TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 370nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 428nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Inhibition of bovine brain tubulin assembly using GTP as substrate incubated for 20 mins by spectrophotometric methodMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 681nMAssay Description:Inhibition of recombinant N-terminal His-tagged human iNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization incubated for 15 mins followed by addition of GTP and measured for 20 mins by turbidimetric analysi...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of recombinant human nNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins followed by NADPH addition ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of recombinant human nNOS expressed in Escherichia coli using L-arginine as substrate preincubated for 15 mins followed by NADPH addition ...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human eNOS using L-argininge as substrate preincubated for 15 mins followed by NADPH addition and measured after 20 mins by OPA/NAC rea...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of iNOS assessed as conversion of L-[3H]arginine to L-[3H]-citrulline after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 2.96E+4nMAssay Description:Inhibition of iNOS assessed as conversion of L-[3H]arginine to L-[3H]-citrulline after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of iNOS assessed as conversion of L-[3H]arginine to L-[3H]-citrulline after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 4.10E+4nMAssay Description:Inhibition of iNOS assessed as conversion of L-[3H]arginine to L-[3H]-citrulline after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 4.52E+4nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 5.97E+4nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 1.80E+5nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 1.94E+5nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 2.23E+5nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 3.04E+5nMAssay Description:Inhibition of human eNOS using L-argininge as substrate preincubated for 15 mins followed by NADPH addition and measured after 20 mins by OPA/NAC rea...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 3.25E+5nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibition of recombinant nNOS (unknown origin) assessed as conversion of L-[3H]-arginine to L-[3H]-citrulline after 30 minsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 5.30E+5nMAssay Description:Inhibition of recombinant nNOS (unknown origin) assessed as conversion of L-[3H]-arginine to L-[3H]-citrulline after 30 minsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: 8.80E+5nMAssay Description:Inhibition of recombinant nNOS (unknown origin) assessed as conversion of L-[3H]-arginine to L-[3H]-citrulline after 30 minsMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of N-terminal His-tagged human recombinant iNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
University "G. D'Annunzio" Of Chieti-Pescara
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant nNOS expressed in Escherichia coli assessed as reduction in L-[3H]-citrulline level using L-[3H]-arginine as substrat...More data for this Ligand-Target Pair