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Found 120 with Last Name = 'blommaert' and Initial = 'ag'
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045797(2-[3-(4-Chloro-phenyl)-ureido]-3-(1H-indol-3-yl)-2...)
Affinity DataKi: >0.000100nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.280nMAssay Description:Inhibition of [3H]pCCK-8 binding to Cholecystokinin type A receptor of Guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.600nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.640nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056453(3-(2-{[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  6.10nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  6.5nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  12nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  14nMAssay Description:Tested for binding affinity towards cholecystokinin type A receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  14nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in mouse brain by displacement of [3H]-pBC264 radioligand (icv)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  14nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056449(CHEMBL2371222 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataKi:  18nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056449(CHEMBL2371222 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  18nMAssay Description:Tested for binding affinity towards CCK-B in rat cortex by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50024317(3-{2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-4-...)
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  21nMAssay Description:Tested for binding affinity towards CCK-B in mouse brain by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045796(CHEMBL99939 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  21nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in rat cortex by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056448(CHEMBL2371221 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataKi:  23nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045798(CHEMBL319120 | [1-[2-(2,4-Dichloro-phenyl)-ethylca...)
Affinity DataKi:  27nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045805(CHEMBL318852 | N-Carboxymethyl-N-[2-(2,4-dichloro-...)
Affinity DataKi:  28nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in rat pancreas by displacement of [3H]-pCCK-8 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045810(3-{[2-(Adamantan-2-yloxycarbonylamino)-3-(1H-indol...)
Affinity DataKi:  36nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045816(CHEMBL319880 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  37nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045803(CHEMBL433407 | [1-[2-(4-Chloro-phenyl)-ethylcarbam...)
Affinity DataKi:  39nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056454(CHEMBL2371224 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  40nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in rat cortex by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005459(4-(3,4-Dichloro-benzoylamino)-4-dipentylcarbamoyl-...)
Affinity DataKi:  49nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045806(CHEMBL320399 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  50nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045808(CHEMBL432389 | [1-[2-(4-Bromo-phenyl)-ethylcarbamo...)
Affinity DataKi:  51nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056455(CHEMBL348344 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[...)
Affinity DataKi:  51nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045802(CHEMBL99252 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  70nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(MOUSE)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045800(CHEMBL317999 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  73nMAssay Description:Tested for binding affinity towards cholecystokinin type B receptor in mouse brain by displacement of [3H]-pBC264 radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045813(CHEMBL328852 | {2-(1H-Indol-3-yl)-1-methyl-1-[2-(4...)
Affinity DataKi:  79nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056455(CHEMBL348344 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[...)
Affinity DataKi:  80nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045817(CHEMBL319085 | {[2-(Adamantan-2-yloxycarbonylamino...)
Affinity DataKi:  87nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50005823(CHEMBL291033 | [2-(1H-Indol-3-yl)-1-methyl-1-phene...)
Affinity DataKi:  87nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056453(3-(2-{[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl...)
Affinity DataKi:  87nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045818(CHEMBL95115 | [2-(1H-Indol-3-yl)-1-methyl-1-(2-nap...)
Affinity DataKi:  89nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005456(1-(4-Chloro-phenyl)-3-(3,3-diphenyl-allyl)-urea | ...)
Affinity DataKi:  90nMAssay Description:Inhibition of [3H]-L-364,718 binding to cholecystokinin type A receptor in rat pancreas membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50024317(3-{2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-4-...)
Affinity DataKi:  93nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045804(CHEMBL329088 | {2-(1H-Indol-3-yl)-1-[2-(4-methoxy-...)
Affinity DataKi:  115nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045815(CHEMBL98516 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  134nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056452(CHEMBL2371225 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataKi:  142nMAssay Description:Inhibition of [3H]pCCK-8 binding to Guinea pig cortex membrane Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50056452(CHEMBL2371225 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataKi:  142nMAssay Description:Affinity to inhibit [3H]pCCK-8 specific binding on rat brain Cholecystokinin type B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005471(1H-Indole-2-carboxylic acid (3-phenyl-allyl)-amide...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045814(CHEMBL95793 | [2-(1H-Indol-3-yl)-1-methyl-1-(3-phe...)
Affinity DataKi:  182nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045809(CHEMBL316462 | [1-[2-(3,4-Dichloro-phenyl)-ethylca...)
Affinity DataKi:  184nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005450(1-(4-Chloro-phenyl)-3-(3-pentyl-oct-2-enyl)-urea |...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50005453(1H-Indole-2-carboxylic acid [3,3-bis-(4-chloro-phe...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-L-364,718 from Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50045801(CHEMBL95461 | {[2-(Adamantan-2-yloxycarbonylamino)...)
Affinity DataKi:  224nMAssay Description:Tested for inhibition of [3H]-pCCK-8 specific binding to cholecystokinin type B receptor in guinea pig brain cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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