TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Enzyme inhibitory activity towards Angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 189nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 254nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 333nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 406nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 435nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 2.42E+3nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 3.63E+3nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 4.62E+3nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Antagonistic activity towards Opioid receptor mu 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibitory activity for kappa opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Antagonist activity against mu opioid receptor in guinea-pig ileum assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibitory activity towards Sigma opioid receptor type 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibitory activity towards Sigma opioid receptor type 1More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 78nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain homogenateMore data for this Ligand-Target Pair