Compile Data Set for Download or QSAR
maximum 50k data
Found 75 with Last Name = 'tracey' and Initial = 'wr'
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50006730((R)-2-Hydroxymethyl-5-[6-(1-methyl-2-phenyl-ethyla...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122928(5-{6-[5-Chloro-2-(3-methyl-isoxazol-5-ylmethoxy)-b...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50034171(3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl...)
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182312((2S,3S,4R,5R)-5-(6-(3,5-dichlorobenzylamino)-9H-pu...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182322((2S,3S,4R,5R)-5-(6-(2,5-dimethoxybenzylamino)-9H-p...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82557(I-ABA | IABA | N(6)-(4-Amino-3-iodobenzyl)adenosin...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122927((2S,3S,4R,5R)-3,4-dihydroxy-N-methyl-5-(6-(methyla...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122927((2S,3S,4R,5R)-3,4-dihydroxy-N-methyl-5-(6-(methyla...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM82557(I-ABA | IABA | N(6)-(4-Amino-3-iodobenzyl)adenosin...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122926(3-Amino-5-{6-[5-chloro-2-(3-methyl-isoxazol-5-ylme...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50037785(2-(6-{[2-(4-aminophenyl)ethyl]amino}-9H-purin-9-yl...)
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182326((2S,3S,4R,5R)-5-(6-(2-(2-amino-2-oxoethoxy)-5-chlo...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182313((2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-(4-(dimethylamin...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182324((2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-oxo-2-(piperazin...)
Affinity DataKi:  9.40nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  14nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182323((2S,3S,4R,5R)-5-(6-(5-chloro-2-methoxybenzylamino)...)
Affinity DataKi:  15nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182321((2S,3S,4R,5R)-5-(6-(2-(benzyloxy)-5-chlorobenzylam...)
Affinity DataKi:  16nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182311((2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-oxo-2-(piperidin...)
Affinity DataKi:  18nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50118812((2S,3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-iodo-benzylami...)
Affinity DataKi:  20nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182318((2S,3S,4R,5R)-5-(6-(5-chloro-2-(2-morpholino-2-oxo...)
Affinity DataKi:  20nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Sheep)
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182325((2S,3S,4R,5R)-5-(6-(3,5-dichlorobenzylamino)-9H-pu...)
Affinity DataKi:  25nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50034171(3,4-Dihydroxy-5-[6-(3-iodo-benzylamino)-purin-9-yl...)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A1(Oryctolagus cuniculus (Rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85037(ABA | CAS_14375-45-2)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50037785(2-(6-{[2-(4-aminophenyl)ethyl]amino}-9H-purin-9-yl...)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM25400((2R,3R,4S,5R)-2-[6-(cyclopentylamino)-9H-purin-9-y...)
Affinity DataKi:  49nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50006730((R)-2-Hydroxymethyl-5-[6-(1-methyl-2-phenyl-ethyla...)
Affinity DataKi:  49nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182320((2S,4R,5R)-4-hydroxy-N-methyl-5-(6-(methylamino)-9...)
Affinity DataKi:  59nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122927((2S,3S,4R,5R)-3,4-dihydroxy-N-methyl-5-(6-(methyla...)
Affinity DataKi:  65nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122928(5-{6-[5-Chloro-2-(3-methyl-isoxazol-5-ylmethoxy)-b...)
Affinity DataKi:  68nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122929(3-Amino-4-hydroxy-5-[6-(3-iodo-benzylamino)-purin-...)
Affinity DataKi:  72nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182317((2S,3S,5R)-3-hydroxy-N-methyl-5-(6-(methylamino)-9...)
Affinity DataKi:  87nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM21221((2S,3S,4R,5R)-5-(2-chloro-6-{[(3-iodophenyl)methyl...)
Affinity DataKi:  99nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122930((2S,3S,4R,5R)-3-amino-4-hydroxy-N-methyl-5-(6-(met...)
Affinity DataKi:  120nMAssay Description:Binding affinity using [125I]-ABA against human Adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
Affinity DataKi:  120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50122930((2S,3S,4R,5R)-3-amino-4-hydroxy-N-methyl-5-(6-(met...)
Affinity DataKi:  120nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182319(2-(2-((9-((2R,3R,4S,5S)-4-amino-3-hydroxy-5-(methy...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50182327((2S,3S,4R,5R)-5-(6-(2,5-dimethoxybenzylamino)-9H-p...)
Affinity DataKi:  160nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85037(ABA | CAS_14375-45-2)
Affinity DataKi:  169nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM50207816(CHEMBL273094 | N-(2-Amino-ethyl)-2-[4-(2,6-dioxo-1...)
Affinity DataKi:  329nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Oryctolagus cuniculus (rabbit))
Pfizer

Curated by PDSP Ki Database
LigandPNGBDBM85036(BW-A1433 | BWA1433 | CAS_129447 | NSC_129447)
Affinity DataKi:  746nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Displayed 1 to 50 (of 75 total ) | Next | Last >>
Jump to: