-c3ccc(C(=O)O)cc3)cc2)no1)c1cccc2ccccc12
CC(c1nc(-c2ccc(-c3ccc(C(=O)O)s3)cc2)no1)c1cccc2ccccc12
CC(c1nc(-c2ccc(-c3ccc(C#N)s3)cc2)no1)c1cccc2ccccc12
CONC(=O)c1ccc(-c2ccc(-c3noc(C(C)c4cccc5ccccc45)n3)cc2)cc1
CC(c1noc(-c2ccc(-c3ccc(C#N)s3)cc2)n1)c1cccc2ccccc12
CC(c1noc(-c2ccc(-c3ccc(C(=O)O)s3)cc2)n1)c1cccc2ccccc12
CC(c1ncc(-c2ccc(-c3ccc(C#N)s3)cc2)o1)c1cccc2ccccc12
CC(c1ncc(-c2ccc(-c3ccc(C(=O)O)s3)cc2)o1)c1cccc2ccccc12
Cc1ccc(-c2noc(C(C)c3cccc(-c4ccccc4)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)(C)c3ccc(-c4ccccc4)cc3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)c3ccc(CC(C)C)cc3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)c3cccc(-c4cccs4)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(Cc3cccc(-c4cccs4)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(-c3cccc4ccccc34)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(-c3ccccc3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(-c3ccc(-c4ccccc4)cc3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(c3ccccc3)c3ccccc3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(O)c3ccccc3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)c3cccc(C(O)c4ccccc4)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)c3cccc(Oc4ccccc4)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)c3ccc4c(c3)[nH]c3ccc(Cl)cc34)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc(C(C)c3ccc(N4Cc5ccccc5C4=O)cc3)n2)cc1NCc1ccc(C(=O)O)s1
COc1ccc2cc(C(C)c3nc(-c4ccc(C)c(NCc5ccc(C(=O)O)s5)c4)no3)ccc2c1
COc1ccc2cc([C@@H](C)c3nc(-c4ccc(C)c(NCc5ccc(C(=O)O)s5)c4)no3)ccc2c1
COc1ccc2cc([C@H](C)c3nc(-c4ccc(C)c(NCc5ccc(C(=O)O)s5)c4)no3)ccc2c1
Cc1ccc(-c2noc(C(C)c3ccc(-c4ccccc4)c(F)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc([C@H](C)c3ccc(-c4ccccc4)c(F)c3)n2)cc1NCc1ccc(C(=O)O)s1
Cc1ccc(-c2noc([C@@H](C)c3ccc(-c4ccccc4)c(F)c3)n2)cc1NCc1ccc(C(=O)O)s1
CCCCCC\C=C/CCCCCCCc1cccc(O)c1C(O)=O
O=c1cc(-c2ccc(O)cc2)oc2c([C@@H]3OC[C@H](O)[C@H](O)[C@H]3O)c(O)c([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(O)c12
Oc1cc(cc(O)c1O)C(=O)Oc1cc(cc(O)c1O)C(=O)OC[C@H]1O[C@@H](OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)[C@H](OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)[C@@H](OC(=O)c2cc(O)c(O)c(OC(=O)c3cc(O)c(O)c(O)c3)c2)[C@@H]1OC(=O)c1cc(O)c(O)c(OC(=O)c2cc(O)c(O)c(O)c2)c1 |r|
CCOC(=O)/C=C/[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](N)Cc1ccccc1
CCOC(=O)/C=C/[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1ccc(F)cc1)NC(=O)OC(C)(C)C
CC(C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)N[C@@H](Cc1ccccc1)C(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C=O |r|
CC(C)(c1ccccc1CC[C@H](c2cccc(c2)/C=C/c3ccc4ccc(cc4n3)Cl)SCC5(CC5)CC(=O)O)O
N[C@H]1C(=O)N[C@@H]2Cc3ccc(c(Cl)c3)Oc3cc4cc(c3O)Oc3ccc(cc3Cl)[C@@H](O)[C@@H]3NC(=O)[C@H](NC(=O)[C@@H]4NC(=O)[C@@H](NC2=O)c2cc(O)cc(c2)Oc2cc1ccc2O)c1ccc(O)c(c1)-c1c(O)cc(O)cc1[C@@H](C(=O)O)NC3=O
CC(=O)N[C@H](CC(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@H](C=O)CCCN=C(N)N
COc1ccc2C[C@H]3N(C)CCc4cc(OC)c(Oc5c6OCOc6cc6CCN(C)[C@@H](Cc7ccc(Oc1c2)cc7)c56)cc34 |r|
CC(C)c1c(O)c(O)c(C=O)c2c(O)c(c(C)cc12)-c1c(C)cc2c(C(C)C)c(O)c(O)c(C=O)c2c1O |(-4.44,-1.63,;-5.78,-.86,;-7.11,-1.63,;-5.78,.68,;-7.11,1.45,;-8.44,.68,;-7.11,2.99,;-8.44,3.76,;-5.78,3.76,;-5.78,5.3,;-4.44,6.07,;-4.44,2.99,;-3.11,3.76,;-3.11,5.3,;-1.77,2.99,;-1.77,1.45,;-.44,.68,;-3.11,.68,;-4.44,1.45,;-.44,3.76,;-.44,5.3,;-1.77,6.07,;.89,6.07,;2.23,5.3,;3.56,6.07,;3.56,7.61,;4.89,8.38,;2.23,8.38,;4.89,5.3,;6.23,6.07,;4.89,3.76,;6.23,2.99,;3.56,2.99,;3.56,1.45,;4.89,.68,;2.23,3.76,;.89,2.99,;.89,1.45,)|
CC1=NN(c2ccc(Cl)cc2)C(=O)/C1=Cc1ccc(OCc2cn(CC(=O)NCc3ccc(C(=O)O)cc3)nn2)cc1
Cc1cc(C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C=O)C[C@@H]2CCCNC2=O)no1
CC(C)[C@H]1C(=O)N2C[C@]3(C[C@H]2C#N)C(=O)Nc2ccc(cc23)CCCCCN1C(=O)C1CN(c2ccccc2)N=N1
N#C[C@@H]1C[C@]23CN1C(=O)[C@H](c1ccccc1)N(C(=O)C1CN(c4ccc(F)cc4)N=N1)CCCCCc1ccc(c2c1)NC3=O
CCC[C@H]1C(=O)N2C[C@]3(C[C@H]2C#N)C(=O)Nc2ccc(cc23)CCCCCN1C(=O)c1cc2c(F)cc(F)c(F)c2[nH]1
CC(C)[C@H]1C(=O)N2C[C@]3(C[C@H]2C#N)C(=O)Nc2ccc(cc23)CCCCCN1C(=O)c1cc2c(F)cc(F)cc2[nH]1
CC(C)[C@H]1C(=O)N2C[C@]3(C[C@H]2C#N)C(=O)Nc2ccc(cc23)CCCCCN1C(=O)c1cc2ccc(C(F)(F)F)cc2[nH]1
CC(C)[C@H]1C(=O)N2C[C@]3(C[C@H]2C#N)C(=O)Nc2ccc(cc23)CCCCCN1C(=O)c1cc2c(F)cc(F)c(F)c2[nH]1
CC1(C)[C@@H]2[C@H]1CN(C(=O)COc1ccc(OC(F)(F)F)cc1)[C@H]2C(=O)N[C@@H](C=O)C[C@H]1CCNC1=O
O=C[C@@H](C[C@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@@H]2CN1C(=O)COc1ccc(Cl)cc1Cl
CC1(C)[C@@H]2[C@H]1CN(C(=O)OCc1ccccc1)[C@H]2C(=O)N[C@@H](C=O)C[C@H]1CCNC1=O
O=C[C@@H](C[C@H]1CCNC1=O)NC(=O)[C@H]1[C@@H]2CCC[C@@H]2CN1C(=O)OCc1ccccc1
C=CS(=O)(=O)N(c1ccc(-c2ccccc2)cc1)[C@@H](C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
CCOc1cc(O)c2c(=O)c(O)c(-c3cc(O)c(O)c(O)c3)oc2c1
CC(C)CCOc1cc(O)c2c(=O)c(O)c(-c3cc(O)c(O)c(O)c3)oc2c1
O=c1c(O)c(-c2cc(O)c(O)c(O)c2)oc2cc(OCC3CCCC3)cc(O)c12
CC1COP(=O)(Oc2cc(O)c3c(=O)c(O)c(-c4cc(O)c(O)c(O)c4)oc3c2)OC1
O=c1c(O)c(-c2cc(O)c(O)c(O)c2)oc2cc(OP(=O)(Oc3ccccc3)Oc3ccccc3)cc(O)c12
O=C1c2c(O)cc(O)c([Se][Se]c3c(O)cc(O)c4c3OC(c3cc(O)c(O)c(O)c3)C(O)C4=O)c2CC(c2cc(O)c(O)c(O)c2)C1O
O[C@@H]1[C@H](Oc2cc(O)cc(O)c2C1=O)c1cc(O)c(O)c(O)c1
O=C1c2c(O)cc(OP(=O)(Oc3ccccc3)Oc3ccccc3)cc2O[C@H](c2cc(O)c(O)c(O)c2)[C@H]1O
C#CC(=O)N(c1ccc(-c2ccccc2)cc1)[C@@H](C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)CC#N)c1ccc(-c2ccccc2)cc1)c1ccccc1
COc1ccc(/C=C(C#N)C(=O)N(c2ccc(-c3ccccc3)cc2)[C@@H](C(=O)N[C@@H](C)c2ccccc2)c2cccnc2)cc1
CCOC(=O)/C=C/C(=O)N(c1ccc(-c2ccccc2)cc1)[C@@H](C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C=C(Cl)C(=O)N(c1ccc(-c2ccccc2)cc1)[C@@H](C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)CCl)c1ccc(-c2ccccc2)cc1)c1ccccc1
O=C1NCC[C@H]1C[C@H](NC(=O)[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1Cl)C(=O)CF
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)COc1ccc(Cl)cc1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)COc3ccc(Cl)cc3)C[C@@H]21
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@H](Cc1ccc(F)cc1)NC(=O)c1cc2ccccc2[nH]1
CC(C)(C)c1ccc(N(C(=O)c2ccco2)[C@@H](C(=O)NC2CC2)c2cccnc2)cc1
CC(C)(C)c1ccc(N(C(=O)c2ccco2)[C@@H](C(=O)NC2CCCC2)c2cccnc2)cc1
CC(C)(C)c1ccc(N(C(=O)c2ccco2)[C@@H](C(=O)NC2CCCCC2)c2cccnc2)cc1
C[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)c1ccco1)c1ccc(C(C)(C)C)cc1)c1ccccc1
C[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)c1ccco1)c1ccc(-n2cccc2)cc1)c1ccccc1
CC(C)(C)NC(=O)[C@@H](c1cccnc1)N(C(=O)c1c[nH]cn1)c1ccc(C(C)(C)C)cc1
CC(C)(C)NC(=O)[C@@H](c1cccnc1)N(C(=O)c1ccno1)c1ccc(-c2ccccc2)cc1
CC(C)(C)NC(=O)[C@@H](c1cccnc1)N(C(=O)c1cnco1)c1ccc(-c2ccccc2)cc1
CC(C)(C)NC(=O)[C@@H](c1cnccn1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1
Cn1cc2cc(\N=c3/[nH]c(=O)n(Cc4nnn[nH]4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
CCn1nnnc1Cn1c(=O)[nH]\c(=N/c2cc3cn(C)nc3cc2Cl)n(Cc2cc(F)c(F)cc2F)c1=O
COc1ccc(Nc2nc(=O)n(Cc3ccc[nH]c3=O)c(=O)n2Cc2cc(F)c(F)c(F)c2)c(OC)c1
O=C(O)c1ccc(Nc2nc(=O)n(Cc3ccc[nH]c3=O)c(=O)n2Cc2cc(F)c(F)c(F)c2)cc1
COc1ccc(Nc2nc(=O)n(Cc3ccc[nH]c3=O)c(=O)n2Cc2cc(F)c(F)c(F)c2)cc1
Cn1cnc(Cn2c(=O)nc(Nc3cc4sc(N)nc4cc3Cl)n(Cc3cc(F)c(F)c(Cl)c3)c2=O)n1
Cc1nc2cc(Br)c(Nc3nc(=O)n(Cc4ncn(C)n4)c(=O)n3Cc3cc(F)c(F)c(F)c3)cc2s1
Cn1cnc(Cn2c(=O)nc(Nc3cc4sc(NCC(F)F)nc4cc3Cl)n(Cc3cc(F)c(F)c(F)c3)c2=O)n1
CC(=O)Nc1nc2cc(Cl)c(Nc3nc(=O)n(Cc4ncn(C)n4)c(=O)n3Cc3cc(F)c(F)c(Cl)c3)cc2s1
CN(C)CCn1cc2cc(Nc3nc(=O)n(Cc4ccc[nH]c4=O)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
CC(C)(O)Cn1cc2cc(Nc3nc(=O)n(Cc4ccc[nH]c4=O)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
Cn1cc2cc(Nc3nc(=O)n(Cc4ccc[nH]c4=O)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
O=c1[nH]cccc1Cn1c(=O)nc(Nc2cc3cn(C4CCOCC4)nc3cc2Cl)n(Cc2cc(F)c(F)c(F)c2)c1=O
CC(=O)NCCn1cc2cc(Nc3nc(=O)n(Cc4ccc[nH]c4=O)c(=O)n3Cc3cc(F)c(F)c(F)c3)c(Cl)cc2n1
CCn1cc2cc(Nc3nc(=O)n(-c4cncc(Cl)c4)c(=O)n3Cc3cc(C#N)ccc3Cl)ccc2n1
CCn1cc2cc(Nc3nc(=O)n(-c4cncc(Cl)c4)c(=O)n3Cc3cc(C#N)ccc3C)ccc2n1
Cn1cnc(Cn2c(=O)cc(Nc3cc4cn(C)nc4cc3Cl)n(Cc3cc(F)c(F)cc3F)c2=O)n1
Cn1cnc(Cn2c(=O)cc(Nc3cc4cn(C)nc4cc3OC(F)(F)F)n(Cc3cc(F)c(F)cc3F)c2=O)n1
Cn1cnc(Cn2c(=O)cc(Nc3cc4cn(C)nc4cc3F)n(Cc3cc(Cl)c(F)cc3F)c2=O)n1
Cc1cc(Cn2c(Nc3cc4cn(C)nc4cc3Cl)cc(=O)n(Cc3ncn(C)n3)c2=O)c(F)cc1F
Cn1cnc(Cn2c(=O)cc(Nc3cc4cn(C)nc4cc3C(F)(F)F)n(Cc3cc(Cl)c(Cl)cc3F)c2=O)n1
CNC(=O)[C@@H](Cc1cccc(F)c1)NC(=O)C1CN(C(=O)c2cncc3cccc(O)c23)CCN1Cc1ccc(Cl)cc1Cl
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@H]1CCCC[C@H]1NC(=O)c1cncc2ccccc12
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@H]1CCCC[C@H]1NC(=O)c1cncc2cc(O)ccc12
CNC(=O)c1cc(C)cc([N+](=O)[O-])c1N1CC[C@]2(CCN(C(=O)c3cncc4cc(O)ccc34)C2)C1
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCC[C@H](NC(=O)c2cncc3cccc(O)c23)C1
Cc1ccncc1N1C(=O)N[C@@H](CC2CCCCC2)C1=O
Cc1c(Br)cncc1NC[C@@H](N)CC1CCCCC1
O=C1N[C@@H](CC2CCCCC2)C(=O)N1c1cncc2ccccc12
CC(C)(C)C1CC2(C1)NC(=O)N(c1cncc3ccccc13)C2=O
CC1(CC2(C1)NC(=O)N(C2=O)c1cncc2ccccc12)c1ccccc1 |(.27,-3.52,;1.35,-2.43,;-.17,-2.19,;.07,-.66,;1.6,-.91,;-1.47,-.66,;-1.94,.8,;-3.41,1.28,;-.7,1.71,;.55,.8,;2.02,1.28,;-.7,3.25,;.64,4.02,;.64,5.56,;-.7,6.33,;-2.03,5.56,;-3.36,6.33,;-4.7,5.56,;-4.7,4.02,;-3.36,3.25,;-2.03,4.02,;2.26,-3.67,;3.79,-3.51,;4.7,-4.76,;4.07,-6.16,;2.54,-6.33,;1.63,-5.08,)|
O=c1n([se]c2ccccc12)-c1ccccc1
Cc1cccc2c(=O)n(-c3ccccc3)sc12
O=c1c2cccc(Br)c2sn1-c1ccccc1
O=c1c2cccc(-c3ccccc3)c2sn1-c1ccccc1
O=c1c2cnccc2sn1-c1ccccc1
Cc1cccc2c(=O)n(CCC(C)C)sc12
CC(C)CCn1sc2c(Br)cccc2c1=O
O=c1c2ccccc2sn1-c1ccccn1
O=C1C[C@H](Cn2sc3ccccc3c2=O)CN1
COCCn1sc2ccccc2c1=O
COC(=O)CCn1sc2ccccc2c1=O
COC(=O)Cn1sc2ccccc2c1=O
N#Cc1ccccc1-c1cc(-c2cccc(Cl)c2)cn(-c2cccnc2)c1=O
c1ccc(c(c1)C#N)C2=CN(C(=O)C(=C2)c3cc(cc(c3)Cl)Cl)c4cccnc4
COCCCc1cc(Cl)cc(-c2cc(-c3ccccc3C#N)cn(-c3cccnc3)c2=O)c1
COCCOc1cc(cc(c1)Cl)C2=CC(=CN(C2=O)c3cccnc3)c4ccccc4C#N
Clc1cc(OCc2ccccc2)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1ccccc1C#N
Clc1cc(OCCc2ccccc2)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1ccccc1C#N
COc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
CCCCOc1cc(Cl)cc(c1)-c1cc(cn(-c2cccnc2)c1=O)-c1c[nH]c(=O)[nH]c1=O
CC(C)COc1cc(Cl)cc(-c2cc(-c3c[nH]c(=O)[nH]c3=O)cn(-c3cccnc3)c2=O)c1
c1ccc(cc1)CCOc2cc(cc(c2)Cl)C3=CC(=CN(C3=O)c4cccnc4)C5=CNC(=O)NC5=O
COCCCc1cc(Cl)cc(-c2cc(-c3c[nH]c(=O)[nH]c3=O)cn(-c3cccnc3)c2=O)c1
O=c1[nH]cc(-c2cc(-c3cc(Cl)cc(COc4ccccc4)c3)c(=O)n(-c3cccnc3)c2)c(=O)[nH]1
Cc1ccccc1OCc1cc(Cl)cc(-c2cc(-c3c[nH]c(=O)[nH]c3=O)cn(-c3cccnc3)c2=O)c1
Cc1cccc(OCc2cc(Cl)cc(-c3cc(-c4c[nH]c(=O)[nH]c4=O)cn(-c4cccnc4)c3=O)c2)c1
O=c1[nH]cc(-c2cc(-c3cc(Cl)cc(COc4ccccc4F)c3)c(=O)n(-c3cccnc3)c2)c(=O)[nH]1
O=c1[nH]cc(-c2cc(-c3cc(Cl)cc(COc4cccc(F)c4)c3)c(=O)n(-c3cccnc3)c2)c(=O)[nH]1
O=c1[nH]cc(-c2cc(-c3cc(Cl)cc(COc4c(F)cccc4F)c3)c(=O)n(-c3cccnc3)c2)c(=O)[nH]1
O=c1[nH]cc(-c2cc(-c3cc(Cl)cc(COc4ccccc4Cl)c3)c(=O)n(-c3cccnc3)c2)c(=O)[nH]1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCCCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCCCCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCCCCCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCCCCCCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCOCCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cn1cc2cc(/N=c3[nH]c(=O)n(Cc4cn(CCOCCOCCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6)nn4)c(=O)n3Cc3cc(F)c(F)cc3F)c(Cl)cc2n1
Cc1c(c2cc(ccc2n1C(=O)c3ccc(cc3)Cl)OC)CC(=O)O
O=C(NCCc1cccc(F)c1)[C@H](c1cncnc1)N(C(=O)[C@H](F)Cl)c1ccc(S(F)(F)(F)(F)F)cc1
O=C(NCCc1cccc(F)c1)[C@@H](c1cncnc1)N(C(=O)[C@@H](F)Cl)c1ccc(S(F)(F)(F)(F)F)cc1
C[C@@H](NC(=O)[C@H](c1cccnc1)N(C(=O)C(Cl)Cl)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@@H](NC(=O)[C@H](c1cccnc1)N(C(=O)C(Br)(Br)Br)c1ccc(-c2ccccc2)cc1)c1ccccc1
CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S([O-])(=O)=O
CCCSc1nc2sc3c(c2c(=O)n1CC)CCc1ccccc1-3
CCSc1nc2sc3c(c2c(=O)n1CC)CCc1ccccc1-3
CCn1c(SCC=C)nc2sc-3c(CCc4ccccc-34)c2c1=O
O=C[C@H](CC1CCNC1=O)NC(=O)[C@H](CC1CCCCC1)NC(=O)c1cc2ccccc2[nH]1
O=C[C@H](CC1CCNC1=O)NC(=O)[C@H](Cc1cccc(F)c1)NC(=O)c1cc2ccccc2[nH]1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccccc1F
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccccc1Cl
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccccc1Br
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1cccc(F)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1cccc(Cl)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1cccc(Br)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(F)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Br)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc([N+](=O)[O-])cc1
COc1ccc(CN(C#N)N(C)C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1cccc(Cl)c1F
COc1cccc(CN(C#N)N(C)C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1F
COc1c(Cl)cccc1CN(C#N)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1cc(Cl)ccc1F
COc1ccc(OC)c(CN(C#N)N(C)C(=O)[C@H](Cc2ccccc2)NC(=O)OCc2ccccc2)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Br)cc1F
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Br)cc1Cl
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Br)c(F)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Br)c(Cl)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccc(Br)c(Cl)c1F
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1c(F)cc(Br)cc1F
COc1ccc(Cl)c(F)c1CN(C#N)N(C)C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccco1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)N(C#N)Cc1ccsc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1cccc(Cl)c1)N(C#N)Cc1ccc(Cl)cc1
COc1cccc(OCC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)N(C#N)Cc2ccc(Cl)cc2)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1ccc(F)cc1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1ccc(Cl)cc1)N(C#N)Cc1ccc(Cl)cc1
COc1ccc(OCC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)N(C#N)Cc2ccc(Cl)cc2)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1cccc(F)c1Br)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1ccc(F)c(F)c1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1ccc(Cl)cc1Cl)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1cccc2ccccc12)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)COc1ccc2c(c1)NC(=O)CC2)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)CCc1ccc(F)c(F)c1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)CNc1ccc(F)c(F)c1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)CNc1c(F)cccc1F)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)CNc1ccc(F)cc1F)N(C#N)Cc1ccc(Cl)cc1
COc1ccc(NCC(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)N(C#N)Cc2ccc(Cl)cc2)c(Cl)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)c1cccs1)C1CCCCC1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)C1(NC(=O)c2cccs2)CC1)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)c1cc2cc(Cl)ccc2[nH]1)N(C#N)Cc1ccc(Cl)cc1
COc1cccc2[nH]c(C(=O)N[C@@H](Cc3ccccc3)C(=O)N(C)N(C#N)Cc3ccc(Cl)cc3)cc12
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Nc1ccc([N+](=O)[O-])cc1[N+](=O)[O-])C(C)(C)C)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)C(F)(F)F)C(C)(C)C)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)C1(F)CC1)C(C)(C)C)N(C#N)Cc1ccc(Cl)cc1
CCCS(=O)(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)N(C)N(C#N)Cc1ccc(Cl)cc1)C(C)(C)C
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)C1CCCC1)C(C)(C)C)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1ccc(Cl)cc1
Cc1csc(C(=O)N[C@H](C(=O)N[C@@H](Cc2ccccc2)C(=O)N(C)N(C#N)Cc2ccc(Cl)cc2)C(C)(C)C)c1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)c1ccc(-c2cccs2)s1)C(C)(C)C)N(C#N)Cc1ccc(Cl)cc1
CN(C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN(C(=O)[C@H](Cc1ccccc1F)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN(C(=O)[C@H](Cc1ccccc1Cl)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN(C(=O)[C@H](Cc1cccc(F)c1)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN(C(=O)[C@H](Cc1cccc(Cl)c1)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN(C(=O)[C@H](Cc1ccc(F)cc1)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN(C(=O)[C@H](Cc1cccs1)NC(=O)[C@@H](NC(=O)c1cccs1)C(C)(C)C)N(C#N)Cc1cccc(Cl)c1F
CN1C(=O)[C@H](Cc2ccccc2)NC(=O)COCCOCCOc2ccc(F)cc2CN1C#N
CN1C(=O)[C@H](CCc2ccccc2)NC(=O)COCCOc2ccc(F)cc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)NC(=O)COCCOc2ccc(F)cc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)COc2ccc(Cl)cc2Cl)CCCCCOc2ccc(F)cc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)COc2ccc(Cl)cc2Cl)CCCCOc2ccc(F)cc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)COc2ccc(Cl)cc2Cl)CCCOc2ccc(F)cc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)COc2ccc(Cl)cc2Cl)CCCOc2ccc(Cl)c(F)c2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)COc2ccc(Cl)cc2Cl)CCCOc2c(Cl)cccc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)CNC(=O)c2cccs2)CCCOc2c(Cl)cccc2CN1C#N
CN1C(=O)[C@H](Cc2ccccc2)N(C(=O)CNC(=O)c2cccs2)CC2(CC2)COc2c(Cl)cccc2CN1C#N
CC(C)C[C@H](NC(=O)OCC1CCN(Cc2ccccc2)C1=O)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CCN(Cc2ccccc2)C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CCN(Cc2cccc(C(F)(F)F)c2)C1=O)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CCN(Cc2cccc(C(F)(F)F)c2)C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CCN(CC2CCCCC2)C1=O)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CCN(CC2CCCCC2)C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CCN(C[C@H]2C[C@H]3CC[C@@H]2C3)C1=O)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CCN(C[C@H]2C[C@H]3CC[C@@H]2C3)C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CCN(C[C@H]2C[C@H]3C=C[C@@H]2C3)C1=O)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CCN(C[C@H]2C[C@H]3C=C[C@@H]2C3)C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CCN(Cc2ccco2)C1=O)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CCN(Cc2ccco2)C1=O)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(Cc2ccccc2)C1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(Cc2ccccc2)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(Cc2cccc(C(F)(F)F)c2)C1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(Cc2cccc(C(F)(F)F)c2)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(CC2CCCCC2)C1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(CC2CCCCC2)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(CC2CC3CCC2C3)C1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(CC2CC3CCC2C3)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(CC2CC3C=CC2C3)C1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(CC2CC3C=CC2C3)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(Cc2ccco2)C1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OCC1CC(=O)N(Cc2ccco2)C1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1ccccc1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1cccc(F)c1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1cccc(F)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1cccc(Cl)c1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1cccc(Cl)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1cccc(C(F)(F)F)c1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1cccc(C(F)(F)F)c1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CCc1ccccc1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CCc1ccccc1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@H]1CCC(=O)N1CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@H]1CCC(=O)N1CC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CCC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CCC1CCCCC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CC1CCC(F)(F)CC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1CC1CCC(F)(F)CC1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1C[C@H]1C[C@@H]2CC[C@H]1C2)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1C[C@H]1C[C@@H]2CC[C@H]1C2)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1C[C@H]1C[C@@H]2C=C[C@H]1C2)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1C[C@H]1C[C@@H]2C=C[C@H]1C2)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1ccc2c(c1)OC(F)(F)O2)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1ccc2c(c1)OC(F)(F)O2)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1ccco1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)C[C@H](NC(=O)OC[C@@H]1CCC(=O)N1Cc1ccco1)C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(O)S(=O)(=O)[O-]
O=C(c1cc(=O)[nH]c2ccccc12)N1CCN(c2ccc(Cl)c(Cl)c2)CC1CN1CCOCC1
O=C(c1cc(=O)[nH]c2ccccc12)N1CCN(c2ccc(Cl)c(Cl)c2)C[C@@H]1CC1CCCCC1
O=C(c1cc(=O)[nH]c2ccccc12)N1CCN(c2ccc(Cl)c(Cl)c2)CC1Cc1ccccc1
O=C(C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12)N1CCOCC1
CN1CCN(C(=O)C2CN(c3ccc(Cl)c(Cl)c3)CCN2C(=O)c2cc(=O)[nH]c3ccccc23)CC1
O=C1CCN(C(=O)C2CN(c3ccc(Cl)c(Cl)c3)CCN2C(=O)c2cc(=O)[nH]c3ccccc23)CC1
CC1(C)C2CN(C(=O)C3CN(c4ccc(Cl)c(Cl)c4)CCN3C(=O)c3cc(=O)[nH]c4ccccc34)CC21
O=C1CC2CN(C(=O)C3CN(c4ccc(Cl)c(Cl)c4)CCN3C(=O)c3cc(=O)[nH]c4ccccc34)CC2C1
O=C1CC2(CCN(C(=O)C3CN(c4ccc(Cl)c(Cl)c4)CCN3C(=O)c3cc(=O)[nH]c4ccccc34)CC2)C1
O=C(C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12)N1CCC2(CC1)COC2
O=C(C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12)N1CC2(COC2)C1
O=C(NCC1CC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCC1CCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCC1CCCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCC1CCCCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCC1CCO1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCC1CCCO1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
CN(CC1COCCO1)C(=O)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCC(F)(F)F)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCC1CC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCC1CCCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCN1CCOCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCC1CCOCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
CCCCNC(=O)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCCC(F)(F)F)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCCN1CCOCC1)C1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
O=C(NCCC(F)(F)F)[C@H]1CN(c2ccc(Cl)c(Cl)c2)CCN1C(=O)c1cc(=O)[nH]c2ccccc12
c1ccc2c(c1)C(=CC(=O)N2)C(=O)N3CCN(C[C@H]3C(=O)NCCC(F)(F)F)c4ccc(c(c4)Cl)Cl
O=C(c1cc(=O)[nH]c2ccccc12)N1CCC(Nc2ccc(Cl)c(Cl)c2)C1
O=C(N[C@@H]1CCC[C@@H]1Nc1ccc(Cl)c(Cl)c1)c1cc(=O)[nH]c2ccccc12
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1NC1CCN(C(=O)c2cc(=O)[nH]c3ccccc23)C1
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@H]1CCC[C@H]1NC(=O)c1cc(=O)[nH]c2ccccc12
O=C(N[C@H]1CCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(Br)cc1[N+](=O)[O-])c1cc(=O)[nH]c2ccccc12
O=C(N[C@H]1CCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(Br)cc1[N+](=O)[O-])c1cc(=O)[nH]c2c(F)cccc12
O=C(N[C@H]1CCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(C2CC2)cc1[N+](=O)[O-])c1cc(=O)[nH]c2ccccc12
COc1ccc2[nH]c(=O)cc(C(=O)N[C@H]3CCC[C@H]3Nc3c(C(=O)N4CCOCC4)cc(C4CC4)cc3[N+](=O)[O-])c2c1
O=C(N[C@H]1CCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(C2CC2)cc1[N+](=O)[O-])c1cc(=O)[nH]c2c(F)cccc12
CN1CCN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCC[C@@H]2NC(=O)c2cc(=O)[nH]c3ccccc23)CC1
CN1CCN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCC[C@@H]2NC(=O)c2cc(=O)[nH]c3c(F)cccc23)CC1
CN1CCN(C(=O)c2cc(C3CC3)cc([N+](=O)[O-])c2N[C@@H]2CCC[C@@H]2NC(=O)c2cc(=O)[nH]c3ccccc23)CC1
COc1ccc2[nH]c(=O)cc(C(=O)N[C@H]3CCC[C@H]3Nc3c(C(=O)N4CCN(C)CC4)cc(C4CC4)cc3[N+](=O)[O-])c2c1
CN1CCN(C(=O)c2cc(C3CC3)cc([N+](=O)[O-])c2N[C@@H]2CCC[C@@H]2NC(=O)c2cc(=O)[nH]c3c(F)cccc23)CC1
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCC[C@@H]1NC(=O)c1cc(=O)[nH]c2ccccc12
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCC[C@@H]1NC(=O)c1cc(=O)[nH]c2ccc(F)cc12
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCC[C@@H]1NC(=O)c1cc(=O)[nH]c2cc(F)ccc12
CNC(=O)c1cc(Br)cc([N+](=O)[O-])c1N[C@@H]1CCCC[C@@H]1NC(=O)c1cc(=O)[nH]c2c(F)cccc12
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(Br)cc1[N+](=O)[O-])c1cc(=O)[nH]c2cc(F)ccc12
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(Br)cc1[N+](=O)[O-])c1cc(=O)[nH]c2c(F)cccc12
COc1ccc2[nH]c(=O)cc(C(=O)N[C@H]3CCCC[C@H]3Nc3c(C(=O)N4CCOCC4)cc(Br)cc3[N+](=O)[O-])c2c1
COc1ccc2[nH]c(=O)cc(C(=O)N[C@H]3CCCC[C@H]3Nc3c(C(=O)N4CCN(C)CC4)cc(Br)cc3[N+](=O)[O-])c2c1
CN1CCN(C(=O)c2cc(Br)cc([N+](=O)[O-])c2N[C@@H]2CCCC[C@@H]2NC(=O)c2cc(=O)[nH]c3c(F)cccc23)CC1
CNC(=O)c1cccc([N+](=O)[O-])c1N[C@@H]1CCCC[C@@H]1NC(=O)c1cc(=O)[nH]c2ccccc12
CNC(=O)c1cc(cc(c1N[C@@H]2CCCC[C@@H]2NC(=O)C3=CC(=O)Nc4c3cccc4)[N+](=O)[O-])C5CC5
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(C2CC2)cc1[N+](=O)[O-])c1cc(=O)[nH]c2ccccc12
COc1ccc2[nH]c(=O)cc(C(=O)N[C@H]3CCCC[C@H]3Nc3c(C(=O)N4CCOCC4)cc(C4CC4)cc3[N+](=O)[O-])c2c1
O=C(N[C@H]1CCCC[C@H]1Nc1c(C(=O)N2CCOCC2)cc(C2CC2)cc1[N+](=O)[O-])c1cc(=O)[nH]c2c(F)cccc12
C[C@H](c1cccc2ccccc12)N(C)Cc1ccc(O)cc1F
C[C@H](c1cccc2ccccc12)N(C)Cc1cc[nH]c1
C[C@H](c1cccc2ccccc12)N(C)Cc1ccc(O)cc1O
C[C@H](c1cccc2ccccc12)N(C)Cc1ccc(N)cc1
C[C@H](c1cccc2ccccc12)N(C)Cc1cccc(N)c1
C[C@H](c1cccc2ccccc12)N(C)Cc1ccc(C(=O)O)cc1
C[C@H](c1cccc2ccccc12)N(C)Cc1cccc(C(=O)O)c1
Cc1ccc([N+](=O)[O-])cc1CN(C)[C@H](C)c1cccc2ccccc12
C[C@H](c1cccc2ccccc12)N(C)Cc1cc([N+](=O)[O-])ccc1O
COc1cc([N+](=O)[O-])ccc1CN(C)[C@H](C)c1cccc2ccccc12
C[C@H](c1cccc2ccccc12)N(C)Cc1c[nH]c2cc(F)ccc12
C[C@H](c1cccc2ccccc12)N(C)Cc1c[nH]c2ccc(F)cc12
C[C@H](c1cccc2ccccc12)N(C)Cc1cc2ccccc2[nH]1
C[C@H](c1cccc2ccccc12)N(C)Cc1cccc2cc[nH]c12
C[C@H](c1cccc2ccccc12)N(C)Cc1ccc2cn[nH]c2c1
Cc1ccc(NC2CNC2)cc1CN(C)[C@H](C)c1cccc2ccccc12
Cc1ccc(NC2CCNCC2)cc1CN(C)[C@H](C)c1cccc2ccccc12
Cc1ccc(NCCN)cc1CN(C)[C@H](C)c1cccc2ccccc12
Cc1ccc(NCCNC(=N)N)cc1CN[C@H](C)c1cccc2ccccc12
C[C@H](c1cccc2ccccc12)N(C)Cc1cc(NC2CCNCC2)ccc1O
C[C@H](c1cccc(-c2cccs2)c1)N(C)Cc1c[nH]c2ccccc12
C[C@H](c1cccc(-c2ccc(CN3CCCC3)s2)c1)N(C)Cc1c[nH]c2ccccc12
C[C@H](c1cccc(-c2cccs2)c1)N(C)Cc1ccc(O)cc1
C[C@H](c1cccc(-c2ccc(CN3CCCC3)s2)c1)N(C)Cc1ccc(O)cc1
C[C@H](c1cccc(-c2cccs2)c1)N(C)Cc1c[nH]c2ccc(F)cc12
C[C@H](c1cccc(-c2cccs2)c1)N(C)Cc1c[nH]c2cc(F)ccc12
C[C@H](c1cccc(-c2cccs2)c1)N(C)Cc1ccc(O)cc1O
C[C@H](c1cccc(-c2cccs2)c1)N(C)Cc1ccc2cn[nH]c2c1
COc1cc(O)ccc1CN(C)[C@@H](C)c1cccc(-c2ccc(CN3CCCC3)s2)c1
C[C@H](c1cccc(-c2ccc(CN3CCCC3)s2)c1)N(C)Cc1ccc2[nH]ncc2c1
C[C@H](c1cccc(-c2ccc(CN3CCCC3)s2)c1)N(C)Cc1cccc2[nH]ccc12
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc2ccccc12
Cc1ccc(OCCNC(=N)N)cc1C(=O)N[C@H](C)c1cccc2ccccc12
Cc1ccc(OCC(=O)NC(=N)N)cc1C(=O)N[C@H](C)c1cccc2ccccc12
Cc1ccc(OC2CNC2)cc1C(=O)N[C@H](C)c1cccc2ccccc12
Cc1ccc(OC2CN(C(=N)N)C2)cc1C(=O)N[C@H](C)c1cccc2ccccc12
C#CCCC(=O)NCCOc1ccc(C)c(C(=O)N[C@H](C)c2cccc3ccccc23)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(F)cc2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(F)cc2F)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(O)cc2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccccc2O)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(C#N)cc2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2cnc(N(C)C)nc2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc3c(c2)CCO3)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc3c(c2)OCCO3)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2cccs2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccsc2)c1
C[C@@H](NC(=O)c1cccc(OCCN)c1)c1cccc(-c2cccs2)c1
Cc1ccc(OCC[N+](C)(C)C)cc1C(=O)N[C@H](C)c1cccc(-c2cccs2)c1
Cc1cc(OCCN)ccc1C(=O)N[C@H](C)c1cccc(-c2cccs2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(C#N)s2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC3CC3)s2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccoc2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2cnn(C)c2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2cnn(C(F)F)c2)c1
COCCn1cc(-c2cccc([C@@H](C)NC(=O)c3cc(OCCN)ccc3C)c2)cn1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2c(C)noc2C)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccn[nH]2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccn(C)c2C)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2cn[nH]c2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2cnn(Cc3ccccc3)c2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2c[nH]nc2C)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccnn2C)c1
O=C1N[C@@H](Cc2ccccc2)C(=O)N1c1cncc(F)c1
CC(F)(F)CC[C@H](NC(=O)[C@@H]1[C@@H]2[C@H](CN1C(=O)[C@@H](NC(=O)NC1(CS(=O)(=O)C(C)(C)C)CCCCC1)C(C)(C)C)C2(C)C)C(=O)C(=O)NC1CC1
CNC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
CC(F)(F)CC[C@H](NC(=O)[C@@H]1CC2(CCCCC2)CN1C(=O)c1cc2ccccc2[nH]1)C(=O)C(=O)NC1CC1
CC(F)(F)CC[C@H](NC(=O)[C@@H]1CC2(CCCCC2)CN1C(=O)C(O)c1cccc(F)c1)C(=O)C(=O)NC1CC1
CC(C)(C)CC(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1
CC(F)(F)CC[C@H](NC(=O)[C@@H]1CC2(CCCCC2)CN1C(=O)[C@@H](NC(=O)OCc1ccccc1)C1CCCCC1)C(=O)C(=O)NC1CC1
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(N)=O)C(C)(C)C
CNC(=O)C(=O)[C@H](CCC(C)(F)F)NC(=O)[C@@H]1CC2(CCCCC2)CN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NCc1ccccc1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CCCCC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NCc1ccncc1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCC(F)(F)CC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCOCC2)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)CC2(F)F)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C21CCOCC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC[C@@H](C(F)(F)F)C[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
CNC(=O)C(=O)[C@H](CCC(C)(F)F)NC(=O)[C@@H]1C[C@H](C(F)(F)F)CCN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](CCC(C)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
CNC(=O)C(=O)[C@H](CCC(C)(F)F)NC(=O)[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C
CCCC[C@H](NC(=O)[C@@H]1CC2(CCCCC2)CN1C(=O)[C@@H](NC(=O)OC)C(C)(C)C)C(=O)C(=O)NC1CC1
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CCC(F)(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1CC2(CCCCC2)C[C@H]1C(=O)N[C@@H](CC1CC1(F)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](CCC(C)(C)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](CC[C@@H](C)F)C(=O)C(=O)NC1CC1)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@@H]2CCC[C@@H]2[C@H]1C(=O)N[C@@H](CC[C@H](C)F)C(=O)C(=O)NC1CC1)C(C)(C)C
CCCCCCCCCC(C)CCC(C)C(=O)O
CCCCCCCCCC(C)CCC(C)C(=O)OC
CCCCCCCCCC(C)CCC(C)C(=O)OCc1ccccc1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)OC(c3ccccc3)c3ccccc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)OC(c3ccc(F)cc3)c3ccc(F)cc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C(c3ccc(Cl)cc3)c3ccc(Cl)cc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)N(c3ccc(Cl)cc3)c3ccc(Cl)cc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C(Oc3ccc(Cl)cc3)Oc3ccc(Cl)cc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)[C@H](Cc3ccccc3)NC(=O)OCc3ccccc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)[C@H](CC3CCCCC3)NC(=O)OCc3ccccc3)C[C@@H]21
CC(C)(C)C[C@H](NC(=O)OCc1cccnc1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)OCc3cccnc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)N(C(=O)OCc3cccnc3)C[C@@H]21
CC(C)(C)C[C@H](NC(=O)[C@@H]1CC[C@@H]1c1ccccc1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)(C)C[C@H](NC(=O)N1CC[C@@H]1c1ccccc1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)N(C(=O)[C@@H](NC(=O)C(F)(F)F)c3ccc(Cl)cc3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)N(C(=O)[C@@H](NC(=O)C(F)(F)F)c3ccc(Cl)c(Cl)c3)C[C@@H]21
O=C(c1cncc2ccc(F)cc12)N1CCN(Cc2ccc(Cl)cc2Cl)CC1
O=C(c1cccnc1)N1CCN(Cc2cc(Cl)cc(Cl)c2OC(F)F)CC1
O=C(c1cccnc1)N1CCN(Cc2cccc(Cl)c2Cl)CC1
O=C(Nn1cnc2c(F)cc(F)cc21)C1COc2cc(Cl)c(Cl)cc21
Cc1cc(cnc1)CC(=O)N2CCC[C@H]2c3cccc(c3)Cl
c1ccc(c(c1)CN2CCCN(CC2)C(=O)c3cc(cnc3)Cl)C#N
O=C1N[C@@H](Cc2cc(Cl)ccc2F)C(=O)N1c1cncc(F)c1
O=C(Cc1cccnc1)N1CCc2c(Cl)cc(Cl)cc2C1
c1ccc(c(c1)CN2CCCN(CC2)C(=O)c3cc(cnc3)Cl)Cl
Cc1cc(cnc1)CC(=O)N2CCc3cc(c(cc3C2)Cl)Cl
CCn1cncc1NC(=O)C1c2cc(Cl)cc(Cl)c2OCC1C
O=C1N(Cc2ccccc2Cl)CCN1c1cncc2ccc(Cl)cc12
O=C1N(Cc2ccc(Cl)cc2Cl)CCN1c1cncc2ccccc12
[#6]-[#8]-c1cc(-[#8])c(-[#6](=O)-[#6@@H]-2-[#6@H](-[#6]\[#6]=[#6](/[#6])-[#6])-[#6](-[#6])=[#6]-[#6]-[#6@H]-2-c2ccccc2)c(-[#8])c1 |r,c:17|
[#6]\[#6](-[#6])=[#6]\[#6]-[#6]\[#6](-[#6])=[#6]\[#6]-[#8]-c1c2ccoc2cc2oc(=O)ccc12
CCCCC1CCC(COC(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C=O)C[C@@H]2CCNC2=O)CC1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)COc3ccccc3)C[C@@H]21
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C[C@@H]1CCNC1=O)C(=O)C(N)=O)C2(C)C)C(C)(C)C
COC[C@@H](NC(=O)C1CCCC(F)(F)C1)C(=O)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1nccs1
C=CC(=O)N(CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)OCc1ccccc1)[C@@H](C)OC(C)(C)C
CC(C)c1nc(cs1)CN(C)C(=O)N[C@@H](CCN2CCOCC2)C(=O)N[C@H](CC[C@H](Cc3ccccc3)NC(=O)OCc4cncs4)Cc5ccccc5
COc1ccc(C(=O)\C=C\c2ccc(O)cc2)c(O)c1CC(OO)C(C)=C
C[C@@]12CC[C@]3(CCC(C[C@H]3[C@H]1C(=O)C=C4[C@]2(CC[C@@H]5[C@@]4(C=C(C(=O)C5(C)C)C#N)C)C)(C)C)C(=O)OC
CC(=C)[C@@H]1CC[C@]2([C@H]1[C@H]3CC[C@@H]4[C@]5(CC[C@@H](C([C@@H]5CC[C@]4([C@@]3(CC2)C)C)(C)C)O)C)C(=O)O
O=C(Oc1cncc(Cl)c1)c1sccc1Cl
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](CC1CCCCC1)C(=O)NN(CCC(N)=O)C(=O)C(Cl)Cl
Oc1c(Cl)c(N=CCN2CCOCC2)c(O)c2ncccc12 |w:6.6|
C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)[C@H]1CO1
C=CC(=O)N[C@H](CC(=C)C)C(=O)N1C[C@@H](C(=O)N[C@H](Cc2ccccc2)C(=O)NC)[C@H](c2cccc(C(F)(F)F)c2)C1
O=C(NCc1ccc(O)c(F)c1)N1CCC(CN2CCc3ccccc32)CC1
CNC(=O)c1ccc([C@H]2CCCCN2Cc2cccc(C(=O)N(C)C)c2)n1C
C1CCN(CC1)c2c3c(c(nc(n3)N(CCO)CCO)N4CCCCC4)nc(n2)N(CCO)CCO
C[C@H](c1cccc2c1cccc2)NCCCc3cccc(c3)C(F)(F)F
CCOc1ccc(C(=O)Nc2ccc(CN3CC(N(C)C)C3)c(C(F)(F)F)c2)cc1[N+](=O)[O-]
CN(C)C1CN(Cc2ccc(NC(=O)c3ccc(OCCC(F)(F)F)c([N+](=O)[O-])c3)cc2C(F)(F)F)C1
C=C[C@@H]1C[C@]1(NC(=O)[C@@H]1C[C@@H](Oc2cc(-c3csc(NC(C)C)n3)nc3c(C(C)C)c(OC)ccc23)CN1C(=O)[C@@H](NC(=O)OC1CCCC1)C(C)(C)C)C(=O)O
C=C[C@@H]1C[C@]1(NC(=O)[C@@H]1C[C@@H](Oc2cc(-c3csc(C(=O)CC)n3)nc3c(C)c(OC)ccc23)CN1C(=O)[C@@H](NC(=O)OC1CCCC1)C(C)(C)C)C(=O)O
C=C[C@@H]1C[C@]1(NC(=O)[C@@H]1C[C@@H](Oc2cc(-c3csc(NC(C)C)n3)nc3cc(OC)ccc23)CN1C(=O)[C@@H](NC(=O)OC1CCCC1)C(C)(C)C)P(=O)(O)O
COc1ccc2c(O[C@@H]3C[C@H]4C(=O)N[C@]5(P(=O)(O)Cc6ccccc6)C[C@H]5CCCCCCC[C@H](NC(=O)OC5CCCC5)C(=O)N4C3)cc(-c3csc(NC(C)C)n3)nc2c1
COc1ccc2nc3c4c(c2c1)CC[C@]1(C[C@H]2C(=O)N[C@]5(C(=O)NS(=O)(=O)C6(C)CC6)C[C@H]5/C=C/CCCCC[C@H](NC(=O)O[C@@H]5CCC[C@H]5CCCCC3)C(=O)N2C1)O4
ClCC(=O)N[C@@H](CC=C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1 |r|
CC(C)C[C@H](NC(=O)CCl)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
C=CC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
CC(C)C[C@@H](NC(=O)CCl)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
O=C(CCl)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
O=C(CCl)NCC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
O=C(CS)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
O=C(CCl)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
C=CC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
CC(C)C[C@H](NC(=O)CCl)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
CC(C)C[C@H](NC(=O)CCl)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
C=CC[C@H](NC(=O)CCl)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCN1CCOCC1
CC(C)C[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCl)C(=O)NCc1ccccc1
COC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CCl
C=CC[C@H](NC(=O)CCl)C(=O)N[C@@H](CC=C)C(=O)N[C@H](CNCc1ccccc1)Cc1c[nH]c2ccccc12
COC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(C)C)NC(=O)CCl
CC(C)C[C@@H](C(=O)NCC12CC3CC(CC(C3)C1)C2)N(Cc1ccccc1)C(=O)CCl
CC(C)(C)[C@H](NC(=O)C(Cl)(Cl)Cl)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)C(Cl)(Cl)Cl)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCCNC1=O)C2(C)C
CC(C)(C)OC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C)C(C)(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N(C(=O)C(F)(F)F)[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)OCc1ccccn1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)OCc1cccnc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)OCc1ccncc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C2(C)C)C(C)(C)C
CC(C)(C)[C@H](NC(=O)OCc1cccnc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCCNC1=O)C2(C)C
CC(C)(C)[C@H](NC(=O)OCc1ccncc1)C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCCNC1=O)C2(C)C
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cccc(OCCCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cccc(OCCCCCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cccc(OCCCCCCCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cccc(OCCCCCCN(C)CCN(C)c2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cn(CCOCCOCCOCCC(=O)Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nn1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
C[C@@H](OC(C)(C)C)[C@H](NC(=O)OCc1cn(CCOCCOCCOCCC(=O)N(C)CCN(C)c2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nn1)C(=O)N[C@@H](CC1CCCCC1)C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O
CC(C)(COCCCCCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)C(C)(C)C
CC(C)(CCOCCCCCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)C(C)(C)C
CN(CCN(C)c1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)CCC(C)(C)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)C(C)(C)C
CC(C)(CCC(=O)NCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)N[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)C(C)(C)C
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1CCCN1C(=O)c1cc2ccccc2[nH]1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1CC(F)(F)CN1C(=O)c1cc2ccccc2[nH]1
CC1(C)C[C@@H](C(=O)N[C@H](C=O)C[C@@H]2CCNC2=O)N(C(=O)c2cc3ccccc3[nH]2)C1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1CC2(CC2)CN1C(=O)c1cc2ccccc2[nH]1
O=C[C@H](C[C@@H]1CCNC1=O)NC(=O)[C@@H]1C[C@@H](C2CCCCC2)CN1C(=O)c1cc2ccccc2[nH]1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4ccccc4[nH]3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4c(F)cccc4[nH]3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4cc(F)ccc4[nH]3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4ccc(F)cc4[nH]3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4cccc(F)c4[nH]3)C[C@@H]21
Cc1cccc2cc(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)[nH]c12
COc1cccc2cc(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)[nH]c12
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4cccc(C#N)c4[nH]3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4cccc(C(F)(F)F)c4[nH]3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4cccc(Cl)c4[nH]3)C[C@@H]21
Cc1cccc2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
CCc1cccc2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
CC(C)c1cccc2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
COc1cccc2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
CC(C)Oc1cccc2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)c3cc4c(C#N)cccc4[nH]3)C[C@@H]21
CC(C)c1ccc(Cl)c2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
CC(C)c1ccc(F)c2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)C4(C)C)cc12
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C3CCCC3)C[C@@H]21
CC1CC(C(=O)N2C[C@H]3[C@@H]([C@H]2C(=O)N[C@H](C=O)C[C@@H]2CCNC2=O)C3(C)C)C1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C3(O)CCCCC3)C[C@@H]21
CC(C)(C)CC(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C
CC(C)(C)CCC(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)CC3CCCCC3)C[C@@H]21
C[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)C1CCCCC1
C[C@@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)C1CCCCC1
CC1CCC(CC(=O)N2C[C@H]3[C@@H]([C@H]2C(=O)N[C@H](C=O)C[C@@H]2CCNC2=O)C3(C)C)CC1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)Cc3ccccc3)C[C@@H]21
C[C@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)c1ccccc1
C[C@@H](C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)c1ccccc1
Cc1cccc([C@@H](C)C(=O)N2C[C@H]3[C@@H]([C@H]2C(=O)N[C@H](C=O)C[C@@H]2CCNC2=O)C3(C)C)c1
CC(C)(C(=O)N1C[C@H]2[C@@H]([C@H]1C(=O)N[C@H](C=O)C[C@@H]1CCNC1=O)C2(C)C)c1ccccc1
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C3(c4ccccc4)CC3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C3(c4cccc(Cl)c4)CC3)C[C@@H]21
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C=O)C[C@@H]3CCNC3=O)N(C(=O)C3(c4ccccc4)CCCC3)C[C@@H]21
CC(C)c1cccc2[nH]c(C(=O)N3C[C@H]4[C@@H]([C@H]3C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)C4(C)C)cc12
CC1(C)[C@@H]2[C@@H](C(=O)N[C@H](C#N)C[C@@H]3CCNC3=O)N(C(=O)C3(c4cccc(Cl)c4)CC3)C[C@@H]21
O=C[C@H](C[C@@H]1CNCC1=O)NC(=O)[C@H](Cc1cccc(F)c1)NC(=O)c1cc2ccccc2[nH]1
CN1C(=O)/C(=C2/C(=O)Nc3ccccc32)c2ccccc21
O=C1Nc2ccccc2\C1=C1/C(=O)Nc2ccccc12
CN1C(=O)/C(=C2/C(=O)N(CCN3CCCC3)c3ccccc32)c2ccccc21
O=C(O)CCCCCCCN1C(=O)/C(=C2/C(=O)Nc3ccccc32)c2cc(Br)ccc21
COc1ccc2c(c1)/C(=C1C(=O)Nc3ccccc31)C(=O)N2CCCCCCCC(=O)O
CN1C(=O)/C(=C2/C(=O)N(CCN)c3ccccc32)c2cc(Br)ccc21
CN1C(=O)/C(=C2/C(=O)N(CCCN)c3ccc(Br)cc32)c2ccccc21
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H](OC(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O
COC(=O)N[C@H](C(=O)N1C[C@H](OC(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C(C)(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H](OC(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O
COC(=O)N[C@H](C(=O)N1C[C@H](OC(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C(C)(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1C[C@H](C(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O
COC(=O)N[C@H](C(=O)N1C[C@H](C(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@H](C(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCCNC1=O)C(C)(C)C
COC(=O)N[C@H](C(=O)N1C[C@H](C(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)C(C)C
COC(=O)N[C@H](C(=O)N1C[C@H](C(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCCNC1=O)C(C)C
COC(=O)N[C@H](C(=O)N1C[C@H](C(F)(F)F)C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CC(O)NC1=O)C(C)(C)C
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2cc(C)c(CN3CCCC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2cc(C)c(CNC3CCCC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2cc(C)c(CN[C@H]3CC[C@@H](O)C3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2sc(CN[C@H]3CC[C@@H](O)C3)cc2C)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2sc(CNC3CCCC3)cc2C)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2sc(CN3CCCC3)cc2C)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2cc3ccccc3s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(C#N)s2)c1
Cc1csc(-c2cccc([C@@H](C)NC(=O)c3cc(NC4CNC4)ccc3C)c2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2sccc2C)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(-c3ccccc3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(-c3cccs3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(C(F)(F)F)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(Cl)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2cc3sccc3s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CCCC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CCOCC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CCCO3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CCNCC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CNC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)C3CCC(N)C3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC(=O)[C@@H]3CCCN3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN[C@H]3CC[C@@H](C(=O)O)C3)s2)c1
CCOC(=O)[C@@H]1CC[C@H](NCc2ccc(-c3cccc([C@@H](C)NC(=O)c4cc(NC5CNC5)ccc4C)c3)s2)C1
C[C@@H](NC(=O)c1cc(OC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CNC2CCCC2)s1 |r|
C[C@@H](NC(=O)c1cc(OC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN2CCCC2)s1 |r|
C[C@@H](NC(=O)c1cc(OC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@H]2CC[C@@H](O)C2)s1 |r|
Cc1ccc(OC2CCNCC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC3CCCC3)s2)c1
Cc1ccc(OC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN3C(=O)[C@@H]4CC[C@H]3C4)s2)c1
C[C@@H](NC(=O)c1cc(OC2CNC2)ccc1C)c1cccc(c1)-c1ccc(CN[C@H]2CC[C@H](C2)C(O)=O)s1 |r|
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC3CCCC3)s2)c1
Cc1ccc(OCCN)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN3CCCC3)s2)c1
Cc1ccc(OC2CCNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN3CCCC3)s2)c1
CC(=O)Nc1ccc(C)c(C(=O)N[C@H](C)c2cccc(-c3ccc(CNC4CCCC4)s3)c2)c1
CC(=O)Nc1ccc(C)c(C(=O)N[C@H](C)c2cccc(-c3ccc(CN4CCCC4)s3)c2)c1
Cc1ccc(N)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC3CCCC3)s2)c1
Cc1ccc(N)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN3CCCC3)s2)c1
Cc1ccc(N)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN[C@H]3CC[C@@H](O)C3)s2)c1
Cc1ccc(OC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CNC3CCCC3)o2)c1
Cc1ccc(OC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ncc(CNC3CCCC3)o2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ncc(CNC3CCCC3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2cccn2C)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN[C@H]3CC[C@@H](OC(=O)[C@@H](N)C(C)C)C3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN[C@H]3CC[C@@H](OC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)C(C)C)C3)s2)c1
CC(=O)OC(C)OC(=O)N1CC(Nc2ccc(C)c(C(=O)N[C@H](C)c3cccc(-c4ccc(CNC(=O)C5CCCC5)s4)c3)c2)C1
Cc1ccc(OC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN[C@H]3CC[C@@H](C(=O)OC[C@H]4O[C@@H](n5ccc(N)nc5=O)[C@H](O)[C@@H]4O)C3)s2)c1
Cc1ccc(NC2CNC2)cc1C(=O)N[C@H](C)c1cccc(-c2ccc(CN[C@H]3CC[C@@H](C(=O)OC[C@H]4O[C@@H](n5ccc(NO)nc5=O)[C@H](O)[C@@H]4O)C3)s2)c1
COCCn1c[n+](Cc2cnccn2)c2c1C(=O)c1ccccc1C2=O
c1cc(cc2c1cc3ccc(cc3n2)N)N
Cc1cccc(N2C(=O)C[n+]3ccccc3C2C(=O)Nc2ccccc2)c1
CN1C(=O)C[n+]2ccccc2C1C(=O)Nc1ccccc1
Cc1ccccc1NC(=O)C1c2cccc[n+]2CC(=O)N1C
Cc1cccc(C)c1NC(=O)C1c2cccc[n+]2CC(=O)N1C
O=C(Nc1ccccc1)C1c2cccc[n+]2CC(=O)N1c1ccccc1
CCOc1ccc(NC(=O)C2c3cccc[n+]3CC(=O)N2c2ccccc2)cc1
Cc1ccccc1N1C(=O)C[n+]2ccccc2C1C(=O)Nc1ccccc1
O=C(Nc1ccc(Cl)cc1)C1c2cccc[n+]2CC(=O)N1c1cccc(Cl)c1
Cc1ccc(N2C(=O)C[n+]3ccccc3C2C(=O)Nc2ccccc2C)cc1
O=C(Nc1ccc(Cl)cc1)C1c2cccc[n+]2CC(=O)N1c1ccc(Cl)cc1
O=C(Nc1ccccc1)C1c2cccc[n+]2CC(=O)N1c1ccc(Br)cc1
O=C(Nc1ccc(Cl)cc1)C1c2cccc[n+]2CC(=O)N1c1ccc(Br)cc1
Cc1cc(C)cc(N2C(=O)C[n+]3ccccc3C2C(=O)Nc2ccc(Cl)cc2)c1
Cc1ccc(N2C(=O)C[n+]3ccccc3C2C(=O)Nc2ccc(Cl)cc2)cc1Br
O=C(Nc1ccc(Cl)cc1)C1c2cccc[n+]2CC(=O)N1Cc1ccc2c(c1)OCO2
O=C1C2C3C=CC(CO)(O3)C2C(=O)N1c1cc(C(F)(F)F)ccc1Cl
CC(C)(C)C(=O)N[C@H](C(=O)N1CC2(C[C@H]1C(=O)N[C@H](C#N)C[C@@H]1CCNC1=O)SCCS2)C(C)(C)C
O=C(NC1CCCC1)C(=O)[C@H](CC1CCNC1=O)NC(=O)[C@@H]1[C@H]2CCC[C@H]2CN1C(=O)[C@@H](NC(=O)C(F)(F)F)C1CCCCC1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4ccc5cccc(O)c5n4)oc23)O1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4ccc5ccccc5n4)oc23)O1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4cnc5ccccc5c4)oc23)O1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4ccnc5ccccc45)oc23)O1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4cccc5ncccc45)oc23)O1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4ccc5ncccc5c4)oc23)O1
CC1(C)C=Cc2c(ccc3cc(C(=O)N/N=C/c4cccc5cccnc45)oc23)O1
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCn2cc(COc3ccc(COC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C[C@@H]4CCNC4=O)C(O)S(=O)(=O)[O-])cc3)nn2)C(C)(C)C)cc1
Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCn2cc(COc3ccc(COC(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C=O)C[C@@H]4CCNC4=O)cc3)nn2)C(C)(C)C)cc1
COc1ccc(Cl)cc1-n1cnnn1
Cc1cccc(c1)NC(=S)NCCN(C)C
Cc1ccc(C)c(Nc2ncnc3c2cnn3C)c1
Cn1c2c(cn1)c(ncn2)Nc3ccccc3Cl
CC(C)c1cc(O)n2ncc(-c3ccccc3)c2n1
Cc1cc(Nc2ccccc2C)n2ncnc2n1
C#CCNc1c2c(nc3ncnn13)CCC2
Cc1ccc(c(c1)C)Nc2cc(nc3n2cnn3)C
Cc1cc(Nc2cccc(C)c2C)n2ncnc2n1
Cc1cc(NCc2ccccc2Cl)n2cnnc2n1
CCn1ccc(-c2cc(-c3cnn(C)c3)cc([C@@H](C)NC(=O)c3cc(OCCN(C)C)ccc3C)c2)n1
CN1CCN(CC1)c1ccc(C)c(c1)C(=O)NC1(CC1)c1cc(nc2ccccc12)-c1cnn(C)c1
Cc1ccc(NC(=O)[C@H]2CCCCN2)cc1C(=O)N[C@H](C)c1cc(-c2cnn(C)c2)cc(-c2cccs2)c1
Cc1cc(C(=O)NCc2cscn2)ccc1C(=O)N[C@H](C)c1cc(-c2cnn(C)c2)cc(-c2ccns2)c1
Cc1cc(CNCc2cscn2)ccc1C(=O)N[C@H](C)c1cc(-c2cnn(C)c2)cc(-c2ccns2)c1
Cc1ccc(N2CCN(C)CC2)cc1C(=O)N[C@H](C)c1cc(-c2cnn(C)c2)cc(-c2cc(Cl)cnc2N)c1
Cc1ccc(N2CCN(C)CC2)cc1C(=O)N[C@H](C)c1cc(-c2cnn(C)c2)cc(-c2cccs2)c1
Cc1ccc(N2CCNCC2)cc1C(=O)N[C@H](C)c1cc(-c2cnn(C)c2)cc(-c2cc(Cl)cnc2N)c1
Fc1ccc(cc1)-n1[se]c2ccccc2c1=O
O=c1c2ccccc2[se]n1-c1ccc(C(F)(F)F)cc1
O=c1c2ccccc2[se]n1Cc1ccc(F)cc1
COc1ccc(Cn2[se]c3ccccc3c2=O)c(OC)c1
O=c1c2ccccc2[se]n1-c1c(F)cccc1F
COc1ccc2[se]n(-c3ccccc3)c(=O)c2c1
COc1ccc(F)cc1-n1[se]c2ccccc2c1=O
COc1cc(F)ccc1-n1[se]c2ccccc2c1=O
CCc1ccc(-n2[se]c3ccccc3c2=O)cc1
O=c1c2ccccc2[se]n1-c1cccc(Cl)c1
O=c1c2ccccc2[se]n1-c1cc(Cl)cc(Cl)c1
O=c1c2ccccc2[se]n1-c1ccc(Br)cc1
Cc1ccc(cc1)-n1[se]c2ccccc2c1=O
Cc1ccccc1-n1[se]c2ccccc2c1=O
N#Cc1cccc(-n2[se]c3ccccc3c2=O)c1
COc1ccc(cc1)-n1[se]c2ccccc2c1=O
CCCCCCCc1ccc(-n2[se]c3ccccc3c2=O)cc1
CCCCCCCCc1ccc(-n2[se]c3ccccc3c2=O)cc1
O=C(Oc1cncc(Cl)c1)c1ccccc1
O=C(Oc1cncc(Cl)c1)c1ccccc1F
O=C(Oc1cncc(Cl)c1)c1ccccc1Cl
COc1ccccc1C(=O)Oc1cncc(Cl)c1
O=C(Oc1cncc(Cl)c1)c1ccccc1-c1ccccc1
O=C(Oc1cncc(Cl)c1)c1cccc(F)c1
O=C(Oc1cncc(Cl)c1)c1cccc(Cl)c1
O=C(Oc1cncc(Cl)c1)c1cccc(-c2ccccc2)c1
O=C(Oc1cncc(Cl)c1)c1ccc(F)cc1
O=C(Oc1cncc(Cl)c1)c1ccc(I)cc1
COc1ccc(C(=O)Oc2cncc(Cl)c2)cc1
CCOc1ccc(C(=O)Oc2cncc(Cl)c2)cc1
CCCCCCCOc1ccc(C(=O)Oc2cncc(Cl)c2)cc1
CNc1ccc(C(=O)Oc2cncc(Cl)c2)cc1
N=C(N)Nc1ccc(C(=O)Oc2cncc(Cl)c2)cc1
O=C(Oc1cncc(Cl)c1)c1ccc(-c2ccccc2)cc1
O=C(Oc1cncc(Cl)c1)c1ccc(-c2cccnc2)cc1
O=C(Oc1cncc(Cl)c1)c1cccc(Cl)c1Cl
O=C(Oc1cncc(Cl)c1)c1ccc(Cl)c(Cl)c1
O=C(Oc1cncc(Cl)c1)c1ccc(Cl)cc1Cl
Cc1cc(Cl)ccc1C(=O)Oc1cncc(Cl)c1
O=C(Oc1cncc(Cl)c1)c1ccc(Cl)cc1F
COc1c(Cl)ccc(C(=O)Oc2cncc(Cl)c2)c1F
O=C(Oc1cncc(Cl)c1)c1ccc(Br)cc1F
O=C(Oc1cncc(Cl)c1)c1ccc(I)cc1F
N#Cc1ccc(C(=O)Oc2cncc(Cl)c2)c(F)c1
CCOc1ccc(c(c1)F)C(=O)Oc2cc(cnc2)Cl
c1ccc(cc1)COc2ccc(c(c2)F)C(=O)Oc3cc(cnc3)Cl
Nc1ccc(C(=O)Oc2cncc(Cl)c2)c(F)c1
COc1cc(F)ccc1C(=O)Oc1cncc(Cl)c1
COc1ccc(C(=O)Oc2cncc(Cl)c2)c(OC)c1
COc1ccc(C(=O)Oc2cncc(Cl)c2)cc1Cl
COc1cccc(C(=O)Oc2cncc(Cl)c2)c1OC
O=C(Oc1cncc(Cl)c1)c1cc(F)cc(F)c1
O=C(Oc1cncc(Cl)c1)c1cc(Cl)cc(Cl)c1
O=C(Oc1cncc(Cl)c1)c1c(F)cccc1F
COc1ccc(F)c(C(=O)Oc2cncc(Cl)c2)c1F
O=C(Oc1cncc(Br)c1)c1ccccc1
O=C(Oc1cncc(Br)c1)c1ccccc1F
O=C(Oc1cncc(Br)c1)c1ccccc1Cl
O=C(Oc1cncc(Br)c1)c1cccc(Cl)c1
COc1cccc(C(=O)Oc2cncc(Br)c2)c1
O=C(Oc1cncc(Br)c1)c1ccc(Cl)cc1
COc1ccc(C(=O)Oc2cncc(Br)c2)cc1
O=C(Oc1cncc(Br)c1)c1ccc(Cl)c(Cl)c1
O=C(Oc1cncc(Br)c1)c1ccc(Cl)cc1Cl
O=C(Oc1cncc(Br)c1)c1ccc(Cl)cc1F
O=C(Oc1cncc(Br)c1)c1ccc(I)cc1F
CCOc1ccc(C(=O)Oc2cncc(Br)c2)c(F)c1
O=C(Oc1cncc(Br)c1)c1ccc(OCc2ccccc2)cc1F
COc1cccc(C(=O)Oc2cncc(Br)c2)c1OC
CSc1nc2cc3OCCOc3cc2n1C(=O)c1ccc(C)cc1
CSc1nc2ccccc2n1C(=O)c1ccc(C)cc1
CSc1nc2ccccc2n1C(=O)Cc1ccccc1
CSc1nc2ccccc2n1C(C)=O
CSc1nc2ccccc2n1Cc1ccc(C)cc1
CSc1nc2ccccc2n1S(=O)(=O)c1ccc(C)cc1
CSc1nc2ccccc2n1C(=O)Oc1ccccc1
CSc1nc2ccccc2n1C(=O)NCc1ccc(C)cc1
Cc1ccc(C(=O)n2cnc3ccccc32)cc1
Cc1ccc(C(=O)n2ccc3ccccc32)cc1
Cc1ccc(C(=O)n2ncc3ccccc32)cc1
Cc1ccc(cc1)C(=O)n1nnc2ccccc12
CCSc1nc2ccccc2n1C(=O)c1ccc(C)cc1
C=CCSc1nc2ccccc2n1C(=O)c1ccc(C)cc1
Cc1ccc(C(=O)n2c(S)nc3ccccc32)cc1
COc1nc2ccccc2n1C(=O)c1ccc(C)cc1
Cc1ccc(C(=O)n2c(C)nc3ccccc32)cc1
CCc1nc2ccccc2n1C(=O)c1ccc(C)cc1
Cc1ccc(C(=O)n2c(C(F)(F)F)nc3ccccc32)cc1
Cc1ccc(C(=O)n2c(-c3ccccc3)nc3ccccc32)cc1
Cc1ccc(cc1)C(=O)n1c(N)nc2ccccc12
Cc1ccc(C(=O)n2c(C#N)nc3ccccc32)cc1
CSc1nc2ccccc2n1C(=O)c1cccc(C)c1
CSc1nc2ccccc2n1C(=O)c1ccccc1C
CSc1nc2ccccc2n1C(=O)c1ccc(C(F)(F)F)cc1
CSc1nc2ccccc2n1C(=O)c1cccc(C(F)(F)F)c1
CSc1nc2ccccc2n1C(=O)c1ccccc1C(F)(F)F
COc1ccc(C(=O)n2c(SC)nc3ccccc32)cc1
CCc1ccc(C(=O)n2c(SC)nc3ccccc32)cc1
CSc1nc2ccccc2n1C(=O)c1ccc(C(C)(C)C)cc1
CSc1nc2ccccc2n1C(=O)c1ccc(F)cc1
CSc1nc2ccccc2n1C(=O)c1ccc(Cl)cc1
CSc1nc2ccccc2n1C(=O)c1ccccc1
CSc1nc2ccccc2n1C(=O)c1ccncc1
CSc1nc2ccccc2n1C(=O)c1ccsc1
COc1ccc(C(=O)n2c(SC)nc3ccccc32)cc1OC
CSc1nc2ccccc2n1C(=O)c1ccc(C)c(C)c1
CSc1nc2ccccc2n1C(=O)c1ccc(C)c(F)c1
CSc1nc2ccccc2n1C(=O)c1ccc(C)c(Cl)c1
COc1cc(C(=O)n2c(SC)nc3ccccc32)ccc1C
CSc1nc2ccccc2n1C(=O)c1ccc2c(c1)OCCO2
CSc1nc2cc3c(cc2n1C(=O)c1ccc(C)c(F)c1)OCCO3
COc1cc2nc(SC)n(C(=O)c3ccc(C)cc3)c2cc1OC
CSc1nc2cc(Cl)ccc2n1C(=O)c1ccc(C)cc1
CSc1nc2ccc(Cl)cc2n1C(=O)c1ccc(C)cc1
CSc1nc2cc(F)ccc2n1C(=O)c1ccc(C)cc1
CSc1nc2ccc(F)cc2n1C(=O)c1ccc(C)cc1
CSc1nc2ccc(F)cc2n1C(=O)c1ccc(C)c(F)c1
CSc1nc2cc3c(cc2n1C(=O)c1ccc(C)cc1)OCO3
CSc1nc2cc3c(cc2n1C(=O)c1ccc(C)c(F)c1)OCO3
CSc1nc2cc(C#N)ccc2n1C(=O)c1ccc(C)c(F)c1
CSc1nc2ccc(C#N)cc2n1C(=O)c1ccc(C)c(F)c1
Cc1ccc(C(=O)n2c(C)nc3cc4c(cc32)OCCO4)cc1
Cc1ccc(C(=O)n2c(C)nc3ccccc32)cc1F
CSc1nc2cc(F)ccc2n1C(=O)c1ccc(C)c(F)c1
N#C[C@@]1(c2ccc3c(NC(=O)c4ccc(NC(=N)N)cc4)ncnn23)O[C@H](CO)[C@@H](O)[C@H]1O
CC(C)c1cc(=O)oc2ccc(OC(=O)c3ccc(NC(=N)N)cc3)cc12
N#C[C@@]1(c2ccc3c(NC(=O)c4ccc(Nc5ncccn5)cc4)ncnn23)O[C@H](CO)[C@@H](O)[C@H]1O
CC(C)(C)OC(=O)N[C@H](C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)C(C)(C)C
CC(C)(C)[C@H](NC(=O)C(F)(F)F)C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CC(C)(F)C(=O)N[C@H](C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)C(C)(C)C
[2H]C([2H])([2H])C(=O)N[C@H](C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)C(C)(C)C
CC(C)(C)[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
CN(C)S(=O)(=O)N[C@H](C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1)C(C)(C)C
CC(C)(C)OC[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N1[C@@H]2CC[C@@H](C2)[C@H]1C(=O)N[C@@H](C[C@@H]1CCNC1=O)C(=O)c1nc2ccccc2s1
COc1ccc(C[C@H](NS(=O)(=O)C(F)(F)F)C(=O)N2[C@@H]3CC[C@@H](C3)[C@H]2C(=O)N[C@@H](C[C@@H]2CCNC2=O)C(=O)c2nc3ccccc3s2)cc1
O=C1NCC[C@H]1C[C@H](NC(=O)[C@@H]1[C@H]2CC[C@H](C2)N1C(=O)[C@H](CC1CCCCC1)NS(=O)(=O)C(F)(F)F)C(=O)c1nc2ccccc2s1
O=C1NCC[C@H]1C[C@H](NC(=O)[C@@H]1[C@H]2CC[C@H](C2)N1C(=O)[C@@H](NS(=O)(=O)C(F)(F)F)C12CC3CC(CC(C3)C1)C2)C(=O)c1nc2ccccc2s1
CN1C[C@@H](c2ccccc2)[C@@]2(CN(P(=O)(CO)CO)C/C(=Cc3ccccc3)C2=O)[C@@]12C(=O)Nc1ccc(Cl)cc12
CN1C[C@@H](c2ccc(F)cc2)[C@@]2(CN(P(=O)(CO)CO)C/C(=Cc3ccccc3)C2=O)[C@@]12C(=O)Nc1ccc(Cl)cc12
CN1C[C@@H](c2ccc(Br)cc2)[C@@]2(CN(P(=O)(CO)CO)C/C(=Cc3ccccc3)C2=O)[C@@]12C(=O)Nc1ccccc12
CCC[C@@]1(CCc2ccccc2)CC(O)=C([C@H](CC)c2cccc(NS(=O)(=O)c3ccc(cn3)C(F)(F)F)c2)C(=O)O1 |t:15|
C=C(F)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C=C(Br)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C=C(C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1)C(F)(F)F
C=C(C)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C=C(C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1)c1ccccc1
C=C(NC(C)=O)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)/C=C/Br)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)/C=C/Cl)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)/C=CI)c1ccc(-c2ccccc2)cc1)c1ccccc1
C/C=C(C)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
CC(C)=CC(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)/C=C/C(=O)O)c1ccc(-c2ccccc2)cc1)c1ccccc1
COC(=O)/C=C/C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
CC(=O)/C=C/C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)/C=C/c1ccco1)c1ccc(-c2ccccc2)cc1)c1ccccc1
CO/C=C/C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C1=CC(=O)CC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C1=CCCCC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
C=CS(=O)(=O)N(c1ccc(-c2ccccc2)cc1)[C@H](C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C#CC(=O)N(c1ccc(-c2ccccc2)cc1)[C@H](C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
CCC#CC(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
CC(C)C#CC(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C#CC(C)(C)F)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C#CC1CC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
CCCC#CC(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C#CC(C)(C)C)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C#CC(C)(C)O)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)C#CCCl)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)[C@H](c1cccnc1)N(C(=O)C#CCCl)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)C#CCC#N)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)[C@H](c1cccnc1)N(C(=O)C#CCC#N)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C1(C#N)CC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C1(C#N)CCN(C(=O)OC(C)(C)C)CC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C1(C#N)CCOCC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
CC(C)/C=C(C#N)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)/C(C#N)=C/C1CC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C(C#N)=C1CCCCC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
CCC(=O)C(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C(=O)N1CCN(C)CC1)c1ccc(-c2ccccc2)cc1)c1ccccc1
C#CCC(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C#CCCC(=O)N(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C#CCN(c1ccc(-c2ccccc2)cc1)C(C(=O)N[C@@H](C)c1ccccc1)c1cccnc1
C[C@H](NC(=O)C(c1cccnc1)N(C(=O)C(F)(F)S(=O)(=O)F)c1ccc(-c2ccccc2)cc1)c1ccccc1
COc1ccc(/C=C(C#N)C(=O)N(c2ccc(-c3ccccc3)cc2)[C@H](C(=O)N[C@@H](C)c2ccccc2)c2cccnc2)cc1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)N1Cc1ccccc1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccccc1
O=C(Cc1ccccc1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CCc1ccccc1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(COc1ccccc1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CCCc1ccccc1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CNC(=O)c1ccccc1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CNC(=O)c1ccc(Cl)cc1)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)c1ccc(Cl)c(Cl)c1)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)c1ccc(Cl)c(F)c1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
N#Cc3cc(F)cc(C(=O)NCC(=O)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc2ccccn2)c3
N#Cc1cc(C(=O)NCC(=O)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc2ccccn2)ccc1F
O=C(CNC(=O)c2cc1ccccc1o2)N[C@H](Cc3ccccc3)C(=O)C(=O)NCc4ccccn4
O=C(CNC(=O)C1CCCCC1)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)C1CCOCC1)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)C1CCC(F)(F)CC1)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CC1CCC(F)(F)CC1)NCC(=O)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CNC(=O)[C@@H]1C[C@@H]2[C@H](C1)C2(F)F)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(CNC(=O)C1CCC(F)(F)CC1)N[C@H](Cc2ccc(Cl)cc2)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)C1CCC(F)(F)CC1)N[C@H](Cc2cccc(Cl)c2)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)C1CCC(F)(F)CC1)N[C@H](Cc2ccccc2Cl)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)C1CCC(F)(F)CC1)N[C@H](Cc2ccc(Cl)cc2Cl)C(=O)C(=O)NCc3ccccn3
O=C(CNC(=O)C1CCC(F)(F)CC1)N[C@H](Cc1ccc(Cl)c(Cl)c1)C(=O)C(=O)NCc1ccccn1
C[C@H](NC(=O)C1CCC(F)(F)CC1)C(=O)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
C[C@@H](NC(=O)C1CCC(F)(F)CC1)C(=O)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
CC[C@@H](NC(=O)C1CCC(F)(F)CC1)C(=O)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
COC[C@@H](NC(=O)C1CCC(F)(F)CC1)C(=O)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
CC(C)[C@@H](NC(=O)C1CCC(F)(F)CC1)C(=O)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)C1(NC(=O)C2CCC(F)(F)CC2)CC1
CN(CC(=O)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1)C(=O)C1CCC(F)(F)CC1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1CC(F)(F)CN1C(=O)C1CCC(F)(F)CC1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COCCN1C(=O)C1CCC(F)(F)CC1
C[C@@H](NC(=O)CC1CCC(F)(F)CC1)C(=O)N[C@H](Cc2ccccc2)C(=O)C(=O)NCc3ccccn3
C[C@@H](NC(=O)[C@@H]1C[C@@H]2[C@H](C1)C2(F)F)C(=O)N[C@H](Cc1ccccc1)C(=O)C(=O)NCc1ccccn1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1CC(F)(F)CN1C(=O)CC1CCC(F)(F)CC1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1CC(F)(F)CN1C(=O)[C@@H]1C[C@@H]2[C@H](C1)C2(F)F
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COCCN1C(=O)CC1CCC(F)(F)CC1
O=C(NCc1ccccn1)C(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COCCN1C(=O)[C@@H]1C[C@@H]2[C@H](C1)C2(F)F
[2H][C@](C(=O)N[C@@H](C)c1ccc(F)cc1)(c1ccccc1)N(C(=O)C(C)=O)c1ccc2c(c1)oc1ccccc12
O=C(NCCC1CCCC1)n1cc(F)c(=O)[nH]c1=O
O=C(NCCC1CCCCC1)n1cc(F)c(=O)[nH]c1=O
O=C(NCCCC1CCCCC1)n1cc(F)c(=O)[nH]c1=O
O=C(NCCCCc1ccccc1)n1cc(F)c(=O)[nH]c1=O
O=C(NCCCCCCc1ccccc1)n1cc(F)c(=O)[nH]c1=O
CC(C)(C)OC(=O)N1CCC(CCCNC(=O)n2cc(F)c(=O)[nH]c2=O)CC1
CC(C)(C)CC(=O)N1CCC(CCCNC(=O)n2cc(F)c(=O)[nH]c2=O)CC1
O=C(CC1CCCCC1)N1CCC(CCCNC(=O)n2cc(F)c(=O)[nH]c2=O)CC1
O=C(Cc1ccccc1)N1CCC(CCCNC(=O)n2cc(F)c(=O)[nH]c2=O)CC1
O=C(c1ccc2cc[nH]c2c1)N1CCC(CCCNC(=O)n2cc(F)c(=O)[nH]c2=O)CC1
O=C(NCCCNC(=O)n1cc(F)c(=O)[nH]c1=O)c1ccc2cc[nH]c2c1
Cn1ccc2ccc(C(=O)NCCCNC(=O)n3cc(F)c(=O)[nH]c3=O)cc21
O=C(NCCCNC(=O)n1cc(F)c(=O)[nH]c1=O)c1cc2ccccc2[nH]1
Cn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2ccccc21
CC(C)C[C@H](CNC(=O)c1cc2ccccc2[nH]1)CNC(=O)n1cc(F)c(=O)[nH]c1=O
CCn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2ccccc21
CC(C)Cn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2ccccc21
O=C(NCCCNC(=O)n1cc(F)c(=O)[nH]c1=O)c1cc2ccccc2n1Cc1ccccc1
Cc1ccc2c(c1)cc(C(=O)NCCCNC(=O)n1cc(F)c(=O)[nH]c1=O)n2CC(C)C
COc1ccc2c(c1)cc(C(=O)NCCCNC(=O)n1cc(F)c(=O)[nH]c1=O)n2CC(C)C
CC(C)Cn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2cc(Cl)ccc21
CC(C)Cn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2cc(F)ccc21
CC(C)Cn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2cc(C(F)(F)F)ccc21
CC(C)Cn1c(C(=O)NCCCNC(=O)n2cc(F)c(=O)[nH]c2=O)cc2cc(OC(F)(F)F)ccc21
CCCCCCNC(=O)n1ccc(=O)[nH]c1=O
CCCCCCNC(=O)n1cc(C)c(=O)[nH]c1=O
CCCCCCNC(=O)n1cc(CC)c(=O)[nH]c1=O
CCCCCCNC(=O)n1cc(Cl)c(=O)[nH]c1=O
CCCCCCNC(=O)n1cc(Br)c(=O)[nH]c1=O
CCCCCCNC(=O)n1cc(c(=O)[nH]c1=O)C(F)(F)F
CC(C)Cn1c(C(=O)NCCCNC(=O)n2ccc(=O)[nH]c2=O)cc2cc(Cl)ccc21
Cc1cn(C(=O)NCCCNC(=O)c2cc3cc(Cl)ccc3n2CC(C)C)c(=O)[nH]c1=O
CC(C)Cn1c(C(=O)NCCCNC(=O)n2ccc(=O)[nH]c2=O)cc2cc(F)ccc21
Cc1cn(C(=O)NCCCNC(=O)c2cc3cc(F)ccc3n2CC(C)C)c(=O)[nH]c1=O
CCSC1=CC(=O)c2ccccc2C1=O |t:3|
O=C1C=C(Sc2ccccc2)C(=O)c2ccccc21
COc1ccc(C(=C[C@@H]2COC[C@H]2S(=O)(=O)c2nnc(-c3ccc(Cl)cc3)o2)c2ccc(OC)cc2)cc1
COc1ccc(C(=C[C@@H]2COC[C@H]2S(=O)(=O)c2nnc(-c3ccc(Cl)cc3)[nH]2)c2ccc(OC)cc2)cc1
COc1ccc(C(=C[C@@H]2COC[C@H]2S(=O)(=O)c2nc(-c3ccc(Cl)cc3)cs2)c2ccc(OC)cc2)cc1
CS(=O)(=O)c1nnc(-c2ccc(Cl)cc2)o1
CCS(=O)(=O)c1nnc(-c2ccc(Cl)cc2)o1
COCCS(=O)(=O)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(CC1CC1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(c1nnc(-c2ccc(Cl)cc2)o1)C1COC1
O=S(=O)(c1nnc(-c2ccc(Cl)cc2)o1)C1CCOC1
O=S(=O)(c1ccccc1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1ccccc1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1cscn1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1ccccn1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1cccnc1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1ccncc1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1ncccn1)c1nnc(-c2ccc(Cl)cc2)o1
O=S(=O)(Cc1ccc2cnccc2c1)c1nnc(-c2ccc(Cl)cc2)o1
C[S+]([O-])c1nnc(-c2ccc(Cl)cc2)o1
CC[S+]([O-])c1nnc(-c2ccc(Cl)cc2)o1
COCC[S+]([O-])c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](CC1CC1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](c1nnc(-c2ccc(Cl)cc2)o1)C1COC1
[O-][S+](c1nnc(-c2ccc(Cl)cc2)o1)C1CCOC1
[O-][S+](c1ccccc1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1ccccc1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1cscn1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1ccccn1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1ccncc1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1ncccn1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1ccc2cnccc2c1)c1nnc(-c2ccc(Cl)cc2)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccccc2)o1
Cc1ccc(-c2nnc([S+]([O-])Cc3cccnc3)o2)cc1
N#Cc1ccc(-c2nnc([S+]([O-])Cc3cccnc3)o2)cc1
CC(C)(C)c1ccc(-c2nnc([S+]([O-])Cc3cccnc3)o2)cc1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccc(F)cc2)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccc(Br)cc2)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccc(OC(F)F)cc2)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccc(C(F)(F)F)cc2)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2ccccc2Br)o1
[O-][S+](Cc1cccnc1)c1nnc(-c2cccc(Br)c2)o1
OC(=O)C(=O)CC(=O)c1ccc(OCc2ccccc2)cc1
OC(=O)C(=O)CC(=O)c1cccc(NCc2ccc(Cl)cc2)c1
OC(=O)C(=O)CC(=O)c1cccc(NCc2ccccc2)c1
OC(=O)C(=O)CC(=O)c1ccc(OCc2ccc(Cl)cc2)cc1
OC(=O)C(=O)CC(=O)c1ccccc1OCc1ccc(Cl)cc1
OC(=O)C(=O)CC(=O)c1cccc(OCc2ccccc2)c1
OC(=O)C(=O)CC(=O)c1ccccc1OCc1ccccc1
OC(=O)C(=O)CC(=O)c1cccc(OCc2ccc(Cl)cc2)c1
Oc1cc(OCc2cccc(Cl)c2)cc2oc(c(O)c(=O)c12)-c1ccc2OCOc2c1
Oc1ccc(cc1O)-c1oc2cc(OCc3ccc(Cl)cc3)cc(O)c2c(=O)c1O
Oc1ccc(cc1O)-c1oc2cc(OCc3cccc(c3)C#N)cc(O)c2c(=O)c1O
Oc1ccc(cc1O)-c1oc2cc(OCc3cccc(Cl)c3)cc(O)c2c(=O)c1O
Oc1cc(CNCc2cccc(Cl)c2)oc2ccc(O)c(=O)c12
Oc1cc(OCc2cccc(c2)C#N)cc2oc(c(O)c(=O)c12)-c1ccc2OCOc2c1
Oc1cc(OCc2ccc(Cl)cc2)cc2oc(c(O)c(=O)c12)-c1ccc2OCOc2c1
Oc1cc(O)c2c(c1)oc(-c1ccc3OCOc3c1)c(O)c2=O
Oc1cc(CNCc2ccc(Cl)cc2)oc2ccc(O)c(=O)c12
Oc1cc(CNCc2cccc(c2)C#N)oc2ccc(O)c(=O)c12
Cc1nc(C)c(s1)C(=O)C1C(N(CCCN2CCOCC2)C(=O)C1=O)c1cccc(c1)[N+]([O-])=O
COc1cc(\C=N\NC(=O)C(\NC(=O)c2ccccc2)=C/c2ccccc2)cc(OC)c1O
COc1cc(ccc1O)C1C(C(=O)c2ccc(OCC(C)C)cc2C)C(=O)C(=O)N1CCN(C)C
CC1=NN(C(=O)\C1=C/c1ccc(o1)-c1cc(Cl)ccc1C(O)=O)c1cccc(c1)C(O)=O |t:1|
OC(=O)c1cccc(c1)N1N=C(\C(=C\c2ccc(o2)-c2cc(Cl)ccc2C(O)=O)C1=O)C(F)(F)F |c:11|
OC(=O)c1cccc(c1)N1N=C(\C(=C/c2ccc(o2)-c2ccccc2C(O)=O)C1=O)C(F)(F)F |c:11|
OC(=O)c1cccc(c1)N1N=C(\C(=C\c2ccc(o2)-c2cc(Cl)ccc2C(O)=O)C1=O)c1ccccc1 |c:11|
CC1=NN(C(=O)\C1=C/c1ccc(o1)-c1cc(Cl)ccc1C(O)=O)c1ccccc1 |t:1|
OC(=O)c1ccc(Cl)cc1-c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccccc2)o1 |c:20|
OC(=O)c1ccc(Cl)cc1-c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(F)cc2)o1 |c:20|
CC(C)c1ccc(cc1)N1N=C(\C(=C\c2ccc(o2)-c2cc(Cl)ccc2C(O)=O)C1=O)c1ccccc1 |c:11|
CC(C)(C)c1ccc(cc1)N1N=C(\C(=C\c2ccc(o2)-c2cc(Cl)ccc2C(O)=O)C1=O)c1ccccc1 |c:12|
O=C1N(N=C(\C1=C\c1ccc(o1)-c1ccccc1)c1ccccc1)c1ccccc1 |c:3|
OC(=O)c1cccc(c1)N1N=C(\C(=C\c2ccc(o2)-c2ccccc2)C1=O)c1ccccc1 |c:11|
CC1=NN(C(=O)\C1=C/c1ccc(o1)-c1ccccc1)c1cccc(c1)C(O)=O |t:1|
OC(=O)c1ccccc1-c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccccc2)o1 |c:19|
OC(=O)c1ccccc1-c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(F)cc2)o1 |c:19|
CC(C)c1ccc(cc1)N1N=C(\C(=C\c2ccc(o2)-c2ccccc2C(O)=O)C1=O)c1ccccc1 |c:11|
CC(C)(C)c1ccc(cc1)N1N=C(\C(=C\c2ccc(o2)-c2ccccc2C(O)=O)C1=O)c1ccccc1 |c:12|
OC(=O)c1ccccc1-c1ccc(\C=C2/C(=O)N(N=C2c2ccccc2)c2ccc(cc2)C#N)o1 |c:19|
COc1ccc(cc1)N1N=C(\C(=C\c2ccc(o2)-c2ccccc2C(O)=O)C1=O)c1ccccc1 |c:10|
OC(=O)c1cccc(c1)N1N=C(\C(=C\c2ccco2)C1=O)c1ccccc1 |c:11|
OC(=O)c1cccc(c1)N1N=C(\C(=C\c2ccc(cc2)-c2ccccc2)C1=O)c1ccccc1 |c:11|
OC(=O)c1cccc(c1)N1N=C(\C(=C\c2ccc(OCc3ccccc3)cc2)C1=O)c1ccccc1 |c:11|