Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 10891
TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576437BDBM576437(WO2022115301, Example 23)
Affinity DataEC50:  0.410nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576435BDBM576435(WO2022115301, Example 21)
Affinity DataEC50:  0.910nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576438BDBM576438(WO2022115301, Example 24)
Affinity DataEC50:  0.930nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576417BDBM576417(WO2022115301, Example 3 | (R)-2-(1-Cyclopropyl-2-h...)
Affinity DataEC50:  2nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576416BDBM576416(WO2022115301, Example 2 | (R or S)-2-(1-Cyclopropy...)
Affinity DataEC50:  2.60nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576424BDBM576424(WO2022115301, Example 10)
Affinity DataEC50:  2.80nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576421BDBM576421(WO2022115301, Example 7)
Affinity DataEC50:  3.60nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576420BDBM576420(WO2022115301, Example 6)
Affinity DataEC50:  4.5nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576425BDBM576425(WO2022115301, Example 11)
Affinity DataEC50:  4.90nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576429BDBM576429(WO2022115301, Example 15)
Affinity DataEC50:  6.40nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576436BDBM576436(WO2022115301, Example 22)
Affinity DataEC50:  6.90nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576422BDBM576422(WO2022115301, Example 8)
Affinity DataEC50:  7.5nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576415BDBM576415(WO2022115301, Example 1 | (R)-2-(1-Cyclopropyl-2-h...)
Affinity DataEC50:  7.90nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576439BDBM576439(WO2022115301, Example 25)
Affinity DataEC50:  9.20nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576426BDBM576426(WO2022115301, Example 12)
Affinity DataEC50:  13nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576423BDBM576423(WO2022115301, Example 9)
Affinity DataEC50:  24nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576433BDBM576433(WO2022115301, Example 19)
Affinity DataEC50:  28nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576430BDBM576430(WO2022115301, Example 16)
Affinity DataEC50:  39nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576432BDBM576432(WO2022115301, Example 18)
Affinity DataEC50:  45nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576428BDBM576428(WO2022115301, Example 14)
Affinity DataEC50:  48nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576419BDBM576419(WO2022115301, Example 5)
Affinity DataEC50:  52nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576434BDBM576434(WO2022115301, Example 20)
Affinity DataEC50:  67nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576427BDBM576427(WO2022115301, Example 13)
Affinity DataEC50:  260nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576418BDBM576418(WO2022115301, Example 4 | (R and S)- (E)-2-(1-cycl...)
Affinity DataEC50:  290nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301

TargetCeramide glucosyltransferase(Human)
Merck Sharp &Amp

WIPO
LigandChemical structure of BindingDB Monomer ID 576431BDBM576431(WO2022115301, Example 17)
Affinity DataEC50:  580nMAssay Description: Using Promega s UDP-Glo Glycosyltransferase assay kit (Promega Corporation, Madison, WI, USA (Promega)), GCS activity was indirectly measured by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2022
Entry Details
WIPO WO2022115301