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Found 701 with Last Name = 'oyama' and Initial = 'y'
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260267(CHEMBL2059382)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260248(CHEMBL4092119)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454798(7-Benzylidenenaltrexone | BNTX)
Affinity DataKi:  2.80nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260257(CHEMBL4105306)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260244(CHEMBL3632690)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260242(CHEMBL4071324)
Affinity DataKi:  4.20nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260242(CHEMBL4071324)
Affinity DataKi:  5nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260267(CHEMBL2059382)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260243(CHEMBL4070277)
Affinity DataKi:  6.10nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260243(CHEMBL4070277)
Affinity DataKi:  8.20nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260249(CHEMBL4081053)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454798(7-Benzylidenenaltrexone | BNTX)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260249(CHEMBL4081053)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260257(CHEMBL4105306)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260244(CHEMBL3632690)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260258(CHEMBL4089193)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260248(CHEMBL4092119)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260247(CHEMBL2059381)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against binding of Fibrinogen to thrombocyte alpha IIb beta-3 integrinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260267(CHEMBL2059382)
Affinity DataKi:  28nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260244(CHEMBL3632690)
Affinity DataKi:  29nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260258(CHEMBL4089193)
Affinity DataKi:  33nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50454798(7-Benzylidenenaltrexone | BNTX)
Affinity DataKi:  33nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260247(CHEMBL2059381)
Affinity DataKi:  35nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260257(CHEMBL4105306)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260249(CHEMBL4081053)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260242(CHEMBL4071324)
Affinity DataKi:  70nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260243(CHEMBL4070277)
Affinity DataKi:  79nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260262(CHEMBL4061882)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260263(CHEMBL4090365)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260247(CHEMBL2059381)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260248(CHEMBL4092119)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260262(CHEMBL4061882)
Affinity DataKi:  176nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260262(CHEMBL4061882)
Affinity DataKi:  192nMAssay Description:Inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260258(CHEMBL4089193)
Affinity DataKi:  209nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260263(CHEMBL4090365)
Affinity DataKi:  499nMAssay Description:Displacement of [3H]DAMGO from human mu opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50260263(CHEMBL4090365)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]U-69,593 from human kappa opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Toho University

Curated by ChEMBL
LigandPNGBDBM50013804(10,13-Dimethyl-hexadecahydro-cyclopenta[a]phenanth...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant IDO assessed as inhibition of indoleamine 2,3-dioxygenase to kynurenine conversion after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Toho University

Curated by ChEMBL
LigandPNGBDBM36371(5-(1H-indol-3-ylmethyl)-3-methyl-2-thioxo-4-Imidaz...)
Affinity DataKi:  1.14E+4nMAssay Description:Inhibition of human recombinant IDO assessed as inhibition of indoleamine 2,3-dioxygenase to kynurenine conversion after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Toho University

Curated by ChEMBL
LigandPNGBDBM21973(1-Methyltryptophan, 1 | 2-amino-3-(1-methyl-1H-ind...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of human recombinant IDO assessed as inhibition of indoleamine 2,3-dioxygenase to kynurenine conversion after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Homo sapiens (Human))
Toho University

Curated by ChEMBL
LigandPNGBDBM24813(Brassinin, 1 | N-(1H-indol-3-ylmethyl)(methylsulfa...)
Affinity DataKi:  9.80E+4nMAssay Description:Inhibition of human recombinant IDO assessed as inhibition of indoleamine 2,3-dioxygenase to kynurenine conversion after 60 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataIC50:  0.120nMAssay Description:Displacement of [125I]kisspeptin-15 from GPR54More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM26339((2R,3E)-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carba...)
Affinity DataIC50:  0.120nMAssay Description:Displacement of [125I]kisspeptin-15 from GPR54More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50101132(1,3-Dibenzyl-[1,3]diazetidine-2,4-dione | CHEMBL47...)
Affinity DataIC50:  0.390nMAssay Description:Compound was evaluated for its inhibitory activity against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50101132(1,3-Dibenzyl-[1,3]diazetidine-2,4-dione | CHEMBL47...)
Affinity DataIC50:  0.690nMAssay Description:Compound was evaluated for its inhibitory activity against bovine pancreatic alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM26338((2S)-N-[(1S)-4-carbamimidamido-1-{[(1S)-1-carbamoy...)
Affinity DataIC50:  0.710nMAssay Description:Displacement of [125I]kisspeptin-15 from GPR54More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336911((S)-2-((S)-2-((S)-5-amino-2-((S)-1-((S)-2-((S)-2-(...)
Affinity DataIC50:  0.790nMAssay Description:Displacement of (D-[125I]Tyr1, MePhe3)-NPFF from NPFFR2 after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50101136(1,3-Bis-benzo[1,3]dioxol-5-ylmethyl-[1,3]diazetidi...)
Affinity DataIC50:  0.850nMAssay Description:Compound was evaluated for its inhibitory activity against human Serine protease chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50336911((S)-2-((S)-2-((S)-5-amino-2-((S)-1-((S)-2-((S)-2-(...)
Affinity DataIC50:  1.90nMAssay Description:Displacement of (D-[125I]Tyr1, MePhe3)-NPFF from NPFFR1 after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymase(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50101135(1,3-Bis-(4-methoxy-benzyl)-[1,3]diazetidine-2,4-di...)
Affinity DataIC50:  2nMAssay Description:Compound was evaluated for its inhibitory activity against human Serine protease chymaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50101131(1,3-Di-p-tolyl-[1,3]diazetidine-2,4-dione | CHEMBL...)
Affinity DataIC50:  2.30nMAssay Description:Compound was evaluated for its inhibitory activity against human cathepsin GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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