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Found 28 with Last Name = 'han' and Initial = 'bh'
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18860((2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-di...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor alpha (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18860((2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-di...)
Affinity DataKi:  0.550nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242403((3,5-dimethyl-4-(4-hydroxy-3-isopropylbenzyl)pheno...)
Affinity DataKi:  2.17nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM18869(2-{3,5-dichloro-4-[4-hydroxy-3-(propan-2-yl)phenox...)
Affinity DataKi:  7.18nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor alpha (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242403((3,5-dimethyl-4-(4-hydroxy-3-isopropylbenzyl)pheno...)
Affinity DataKi:  35.2nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor alpha (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242404((4S)-4-(3-chlorophenyl)-2-[(3,5-dimethyl-4-(4-hydr...)
Affinity DataKi:  1.25E+4nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor alpha (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics

Curated by ChEMBL
LigandPNGBDBM50242404((4S)-4-(3-chlorophenyl)-2-[(3,5-dimethyl-4-(4-hydr...)
Affinity DataKi:  1.46E+4nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065348((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065336((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065344(CHEMBL89088 | methyl 5,8a-dimethyl-1-[2-(2-oxo-2,5...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065343((1S,4aR,5S,6S)-6-Hydroxymethyl-1,4a-dimethyl-5-[2-...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065347(3-[2-((1S,5S,8aR)-5-Methoxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065339((1S,4aS)-6-Formyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065352((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065335((1S,4aS,5R,6S)-6-Hydroxy-1,4a-dimethyl-5-[2-(2-oxo...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065342((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-tetrah...)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065333(6-Hydroxymethyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-dihy...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065345((1S,4aR,5S)-1,4a,6-Trimethyl-5-[2-(2-oxo-tetrahydr...)
Affinity DataIC50:  4.80E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065346((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(5-oxo-...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065341((1R,6S,9aS)-6,9a-Dimethyl-3-oxo-1-[2-(5-oxo-2,5-di...)
Affinity DataIC50:  8.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065337((1S,4aR,5S)-5-((Z)-5-Hydroxy-3-hydroxymethyl-pent-...)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065351((Z)-2-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethy...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065350((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065338(3-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065349(4-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065340((1S,4aR,5S)-5-(2-Furan-3-yl-ethyl)-1,4a-dimethyl-6...)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065334((1S,4aS,5R,6R)-6-Hydroxy-6-hydroxymethyl-1,4a-dime...)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed