Affinity DataKi: 8nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 8nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 10nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 13nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 14nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 16nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 26nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 43nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
Affinity DataKi: 50nMpH: 7.4Assay Description:The radioligand EP4 binding assay was performed using ChemiScreen recombinant human EP4 receptor membrane preparations from Millipore, according to m...More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 73nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 108nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetInterstitial collagenase(Homo sapiens (Human))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase 1More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 121nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetInterstitial collagenase(Homo sapiens (Human))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase 1More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 139nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 187nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 207nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMetalloproteinase inhibitor 3(Rattus norvegicus)
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 223nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Rattus norvegicus (Rat))
Novartis Biomedical Research Institute
Curated by ChEMBL
Novartis Biomedical Research Institute
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory activity against matrix metalloproteinase-9More data for this Ligand-Target Pair