TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: <1.20nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 35nMAssay Description:Binding affinity to Bcl-2 (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 153nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 298nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 660nMAssay Description:Binding affinity to Bcl-XL (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 1.79E+3nMAssay Description:Binding affinity to Bak/Mcl-1 (unknown origin) protein protein interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 6.90E+3nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 7.77E+3nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to Bcl-2 (unknown origin) assessed as inhibition constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
TargetBcl-2-like protein 1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to Bcl-xL (unknown origin) assessed as inhibition constant by fluorescence polarisation assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 1.14E+4nMAssay Description:Binding affinity to Mcl-1/Bak protein protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Binding affinity to Bcl-2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Binding affinity to Mcl-1 (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 4.40E+4nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKi: 2.61E+5nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of Mcl-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibition of Mcl-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibition of Mcl-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of Mcl-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 162nMAssay Description:Inhibition of Mcl-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of Mcl-1/Bak (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of Mcl-1/Bak (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 620nMAssay Description:Inhibition of Mcl-1/Bak (unknown origin)More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of Mcl-1 (unknown origin) measured after 5 mins by spectramax M5 microplate reader methodMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of FITC-MCL-1 SAHBa binding to recombinant MCL-1 (172 - 327 residues) (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of Bak/Mcl-1 (unknown origin) protein protein interaction by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibition of Mcl-1/Bak (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of Mcl-1/Bak (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of Mcl-1/Bak (unknown origin)More data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 430nMAssay Description:Binding affinity to wildtype Mcl-1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding affinity to wildtype Mcl-1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding affinity to wildtype Mcl-1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 8.40E+4nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 0.190nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetBcl-2 homologous antagonist/killer(Homo sapiens)
National University Of Ireland Galway
Curated by ChEMBL
National University Of Ireland Galway
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Binding affinity to Mcl-1/Bak (unknown origin) assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair