Affinity DataIC50: 0.130nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.260nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.390nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.690nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Selectivity against rhesus monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 0.790nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Selectivity against guinea pig plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Selectivity against sheep plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Concentration required for 50% inhibition of human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Concentration required for 50% inhibition of human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Concentration required for 50% inhibition of human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Concentration required for 50% inhibition of human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Concentration required for 50% inhibition of human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Concentration required for 50% inhibition of human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Selectivity against dog plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Concentration required for 50% inhibition of sheep plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Concentration required for 50% inhibition of rhesus monkey plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Concentration required for 50% inhibition of human plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required for 50% inhibition of human kidney reninMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Concentration required for 50% inhibition of dog plasma reninMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Concentration required for 50% inhibition of human kidney reninMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibitory effect against human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Concentration required for 50% inhibition of human plasma reninMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibitory effect against human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland
Curated by ChEMBL
Aventis Pharma Deutschland
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibitory effect against human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair