Compile Data Set for Download or QSAR
Report error Found 1927 Enz. Inhib. hit(s) with Target = 'Neuropeptide Y receptor type 5'
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417035(CHEMBL1257993)
Affinity DataKi:  0.0251nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417033(CHEMBL1258111)
Affinity DataKi:  0.0316nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417056(CHEMBL1258225)
Affinity DataKi:  0.0398nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417045(CHEMBL1258341)
Affinity DataKi:  0.0631nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417051(CHEMBL1258787)
Affinity DataKi:  0.0631nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417036(CHEMBL1257992)
Affinity DataKi:  0.0631nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417032(CHEMBL1258110)
Affinity DataKi:  0.0794nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417046(CHEMBL1258453)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417044(CHEMBL1258340)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417050(CHEMBL1258674)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417042(CHEMBL1257636)
Affinity DataKi:  0.100nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417041(CHEMBL1257637)
Affinity DataKi:  0.126nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141347(US8916594, I-024)
Affinity DataIC50: 0.130nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417390(CHEMBL1289154)
Affinity DataKi:  0.158nMAssay Description:Antagonistic activity at human NPY Y5 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417054(CHEMBL1258673)
Affinity DataKi:  0.158nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417039(CHEMBL1257761)
Affinity DataKi:  0.158nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417040(CHEMBL1257760)
Affinity DataKi:  0.158nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50390216(CHEMBL2070151)
Affinity DataIC50: 0.160nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50390219(CHEMBL2070148)
Affinity DataIC50: 0.160nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141350(US8916594, I-034)
Affinity DataIC50: 0.180nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50390213(CHEMBL2069316)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50258001(N-(3,4-dichlorophenyl)-1-(methylsulfonyl)spiro[ind...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I]PYY from human recombinant Y5 receptor expressed in mouse LMtk cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417047(CHEMBL1258454)
Affinity DataKi:  0.200nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141345(US8916594, I-018)
Affinity DataIC50: 0.200nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417048(CHEMBL1258562)
Affinity DataKi:  0.200nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417407(CHEMBL1289153)
Affinity DataKi:  0.200nMAssay Description:Antagonistic activity at human NPY Y5 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50093652(2-Methyl-6-pentyl-4-piperidin-1-yl-5H-pyrrolo[3,2-...)
Affinity DataIC50: 0.200nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]PYY binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Chicken)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM82276(NPY [Leu31, Pro34], human | NPY,[leu31,Pro34], por...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50394224(CHEMBL2159167)
Affinity DataIC50: 0.210nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141349(US8916594, I-029)
Affinity DataIC50: 0.220nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141344(US8916594, I-017)
Affinity DataIC50: 0.220nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM141351(US8916594, I-053)
Affinity DataIC50: 0.230nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding a mouse NPY Y5 receptor (Biochim. Biophys. Acta 1328:83-89, 1997) was cloned in a vector (pME18S, Takebe et al. Mol. Cell. Bio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2015
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50111656(FR-236478 | 1-[2-(5-Chloro-2-oxo-benzothiazol-3-yl...)
Affinity DataIC50: 0.230nMAssay Description:Tested for the inhibition of [125I]PYY binding to HEK 293 cells stably expressed with human neuropeptide NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Chicken)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM50089038(CGP 71683 | CHEMBL17645 | Naphthalene-1-sulfonic a...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM85680(PP [cPP(1-7), NPY(19-23), Ala31, Aib32, Gln34], hu...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417055(CHEMBL1258788)
Affinity DataKi:  0.251nMAssay Description:Antagonist activity at human NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM118179(US8653125, Ia-40)
Affinity DataIC50: 0.260nMpH: 7.4 T: 2°CAssay Description:cDNA sequence encoding mouse NPY Y5 receptor (Biochem. Biophys. Acta 1328: 83-89, 1997) was cloned in the expression vector (pME18S, Takebe et al. Mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2014
Entry Details
US Patent

TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50394211(CHEMBL2159165)
Affinity DataIC50: 0.280nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Chicken)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM50005530(Tyr-Pro-Ser-Lys-Pro-Asp-Asn-pro-Gly-Glu-Asp-Ala-Pr...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50394221(CHEMBL2159158)
Affinity DataIC50: 0.290nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50390228(CHEMBL2070161)
Affinity DataIC50: 0.290nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50379608(CHEMBL2013020)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]peptide YY from human NPY5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50093664(6-(4-Fluoro-phenyl)-2-methyl-4-piperidin-1-yl-5H-p...)
Affinity DataIC50: 0.300nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]PYY binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50093646(6-Benzofuran-2-yl-2-methyl-4-piperidin-1-yl-5H-pyr...)
Affinity DataIC50: 0.300nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]PYY binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50353148(CHEMBL1829320)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]peptide YY from human NPY5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50093696(6-(3-Fluoro-phenyl)-2-methyl-4-piperidin-1-yl-5H-p...)
Affinity DataIC50: 0.300nMAssay Description:Affinity for human neuropeptide Y receptor Y5, binding was evaluated in an in vitro radioligand [125I]PYY binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50128931(N-(9-Isobutyl-9H-carbazol-3-yl)-3-pyrrolidin-1-yl-...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity towards human neuropeptide Y receptor type 5 using 125[I]-PYY as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Chicken)
Uppsala University

Curated by PDSP Ki Database
LigandPNGBDBM84998(NPY 3-36, porcine)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2012
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Mouse)
Shionogi

US Patent
LigandPNGBDBM50390232(CHEMBL2070157)
Affinity DataIC50: 0.310nMAssay Description:Displacement of [125I]PYY from mouse NPY Y5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417405(CHEMBL1289267)
Affinity DataKi:  0.316nMAssay Description:Antagonistic activity at human NPY Y5 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
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