TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 2.20nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 2.70nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
Affinity DataIC50: 13nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
Affinity DataIC50: 22nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Affinity DataIC50: 58nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 60nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 70nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 80nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 100nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 100nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 190nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
Affinity DataIC50: 280nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Affinity DataIC50: 400nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 490nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 560nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 730nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 790nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 1.00E+3nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 1.40E+3nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargetPhenylalanine--tRNA ligase alpha/beta subunit(Escherichia coli (Enterobacteria))
Astrazeneca R&D Boston
Astrazeneca R&D Boston
Affinity DataIC50: 1.40E+3nMpH: 8.0Assay Description:Compounds were solubilized in DMSO. Serial 2-fold dilutions covering two concentration ranges, 10 mM to 19.5 μM and 100 μM to 195 nM, were ...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22...)
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Singapore-Mit Alliance For Research And Technology
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair