Compile Data Set for Download or QSAR
maximum 50k data
Found 132 with Last Name = 'cantarella' and Initial = 'g'
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528960(CHEMBL4450250)
Affinity DataKi:  0.0109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528965(CHEMBL4550234)
Affinity DataKi:  0.0109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528966(CHEMBL4521879)
Affinity DataKi:  0.0109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528967(CHEMBL4439415)
Affinity DataKi:  0.0109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269634(CHEMBL4079574)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269634(CHEMBL4079574)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269637(CHEMBL4102093)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50518036(CHEMBL4467777 | US11484525, Compound BD-122LS-PZM2...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of mu opioid receptor (unknown origin) assessed as reduction in intracellular cAMP accumulationMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269634(CHEMBL4079574)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269638(CHEMBL4066846)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269637(CHEMBL4102093)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474153(CHEMBL61630)
Affinity DataKi:  7.20nMAssay Description:Inhibition of mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269638(CHEMBL4066846)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269638(CHEMBL4066846)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269633(CHEMBL4077833)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474152(CHEBI:6956 | CHEMBL299031)
Affinity DataKi:  13nMAssay Description:Inhibition of mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269637(CHEMBL4102093)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50518026(CHEMBL4449152)
Affinity DataKi:  42nMAssay Description:Inhibition of mu opioid receptor (unknown origin) assessed as reduction in intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269633(CHEMBL4077833)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474152(CHEBI:6956 | CHEMBL299031)
Affinity DataKi:  123nMAssay Description:Inhibition of kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269633(CHEMBL4077833)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528970(CHEMBL4522339)
Affinity DataKi:  720nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) expressed in CHO cells by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474153(CHEMBL61630)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269639(CHEMBL4060120)
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269639(CHEMBL4060120)
Affinity DataKi:  2.19E+3nMAssay Description:Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269639(CHEMBL4060120)
Affinity DataKi:  2.28E+3nMAssay Description:Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50518058(CHEMBL4463417)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of mu opioid receptor (unknown origin) assessed as reduction in intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataIC50:  0.282nMAssay Description:Inhibition of mu opioid receptor (unknown origin) in presence of DPDPE by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of delta opioid receptor (unknown origin) in presence of DPDPE by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of delta opioid receptor (unknown origin) in presence of DAMGO by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetKappa-type/Mu-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50142692(CHEMBL3759092)
Affinity DataIC50:  1.90nMAssay Description:Agonist activity at MOR/KOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of mu opioid receptor (unknown origin) in presence of DAMGO by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetKappa-type/Mu-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269634(CHEMBL4079574)
Affinity DataIC50:  9.90nMAssay Description:Agonist activity at MOR/KOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type/Mu-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269637(CHEMBL4102093)
Affinity DataIC50:  22nMAssay Description:Agonist activity at MOR/KOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type/Mu-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269638(CHEMBL4066846)
Affinity DataIC50:  49nMAssay Description:Agonist activity at MOR/KOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataIC50:  132nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) in presence of DPDPE by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataIC50:  132nMAssay Description:Inhibition of kappa opioid receptor (unknown origin) in presence of DAMGO by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetKappa-type/Mu-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50269633(CHEMBL4077833)
Affinity DataIC50:  194nMAssay Description:Agonist activity at MOR/KOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528962(CHEMBL4563548)
Affinity DataIC50:  900nMAssay Description:Inhibition of delta opioid receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528962(CHEMBL4563548)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of full length delta opioid receptor (unknown origin) assessed as inhibition of forskolin-stimulated intracellular cAMP accumulationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528971(CHEMBL4582676)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of delta opioid receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528971(CHEMBL4582676)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of full length delta opioid receptor (unknown origin) assessed as inhibition of forskolin-stimulated intracellular cAMP accumulationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528962(CHEMBL4563548)
Affinity DataIC50:  2.44E+4nMAssay Description:Inhibition of delta opioid receptor (unknown origin) by MVD assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528971(CHEMBL4582676)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of delta opioid receptor (unknown origin) by MVD assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528971(CHEMBL4582676)
Affinity DataIC50:  1.09E+6nMAssay Description:Inhibition of mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50528962(CHEMBL4563548)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition of mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 132 total ) | Next | Last >>
Jump to: