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Found 111 with Last Name = 'iyer' and Initial = 'v'
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404964(CHEMBL2367720)
Affinity DataKi:  250nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405380(CHEMBL1627565)
Affinity DataKi:  2.43E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50028411(3-Methoxy-13-methyl-4-nitro-6,7,8,9,11,12,13,14,15...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405376(CHEMBL1627689)
Affinity DataKi:  7.51E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405378(CHEMBL1627562)
Affinity DataKi:  9.76E+3nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405374(CHEMBL1627977)
Affinity DataKi:  1.02E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405382(CHEMBL1627685)
Affinity DataKi:  1.05E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405377(CHEMBL1627697)
Affinity DataKi:  1.19E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405383(CHEMBL1627683)
Affinity DataKi:  1.36E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405381(CHEMBL1627690)
Affinity DataKi:  1.48E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405375(CHEMBL194749)
Affinity DataKi:  1.63E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50405379(CHEMBL1627698)
Affinity DataKi:  2.51E+4nMAssay Description:Compound was tested for inhibition of porcine endometrial estrogen sulfotransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367130(CHEMBL1628097)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367129(CHEMBL1628095)
Affinity DataKi:  8.40E+4nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404963(CHEMBL2067995)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50367131(CHEMBL1628164)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404965(CHEMBL2067994)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSulfotransferase 1E1(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50404966(CHEMBL2067996)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition of bovine estrogen sulfotransferase by the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213578(US9278981, 170)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213594(US9278981, 186)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50459091(ABL-001 | ABL001 | ABL001-NX | Asciminib | NVP-ABL...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213656(US9278981, 248)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50459090(CHEMBL4213152)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50459089(CHEMBL4217559)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM230760(US9340537, 14 | US9896444, Example 14)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213441(US9278981, 33)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213443(US9278981, 35)
Affinity DataIC50:  4nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213434(US9278981, 26)
Affinity DataIC50:  7nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM222504(US9315489, 40)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]dofetilide from human ERG by high throughput assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50325999(3-(6-(4-(trifluoromethoxy)phenylamino)pyrimidin-4-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human c-ABL SH3/SH2/SH1 domain (46 to 531 residues) expressed in sf9 insect cells after 30 mins in presence of [gamma-32P]A...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM222494(US9315489, 30)
Affinity DataIC50:  11nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50328152(CHEMBL1257423 | N-(2-hydroxyethyl)-3-(6-(4-(triflu...)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant human c-ABL SH3/SH2/SH1 domain (46 to 515 residues) expressed in bacterial expression system using EAIYAAPFAKKK as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213569(US9278981, 161)
Affinity DataIC50:  18nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM222465(US9315489, 1)
Affinity DataIC50:  18nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM222504(US9315489, 40)
Affinity DataIC50:  19nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM222506(US9315489, 42)
Affinity DataIC50:  24nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213434(US9278981, 26)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]dofetilide from human ERG by high throughput assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50459086(CHEMBL4217428)
Affinity DataIC50:  550nMAssay Description:Inhibition of ABL1 (64 to 515 residues)(unknown origin) expressed in Escherichia coli using FITC-Ahx-EAIYAAPFAKKK-NH2 peptide as substrate after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50558881(CHEMBL4761836)
Affinity DataIC50:  900nMAssay Description:Inhibition of human ERG transfected in HEK293 cells assessed as reduction in channel current at -80 mV holding potential by whole-cell patch clamp me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM222494(US9315489, 30)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by high throughput assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213594(US9278981, 186)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human ERG by automated patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213569(US9278981, 161)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by high throughput assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213578(US9278981, 170)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human ERG by automated patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50357206(CHEMBL1915083 | CHEMBL1962378)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50558880(CHEMBL4533529)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human ERG transfected in HEK293 cells assessed as reduction in channel current at -80 mV holding potential by whole-cell patch clamp me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50357204(CHEMBL1914835 | CHEMBL1963280)
Affinity DataIC50:  3.46E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213578(US9278981, 170)
Affinity DataIC50:  3.60E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by high throughput assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50459086(CHEMBL4217428)
Affinity DataIC50:  3.70E+3nMAssay Description:Displacement of [3H]dofetilide from human ERG by high throughput assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM213441(US9278981, 33)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human ERG by automated patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50357205(CHEMBL1914844 | CHEMBL1963594)
Affinity DataIC50:  4.31E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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