TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.214nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.240nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.288nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.295nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.339nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.347nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.355nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against Alpha-1 adrenergic receptor was determined using [3H]WB-4101 radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.447nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.589nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.603nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.692nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 0.891nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Concentration of the compound necessary to achieve half maximal inhibition of [3H]-clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 3.67nMAssay Description:Displacement of [3H]MK9112 from human recombinant adrenergic alpha2A receptor expressed in insect Sf9 cells after 60 minsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 7.70nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 9.90nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Binding affinity for human cloned Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]-clonidine binding to alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]-clonidine binding to alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]-clonidine binding to alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Binding affinity at human Alpha-2A adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]-clonidine binding to alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465](Rattus norvegicus (rat))
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Hoechst-Roussel Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen Research Foundation
Curated by ChEMBL
Janssen Research Foundation
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibitory activity against constitutively activated human Alpha-2A adrenergic receptor transiently expressed in COS-1 cells using [3H]-MK912More data for this Ligand-Target Pair