Compile Data Set for Download or QSAR
Report error Found 206 Enz. Inhib. hit(s) with all data for entry = 9291
TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455983BDBM455983(4-(3- (cyclopropylethynyl)-2- (1-(hydroxyamino)-1-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455984BDBM455984(4-(3- (cyclopropylethynyl)-2- (1-(hydroxyamino)-1-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455981BDBM455981(4-(3-(cyclopropylethynyl)-2- (1-(hydroxyamino)-1-o...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456045BDBM456045(US10723705, No. I-0202)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455982BDBM455982(4-(3-(cyclopropylethynyl)-2- (1-(hydroxyamino)-1-o...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455979BDBM455979(2-(7-chloro-3- (cyclopropylethynyl)- 2H-indazol-2-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455980BDBM455980(2-(3-(cyclopropylethynyl)-7- (1-methyl-1H-pyrazol-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456041BDBM456041(N-hydroxy-3-phenyl- 2-(7-(pyrimidin-5- yl)-2H- pyr...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455849BDBM455849(US10723705, No. I-0005)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456042BDBM456042(N-hydroxy-2-(7-(1- methyl-1H-pyrazol- 5-yl)-2H- py...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456040BDBM456040(US10723705, No. I-0197)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455971BDBM455971(US10723705, No. I-0128)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455970BDBM455970(US10723705, No. I-0127)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455999BDBM455999(2-(3-(cyclopropylethynyl)-7- (pyrimidin-5-yl)-2H-i...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456000BDBM456000(3-(3-(cyclopropylethynyl)-2- (1-(hydroxyamino)-1-o...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455872BDBM455872(2-(3-(cyclopropylethynyl)-5- (1-methyl-1H-pyrazol-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455997BDBM455997(2-(3-(cyclopropylethynyl)-7- (pyridin-4-yl)-2H-ind...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455998BDBM455998(2-(3-(cyclopropylethynyl)-7- (pyridin-3-yl)-2H-ind...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455870BDBM455870(4-(3-(cyclopropylethynyl)-2- (1-(hydroxyamino)-1-o...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455985BDBM455985(4-(3- (cyclopropylethynyl)-2- (1-(hydroxyamino)-1-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456049BDBM456049(2-(3- (cyclopropylethynyl)- 4,5,6,7-tetrahydro- 2H...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456050BDBM456050(2-(3- (cyclopropylethynyl)-7- (pyrimidin-5-yl)-2H-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456009BDBM456009(2-(3-(cyclopropylethynyl)-7- (3-methyl-1H-pyrazol-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456008BDBM456008(2-(3-(cyclopropylethynyl)-7- (1-(2-methoxyethyl)-3...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456003BDBM456003(2-(7-cyclopropyl-3- (cyclopropylethynyl)-2H- indaz...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455875BDBM455875(2-(3-(cyclopropylethynyl)-5- (2-methoxypyrimidin-5...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456004BDBM456004(2-(3-(cyclopropylethynyl)-7- methyl-2H-indazol-2-y...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455876BDBM455876(2-(3-(cyclopropylethynyl)-5- methyl-2H-indazol-2-y...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456001BDBM456001(3-(3-(cyclopropylethynyl)-2- (1-(hydroxyamino)-1-o...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455937BDBM455937(US10723705, No. I-0093)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456002BDBM456002(3-(3-(cyclopropylethynyl)-2- (1-(hydroxyamino)-1-o...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455874BDBM455874(2-(3-(cyclopropylethynyl)-5- (pyrimidin-5-yl)-2H-i...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456021BDBM456021(2-(1-(hydroxyamino)-1-oxo- 3-phenylpropan-2-yl)-N-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456020BDBM456020(2-(1-(hydroxyamino)-1-oxo- 3-phenylpropan-2-yl)-N-...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455953BDBM455953(4-(2-(1- (hydroxyamino)-1- oxo-3-phenylpropan- 2-y...)
Affinity DataIC50: 50nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456047BDBM456047(US10723705, No. I-0204)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455855BDBM455855(US10723705, No. I-0011)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456048BDBM456048(N-hydroxy-2-(1-methyl-6-(pyridin-4- yl)-1H-indazol...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455856BDBM455856(N-hydroxy-3- phenyl-2-(5- (pyrimidin-5-yl)-1H- i...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455920BDBM455920(2-(5-chloro-1H- pyrazolo[4,3-b]pyridin-1-yl)- N-hy...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455853BDBM455853(2-(5-chloro-3- (cyclopropylethynyl)- 1H-indazol-1-...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456046BDBM456046(N-hydroxy-2-(1-methyl-6-(1-methyl- 1H-pyrazol-5-yl...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455854BDBM455854(N-hydroxy-2-(5-(1- methyl-1H-pyrazol- 5-yl)-1H-ind...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455918BDBM455918(N-hydroxy-3- phenyl-2-(5- (pyrimidin-5-yl)-1H- pyr...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455915BDBM455915(N-hydroxy-3- phenyl-2-(4- (pyrimidin-5-yl)- 1H-pyr...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455913BDBM455913(N-hydroxy-2-(4-(1- methyl-1H-pyrazol- 5-yl)-1H- py...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455914BDBM455914(N-hydroxy-3- phenyl-2-(4- (pyridin-4-yl)-1H- pyraz...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455911BDBM455911(N-hydroxy-2-(7-(1- methyl-1H-pyrazol- 5-yl)-2H-ind...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 455845BDBM455845(US10723705, No. I-0001)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

TargetHistone deacetylase 8(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 456035BDBM456035(N-hydroxy-2-(7-((4-methyl-3- oxopiperazin-1-yl)met...)
Affinity DataIC50: 125nMAssay Description:HDAC-Glo I/II Assay Kit was purchased from Promega Corporation (Madison, Wis.), including the following components: HDAC-Glo I/II Buffer (25 mM Tris ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2021
Entry Details
US Patent

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