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Found 90 with Last Name = 'go' and Initial = 'hj'
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231553(CHEMBL1203032)
Affinity DataIC50:  0.630nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231400(CHEMBL1203053)
Affinity DataIC50:  0.810nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231339(CHEMBL1203039)
Affinity DataIC50:  0.810nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231552(CHEMBL1203031)
Affinity DataIC50:  0.840nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231396(CHEMBL1203034)
Affinity DataIC50:  1nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231560(CHEMBL1203083)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231551(CHEMBL1203086)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231546(CHEMBL1203024)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231537(CHEMBL1203019)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231511(CHEMBL1203063)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231541(CHEMBL1203069)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231465(CHEMBL1203057)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231463(CHEMBL1203091)
Affinity DataIC50:  5nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231517(CHEMBL1203068)
Affinity DataIC50:  5.10nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231464(CHEMBL1203092)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of human platelet aggregation cAMP PDE in vitroMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50231555(CHEMBL1203084)
Affinity DataIC50: >10nMAssay Description:Inhibition of human blood platelet c-AMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065348((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065336((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50:  260nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065344(CHEMBL89088 | methyl 5,8a-dimethyl-1-[2-(2-oxo-2,5...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065343((1S,4aR,5S,6S)-6-Hydroxymethyl-1,4a-dimethyl-5-[2-...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065347(3-[2-((1S,5S,8aR)-5-Methoxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065339((1S,4aS)-6-Formyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-di...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065352((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065335((1S,4aS,5R,6S)-6-Hydroxy-1,4a-dimethyl-5-[2-(2-oxo...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065342((1S,4aS,5R)-1,4a-Dimethyl-6-oxo-5-[2-(2-oxo-tetrah...)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065333(6-Hydroxymethyl-1,4a-dimethyl-5-[2-(2-oxo-2,5-dihy...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065345((1S,4aR,5S)-1,4a,6-Trimethyl-5-[2-(2-oxo-tetrahydr...)
Affinity DataIC50:  4.80E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065346((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(5-oxo-...)
Affinity DataIC50:  6.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065341((1R,6S,9aS)-6,9a-Dimethyl-3-oxo-1-[2-(5-oxo-2,5-di...)
Affinity DataIC50:  8.00E+3nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065337((1S,4aR,5S)-5-((Z)-5-Hydroxy-3-hydroxymethyl-pent-...)
Affinity DataIC50:  1.20E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065351((Z)-2-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethy...)
Affinity DataIC50:  2.10E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065350((1S,4aR,5S)-1,4a-Dimethyl-6-methylene-5-[2-(2-oxo-...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065338(3-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  3.00E+4nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50613929(CHEMBL5270848)
Affinity DataIC50: >1.00E+5nMAssay Description:Binding affinity to human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065349(4-[2-((1S,5S,8aR)-5-Hydroxymethyl-5,8a-dimethyl-2-...)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065340((1S,4aR,5S)-5-(2-Furan-3-yl-ethyl)-1,4a-dimethyl-6...)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50065334((1S,4aS,5R,6R)-6-Hydroxy-6-hydroxymethyl-1,4a-dime...)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against PAF receptor using [3H]-PAF as radioligand in rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50456020(CHEMBL2368531)
Affinity DataKd:  22nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047265(3-(2-{3-[4-(5-Hydroxy-pentylcarbamoyl)-oxazol-2-yl...)
Affinity DataKd:  20nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047266(3-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  0.100nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047267(2-{3-[2-(3-Hydroxy-propyl)-benzyl]-7-oxa-bicyclo[2...)
Affinity DataKd:  112nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047268(3-(2-{3-[4-(4-Cyclohexylcarbamoyl-butylcarbamoyl)-...)
Affinity DataKd:  22nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047270(3-[2-(3-{4-[4-(4-Methoxy-phenyl)-butylcarbamoyl]-o...)
Affinity DataKd:  0.300nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047269(3-(2-{3-[4-(5,5,5-Trifluoro-pentylcarbamoyl)-oxazo...)
Affinity DataKd:  4.80nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047271(3-{2-[3-(4-tert-Butylcarbamoyl-oxazol-2-yl)-7-oxa-...)
Affinity DataKd:  19nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047272(3-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  36nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047273(2-{3-[2-(2-Carboxy-ethyl)-benzyl]-7-oxa-bicyclo[2....)
Affinity DataKd:  1nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047275(3-{2-[3-(4-Methylcarbamoyl-oxazol-2-yl)-7-oxa-bicy...)
Affinity DataKd:  45nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047274(3-{2-[3-(4-Pentylcarbamoyl-oxazol-2-yl)-7-oxa-bicy...)
Affinity DataKd:  4nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047276(3-(2-{3-[4-(Methyl-pentyl-carbamoyl)-oxazol-2-yl]-...)
Affinity DataKd:  11nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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