Affinity DataKi: 0.0150nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0850nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:In vitro inhibition of rat liver dihydrofolate reductase.More data for this Ligand-Target Pair
Affinity DataKi: 0.261nMAssay Description:In vitro inhibition of rat liver dihydrofolate reductase.More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University
Curated by ChEMBL
New York University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]-haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University
Curated by ChEMBL
New York University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]- haloperidolMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
New York University
Curated by ChEMBL
New York University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]- haloperidolMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 82nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 168nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 491nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 507nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: 770nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 820nMAssay Description:In vivo compound was evaluated for binding towards Dopamine receptor D2 in rat striatal membranes using competitive binding assay and [125I]IBZM radi...More data for this Ligand-Target Pair
Affinity DataKi: 843nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: 1.24E+3nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:The compound was tested for competition binding with [3H]NKA against the CHO cells from cloned human Tachykinin receptor 2More data for this Ligand-Target Pair
TargetSubstance-K receptor(Homo sapiens (Human))
Creighton University School Of Medicine
Curated by ChEMBL
Creighton University School Of Medicine
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity towards NK-2 receptors using [3H]NKA as radioligand in cloned human CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibition of human ABL by radiometric assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Washington
Curated by ChEMBL
University Of Washington
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human SRC by radiometric assayMore data for this Ligand-Target Pair