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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
97
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Target
Metabotropic glutamate receptor 8
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
Ki: 61nM
Assay Description:
Agonist potency against cloned Metabotropic glutamate receptor 8 (mGluR-8).
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
Ki: 160nM
Assay Description:
Displacement of [3H]L-AP4 from rat recombinant mGluR4 expressed in BHK cells by SPA assay
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 160nM
Assay Description:
Displacement of [3H]L-AP4 from rat mGluR4 expressed in BHK cells
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 160nM
Assay Description:
Displacement of [3H]Quisqualate from human mGluR4 receptor expressed in BHK cells
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 470nM
Assay Description:
Binding affinity at Metabotropic glutamate receptor 4
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Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 900nM
Assay Description:
Agonist potency against cloned Metabotropic glutamate receptor 6 (mGluR-6).
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 910nM
Assay Description:
Agonist potency against cloned human Metabotropic glutamate receptor 4 (mGluR-4)
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Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
University of Minnesota
Curated by
PDSP K
i
Database
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
Ki: 1.50E+3nM
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
Ki: 1.90E+3nM
Assay Description:
Displacement of [3H]LY341495 from rat mGluR8 expressed in BHK cells
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.90E+3nM
Assay Description:
Displacement of [3H]LY341495 from rat recombinant mGluR8 expressed in BHK cells by SPA assay
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
Ki: 2.70E+3nM
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
Ki: 1.29E+5nM
Assay Description:
Binding affinity at Metabotropic glutamate receptor 2
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
Ki: 1.75E+5nM
Assay Description:
Agonist potency against cloned Metabotropic glutamate receptor 7 (mGluR-7).
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Agonist potency against cloned human metabotropic glutamate receptor 1
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Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Agonist potency against cloned metabotropic glutamate receptor 5
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Agonist potency against cloned Metabotropic glutamate receptor 2 (mGluR-2).
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 3
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Agonist potency against cloned Metabotropic glutamate receptor 3 (mGluR-3).
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Binding affinity at Metabotropic glutamate receptor 1
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Displacement of [3H]Quisqualate from human mGluR1A receptor expressed in BHK cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Displacement of [3H]Quisqualate from human mGluR5 receptor expressed in BHK cells
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: >1.00E+6nM
Assay Description:
Displacement of [3H]Quisqualate from human mGluR2 receptor expressed in BHK cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 130nM
Assay Description:
Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...
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Target
Metabotropic glutamate receptor 8
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 290nM
Assay Description:
Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 100nM
Assay Description:
Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...
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Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 2.40E+3nM
Assay Description:
Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.49E+5nM
Assay Description:
Agonist activity at mGlu7 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...
More data for this Ligand-Target Pair
Target Info
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Copy BDB DOI
Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.37E+5nM
Assay Description:
Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.00E+3nM
Assay Description:
Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 8
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 290nM
Assay Description:
Agonist activity at mGlu8 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as increase in intracellular calcium...
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 130nM
Assay Description:
Agonist activity at mGlu6 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...
More data for this Ligand-Target Pair
Target Info
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 310nM
Assay Description:
Activation of human metabotropic glutamate 4 receptor expressed in golden hamster AV12-664 cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 8
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 60nM
Assay Description:
Activation of human metabotropic glutamate 8 receptor expressed in golden hamster AV12-664 cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 55nM
Assay Description:
Activation of human metabotropic glutamate 6 receptor expressed in golden hamster AV12-664 cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 500nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR4a in rat
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 1.60E+5nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR7 in rat
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR2 in rat
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 500nM
Assay Description:
Agonistic activity at Metabotropic glutamate receptor 4 expressed in mammalian cells by GTPgammaS binding assay
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 55nM
Assay Description:
Metabotropic glutamate receptor 6 agonist activity to influence forskolin stimulated c-AMP formation in rat nonneuronal cells
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+5nM
Assay Description:
Metabotropic glutamate receptor 1 agonist activity as basal [3H]- IP formation in rat
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 320nM
Assay Description:
Metabotropic glutamate receptor 4 agonist activity to influence forskolin stimulated c-AMP formation in rat nonneuronal cells
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 4.48E+5nM
Assay Description:
Metabotropic glutamate receptor 2 agonist activity against forskolin stimulated c-AMP formation in rat nonneuronal cells
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 60nM
Assay Description:
Metabotropic glutamate receptor 8 agonist activity against forskolin stimulated c-AMP formation in rat nonneuronal cells
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+5nM
Assay Description:
Metabotropic glutamate receptor 5 agonist activity as basal [3H]- IP formation in rat
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Target
Metabotropic glutamate receptor 3
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+5nM
Assay Description:
Metabotropic glutamate receptor 3 agonist activity against forskolin stimulated c-AMP formation in rat nonneuronal cells
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 1.75E+5nM
Assay Description:
Metabotropic glutamate receptor 7 agonist activity to influence forskolin stimulated c-AMP formation in rat nonneuronal cells
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 30nM
Assay Description:
Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assay
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 3.45E+3nM
Assay Description:
Agonist activity at rat mGluR6 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assay
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 4.26E+5nM
Assay Description:
Agonist activity at rat mGluR7 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assay
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 110nM
Assay Description:
Agonist activity at rat mGluR8 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assay
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 2.08E+3nM
Assay Description:
Agonist activity at rat mGluR6 receptor expressed HEK293 cells assessed as effect on inositol phosphate production
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 80nM
Assay Description:
Agonist activity at rat mGluR4 receptor expressed HEK293 cells assessed as effect on inositol phosphate production
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 4.40E+5nM
Assay Description:
Agonist activity at rat mGluR7 receptor expressed HEK293 cells assessed as effect on inositol phosphate production
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Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 128nM
Assay Description:
Agonist activity at rat mGluR8 receptor expressed HEK293 cells assessed as effect on inositol phosphate production
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 690nM
Assay Description:
Agonist activity at mGlu4 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate production
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Metabotropic glutamate receptor 8
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 560nM
Assay Description:
Agonist activity at mGlu8 receptor expressed in HEK 293 cells assessed as effect on inositol phosphate production
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 30nM
Assay Description:
Agonist activity at rat mGlu4 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assay
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 1.91E+3nM
Assay Description:
Agonist activity at rat mGlu6 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assay
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 3.40E+5nM
Assay Description:
Agonist activity at rat mGlu7 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assay
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 70nM
Assay Description:
Agonist activity at rat mGlu8 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assay
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR2 in human
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Target
Metabotropic glutamate receptor 8
(Mus musculus)
Cns Research
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 400nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR8 in mouse
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Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Universit£
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ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 200nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR4a in human
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR1c in rat
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 500nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR4a in rat
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 900nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR6 in rat
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 1.60E+5nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR7 in rat
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR2 in rat
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 2.00E+5nM
Assay Description:
Concentration for half maximal activation of metabotropic glutamate mGluR7 in human
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 910nM
Assay Description:
Effect on Metabotropic glutamate receptor 4
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 2.52E+5nM
Assay Description:
Effect on Metabotropic glutamate receptor 7
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 1.00E+6nM
Assay Description:
Effect on Metabotropic glutamate receptor 2
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Effect on Metabotropic glutamate receptor 5
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 1.00E+6nM
Assay Description:
Effect on Metabotropic glutamate receptor 1
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 570nM
Assay Description:
Effect on Metabotropic glutamate receptor 6
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 320nM
Assay Description:
Stimulation od [3H]phosphatidylinositol accumulation by rat Metabotropic glutamate receptor 4 co-expressed with Gqi9 protein in HEK 293 cells
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: 1.29E+5nM
Assay Description:
Effective concentration against D309A mutant Metabotropic glutamate receptor 4
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 200nM
Assay Description:
Effective concentration against Metabotropic glutamate receptor 4
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 510nM
Assay Description:
Functional activity at rat mGluR4
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 340nM
Assay Description:
Activity at rat mGluR6 by measuring cAMP formation in CHO cells
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Activity at rat mGluR1 by measuring intracellular calcium concentration in CHO cells
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Activity at human mGluR2 from BHK cells in [35S]GTP-gamma-S stimulation assay
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 1.88E+5nM
Assay Description:
Activity at human mGluR7 by measuring cAMP formation in BHK cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Activity at rat mGluR5 by measuring intracellular calcium concentration in CHO cells
More data for this Ligand-Target Pair
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Target
Metabotropic glutamate receptor 1
(RAT)
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Activity at rat recombinant mGluR1 expressed in CHO cells assessed as intracellular calcium concentration
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Target
Metabotropic glutamate receptor 5
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Activity at rat recombinant mGluR5 expressed in CHO cells assessed as intracellular calcium concentration
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 510nM
Assay Description:
Agonist activity at rat recombinant mGluR4 expressed in BHK cells
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Target
Metabotropic glutamate receptor 7
(Homo sapiens (Human))
The Royal Danish School Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 1.88E+5nM
Assay Description:
Activity at human recombinant mGluR7 expressed in BHK cells assessed as cAMP production
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Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Parc Club Orsay Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: >1.00E+6nM
Assay Description:
Activity at human recombinant mGluR2 expressed in BHK cells assessed as stimulation of [35S]GTP-gamma-S binding
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 340nM
Assay Description:
Activity at rat recombinant mGluR6 expressed in CHO cells assessed as cAMP production
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 3.06E+5nM
Assay Description:
Agonist activity at rat mGlu7 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 300nM
Assay Description:
Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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3D Structure (crystal)
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Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 240nM
Assay Description:
Agonist activity at rat mGlu8 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 130nM
Assay Description:
Agonist activity at rat mGlu4 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 96nM
Assay Description:
Agonist activity at rat mGlu4 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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Target Info
PDB
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 1.00E+3nM
Assay Description:
Agonist activity at rat mGlu6 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.30E+3nM
Assay Description:
Agonist activity at rat mGlu6 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
Cns Research
Curated by
ChEMBL
Ligand
BDBM50007548
((S)-2-Amino-4-phosphono-butyric acid | (S)-2-amino...)
Copy SMILES
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Affinity Data
EC50: 2.49E+5nM
Assay Description:
Agonist activity at rat mGlu7 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...
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