Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 50049313
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238882BDBM50238882(CHEMBL4094600)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238893BDBM50238893(CHEMBL4096379)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human CLK4 expressed in baculovirus infected Sf21 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026622BDBM50026622(CHEMBL408982)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238868BDBM50238868(CHEMBL4072795)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238881BDBM50238881(CHEMBL4067143)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238884BDBM50238884(CHEMBL4060440)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238887BDBM50238887(CHEMBL4093503)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human CLK2 (144 to 498 residues) expressed in insect cells using S6 kinase/Rsk2 substrate peptide 2 in presence of [gamma-3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238892BDBM50238892(CHEMBL4104765)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238883BDBM50238883(CHEMBL4088668)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238885BDBM50238885(CHEMBL4069124)
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238886BDBM50238886(CHEMBL4104122)
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50026622BDBM50026622(CHEMBL408982)
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238893BDBM50238893(CHEMBL4096379)
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 138nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238866BDBM50238866(CHEMBL4079878)
Affinity DataIC50: 139nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238892BDBM50238892(CHEMBL4104765)
Affinity DataIC50: 141nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238879BDBM50238879(CHEMBL4064426)
Affinity DataIC50: 155nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238880BDBM50238880(CHEMBL4086890)
Affinity DataIC50: 173nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238882BDBM50238882(CHEMBL4094600)
Affinity DataIC50: 177nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238874BDBM50238874(CHEMBL4100703)
Affinity DataIC50: 186nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238876BDBM50238876(CHEMBL4081470)
Affinity DataIC50: 189nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238883BDBM50238883(CHEMBL4088668)
Affinity DataIC50: 194nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238881BDBM50238881(CHEMBL4067143)
Affinity DataIC50: 245nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238868BDBM50238868(CHEMBL4072795)
Affinity DataIC50: 257nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238888BDBM50238888(CHEMBL4063617)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238886BDBM50238886(CHEMBL4104122)
Affinity DataIC50: 283nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238885BDBM50238885(CHEMBL4069124)
Affinity DataIC50: 404nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238866BDBM50238866(CHEMBL4079878)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238890BDBM50238890(CHEMBL4092984)
Affinity DataIC50: 430nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238875BDBM50238875(CHEMBL4072220)
Affinity DataIC50: 439nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238889BDBM50238889(CHEMBL4082710)
Affinity DataIC50: 529nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 690nMAssay Description:Inhibition of human DYRK1BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238870BDBM50238870(CHEMBL4104093)
Affinity DataIC50: 993nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238876BDBM50238876(CHEMBL4081470)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238884BDBM50238884(CHEMBL4060440)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238887BDBM50238887(CHEMBL4093503)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238880BDBM50238880(CHEMBL4086890)
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of recombinant human CDK9 expressed in fall armyworm sf21 cells using PDKtide as substrate in presence of [gamma-32]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of recombinant human GSK3beta expressed in fall armyworm sf21 cells using Phospho-glycogen synthase peptide-2 as substrate in presence of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238879BDBM50238879(CHEMBL4064426)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238890BDBM50238890(CHEMBL4092984)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238888BDBM50238888(CHEMBL4063617)
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238889BDBM50238889(CHEMBL4082710)
Affinity DataIC50: 3.36E+3nMAssay Description:Inhibition of recombinant human DYRK1A expressed in insect cells using RRRFRPASPLRGPPK peptide as substrate after 40 mins in presence of [gamma-33P]-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238878BDBM50238878(CHEMBL4078073)
Affinity DataIC50: 4.99E+3nMAssay Description:Inhibition of recombinant human CLK1 expressed in insect cells using ERMRPRKRQGSVRRRV peptide as substrate after 40 mins in presence of [gamma-33P]-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 5.59E+3nMAssay Description:Inhibition of human CLK3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human JAK2 expressed in insect cells using Poly(Glu:Tyr) as substrate in presence of [gamma-32]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Human)
Sichuan University and Collaborative Innovation Center For Biotherapy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50238867BDBM50238867(CHEMBL4083249)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DYRK3More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
Displayed 1 to 50 (of 73 total ) | Next | Last >>
Jump to: