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Found 44 for UniProtKB: P28471
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM26267(RO-154513 | Ro15-4513 | [3H]Ro15-4513 | ethyl 12-a...)
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50044941(8-Azido-5-methyl-6-oxo-5,6-dihydro-4H-2,5,10b-tria...)
Affinity DataKi:  5.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50034835(5-Methyl-6-oxo-5,6-dihydro-4H-7-thia-2,5,9b-triaza...)
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM84956(2-(4-Methoxy-phenyl)-2,5-dihydro-pyrazolo[4,3-c]qu...)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50017009(2-Phenyl-2,3a-dihydro-pyrazolo[4,3-c]quinolin-3-on...)
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50034816(8-Chloro-5-methyl-6-oxo-5,6-dihydro-4H-2,5,10b-tri...)
Affinity DataKi:  9.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50049739(8-Ethyl-5-methyl-6-oxo-5,6-dihydro-4H-2,5,10b-tria...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85038(CHEMBL43948 | PZII-029)
Affinity DataKi:  11.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85042(CHEMBL44613 | PW-007A)
Affinity DataKi:  22.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM81951(CAS_104999 | DMCM | NSC_104999)
Affinity DataKi:  38.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM26263(Anexate | CHEMBL407 | FLUMAZENIL | Ro15-1788 | Rom...)
Affinity DataKi:  118nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85041(DM 236 | DM-236)
Affinity DataKi:  188nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM84957(CGS 9896 | CHEMBL20042)
Affinity DataKi:  214nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50243981(Beta CCM | CHEMBL453066 | Methyl Beta-carboline-3 ...)
Affinity DataKi:  436nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85040(CAS_123700 | NSC_123700 | ZK 91296)
Affinity DataKi:  573nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50244036(Beta-CCT | CHEMBL509197 | tert-butyl 9H-pyrido[3,4...)
Affinity DataKi:  897nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50045050(1-(3-Hydroxy-10,13-dimethyl-hexadecahydro-cyclopen...)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85683(Co 2-6749 | Co-2-6749 | GMA-839 | WAY-141839)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM85039(CAS_121926 | NSC_121926 | ZK 93423)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235902(US9365502, MQ-87)
Affinity DataIC50:  14nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235905(US9365502, MQ-85)
Affinity DataIC50:  29nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235901(US9365502, MQ-86)
Affinity DataIC50:  43nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235900(US9365502, MQ-37)
Affinity DataIC50:  46nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235898(US9365502, MQ-38)
Affinity DataIC50:  52nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235894(US9365502, MQ-31)
Affinity DataIC50:  61nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235897(US9365502, MQ-33)
Affinity DataIC50:  62nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235907(US9365502, MQ-39)
Affinity DataIC50:  65nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235896(US9365502, MQ-32)
Affinity DataIC50:  147nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235904(US9365502, MQ-48)
Affinity DataIC50:  282nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3/delta(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataIC50:  510nMAssay Description:Displacement of [3H]EBOB from rat GABA-A receptor alpha4beta3delta expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235899(US9365502, MQ-83)
Affinity DataIC50:  748nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235910(US9365502, MQ-50)
Affinity DataIC50:  1.06E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235903(US9365502, MQ-47)
Affinity DataIC50:  1.33E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235906(US9365502, MQ-49)
Affinity DataIC50:  1.58E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235895(US9365502, MQ-36)
Affinity DataIC50:  1.73E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataIC50:  1.86E+3nMAssay Description:Displacement of [3H]EBOB from rat GABA-A receptor alpha4beta3 expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235911(US9365502, MQ-54)
Affinity DataIC50:  1.99E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3/gamma-2(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataIC50:  3.29E+3nMAssay Description:Displacement of [3H]EBOB from rat GABA-A receptor alpha4beta3gamma2 expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235908(US9365502, MQ-53)
Affinity DataIC50:  3.63E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM235909(US9365502, MQ-51)
Affinity DataIC50:  5.86E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3/delta(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataEC50:  150nMAssay Description:Modulation of rat eGFP-fused GABA-A receptor alpha4beta3delta expressed in HEK293 cells in presence of GABA by patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3/delta(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457445(CHEMBL4212818)
Affinity DataEC50:  970nMAssay Description:Modulation of rat eGFP-fused GABA-A receptor alpha4beta3delta expressed in HEK293 cells in presence of GABA by patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rattus norvegicus (Rat))
National Institute Of Diabetes, Digestive And Kidney Diseases

Curated by PDSP Ki Database
LigandPNGBDBM50273002(5-Aminomethyl-3H-[1,3,4]oxadiazol-2-one Hydrochlor...)
Affinity DataEC50:  1.28E+5nMAssay Description:Agonist activity at rat recombinant GABAAalpha4beta3gamma2 receptor expressed in HEK293 cells assessed as normalization of GABA-induced current by wh...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-4/beta-3(Rattus norvegicus (Rat))
Johannes Gutenberg University Mainz

Curated by ChEMBL
LigandPNGBDBM50457439(CHEMBL4213357)
Affinity DataEC50:  60nMAssay Description:Modulation of rat eGFP-fused GABA-A receptor alpha4beta3 expressed in HEK293 cells in presence of GABA by patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed