Compile Data Set for Download or QSAR
maximum 50k data
Found 59 with Last Name = 'matsumizu' and Initial = 'm'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348115(CHEMBL1800654)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348114(CHEMBL1800653)
Affinity DataKi: >1.94E+4nMAssay Description:Binding affinity at human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348122(CHEMBL1800168)
Affinity DataKi: >2.00E+4nMAssay Description:Binding affinity at human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220714(CHEMBL237751 | N-((1s,4s)-4-hydroxy-4-(5-hydroxypy...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220726(CHEMBL237533 | N-((1s,4s)-4-(3-fluoro-4-hydroxyphe...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220729(CHEMBL237320 | N-((1s,4s)-4-hydroxy-4-(4-hydroxyph...)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220712(CHEMBL395904 | N-((1s,4s)-4-hydroxy-4-(4-hydroxy-2...)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220716(CHEMBL236893 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50:  30nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220727(CHEMBL237534 | N-((1r,4r)-4-(3-fluoro-4-hydroxyphe...)
Affinity DataIC50:  59nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220720(CHEMBL237752 | N-((1s,4s)-4-hydroxy-4-(2-oxo-2,3-d...)
Affinity DataIC50:  85nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220725(CHEMBL237101 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50:  96nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220728(CHEMBL237962 | N-((1s,4s)-4-hydroxy-4-(5-hydroxy-4...)
Affinity DataIC50:  116nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220715(CHEMBL237321 | N-((1s,4s)-4-hydroxy-4-(4-hydroxy-3...)
Affinity DataIC50:  189nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220713(CHEMBL237323 | N-((1r,4r)-4-(4-hydroxy-2-methylphe...)
Affinity DataIC50:  722nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220718(CHEMBL236895 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50:  856nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220723(CHEMBL237102 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220731(CHEMBL393609 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220734(2-(dimethylamino)-N-((1r,4r)-4-(4-hydroxyphenyl)cy...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220719(CHEMBL236894 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220730((R)-6-(2-(4-(3-fluorophenyl)-4-hydroxypiperidin-1-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220732(CHEMBL237965 | N-((1s,4s)-4-hydroxy-4-(1H-pyrazol-...)
Affinity DataIC50:  2.44E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348122(CHEMBL1800168)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220735(CHEMBL238184 | N-((1s,4s)-4-(1H-benzo[d]imidazol-5...)
Affinity DataIC50:  4.96E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220722(CHEMBL237322 | N-((1r,4r)-4-(4-hydroxy-3-methylphe...)
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220717(CHEMBL237964 | N-((1s,4s)-4-(6-aminopyridin-3-yl)-...)
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220721(CHEMBL398127 | N-((1s,4s)-4-hydroxy-4-(1H-imidazol...)
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 2B(Rattus norvegicus (Rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220724(CHEMBL237963 | N-((1s,4s)-4-hydroxy-4-(6-(methylsu...)
Affinity DataIC50: >5.00E+3nMAssay Description:Displacement of [3H]CP101,606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220725(CHEMBL237101 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220716(CHEMBL236893 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220729(CHEMBL237320 | N-((1s,4s)-4-hydroxy-4-(4-hydroxyph...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220714(CHEMBL237751 | N-((1s,4s)-4-hydroxy-4-(5-hydroxypy...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220733(4-benzyl-1-(2-hydroxy-2-(4-hydroxyphenyl)ethyl)pip...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220726(CHEMBL237533 | N-((1s,4s)-4-(3-fluoro-4-hydroxyphe...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220723(CHEMBL237102 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220719(CHEMBL236894 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220718(CHEMBL236895 | N-((1r,4r)-4-(4-hydroxyphenyl)cyclo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50220713(CHEMBL237323 | N-((1r,4r)-4-(4-hydroxy-2-methylphe...)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348117(CHEMBL1800163)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348116(CHEMBL1800655)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348119(CHEMBL1800165)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348120(CHEMBL1800166)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348121(CHEMBL1800167)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348122(CHEMBL1800168)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348115(CHEMBL1800654)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348114(CHEMBL1800653)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348123(CHEMBL1800169)
Affinity DataEC50:  132nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348124(CHEMBL1800170)
Affinity DataEC50:  199nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348125(CHEMBL1800171)
Affinity DataEC50:  425nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348126(CHEMBL1800172)
Affinity DataEC50:  82nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50348127(CHEMBL1800173)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human recombinant CB2 receptor expressed in CHO cells assessed as inhibition forskolin-induced cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 59 total ) | Next | Last >>
Jump to: