Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50021061
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50007517(CHEMBL76402 | 3-Bromo-N-(1-ethyl-pyrrolidin-2-ylme...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220542(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2,3-...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220543(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2,3...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50007517(CHEMBL76402 | 3-Bromo-N-(1-ethyl-pyrrolidin-2-ylme...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220542(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2,3-...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220542(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2,3-...)
Affinity DataKi:  0.740nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220543(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2,3...)
Affinity DataKi:  0.850nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220543(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2,3...)
Affinity DataKi:  0.880nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220541(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50007517(CHEMBL76402 | 3-Bromo-N-(1-ethyl-pyrrolidin-2-ylme...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220541(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220541(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50012961(N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-3-iodo...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50012961(N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-3-iodo...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50012961(N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-3-iodo...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220546(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2-me...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220546(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2-me...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220546(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2-me...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220545(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2-m...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220545(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2-m...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220545(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2-m...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220544(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220544(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220544(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50012961(N-(1-Ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-3-iodo...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220546(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2-me...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220543(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2,3...)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50007517(CHEMBL76402 | 3-Bromo-N-(1-ethyl-pyrrolidin-2-ylme...)
Affinity DataKi:  1.50E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220545(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-bromo-2-m...)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220541(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220542(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-iodo-2,3-...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50220544(N-(((S)-1-allylpyrrolidin-2-yl)methyl)-5-(3-fluoro...)
Affinity DataKi:  3.00E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Pig)
Johannes Gutenberg University

Curated by ChEMBL
LigandPNGBDBM50005118(3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-h...)
Affinity DataKi:  3.70E+4nMAssay Description:Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed