Found 29 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein phosphatase 2A catalytic subunit alpha isoform'
Affinity DataIC50: 0.25nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration of the compound against Protein phosphatase 2A (25 nM) isolated from bovine myocardial tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Antagonist activity at rat H3 receptor expressed in human SK-N-MC cells assessed as inhibition of forskolin-induced cAMP accumulation after 6 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of PP2A alpha (unknown origin) pre-incubated for 20 mins followed by fluorescence substrate addition and measured after 120 mins by DiFMUP...More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 304nMAssay Description:Inhibitory concentration of the compound against Protein phosphatase 2A (25 nM) isolated from bovine myocardial tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human H-PGDS expressed in Escherichia coli BL21 DE2 by enzyme immuno assay at 50 uMMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Inhibition of recombinant human PP2A catalytic subunit L309 deletion mutant using DIFMUP as substrate pretreated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 2A (PP2A) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >3.90E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >6.30E+4nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against protein phosphatase 2A (PP2A) using pNPP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Homo sapiens (Human))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration of the compound against Protein phosphatase 2A (25 nM) isolated from bovine myocardial tissueMore data for this Ligand-Target Pair