Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50008869
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523020BDBM50523020(CHEMBL4466171)
Affinity DataEC50:  5nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataEC50:  6nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523029BDBM50523029(CHEMBL4450117)
Affinity DataEC50:  7nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523013BDBM50523013(CHEMBL4458134)
Affinity DataEC50:  25nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523025BDBM50523025(CHEMBL4525262)
Affinity DataEC50:  27nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523024BDBM50523024(CHEMBL4515029)
Affinity DataEC50:  27nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523021BDBM50523021(CHEMBL4441437)
Affinity DataEC50:  29nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523028BDBM50523028(CHEMBL4456673)
Affinity DataEC50:  31nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523016BDBM50523016(CHEMBL4441091)
Affinity DataEC50:  44nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523019BDBM50523019(CHEMBL4440715)
Affinity DataEC50:  64nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523012BDBM50523012(CHEMBL4476507)
Affinity DataEC50:  69nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523023BDBM50523023(CHEMBL4454946)
Affinity DataEC50:  86nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50508029BDBM50508029(CHEMBL4467856)
Affinity DataEC50:  89nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523015BDBM50523015(CHEMBL4465577)
Affinity DataEC50:  261nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523027BDBM50523027(CHEMBL4466588)
Affinity DataEC50:  301nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523018BDBM50523018(CHEMBL4577659)
Affinity DataEC50:  426nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523017BDBM50523017(CHEMBL4583270)
Affinity DataEC50:  430nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523022BDBM50523022(CHEMBL4549349)
Affinity DataEC50:  720nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523026BDBM50523026(CHEMBL4442686)
Affinity DataEC50:  2.46E+3nMAssay Description:Agonist activity at recombinant human GPR119 expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Japan Tobacco

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50523014BDBM50523014(CHEMBL4548931)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed