Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50016153
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165669(2-(2-(4-(3-(3-bromophenylamino)-3-oxoprop-1-enyl)-...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165653(2-(2-(4-(3-(3,4-dichlorophenylamino)-3-oxoprop-1-e...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165660(2-(3-(5-(4-chlorophenyl)benzo[d]oxazol-2-yl)-4-(pr...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165639(2-(2-(4-(3-(2,4-dichlorophenylamino)-3-oxoprop-1-e...)
Affinity DataIC50: 200nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165627(2-(2-(4-(3-(3-fluoro-4-methoxyphenylamino)-3-oxopr...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165640(2-(4-(5-(2-chloro-4-(3-(2,4-dichlorophenyl)acrylam...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165614((2-{4-[3-((E)-3-Chloro-2-fluoro-phenyl)-acryloylam...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165638(2-(2-(4-(3-(4-cyanophenylamino)-3-oxoprop-1-enyl)-...)
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165621((2-{2-Chloro-4-[3-((E)-2,4-dichloro-phenyl)-acrylo...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165624((2-{4-[3-((E)-2,4-Dichloro-phenyl)-acryloylamino]-...)
Affinity DataIC50: 350nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165615((2-{4-[2-(2,4-Dichloro-phenylcarbamoyl)-vinyl]-phe...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165652(2-(2-(4-(3-(4-bromophenyl)acrylamido)-3-fluorophen...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165613(2-(2-(4-(3-(4-bromophenyl)acrylamido)-2-chlorophen...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165663(2-(2-(4-(3-(4-bromophenylamino)-3-oxoprop-1-enyl)-...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165636(2-(4-(5-(4-(3-(4-bromophenyl)acrylamido)-2-chlorop...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165620(2-(4-(5-(2-chloro-4-(3-(4-methoxyphenyl)acrylamido...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165643((2-{2-Fluoro-4-[2-(2-fluoro-4-methoxy-phenylcarbam...)
Affinity DataIC50: 450nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165642((4-{5-[2-Chloro-4-(3-phenyl-acryloylamino)-phenyl]...)
Affinity DataIC50: 450nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165659((2-{4-[2-(3-Bromo-phenylcarbamoyl)-vinyl]-phenyl}-...)
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165657([4-(5-{2-Chloro-4-[3-(4-trifluoromethoxy-phenyl)-a...)
Affinity DataIC50: 600nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165612(2-(2-(4-(3-(4-bromophenyl)acrylamido)phenyl)benzo[...)
Affinity DataIC50: 600nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165634((2-{4-[2-(4-Bromo-phenylcarbamoyl)-vinyl]-phenyl}-...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165623((2-{4-[3-((E)-3-Chloro-phenyl)-acryloylamino]-3-fl...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165607((2-{4-[3-((E)-3-Bromo-phenyl)-acryloylamino]-2-chl...)
Affinity DataIC50: 750nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165629((2-{4-[2-(2,4-Difluoro-phenylcarbamoyl)-vinyl]-2-f...)
Affinity DataIC50: 750nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165662(2-(2-(4-(3-(3-chloro-4-fluorophenyl)acrylamido)-3-...)
Affinity DataIC50: 750nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165619(2-(2-(4-(3-(3-bromophenyl)acrylamido)phenyl)benzo[...)
Affinity DataIC50: 750nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165665((2-{4-[3-((E)-4-Cyano-phenyl)-acryloylamino]-3-flu...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165633(2-(2-(4-(3-(3-bromophenyl)acrylamido)-3-fluorophen...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165667((2-{4-[3-((E)-3,4-Dichloro-phenyl)-acryloylamino]-...)
Affinity DataIC50: 800nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165641((4-{5-[2-Chloro-4-(3,4-dichloro-benzoylamino)-phen...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165668((2-{4-[2-(4-Difluoromethoxy-phenylcarbamoyl)-vinyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165635(2-(4-(5-(2-chloro-4-(4-(trifluoromethoxy)benzamido...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165626((2-{3-Fluoro-4-[3-((E)-4-trifluoromethyl-phenyl)-a...)
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165664((2-{4-[3-((E)-3-Methoxy-phenyl)-acryloylamino]-phe...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165649(2-(2-(4-(3-(2-chlorophenyl)acrylamido)-3-fluorophe...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165646(2-(2-(2-chloro-4-(3-(3-methoxyphenyl)acrylamido)ph...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165632((2-{4-[3-((E)-4-Chloro-phenyl)-acryloylamino]-3-fl...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165609((4-{5-[2-Chloro-4-(4-chloro-benzoylamino)-phenyl]-...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165616(2-(2-(4-(3-(4-fluorophenylamino)-3-oxoprop-1-enyl)...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165617(2-(2-(4-(3-(4-fluorophenyl)acrylamido)phenyl)benzo...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165637((2-{3-Fluoro-4-[3-((E)-4-methoxy-phenyl)-acryloyla...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165647(2-(2-(3-fluoro-4-(3-(4-fluorophenyl)acrylamido)phe...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165648((2-{4-[2-(3-Chloro-4-methoxy-phenylcarbamoyl)-viny...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165644(2-(2-(4-(3-(4-methoxyphenylamino)-3-oxoprop-1-enyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165645(2-(2-(4-cinnamamidophenyl)benzo[d]oxazol-5-yl)acet...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165666(2-(2-(4-(3-(2-chlorophenylamino)-3-oxoprop-1-enyl)...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165656((2-{4-[2-(3-Methoxy-phenylcarbamoyl)-vinyl]-phenyl...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165650((2-{4-[2-(4-Bromo-phenyl)-acetylamino]-2-chloro-ph...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHeparanase(Human)
Celltech R&D

Curated by ChEMBL
LigandPNGBDBM50165661((2-{4-[3-((E)-4-Methoxy-phenyl)-acryloylamino]-phe...)
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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