Compile Data Set for Download or QSAR
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Found 28 with Last Name = 'cai' and Initial = 'rz'
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187196(2'-[(4-fluorophenyl)methyl]-4'-hydroxy-9'-methoxy-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187761(7-(4-fluorobenzyl)-9-hydroxy-5-(morpholine-4-carbo...)
Affinity DataIC50:  36nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187194(7-(4-fluorobenzyl)-6,9-dihydroxy-5-methoxy-6,7-dih...)
Affinity DataIC50:  36nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM23403(7-[(4-fluorophenyl)methyl]-9-hydroxy-5-methoxy-6H,...)
Affinity DataIC50:  50nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM23402(5-(1,1-dioxo-1,2-thiazinan-2-yl)-N-[(4-fluoropheny...)
Affinity DataIC50:  50nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187198(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-6-(3-oxo-3-...)
Affinity DataIC50:  59nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM23403(7-[(4-fluorophenyl)methyl]-9-hydroxy-5-methoxy-6H,...)
Affinity DataIC50:  60nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187191(7-(4-fluorobenzyl)-9-hydroxy-5,6-dimethoxy-6,7-dih...)
Affinity DataIC50:  64nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187760(7-(4-fluorobenzyl)-9-hydroxy-6,7-dihydropyrrolo[3,...)
Affinity DataIC50:  70nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187764(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-6H-pyrrolo[...)
Affinity DataIC50:  80nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187186(7-(4-fluorobenzyl)-5,9-dihydroxy-7H-pyrrolo[3,4-g]...)
Affinity DataIC50:  80nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187190(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-6-methyl-6,...)
Affinity DataIC50:  88nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187185(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-6-methylene...)
Affinity DataIC50:  150nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187759(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-N-(pyridin-2-yl...)
Affinity DataIC50:  190nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187193(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-6,6-dimethy...)
Affinity DataIC50:  210nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187187(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-7,8-dihydro-6H-...)
Affinity DataIC50:  255nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187197(3-(7-(4-fluorobenzyl)-9-hydroxy-5-methoxy-8-oxo-7,...)
Affinity DataIC50:  295nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187188(CHEMBL209641 | methyl 3-(7-(4-fluorobenzyl)-9-hydr...)
Affinity DataIC50:  310nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187765(5-(2,6-difluorophenyl)-7-(4-fluorobenzyl)-9-hydrox...)
Affinity DataIC50:  335nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187767(CHEMBL378395 | ethyl 2-(7-(4-fluorobenzyl)-9-hydro...)
Affinity DataIC50:  350nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187189(2'-[(4-fluorophenyl)methyl]-4'-hydroxy-3'-oxo-2',3...)
Affinity DataIC50:  357nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187192(7-(4-fluorobenzyl)-9-hydroxy-6-methylene-8-oxo-7,8...)
Affinity DataIC50:  420nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187763(7-(4-fluorobenzyl)-9-hydroxy-8-oxo-7,8-dihydro-6H-...)
Affinity DataIC50:  760nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187195(7-(4-fluorobenzyl)-9-hydroxy-6-methyl-8-oxo-7,8-di...)
Affinity DataIC50:  815nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in MT4 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187758(5-(4-ethoxyphenyl)-7-(4-fluorobenzyl)-6H-pyrrolo[3...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187768(CHEMBL209591 | N-(4-fluorobenzyl)-8-hydroxyquinoli...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187762(CHEMBL211275 | ethyl 3-(7-(4-fluorobenzyl)-9-hydro...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50187766(7-(4-fluorobenzyl)-9-hydroxy-6,8-dioxo-7,8-dihydro...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of strand transfer activity of HIV integraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed