Found 505 with Last Name = 'gan' and Initial = 'y' TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 0.420nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nM ΔG°: -54.4kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 0.75nM ΔG°: -54.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 0.850nM ΔG°: -53.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 0.880nM ΔG°: -53.8kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 0.950nM ΔG°: -53.6kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nM ΔG°: -53.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nM ΔG°: -53.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nM ΔG°: -50.9kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nM ΔG°: -52.8kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nM ΔG°: -50.7kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nM ΔG°: -50.7kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nM ΔG°: -50.5kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nM ΔG°: -50.2kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nM ΔG°: -52.2kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nM ΔG°: -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nM ΔG°: -51.8kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nM ΔG°: -49.8kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nM ΔG°: -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nM ΔG°: -51.1kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nM ΔG°: -50.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nM ΔG°: -50.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 3.30nM ΔG°: -48.4kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 3.40nM ΔG°: -48.3kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nM ΔG°: -50.1kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 3.70nM ΔG°: -48.1kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 3.70nM ΔG°: -50.1kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 3.90nM ΔG°: -49.9kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of phosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nM ΔG°: -47.9kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 4.20nM ΔG°: -49.7kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 4.30nM ΔG°: -49.7kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nM ΔG°: -47.6kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nM ΔG°: -47.5kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nM ΔG°: -47.2kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nM ΔG°: -46.8kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
Affinity DataKi: 6.60nM ΔG°: -48.6kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 6.90nM ΔG°: -48.5kJ/molepH: 7.4 T: 2°CAssay Description:A test compound and 150 uM of a DMSO solution of 5-carboxamide tryptamine (5-CT) were added to a 96-well plate at 2 ul/well and suspended in the incu...More data for this Ligand-Target Pair
Affinity DataKi: 7.10nM ΔG°: -46.5kJ/molepH: 7.5 T: 2°CAssay Description:A solution of the compound to be tested and 100 μM 5-CT (5-carboxamidetriptamine) in DMSO was added to a 96-well plate at 2 μl/well, suspen...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
The Reproductive Medicine Special Hospital of The First Hospital of Lanzhou University
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in Wistar rat brain membranes preincubated for 1 hr measured after 1hr by scintillation counting m...More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of unphosphorylated-Kdr after 30 minsMore data for this Ligand-Target Pair
