Compile Data Set for Download or QSAR
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Found 28 Enz. Inhib. hit(s) with all data for entry = 50034758
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50005229(2-{[Acetyl-(5-octadecyloxy-tetrahydro-furan-3-ylme...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM81972((S)-(+)-ALPHA-METHYL-1H-IMIDAZOLE-4-ETHANAMINE DIH...)
Affinity DataIC50:  13nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50041921(5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282029((cis)-3-{3-[5-(3,4,5-Trimethoxy-phenyl)-tetrahydro...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282027(3-{3-[(2S,5R)-5-(3,4-Dimethoxy-phenyl)-tetrahydro-...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282024((cis)-3-{3-[5-(3,4-Dichloro-phenyl)-tetrahydro-fur...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282020((cis)-3-{3-[5-(4-Fluoro-phenyl)-tetrahydro-furan-2...)
Affinity DataIC50:  230nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282007(3-{3-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282014(3-{(E)-3-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-fura...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282028((cis)-3-{3-[5-(4-Bromo-phenyl)-tetrahydro-furan-2-...)
Affinity DataIC50:  800nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282015((cis)-3-{3-[5-(4-Chloro-phenyl)-tetrahydro-furan-2...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282031(3-{3-[(2S,5R)-5-(3,4-Dimethoxy-phenyl)-tetrahydro-...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282010((trans)-3-{3-[5-(3,4,5-Trimethoxy-phenyl)-tetrahyd...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282021(1-[6-(5-Hexyl-tetrahydro-furan-2-yloxy)-hexyl]-pyr...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282019((cis)-3-{3-[5-(4-Methoxy-phenyl)-tetrahydro-furan-...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282018((trans)-3-{3-[5-(3,4-Dichloro-phenyl)-tetrahydro-f...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282023(3-{3-[(2S,5S)-5-(3,4-Dimethoxy-phenyl)-tetrahydro-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282009(3-{5-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282017((trans)-3-{3-[5-(4-Fluoro-phenyl)-tetrahydro-furan...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282026(3-{3-[(2S,5S)-5-(3,4-Dimethoxy-phenyl)-tetrahydro-...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282025((trans)-3-{3-[5-(4-Bromo-phenyl)-tetrahydro-furan-...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282022((trans)-3-{3-[5-(4-Methoxy-phenyl)-tetrahydro-fura...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282013((trans)-3-{3-[5-(4-Chloro-phenyl)-tetrahydro-furan...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282030((trans)-3-[3-(5-Phenyl-tetrahydro-furan-2-yloxy)-p...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282012(3-{4-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282008(3-{2-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-...)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282011(3-{3-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-...)
Affinity DataIC50:  1.80E+4nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282016(3-[5-(3,4-Dimethoxy-phenyl)-tetrahydro-furan-2-ylo...)
Affinity DataIC50:  2.50E+4nMAssay Description:In vitro inhibition of [3H]PAF receptor binding to washed human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article