BDBM300797 US10131645, Compound 5003
BDBM304262 US10143746, Example 5003
US10125111, Compound 5003 BDBM298575
SC-5003 BDBM50084660 CHEMBL445631 {1-[1-(1-Cyclohexylmethyl-2,5-dihydroxy-4-methyl-nonylcarbamoyl)-3-methyl-butylcarbamoyl]-2-phenyl-ethyl}-carbamic acid tert-butyl ester(SC-5003)
BDBM84649 TC-28
TC-107 BDBM84651
TC-34 BDBM84650
BDBM50045047 TC-5214 Dexmecamylamine
BDBM50403808 CHEMBL2370124 TC-14006
CHEMBL2370125 TC-14001 BDBM50403811
CHEMBL2370127 BDBM50403813 TC-14005
CHEMBL2370132 TC-14003 BDBM50403806
CHEMBL2370134 BDBM50403802 TC-14007
CHEMBL2370135 TC-14004 BDBM50403800
CHEMBL2370137 TC-14002 BDBM50403810
BDBM50436713 BUTENAFINE Mentax Mentax-TC
tc-NH2 BDBM85518 trans-cinnamoyl-LIGRLO-NH2
2-Pyridin-3-yl-1-aza-bicyclo[2.2.2]octane CHEMBL105374 TC-2429 BDBM50079456
US9464092, E BDBM253913 US9527857, E
BDBM167074 US9073876, E US9732093, Compound E
US10435361, Example 85(e) BDBM256603 US9481648, 85(e) US9790174, Example 85(e)
US9481648, 83(e) US10435361, Example 83(e) BDBM256588 US9790174, Example 83(e)
US9481648, 84(e) US10435361, Example 84(e) US9790174, Example 84(e) BDBM256595
US10626113, Compound E BDBM480488 US10899756, Compound E
US11267820, Compound e BDBM448075 US10689395, Compound e
(E,E,E)-O-(3,7,11,15-tetramethyl-2,6,10,14-hexadecatetraenyl)-N-(aminosulfonyl)urethane BDBM50051830 CHEMBL28808
BDBM614347 US20230270730, Compound E-13 US20240327355, Compound E-13 US11964950, Compound E-13
US11964950, Compound E-7 US20230270730, Compound E-7 BDBM614341 US20240327355, Compound E-7
US20240327355, Compound E-1 BDBM614335 US11964950, Compound E-1 US20230270730, Compound E-1
SMR000304531 terephthalaldehyde dithiosemicarbazone BDBM95405 [(E)-[4-[(E)-(thiocarbamoylhydrazono)methyl]benzylidene]amino]thiourea 1-[(E)-[4-[(E)-(carbamothioylhydrazinylidene)methyl]phenyl]methylideneamino]thiourea MLS000720002 [(E)-[4-[(E)-(carbamothioylhydrazinylidene)methyl]phenyl]methylideneamino]thiourea cid_9555944
- Tremblay, ML; Penafuerte, C; Feldhammer, M; Zogopoulos, G; Black, C; Kennedy, B TC-PTP inhibitors as APC activators for immunotherapy US Patent US10150787 (2018)
- Tremblay, ML; Pike, K; Perez Quintero, LA Enhancing CD8+ T cells for adoptive T cell therapy by inhibiting PTPN1 (PTP1B) and PTPN2 (TC-PTP) US Patent US11597739 (2023)
- Broekema, M; van Eerd, JJ; Oyen, WJ; Corstens, FH; Liskamp, RM; Boerman, OC; Harris, TD Synthesis of leukotriene B4 antagonists labeled with In-111 or Tc-99m to image infectious and inflammatory foci. J Med Chem 48: 6442-53 (2005)
- Oliveira, BL; Morais, M; Mendes, F; Moreira, IS; Cordeiro, C; Fernandes, PA; Ramos, MJ; Alberto, R; Santos, I; Correia, JD Re(I) and Tc(I) complexes for targeting nitric oxide synthase: influence of the chelator in the affinity for the enzyme. Chem Biol Drug Des 86: 1072-86 (2015)
- Steadman, VA; Pettit, SB; Poullennec, KG; Lazarides, L; Keats, AJ; Dean, DK; Stanway, SJ; Austin, CA; Sanvoisin, JA; Watt, GM; Fliri, HG; Liclican, AC; Jin, D; Wong, MH; Leavitt, SA; Lee, YJ; Tian, Y; Frey, CR; Appleby, TC; Schmitz, U; Jansa, P; Mackman, RL; Schultz, BE J Med Chem 60: 1000-1017 (2017)
- Atack, TC; Raymond, DD; Blomquist, CA; Pasaje, CF; McCarren, PR; Moroco, J; Befekadu, HB; Robinson, FP; Pal, D; Esherick, LY; Ianari, A; Niles, JC; Sellers, WR ACS Med Chem Lett 11: 2131-2138 (2020)
- Mokrosz, MJ; Duszynska, B; Klodzinska, A; Deren-Wesolek, A; Chojnacka-Wójcik, E; Baranowski, TC; Abdou, IM; Redmore, NP; Strekowski, L Bioorg Med Chem Lett 7: 1635-1638 (1997)
- Rennie, GR; Barden, TC; Bernier, SG; Carvalho, A; Deming, R; Germano, P; Hudson, C; Im, GJ; Iyengar, RR; Jia, L; Jung, J; Kim, E; Lee, TW; Mermerian, A; Moore, J; Nakai, T; Perl, NR; Tobin, J; Zimmer, DP; Renhowe, PA Bioorg Med Chem Lett 40: (2021)
- Bastos, MM; Costa, CC; Bezerra, TC; da Silva, Fde C; Boechat, N Eur J Med Chem 108: 455-65 (2016)
- Marhefka, CA; Moore, BM; Bishop, TC; Kirkovsky, L; Mukherjee, A; Dalton, JT; Miller, DD J Med Chem 44: 1729-40 (2001)
- Pagadala, NS; Bjorndahl, TC; Joyce, M; Wishart, DS; Syed, K; Landi, A Bioorg Med Chem 25: 5875-5888 (2017)
- Johnson, MP; Baez, M; Jagdmann, GE; Britton, TC; Large, TH; Callagaro, DO; Tizzano, JP; Monn, JA; Schoepp, DD J Med Chem 46: 3189-92 (2003)
- Yue, EW; Sparks, R; Polam, P; Modi, D; Douty, B; Wayland, B; Glass, B; Takvorian, A; Glenn, J; Zhu, W; Bower, M; Liu, X; Leffet, L; Wang, Q; Bowman, KJ; Hansbury, MJ; Wei, M; Li, Y; Wynn, R; Burn, TC; Koblish, HK; Fridman, JS; Emm, T; Scherle, PA; Metcalf, B; Combs, AP ACS Med Chem Lett 8: 486-491 (2017)
- Collins, JL; Shearer, BG; Oplinger, JA; Lee, S; Garvey, EP; Salter, M; Duffy, C; Burnette, TC; Furfine, ES J Med Chem 41: 2858-71 (1998)
- LINDSLEY, CW; ENGERS, DW; CHILDRESS, ES; BOLLINGER, SR; SCHMITT, J; CHOPKO, TC; DENTON, JS; TANAKA, M; KURATA, H US Patent US20240190824 (2024)
- Ashwell, MA; Lapierre, JM; Brassard, C; Bresciano, K; Bull, C; Cornell-Kennon, S; Eathiraj, S; France, DS; Hall, T; Hill, J; Kelleher, E; Khanapurkar, S; Kizer, D; Koerner, S; Link, J; Liu, Y; Makhija, S; Moussa, M; Namdev, N; Nguyen, K; Nicewonger, R; Palma, R; Szwaya, J; Tandon, M; Uppalapati, U; Vensel, D; Volak, LP; Volckova, E; Westlund, N; Wu, H; Yang, RY; Chan, TC J Med Chem 55: 5291-310 (2012)
- Gray, AP; Platz, RD; Chang, TC; Leverone, TR; Ferrick, DA; Kramer, DN J Med Chem 28: 111-6 (1985)
- Liu, YC; Huang, V; Chao, TC; Hsiao, CD; Lin, A; Chang, MF; Chow, LP Biochem Biophys Res Commun 333: 194-9 (2005)
- Lee, CC; Liu, FL; Chen, CL; Chen, TC; Liu, FC; Ahmed Ali, AA; Chang, DM; Huang, HS Bioorg Med Chem 23: 4522-32 (2015)
- Wong, ILK; Zhu, X; Chan, KF; Liu, Z; Chan, CF; Chow, TS; Chong, TC; Law, MC; Cui, J; Chow, LMC; Chan, TH J Med Chem 64: 14311-14331 (2021)
- Chopko, TC; Han, C; Gregro, AR; Engers, DW; Felts, AS; Poslusney, MS; Bollinger, KA; Morrison, RD; Bubser, M; Lamsal, A; Luscombe, VB; Cho, HP; Schnetz-Boutaud, NC; Rodriguez, AL; Chang, S; Daniels, JS; Stec, DF; Niswender, CM; Jones, CK; Wood, MR; Wood, MW; Duggan, ME; Brandon, NJ; Conn, PJ; Bridges, TM; Lindsley, CW; Melancon, BJ Bioorg Med Chem Lett 29: 2224-2228 (2019)
- Su, TL; Chou, TC; Kim, JY; Huang, JT; Ciszewska, G; Ren, WY; Otter, GM; Sirotnak, FM; Watanabe, KA J Med Chem 38: 3226-35 (1995)
- Coombs, TC; Tanega, C; Shen, M; Wang, JL; Auld, DS; Gerritz, SW; Schoenen, FJ; Thomas, CJ; Aubé, J Bioorg Med Chem Lett 23: 3654-61 (2013)
- Washburn, WN; Sher, PM; Poss, KM; Girotra, RN; McCann, PJ; Gavai, AV; Mikkilineni, AB; Mathur, A; Cheng, P; Dejneka, TC; Sun, CQ; Wang, TC; Harper, TW; Russell, AD; Slusarchyk, DA; Skwish, S; Allen, GT; Hillyer, DE; Frohlich, BH; Abboa-Offei, BE; Cap, M; Waldron, TL; George, RJ; Tesfamariam, B; Ciosek, CP; Ryono, D; Young, DA; Dickinson, KE; Seymour, AA; Arbeeny, CM; Gregg, RE Bioorg Med Chem Lett 11: 3035-9 (2001)
- Huck, BR; Llamas, L; Robarge, MJ; Dent, TC; Song, J; Hodnick, WF; Crumrine, C; Stricker-Krongrad, A; Harrington, J; Brunden, KR; Bennani, YL Bioorg Med Chem Lett 16: 4130-4 (2006)
- Neves, MA; Dinis, TC; Colombo, G; Sá e Melo, ML Eur J Med Chem 44: 4121-7 (2009)
- Eadsforth, TC; Pinto, A; Luciani, R; Tamborini, L; Cullia, G; De Micheli, C; Marinelli, L; Cosconati, S; Novellino, E; Lo Presti, L; Cordeiro da Silva, A; Conti, P; Hunter, WN; Costi, MP J Med Chem 58: 7938-48 (2015)
- Jung, E; Soto-Acosta, R; Xie, J; Wilson, DJ; Dreis, CD; Majima, R; Edwards, TC; Geraghty, RJ; Chen, L ACS Med Chem Lett 13: 1477-1484 (2022)
- Charles, MD; Brookfield, JL; Ekwuru, TC; Stockley, M; Dunn, J; Riddick, M; Hammonds, T; Trivier, E; Greenland, G; Wong, AC; Cheasty, A; Boyd, S; Crighton, D; Olson, MF J Med Chem 58: 8309-13 (2015)
- Fleischer, TC; Murphy, BR; Flick, JS; Terry-Lorenzo, RT; Gao, ZH; Davis, T; McKinnon, R; Ostanin, K; Willardsen, JA; Boniface, JJ Chem Biol 17: 659-64 (2010)
- Gahman, TC; Herbert, MR; Lang, H; Thayer, A; Symons, KT; Nguyen, PM; Massari, ME; Dozier, S; Zhang, Y; Sablad, M; Rao, TS; Noble, SA; Shiau, AK; Hassig, CA Bioorg Med Chem Lett 21: 6888-94 (2011)
- Gallagher, TC; Rego Campello, H US Patent US11667638 (2023)
- Jordan, DB; Lessen, TA; Wawrzak, Z; Bisaha, JJ; Gehret, TC; Hansen, SL; Schwartz, RS; Basarab, GS Bioorg Med Chem Lett 9: 1607-12 (1999)
- Pfefferkorn, JA; Litchfield, J; Hutchings, R; Cheng, XM; Larsen, SD; Auerbach, B; Bush, MR; Lee, C; Erasga, N; Bowles, DM; Boyles, DC; Lu, G; Sekerke, C; Askew, V; Hanselman, JC; Dillon, L; Lin, Z; Robertson, A; Olsen, K; Boustany, C; Atkinson, K; Goosen, TC; Sahasrabudhe, V; Chupka, J; Duignan, DB; Feng, B; Scialis, R; Kimoto, E; Bi, YA; Lai, Y; El-Kattan, A; Bakker-Arkema, R; Barclay, P; Kindt, E; Le, V; Mandema, JW; Milad, M; Tait, BD; Kennedy, R; Trivedi, BK; Kowala, M Bioorg Med Chem Lett 21: 2725-31 (2011)
- Berdini, V; Carr, MG; Congreve, MS; Frederickson, M; Griffiths-Jones, CM; Hamlett, CC; Madin, A; Murray, CW; Benning, RK; Saxty, G; Vickerstaffe, E; Williams, BJ; Woodhead, AJ; Woodhead, SJ; Freyne, EJ; Govaerts, TC; Angibaud, PR US Patent US8796244 (2014)
- YANG, J; MANDEGAR, MA; HOEY, TC US Patent US20230381148 (2023)
- Wang, S; Wan, NC; Harrison, J; Miller, W; Chuckowree, I; Sohal, S; Hancox, TC; Baker, S; Folkes, A; Wilson, F; Thompson, D; Cocks, S; Farmer, H; Boyce, A; Freathy, C; Broadbridge, J; Scott, J; Depledge, P; Faint, R; Mistry, P; Charlton, P J Med Chem 47: 1339-50 (2004)
- Weidner-Wells, MA; Henninger, TC; Fraga-Spano, SA; Boggs, CM; Matheis, M; Ritchie, DM; Argentieri, DC; Wachter, MP; Hlasta, DJ Bioorg Med Chem Lett 14: 4307-11 (2004)
- Ho, TC; Tius, MA; Nikas, SP; Tran, NK; Tong, F; Zhou, H; Zvonok, N; Makriyannis, A Bioorg Med Chem Lett 38: (2021)
- Koyama, K; Hirasawa, Y; Hosoya, T; Hoe, TC; Chan, KL; Morita, H Bioorg Med Chem 18: 4415-21 (2010)
- Singh, SB; Malamas, MS; Hohman, TC; Nilakantan, R; Carper, DA; Kitchen, D J Med Chem 43: 1062-70 (2000)
- Cheng, JH; Huang, AM; Hour, TC; Yang, SC; Pu, YS; Lin, CN Eur J Med Chem 46: 1222-31 (2011)
- Lin, TS; Liw, YW; Song, JS; Hsieh, TC; Yeh, HW; Hsu, LC; Lin, CJ; Wu, SH; Liang, PH Bioorg Med Chem 21: 6282-91 (2013)
- ANDERSON, ED; ARONOW, SD; BOYLES, NA; DAHLGREN, MK; FENG, S; GERASYUTO, AI; HICKEY, ER; IRVIN, TC; KESICKI, EA; KLIPPEL-GIESE, A; KNIGHT, JL; KOLAKOWSKI, GR; KUMAR, M; LONG, KF; MAYNE, CG; MCELLIGOTT, DL; MCLEAN, JA; PUCA, L; RAVI, KK; SEVERANCE, DL; WELCH, MB; WIDJAJA, T US Patent US20230286960 (2023)
- Anderson, ED; Aronow, SD; Boyles, NA; Dahlgren, MK; Feng, S; Gerasyuto, AI; Hickey, ER; Irvin, TC; Kesicki, EA; Klippel-Giese, A; Knight, JL; Kolakowski, GR; Kumar, M; Long, KF; Mayne, CG; McElligott, DL; McLean, JA; Puca, L; Ravi, KK; Severance, DL; Welch, MB; Widjaja, T US Patent US11649227 (2023)
- Green, LS; Bullard, JM; Ribble, W; Dean, F; Ayers, DF; Ochsner, UA; Janjic, N; Jarvis, TC Antimicrob Agents Chemother 53: 86-94 (2008)
- Perry, PJ; Reszka, AP; Wood, AA; Read, MA; Gowan, SM; Dosanjh, HS; Trent, JO; Jenkins, TC; Kelland, LR; Neidle, S J Med Chem 41: 4873-84 (1998)
- Washburn, DG; Holt, DA; Dodson, J; McAtee, JJ; Terrell, LR; Barton, L; Manns, S; Waszkiewicz, A; Pritchard, C; Gillie, DJ; Morrow, DM; Davenport, EA; Lozinskaya, IM; Guss, J; Basilla, JB; Negron, LK; Klein, M; Willette, RN; Fries, RE; Jensen, TC; Xu, X; Schnackenberg, CG; Marino, JP Bioorg Med Chem Lett 23: 4979-84 (2013)
- Jahng, Y; Zhao, LX; Moon, YS; Basnet, A; Kim, EK; Chang, HW; Ju, HK; Jeong, TC; Lee, ES Bioorg Med Chem Lett 14: 2559-62 (2004)
- Jessop, TC; Tarver, JE; Carlsen, M; Xu, A; Healy, JP; Heim-Riether, A; Fu, Q; Taylor, JA; Augeri, DJ; Shen, M; Stouch, TR; Swanson, RV; Tari, LW; Hunter, M; Hoffman, I; Keyes, PE; Yu, XC; Miranda, M; Liu, Q; Swaffield, JC; David Kimball, S; Nouraldeen, A; Wilson, AG; Foushee, AM; Jhaver, K; Finch, R; Anderson, S; Oravecz, T; Carson, KG Bioorg Med Chem Lett 19: 6784-7 (2009)
- Chen, X; Cheng, AC; Connors, RV; Debenedetto, MV; Dransfield, PJ; Fu, Z; Harvey, JS; Heath, JA; Houze, J; Judd, TC; Kopecky, DJ; Lai, S; Ma, Z; Nishimura, N; Olson, SH; Pattaropong, V; Wang, X US Patent US10150760 (2018)
- Ho, W; Tarhan, O; Kiorpes, TC; Tutwiler, GF; Mohrbacher, RJ J Med Chem 30: 1094-7 (1987)
- Hennessy, EJ; Chuaqui, C; Ashton, S; Colclough, N; Cross, DA; Debreczeni, JÉ; Eberlein, C; Gingipalli, L; Klinowska, TC; Orme, JP; Sha, L; Wu, X ACS Med Chem Lett 7: 514-9 (2016)
- Lienau, C; Gräwert, T; Alves Avelar, LA; Illarionov, B; Held, J; Knaab, TC; Lungerich, B; van Geelen, L; Meier, D; Geissler, S; Cynis, H; Riederer, U; Buchholz, M; Kalscheuer, R; Bacher, A; Mordmüller, B; Fischer, M; Kurz, T Eur J Med Chem 181: (2019)
- Okorom, AV; Camacho-Hernandez, GA; Salomon, K; Lee, KH; Ku, TC; Cao, J; Won, SJ; Friedman, J; Lam, J; Paule, J; Rais, R; Klein, B; Xi, ZX; Shi, L; Loland, CJ; Newman, AH J Med Chem 67: 709-727
- Hou, DR; Alam, S; Kuan, TC; Ramanathan, M; Lin, TP; Hung, MS Bioorg Med Chem Lett 19: 1022-5 (2009)
- Le, TC; Yim, CY; Park, S; Katila, N; Yang, I; Song, MC; Yoon, YJ; Choi, DY; Choi, H; Nam, SJ; Fenical, W Bioorg Med Chem Lett 27: 3123-3126 (2017)
- Shi, K; Huang, Q; Huang, Y; Lee, TC; Yu, H J Agric Food Chem 59: 56-61 (2011)
- Geldenhuys, WJ; Yonutas, HM; Morris, DL; Sullivan, PG; Darvesh, AS; Leeper, TC Bioorg Med Chem Lett 26: 5350-5353 (2016)
- Agnihotri, G; Crall, BM; Lewis, TC; Day, TP; Balakrishna, R; Warshakoon, HJ; Malladi, SS; David, SA J Med Chem 54: 8148-60 (2011)
- Zhang, J; Chan, A; Lippa, B; Cross, JB; Liu, C; Yin, N; Romero, JA; Lawrence, J; Heney, R; Herradura, P; Goss, J; Clark, C; Abel, C; Zhang, Y; Poutsiaka, KM; Epie, F; Conrad, M; Mahamoon, A; Nguyen, K; Chavan, A; Clark, E; Li, TC; Cheng, RK; Wood, M; Andersen, OA; Brooks, M; Kwong, J; Barker, J; Parr, IB; Gu, Y; Ryan, MD; Coleman, S; Metcalf, CA Bioorg Med Chem Lett 27: 1670-1680 (2017)
- Lin, SW; Lin, YL; Lin, TC; Yang, DY Bioorg Med Chem Lett 10: 1297-8 (2000)
- Chambers, RJ; Marfat, A; Antognoli, GW; Cheng, JB; Damon, DB; Kuperman, AV; Liston, TC; Mebus, C; Pillar, JS; Shirley, JT; Watson, JW Bioorg Med Chem Lett 9: 2773-8 (1999)
- Wu, CP; Lusvarghi, S; Hsiao, SH; Liu, TC; Li, YQ; Huang, YH; Hung, TH; Ambudkar, SV J Nat Prod 83: 1461-1472 (2020)
- Ghosh, S; Chan, JM; Lea, CR; Meints, GA; Lewis, JC; Tovian, ZS; Flessner, RM; Loftus, TC; Bruchhaus, I; Kendrick, H; Croft, SL; Kemp, RG; Kobayashi, S; Nozaki, T; Oldfield, E J Med Chem 47: 175-87 (2003)
- Sun, L; Liang, C; Shirazian, S; Zhou, Y; Miller, T; Cui, J; Fukuda, JY; Chu, JY; Nematalla, A; Wang, X; Chen, H; Sistla, A; Luu, TC; Tang, F; Wei, J; Tang, C J Med Chem 46: 1116-9 (2003)
- Boschelli, DH; Wu, Z; Klutchko, SR; Showalter, HD; Hamby, JM; Lu, GH; Major, TC; Dahring, TK; Batley, B; Panek, RL; Keiser, J; Hartl, BG; Kraker, AJ; Klohs, WD; Roberts, BJ; Patmore, S; Elliott, WL; Steinkampf, R; Bradford, LA; Hallak, H; Doherty, AM J Med Chem 41: 4365-77 (1998)
- Moradei, OM; Mallais, TC; Frechette, S; Paquin, I; Tessier, PE; Leit, SM; Fournel, M; Bonfils, C; Trachy-Bourget, MC; Liu, J; Yan, TP; Lu, AH; Rahil, J; Wang, J; Lefebvre, S; Li, Z; Vaisburg, AF; Besterman, JM J Med Chem 50: 5543-6 (2007)
- Boral, S; Malone, TC; Wang, S US Patent US9403803 (2016)
- Kehne, JH; Baron, BM; Carr, AA; Chaney, SF; Elands, J; Feldman, DJ; Frank, RA; van Giersbergen, PL; McCloskey, TC; Johnson, MP; McCarty, DR; Poirot, M; Senyah, Y; Siegel, BW; Widmaier, C J Pharmacol Exp Ther 277: 968-81 (1996)
- Bokesch, HR; Cartner, LK; Fuller, RW; Wilson, JA; Henrich, CJ; Kelley, JA; Gustafson, KR; McMahon, JB; McKee, TC Bioorg Med Chem Lett 20: 3848-50 (2010)
- Rodgers, TL; Townsend, PD; Burnell, D; Jones, ML; Richards, SA; McLeish, TC; Pohl, E; Wilson, MR; Cann, MJ PLoS Biol 11: 1-15 (2013)
- Hoang, VH; Trang, NTK; Minh, TC; Long, LTB; Lan, TH; Hue, NT; Tien, LQ; Nguyen, TX; Nguyen, YTK; Yoo, H; Tran, PT Bioorg Med Chem 90: (2023)
- Moon, TC; Quan, Z; Kim, J; Kim, HP; Kudo, I; Murakami, M; Park, H; Chang, HW Bioorg Med Chem 15: 7138-43 (2007)
- Neenan, JP; Opitz, SM; Cooke, CL; Ussery, MA; Morrill, TC; Eckel, LM Bioorg Med Chem Lett 6: 1381-1386 (1996)
- Hicken, EJ; Brown, K; Dwulet, NC; Gaudino, JJ; Hansen, EP; Hartley, DP; Kowalski, JP; Laird, ER; Lazzara, NC; Li, B; Mou, TC; Mutryn, MF; Oko, L; Pajk, S; Pipal, RW; Rosen, RZ; Shelp, R; Singh, A; Wang, J; Wise, CE; Wong, C; Wong, JY J Med Chem 67: 9759-9771
- Chang, YT; Gray, NS; Rosania, GR; Sutherlin, DP; Kwon, S; Norman, TC; Sarohia, R; Leost, M; Meijer, L; Schultz, PG Chem Biol 6: 361-75 (1999)
- Hu, T; Zhang, J; Wang, J; Sha, L; Xia, Y; Ortyl, TC; Tian, X; Chen, L J Med Chem 66: 4434-4467 (2023)
- Merkler, DJ; Asser, AS; Baumgart, LE; Carballo, N; Carpenter, SE; Chew, GH; Cosner, CC; Dusi, J; Galloway, LC; Lowe, AB; Lowe, EW; King, L; Kendig, RD; Kline, PC; Malka, R; Merkler, KA; McIntyre, NR; Romero, M; Wilcox, BJ; Owen, TC Bioorg Med Chem 16: 10061-74 (2008)
- Uprety, R; Váradi, A; Allaoa, A; Redel-Traub, GN; Palmer, TC; Feinberg, EN; Ferris, AC; Pande, VS; Pasternak, GW; Majumdar, S Eur J Med Chem 164: 241-251 (2019)
- Banerjee, S; Norman, DD; Lee, SC; Parrill, AL; Pham, TC; Baker, DL; Tigyi, GJ; Miller, DD J Med Chem 60: 1309-1324 (2017)
- BLANK, BR; GIBBONS, PA; NDUBAKU, C; ROMERO, FA; CHANG, JH; PHAM, JD; ROBERTS, TC; VEKARIYA, RH; JEANNERET, AD; SILVA, H; DADA, RO; McINTOSH, KC; NEIGER, E; BROWN, W; TAKASAKI, H; CRIFAR, CC; POLAT, DE US Patent US20250034159 (2025)
- Antunes, JE; Freitas, MP; da Cunha, EF; Ramalho, TC; Rittner, R Bioorg Med Chem 16: 7599-606 (2008)
- Reddy, NP; Aparoy, P; Reddy, TC; Achari, C; Sridhar, PR; Reddanna, P Bioorg Med Chem 18: 5807-15 (2010)
- de Souza, MM; Andreolla, MC; Ribeiro, TC; Gonçalves, AE; Medeiros, AR; de Souza, AS; Ferreira, LLG; Andricopulo, AD; Yunes, RA; de Oliveira, AS RSC Med Chem 11: 307-316 (2020)
- Ndubaku, CO; Katibah, GE; Roberts, TC; Sung, L; Ciblat, S; Raeppel, F; Ly, VL; Ramtohul, YK; Rybak, T; Zaky, M; Gillard, L; Ismaili, H US Patent US10738056 (2020)
- Hruschka, S; Rosen, TC; Yoshida, S; Kirk, KL; Fröhlich, R; Wibbeling, B; Haufe, G Bioorg Med Chem 16: 7148-66 (2008)
- Kimura, T; Shuto, D; Kasai, S; Liu, P; Hidaka, K; Hamada, T; Hayashi, Y; Hattori, C; Asai, M; Kitazume, S; Saido, TC; Ishiura, S; Kiso, Y Bioorg Med Chem Lett 14: 1527-31 (2004)
- Sanders, TC; Seto, CT J Med Chem 42: 2969-76 (1999)
- Dyckman, AJ; Dodd, DS; Mussari, CP; Sherwood, TC; Haque, TS; Posy, SL; Kumar, SR; Pasunoori, L; Hegde, S; Anumula, RK US Patent US11420973 (2022)
- Matthias, E; Kristina, WM; Juergen, P; Ferenc, K; Leo, T; Siegfried, TC; Dieter, W WIPO WO2022101377 (2022)
- Zhao, LM; Jin, HS; Liu, J; Skaar, TC; Ipe, J; Lv, W; Flockhart, DA; Cushman, M Bioorg Med Chem 24: 5400-5409 (2016)
- Crespo, RA; Dang, Q; Zhou, NE; Guthrie, LM; Snavely, TC; Dong, W; Loesch, KA; Suzuki, T; You, L; Wang, W; O'Malley, T; Parish, T; Olsen, DB; Sacchettini, JC J Med Chem 62: 4483-4499 (2019)
- Rawson, TE; Somers, TC; Marsters, JC; Wan, DT; Reynolds, ME; Burdick, DJ Bioorg Med Chem Lett 5: 1335-1338 (1995)
- Jones, S; Ahmet, J; Ayton, K; Ball, M; Cockerill, M; Fairweather, E; Hamilton, N; Harper, P; Hitchin, J; Jordan, A; Levy, C; Lopez, R; McKenzie, E; Packer, M; Plant, D; Simpson, I; Simpson, P; Sinclair, I; Somervaille, TC; Small, H; Spencer, GJ; Thomson, G; Tonge, M; Waddell, I; Walsh, J; Waszkowycz, B; Wigglesworth, M; Wiseman, DH; Ogilvie, D J Med Chem 59: 11120-11137 (2016)
- Obando, D; Pantarat, N; Handke, R; Koda, Y; Widmer, F; Djordjevic, JT; Ellis, DH; Sorrell, TC; Jolliffe, KA Bioorg Med Chem 17: 6329-39 (2009)
- Ong, HH; Anderson, VB; Wilker, JC; Spaulding, TC; Meyerson, LR J Med Chem 23: 726-9 (1980)
- Turek, TC; Gaon, I; Gamache, D; Distefano, MD Bioorg Med Chem Lett 7: 2125-2130 (1997)
- Möller, D; Banerjee, A; Uzuneser, TC; Skultety, M; Huth, T; Plouffe, B; Hübner, H; Alzheimer, C; Friedland, K; Müller, CP; Bouvier, M; Gmeiner, P J Med Chem 60: 2908-2929 (2017)
- Tosh, DK; Deflorian, F; Phan, K; Gao, ZG; Wan, TC; Gizewski, E; Auchampach, JA; Jacobson, KA J Med Chem 55: 4847-60 (2012)
- Washburn, WN; Sher, PM; Poss, KM; Girotra, RN; McCann, PJ; Gavai, AV; Mikkilineni, AB; Mathur, A; Cheng, P; Dejneka, TC; Sun, CQ; Wang, TC; Harper, TW; Russell, AD; Slusarchyk, DA; Skwish, S; Allen, GT; Hillyer, DE; Frohlich, BH; Abboa-Offei, BE; Cap, M; Waldron, TL; George, RJ; Tesfamariam, B; Ciosek, CP; Ryono, D; Young, DA; Dickinson, KE; Seymour, AA; Arbeeny, CM; Gregg, RE Bioorg Med Chem Lett 11: 3035-9 (2001)
- Kim, DH; Guinosso, CJ; Buzby, GC; Herbst, DR; McCaully, RJ; Wicks, TC; Wendt, RL J Med Chem 26: 394-403 (1983)
- Bennett, JM; Campbell, AD; Campbell, AJ; Carr, MG; Dunsdon, RM; Greening, JR; Hurst, DN; Jennings, NS; Jones, PS; Jordan, S; Kay, PB; O'Brien, MA; King-Underwood, J; Raynham, TM; Wilkinson, CS; Wilkinson, TC; Wilson, FX Bioorg Med Chem Lett 11: 355-7 (2001)
- Carpino, PA; Lefker, BA; Toler, SM; Pan, LC; Hadcock, JR; Murray, MC; Cook, ER; DiBrino, JN; DeNinno, SL; Chidsey-Frink, KL; Hada, WA; Inthavongsay, J; Lewis, SK; Mangano, FM; Mullins, MA; Nickerson, DF; Ng, O; Pirie, CM; Ragan, JA; Rose, CR; Tess, DA; Wright, AS; Yu, L; Zawistoski, MP; Pettersen, JC; DaSilva-Jardine, PA; Wilson, TC; Thompson, DD Bioorg Med Chem Lett 12: 3279-82 (2002)
- Packiarajan, M; Coate, H; Desai, M; Jimenez, HN; Reinhard, EJ; Jubian, VJ; Marzabadi, MR; Chandrasena, G; Wolinski, TC; Walker, MW; Andersen, K Bioorg Med Chem Lett 21: 6500-4 (2011)
- Wu, L; Lu, K; Packiarajan, M; Jubian, V; Chandrasena, G; Wolinsky, TC; Walker, MW Bioorg Med Chem Lett 22: 2167-71 (2012)
- Wallace, EM; Lyssikatos, J; Blake, JF; Seo, J; Yang, HW; Yeh, TC; Perrier, M; Jarski, H; Marsh, V; Poch, G; Livingston, MG; Otten, J; Hingorani, G; Woessner, R; Lee, P; Winkler, J; Koch, K J Med Chem 49: 441-4 (2006)
- Zankel, TC; Isbell, SL; Ko, AA US Patent US10308607 (2019)
- Zhang, G; Wang, F; Li, S; Cheng, KW; Zhu, Y; Huo, R; Abdukirim, E; Kang, G; Chou, TF Bioorg Med Chem 62: (2022)
- Novellino, E; Abignente, E; Cosimelli, B; Greco, G; Iadanza, M; Laneri, S; Lavecchia, A; Rimoli, MG; Settimo, FD; Primofiore, G; Tuscano, D; Trincavelli, L; Martini, C J Med Chem 45: 5030-6 (2002)
- Zuccarello, E; Zhang, H; Acquarone, E; Pham, D; Staniszewski, A; Deng, SX; Landry, DW; Arancio, O; Fiorito, J Bioorg Med Chem Lett 92: (2023)
- La Regina, G; Silvestri, R; Gatti, V; Lavecchia, A; Novellino, E; Befani, O; Turini, P; Agostinelli, E Bioorg Med Chem 16: 9729-40 (2008)
- Alonso, D; Vázquez-Villa, H; Gamo, AM; Martínez-Esperón, MF; Tortosa, M; Viso, A; Fernández de la Pradilla, R; Junquera, E; Aicart, E; Martín-Fontecha, M; Benhamú, B; López-Rodríguez, ML; Ortega-Gutiérrez, S ACS Med Chem Lett 1: 249-253 (2010)
- Johansson, A; Hubatsch, I; Akerblom, E; Lindeberg, G; Winiwarter, S; Danielson, UH; Hallberg, A Bioorg Med Chem Lett 11: 203-6 (2001)
- Aktoudianakis, E; Cho, A; Du, Z; Graupe, M; Lad, LT; Machicao Tello, PA; Medley, JW; Metobo, SE; Mukherjee, PK; Naduthambi, D; Parkhill, EQ; Phillips, BW; Simonovich, SP; Squires, NH; Wang, P; Watkins, WJ; Xu, J; Yang, KS; Ziebenhaus, CA US Patent US10899735 (2021)
- Vaz, RJ; Gao, Z; Pribish, J; Chen, X; Levell, J; Davis, L; Albert, E; Brollo, M; Ugolini, A; Cramer, DM; Cairns, J; Sides, K; Liu, F; Kwong, J; Kang, J; Rebello, S; Elliot, M; Lim, H; Chellaraj, V; Singleton, RW; Li, Y Bioorg Med Chem Lett 14: 6053-6 (2004)
- French, JB; Cen, Y; Vrablik, TL; Xu, P; Allen, E; Hanna-Rose, W; Sauve, AA Biochemistry 49: 10421-39 (2010)
- Altmann, E; Aichholz, R; Betschart, C; Buhl, T; Green, J; Irie, O; Teno, N; Lattmann, R; Tintelnot-Blomley, M; Missbach, M J Med Chem 50: 591-4 (2007)
- Selness, SR; Devraj, RV; Monahan, JB; Boehm, TL; Walker, JK; Devadas, B; Durley, RC; Kurumbail, R; Shieh, H; Xing, L; Hepperle, M; Rucker, PV; Jerome, KD; Benson, AG; Marrufo, LD; Madsen, HM; Hitchcock, J; Owen, TJ; Christie, L; Promo, MA; Hickory, BS; Alvira, E; Naing, W; Blevis-Bal, R Bioorg Med Chem Lett 19: 5851-6 (2009)
- Stockwell, SR; Scott, DE; Fischer, G; Guarino, E; Rooney, TPC; Feng, TS; Moschetti, T; Srinivasan, R; Alza, E; Asteian, A; Dagostin, C; Alcaide, A; Rocaboy, M; Blaszczyk, B; Higueruelo, A; Wang, X; Rossmann, M; Perrior, TR; Blundell, TL; Spring, DR; McKenzie, G; Abell, C; Skidmore, J; Venkitaraman, AR; Hyvönen, M J Med Chem 67: 15521-15536
- Intagliata, S; Salerno, L; Ciaffaglione, V; Leonardi, C; Fallica, AN; Carota, G; Amata, E; Marrazzo, A; Pittalà, V; Romeo, G Eur J Med Chem 183: (2019)
- Amato, E; Bankemper, T; Kidney, R; Do, T; Onate, A; Thowfeik, FS; Merino, EJ; Paula, S; Ma, L Bioorg Med Chem 22: 126-34 (2013)
- Bryk, R; Wu, K; Raimundo, BC; Boardman, PE; Chao, P; Conn, GL; Anderson, E; Cole, JL; Duffy, NP; Nathan, C; Griffin, JH Bioorg Med Chem Lett 21: 4108-14 (2011)
- Prezzavento, O; Arena, E; Parenti, C; Pasquinucci, L; Aricò, G; Scoto, GM; Grancara, S; Toninello, A; Ronsisvalle, S J Med Chem 56: 2447-55 (2013)
- Crowe, DM; Aret, E; Gandhi, K; Lelieveld, RH; Sharp, EK; Todd, RS US Patent US11584735 (2023)
- O'Dowd, CR; Helm, MD; Rountree, JSS; Flasz, JT; Arkoudis, E; Miel, H; Hewitt, PR; Jordan, L; Barker, O; Hughes, C; Rozycka, E; Cassidy, E; McClelland, K; Odrzywol, E; Page, N; Feutren-Burton, S; Dvorkin, S; Gavory, G; Harrison, T ACS Med Chem Lett 9: 238-243 (2018)
- Das, K; Bauman, JD; Rim, AS; Dharia, C; Clark, AD; Camarasa, MJ; Balzarini, J; Arnold, E J Med Chem 54: 2727-37 (2011)
- Meegalla, SK; Huang, H; Martin, T; Xu, J; Zhao, S; Liu, J; Hall, M; Gunnet, J; Wang, Y; Rady, B; Silva, J; Otieno, M; Arnoult, E; Paul Lee, S; Pocai, A; Player, MR Bioorg Med Chem Lett 28: 720-726 (2018)
- Heady, L; Fernandez-Serra, M; Mancera, RL; Joyce, S; Venkitaraman, AR; Artacho, E; Skylaris, CK; Ciacchi, LC; Payne, MC J Med Chem 49: 5141-53 (2006)
- Swahn, BM; Xue, Y; Arzel, E; Kallin, E; Magnus, A; Plobeck, N; Viklund, J Bioorg Med Chem Lett 16: 1397-401 (2006)
- Fässler, A; Rösel, J; Grüther, M; Tintelnot-Blomley, M; Atteri, E; Bold, G; Lang, M Bioorg Med Chem Lett 3: 2837-2842 (1993)
- Pascal, Y; Andrianjara, CR; Auclair, E; Avenel, N; Bertin, B; Calvet, A; Féru, F; Lardon, S; Moodley, I; Ouagued, M; Payne, A; Pruniaux, MP; Szilagyi, C Bioorg Med Chem Lett 10: 35-8 (2000)
- Dowling, JE; Vessels, JT; Haque, S; Chang, HX; van Vloten, K; Kumaravel, G; Engber, T; Jin, X; Phadke, D; Wang, J; Ayyub, E; Petter, RC Bioorg Med Chem Lett 15: 4809-13 (2005)
- Pieroni, M; Annunziato, G; Azzali, E; Dessanti, P; Mercurio, C; Meroni, G; Trifiró, P; Vianello, P; Villa, M; Beato, C; Varasi, M; Costantino, G Eur J Med Chem 92: 377-86 (2015)
- Bacher, E; Boer, C; Bray-French, K; Demnitz, FW; Keller, TH; Mazzoni, L; Müller, T; Walker, C Bioorg Med Chem Lett 8: 3229-34 (1999)
- Haidle, AM; Zabierek, AA; Childers, KK; Rosenstein, C; Mathur, A; Altman, MD; Chan, G; Xu, L; Bachman, E; Mo, JR; Bouthillette, M; Rush, T; Tempest, P; Marshall, CG; Young, JR Bioorg Med Chem Lett 24: 1968-73 (2014)
- Balestrieri, E; Pizzimenti, F; Ferlazzo, A; Giofrè, SV; Iannazzo, D; Piperno, A; Romeo, R; Chiacchio, MA; Mastino, A; Macchi, B Bioorg Med Chem 19: 2084-9 (2011)
- Jagtap, PG; Baloglu, E; Southan, GJ; Mabley, JG; Li, H; Zhou, J; van Duzer, J; Salzman, AL; Szabó, C J Med Chem 48: 5100-3 (2005)
- Ma, B; Metrick, CM; Gu, C; Hoemberger, M; Bajrami, B; Bame, E; Huang, J; Mingueneau, M; Murugan, P; Santoro, JC; Tang, H; Wang, T; Hopkins, BT Bioorg Med Chem Lett 60: (2022)
- Banoglu, E; Çelikoglu, E; Völker, S; Olgaç, A; Gerstmeier, J; Garscha, U; Çaliskan, B; Schubert, US; Carotti, A; Macchiarulo, A; Werz, O Eur J Med Chem 113: 1-10 (2016)
- Xiao, J; Free, RB; Barnaeva, E; Conroy, JL; Doyle, T; Miller, B; Bryant-Genevier, M; Taylor, MK; Hu, X; Dulcey, AE; Southall, N; Ferrer, M; Titus, S; Zheng, W; Sibley, DR; Marugan, JJ J Med Chem 57: 3450-63 (2014)
- Bonifazi, A; Del Bello, F; Mammoli, V; Piergentili, A; Petrelli, R; Cimarelli, C; Pellei, M; Schepmann, D; Wünsch, B; Barocelli, E; Bertoni, S; Flammini, L; Amantini, C; Nabissi, M; Santoni, G; Vistoli, G; Quaglia, W J Med Chem 58: 8601-15 (2015)
- Castellano, S; Taliani, S; Viviano, M; Milite, C; Da Pozzo, E; Costa, B; Barresi, E; Bruno, A; Cosconati, S; Marinelli, L; Greco, G; Novellino, E; Sbardella, G; Da Settimo, F; Martini, C J Med Chem 57: 2413-28 (2014)
- Baston, E; Hartmann, RW Bioorg Med Chem Lett 9: 1601-6 (1999)
- Leblond, B; Chauvignac, C; Taverne, T; Beausoleil, E; Casagrande, A; Desire, L; Pando, MP; Donello, JE; Yang, R US Patent US9670181 (2017)
- Basse, N; Papapostolou, D; Pagano, M; Reboud-Ravaux, M; Bernard, E; Felten, AS; Vanderesse, R Bioorg Med Chem Lett 16: 3277-81 (2006)
- Unzue, A; Jessen-Trefzer, C; Spiliotopoulos, D; Gaudio, E; Tarantelli, C; Dong, J; Zhao, H; Pachmayr, J; Zahler, S; Bernasconi, E; Sartori, G; Cascione, L; Bertoni, F; Śledź, P; Caflisch, A; Nevado, C RSC Med Chem 11: 665-675 (2020)
- Plyasova, AA; Berrino, E; Khan, II; Veselovsky, AV; Pokrovsky, VS; Angeli, A; Ferraroni, M; Supuran, CT; Pokrovskaya, MV; Alexandrova, SS; Gladilina, YA; Sokolov, NN; Hilal, A; Carta, F; Zhdanov, DD J Med Chem 64: 11432-11444 (2021)
- Courme, C; Gresh, N; Vidal, M; Lenoir, C; Garbay, C; Florent, JC; Bertounesque, E Eur J Med Chem 45: 244-55 (2010)
- Sakurai, F; Yukawa, T; Kina, A; Murakami, M; Takami, K; Morimoto, S; Seto, M; Kamata, M; Yamashita, T; Nakashima, K; Narita, N; Bettini, E; Ugolini, A; Corsi, M; Hasui, T Bioorg Med Chem 56: (2022)
- Ontoria, JM; Biancofiore, I; Fezzardi, P; Ferrigno, F; Torrente, E; Colarusso, S; Bianchi, E; Andreini, M; Patsilinakos, A; Kempf, G; Augustin, M; Steinbacher, S; Summa, V; Pacifici, R; Muñoz-Sanjuan, I; Park, L; Bresciani, A; Dominguez, C; Sherman, LT; Harper, S ACS Med Chem Lett 11: 740-746 (2020)
- McKeown, SC; Corbett, DF; Goetz, AS; Littleton, TR; Bigham, E; Briscoe, CP; Peat, AJ; Watson, SP; Hickey, DM Bioorg Med Chem Lett 17: 1584-9 (2007)
- Ahmad, S; Madsen, CS; Stein, PD; Janovitz, E; Huang, C; Ngu, K; Bisaha, S; Kennedy, LJ; Chen, BC; Zhao, R; Sitkoff, D; Monshizadegan, H; Yin, X; Ryan, CS; Zhang, R; Giancarli, M; Bird, E; Chang, M; Chen, X; Setters, R; Search, D; Zhuang, S; Nguyen-Tran, V; Cuff, CA; Harrity, T; Darienzo, CJ; Li, T; Reeves, RA; Blanar, MA; Barrish, JC; Zahler, R; Robl, JA J Med Chem 51: 2722-33 (2008)
- Neelamkavil, S; Arison, B; Birzin, E; Feng, JJ; Chen, KH; Lin, A; Cheng, FC; Taylor, L; Thornton, ER; Smith, AB; Hirschmann, R J Med Chem 48: 4025-30 (2005)
- Hügel, HM; de Silva, NH; Siddiqui, A; Blanch, E; Lingham, A Bioorg Med Chem 43: (2021)
- Bokor, E; Docsa, T; Gergely, P; Somsák, L Bioorg Med Chem 18: 1171-80 (2010)
- Riemer, C; Borroni, E; Levet-Trafit, B; Martin, JR; Poli, S; Porter, RH; Bös, M J Med Chem 46: 1273-6 (2003)
- Vaiana, N; Marzahn, M; Parapini, S; Liu, P; Dell'Agli, M; Pancotti, A; Sangiovanni, E; Basilico, N; Bosisio, E; Dunn, BM; Taramelli, D; Romeo, S Bioorg Med Chem Lett 22: 5915-8 (2012)
- Morere, A; Da Silva, A; Bouffard, E; El Cheikh, K; Durand, J; Maynadier, M; Basile, I US Patent US10894803 (2021)
- Pimková Polidarová, M; Břehová, P; Kaiser, MM; Smola, M; Dračínský, M; Smith, J; Marek, A; Dejmek, M; Šála, M; Gutten, O; Rulíšek, L; Novotná, B; Brázdová, A; Janeba, Z; Nencka, R; Boura, E; Páv, O; Birkuš, G J Med Chem 64: 7596-7616 (2021)
- Kettle, JG; Bagal, SK; Barratt, D; Bodnarchuk, MS; Boyd, S; Braybrooke, E; Breed, J; Cassar, DJ; Cosulich, S; Davies, M; Davies, NL; Deng, C; Eatherton, A; Evans, L; Feron, LJ; Fillery, S; Gleave, ES; Goldberg, FW; Cortés González, MA; Guerot, C; Haider, A; Harlfinger, S; Howells, R; Jackson, A; Johnström, P; Kemmitt, PD; Koers, A; Kondrashov, M; Lamont, GM; Lamont, S; Lewis, HJ; Liu, L; Mylrea, M; Nash, S; Niedbala, MJ; Peter, A; Phillips, C; Pike, K; Raubo, P; Robb, GR; Ross, S; Sanders, MG; Schou, M; Simpson, I; Steward, O J Med Chem 66: 9147-9160 (2023)
- Hoffman, A; Qadri, B; Frant, J; Katz, Y; Bhusare, SR; Breuer, E; Hadar, R; Reich, R J Med Chem 51: 1406-14 (2008)
- Traxler, P; Trinks, U; Buchdunger, E; Mett, H; Meyer, T; Müller, M; Regenass, U; Rösel, J; Lydon, N J Med Chem 38: 2441-8 (1995)
- Skalova, T; Hasek, J; Dohnalek, J; Petrokova, H; Buchtelova, E; Duskova, J; Soucek, M; Majer, P; Uhlikova, T; Konvalinka, J J Med Chem 46: 1636-44 (2003)
- Maurin, C; Bailly, F; Buisine, E; Vezin, H; Mbemba, G; Mouscadet, JF; Cotelle, P J Med Chem 47: 5583-6 (2004)
- de Gaetano, M; Butler, E; Gahan, K; Zanetti, A; Marai, M; Chen, J; Cacace, A; Hams, E; Maingot, C; McLoughlin, A; Brennan, E; Leroy, X; Loscher, CE; Fallon, P; Perretti, M; Godson, C; Guiry, PJ Eur J Med Chem 162: 80-108 (2019)
- Ghinet, A; Moise, IM; Rigo, B; Homerin, G; Farce, A; Dubois, J; Bîcu, E Bioorg Med Chem 24: 2307-17 (2016)
- CHAPEAU, E; CHENE, P; FURET, P; KIEFFER, L; MACHAUER, R; PICARD, A; SCHMELZLE, T; SELLNER, H; SOLDERMANN, N; VOEGTLE, M; WARTMANN, M US Patent US20240382600 (2024)
- Garvey, DS; Wasicak, JT; Chung, JY; Shue, YK; Carrera, GM; May, PD; McKinney, MM; Anderson, D; Cadman, E; Vella-Rountree, L J Med Chem 35: 1550-7 (1992)
- Pike, KG; Hunt, TA; Barlaam, B; Benstead, D; Cadogan, E; Chen, K; Cook, CR; Colclough, N; Deng, C; Durant, ST; Eatherton, A; Goldberg, K; Johnström, P; Liu, L; Liu, Z; Nissink, JWM; Pang, C; Pass, M; Robb, GR; Roberts, C; Schou, M; Steward, O; Sykes, A; Yan, Y; Zhai, B; Zheng, L J Med Chem 67: 3090-3111
- Calleri, E; Ceruti, S; Cristalli, G; Martini, C; Temporini, C; Parravicini, C; Volpini, R; Daniele, S; Caccialanza, G; Lecca, D; Lambertucci, C; Trincavelli, ML; Marucci, G; Wainer, IW; Ranghino, G; Fantucci, P; Abbracchio, MP; Massolini, G J Med Chem 53: 3489-501 (2010)
- Costantino, G; Macchiarulo, A; Entrena-Guadix, A; Camaioni, E; Pellicciari, R Bioorg Med Chem Lett 13: 1865-8 (2003)
- Adonias, M; Anayaba, J; Cámara, J; Canet, E; Gateau-Olesker, A; Gero, SD; Grande, M; Hernando, JI Bioorg Med Chem Lett 3: 2547-2552 (1993)
- Colabufo, NA; Contino, M; Cantore, M; Capparelli, E; Perrone, MG; Cassano, G; Gasparre, G; Leopoldo, M; Berardi, F; Perrone, R Bioorg Med Chem 21: 1324-32 (2013)
- Vidaluc, JL; Calmel, F; Bigg, DC; Carilla, E; Briley, M J Med Chem 38: 2969-73 (1995)
- Seward, EM; Carlson, E; Harrison, T; Haworth, KR; Herbert, R; Kelleher, FJ; Kurtz, MM; Moseley, J; Owen, SN; Owens, AP; Sadowski, SJ; Swain, CJ; Williams, BJ Bioorg Med Chem Lett 12: 2515-8 (2002)
- Meyer, EA; Äänismaa, P; Froidevaux, S; Keller, M; Piali, L; Caroff, E J Med Chem 65: 11513-11532 (2022)
- Carosati, E; Mannhold, R; Wahl, P; Hansen, JB; Fremming, T; Zamora, I; Cianchetta, G; Baroni, M J Med Chem 50: 2117-26 (2007)
- Angiolini, M; Banfi, P; Casale, E; Casuscelli, F; Fiorelli, C; Saccardo, MB; Silvagni, M; Zuccotto, F Bioorg Med Chem Lett 20: 4095-9 (2010)
- Di Fabio, R; St-Denis, Y; Sabbatini, FM; Andreotti, D; Arban, R; Bernasconi, G; Braggio, S; Blaney, FE; Capelli, AM; Castiglioni, E; Di Modugno, E; Donati, D; Fazzolari, E; Ratti, E; Feriani, A; Contini, S; Gentile, G; Ghirlanda, D; Provera, S; Marchioro, C; Roberts, KL; Mingardi, A; Mattioli, M; Nalin, A; Pavone, F; Spada, S; Trist, DG; Worby, A J Med Chem 51: 7370-9 (2009)
- Zlotos, DP; Jockers, R; Cecon, E; Rivara, S; Witt-Enderby, PA J Med Chem 57: 3161-85 (2014)
- Cescon, E; Bolcato, G; Federico, S; Bissaro, M; Valentini, A; Ferlin, MG; Spalluto, G; Sturlese, M; Moro, S ACS Med Chem Lett 11: 1168-1174 (2020)
- Ong, HW; Yang, X; Smith, JL; Dickmander, RJ; Brown, JW; Havener, TM; Taft-Benz, S; Howell, S; Sanders, MK; Capener, JL; Couñago, RM; Chang, E; Krämer, A; Moorman, NJ; Heise, M; Axtman, AD; Drewry, DH; Willson, TM J Med Chem 67: 12261-12313
- Wijeratne, EM; Gunaherath, GM; Chapla, VM; Tillotson, J; de la Cruz, F; Kang, M; U'Ren, JM; Araujo, AR; Arnold, AE; Chapman, E; Gunatilaka, AA J Nat Prod 79: 340-52 (2016)
- Richter, HG; Benson, GM; Bleicher, KH; Blum, D; Chaput, E; Clemann, N; Feng, S; Gardes, C; Grether, U; Hartman, P; Kuhn, B; Martin, RE; Plancher, JM; Rudolph, MG; Schuler, F; Taylor, S Bioorg Med Chem Lett 21: 1134-40 (2011)
- Toure, M; Johnson, T; Li, B; Schmidt, R; Ma, H; Neagu, C; Lopez, AU; Wang, Y; Guler, S; Xiao, Y; Henkes, R; Ho, K; Zhang, S; Chu, CL; Gundra, UM; Porichis, F; Li, L; Maurer, CK; Fang, Z; Musil, D; DiPoto, M; Friis, E; Jones, R; Jones, C; Cummings, J; Chekler, E; Tanzer, EM; Huck, B; Sherer, B Bioorg Med Chem 92: (2023)
- Heightman, TD; Callahan, JF; Chiarparin, E; Coyle, JE; Griffiths-Jones, C; Lakdawala, AS; McMenamin, R; Mortenson, PN; Norton, D; Peakman, TM; Rich, SJ; Richardson, C; Rumsey, WL; Sanchez, Y; Saxty, G; Willems, HMG; Wolfe, L; Woolford, AJ; Wu, Z; Yan, H; Kerns, JK; Davies, TG J Med Chem 62: 4683-4702 (2019)
- Chin, E; Kato, D; Link, JO; Shapiro, N; Yang, Z US Patent US11052087 (2021)
- Ananthan, S; Saini, SK; Zhou, G; Hobrath, JV; Padmalayam, I; Zhai, L; Bostwick, JR; Antonio, T; Reith, ME; McDowell, S; Cho, E; McAleer, L; Taylor, M; Luedtke, RR J Med Chem 57: 7042-60 (2014)
- Richardson, BG; Jain, AD; Potteti, HR; Lazzara, PR; David, BP; Tamatam, CR; Choma, E; Skowron, K; Dye, K; Siddiqui, Z; Wang, YT; Krunic, A; Reddy, SP; Moore, TW J Med Chem 61: 8029-8047 (2018)
- Moree, WJ; Goldman, P; Demaggio, AJ; Christenson, E; Herendeen, D; Eksterowicz, J; Kesicki, EA; McElligott, DL; Beaton, G Bioorg Med Chem Lett 18: 5126-9 (2008)
- Christiansen, E; Due-Hansen, ME; Urban, C; Merten, N; Pfleiderer, M; Karlsen, KK; Rasmussen, SS; Steensgaard, M; Hamacher, A; Schmidt, J; Drewke, C; Petersen, RK; Kristiansen, K; Ullrich, S; Kostenis, E; Kassack, MU; Ulven, T ACS Med Chem Lett 1: 345-349 (2010)
- Liessi, N; Cichero, E; Pesce, E; Arkel, M; Salis, A; Tomati, V; Paccagnella, M; Damonte, G; Tasso, B; Galietta, LJV; Pedemonte, N; Fossa, P; Millo, E Eur J Med Chem 144: 179-200 (2018)
- Zhou, C; Tang, C; Chang, E; Ge, M; Lin, S; Cline, E; Tan, CP; Feng, Y; Zhou, YP; Eiermann, GJ; Petrov, A; Salituro, G; Meinke, P; Mosley, R; Akiyama, TE; Einstein, M; Kumar, S; Berger, J; Howard, AD; Thornberry, N; Mills, SG; Yang, L Bioorg Med Chem Lett 20: 1298-301 (2010)
- O' Donovan, DH; Gregson, C; Packer, MJ; Greenwood, R; Pike, KG; Kawatkar, S; Bloecher, A; Robinson, J; Read, J; Code, E; Hsu, JH; Shen, M; Woods, H; Barton, P; Fillery, S; Williamson, B; Rawlins, PB; Bagal, SK Bioorg Med Chem Lett 39: (2021)
- García-Cárceles, J; Decara, JM; Vázquez-Villa, H; Rodríguez, R; Codesido, E; Cruces, J; Brea, J; Loza, MI; Alén, F; Botta, J; McCormick, PJ; Ballesteros, JA; Benhamú, B; Rodríguez de Fonseca, F; López-Rodríguez, ML J Med Chem 60: 9575-9584 (2017)
- Kesteleyn, B; Bardiot, D; Bonfanti, JF; De Boeck, B; Goethals, O; Kaptein, SJF; Stoops, B; Coesemans, E; Fortin, J; Muller, P; Doublet, F; Carlens, G; Koukni, M; Smets, W; Raboisson, P; Chaltin, P; Simmen, K; Van Loock, M; Neyts, J; Marchand, A; Jonckers, THM J Med Chem 66: 8808-8821 (2023)
- González-Bello, C; Rodríguez, D; Pernas, M; Rodríguez, Á; Colchón, E J Med Chem 63: 1859-1881 (2020)
- Fiorino, F; Perissutti, E; Severino, B; Santagada, V; Cirillo, D; Terracciano, S; Massarelli, P; Bruni, G; Collavoli, E; Renner, C; Caliendo, G J Med Chem 48: 5495-503 (2005)
- Wu, J; Rush, TS; Hotchandani, R; Du, X; Geck, M; Collins, E; Xu, ZB; Skotnicki, J; Levin, JI; Lovering, FE Bioorg Med Chem Lett 15: 4105-9 (2005)
- Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333-8353 (2021)
- Crespan, E; Radi, M; Zanoli, S; Schenone, S; Botta, M; Maga, G Bioorg Med Chem 18: 3999-4008 (2010)
- Kokkonda, S; Deng, X; White, KL; El Mazouni, F; White, J; Shackleford, DM; Katneni, K; Chiu, FCK; Barker, H; McLaren, J; Crighton, E; Chen, G; Angulo-Barturen, I; Jimenez-Diaz, MB; Ferrer, S; Huertas-Valentin, L; Martinez-Martinez, MS; Lafuente-Monasterio, MJ; Chittimalla, R; Shahi, SP; Wittlin, S; Waterson, D; Burrows, JN; Matthews, D; Tomchick, D; Rathod, PK; Palmer, MJ; Charman, SA; Phillips, MA J Med Chem 63: 4929-4956 (2020)
- Matthews, JM; Chen, X; Cryan, E; Hlasta, DJ; Rybczynski, PJ; Strauss, K; Tang, Y; Xu, JZ; Yang, M; Zhou, L; Demarest, KT Bioorg Med Chem Lett 17: 6773-8 (2008)
- Guo, C; Hou, X; Dong, L; Marakovits, J; Greasley, S; Dagostino, E; Ferre, R; Johnson, MC; Humphries, PS; Li, H; Paderes, GD; Piraino, J; Kraynov, E; Murray, BW Bioorg Med Chem Lett 24: 4187-91 (2014)
- Leenders, RGG; Brinch, SA; Sowa, ST; Amundsen-Isaksen, E; Galera-Prat, A; Murthy, S; Aertssen, S; Smits, JN; Nieczypor, P; Damen, E; Wegert, A; Nazaré, M; Lehtiö, L; Waaler, J; Krauss, S J Med Chem 64: 17936-17949 (2021)
- Aspnes, GE; Coffey, SB; Darout, E; Dechert-Schmitt, AM; Dullea, RG; Kamlet, AS; Limberakis, C; Londregan, AT; McClure, KF; Menhaji-Klotz, E; Piotrowski, DW; Polivkova, J; Raymer, B; Ruggeri, RB; Salatto, CT; Tu, M; Wei, L; Xiao, J Bioorg Med Chem Lett 92: (2023)
- Rydzik, AM; Kulis, M; Lukaszewicz, M; Kowalska, J; Zuberek, J; Darzynkiewicz, ZM; Darzynkiewicz, E; Jemielity, J Bioorg Med Chem 20: 1699-710 (2012)
- Valenzano, KJ; Miller, W; Chen, Z; Shan, S; Crumley, G; Victory, SF; Davies, E; Huang, JC; Allie, N; Nolan, SJ; Rotshteyn, Y; Kyle, DJ; Broglé, K J Pharmacol Exp Ther 310: 783-92 (2004)
- Reid, PR; Bridges, TM; Sheffler, DJ; Cho, HP; Lewis, LM; Days, E; Daniels, JS; Jones, CK; Niswender, CM; Weaver, CD; Conn, PJ; Lindsley, CW; Wood, MR Bioorg Med Chem Lett 21: 2697-701 (2011)
- Smith, JM; Barlaam, B; Beattie, D; Bradshaw, L; Chan, HM; Chiarparin, E; Collingwood, O; Cooke, SL; Cronin, A; Cumming, I; Dean, E; Debreczeni, JÉ; Del Barco Barrantes, I; Diene, C; Gianni, D; Guerot, C; Guo, X; Guven, S; Hayhow, TG; Hong, T; Kemmitt, PD; Lamont, GM; Lamont, S; Lynch, JT; McWilliams, L; Moore, S; Raubo, P; Robb, GR; Robinson, J; Scott, JS; Srinivasan, B; Steward, O; Stubbs, CJ; Syson, K; Tan, L; Turner, O; Underwood, E; Urosevic, J; Vazquez-Chantada, M; Whittaker, AL; Wilson, DM; Winter-Holt, JJ J Med Chem 67: 13604-13638
- Gandhi, DM; Rosas, R; Greve, E; Kentala, K; D-R Diby, N; Snyder, VA; Stephans, A; Yeung, THW; Subramaniam, S; DiMilo, E; Kurtenbach, KE; Arnold, LA; Weiler, H; Dockendorff, C Bioorg Med Chem 27: 3788-3796 (2019)
- Kenda, BM; Matagne, AC; Talaga, PE; Pasau, PM; Differding, E; Lallemand, BI; Frycia, AM; Moureau, FG; Klitgaard, HV; Gillard, MR; Fuks, B; Michel, P J Med Chem 47: 530-49 (2004)
- Ahmed, MN; Reyna-González, E; Schmid, B; Wiebach, V; Süssmuth, RD; Dittmann, E; Fewer, DP ACS Chem Biol 12: 1538-1546 (2017)
- Palanki, MS; Dneprovskaia, E; Doukas, J; Fine, RM; Hood, J; Kang, X; Lohse, D; Martin, M; Noronha, G; Soll, RM; Wrasidlo, W; Yee, S; Zhu, H J Med Chem 50: 4279-94 (2007)
- Zehnder, L; Bennett, M; Meng, J; Huang, B; Ninkovic, S; Wang, F; Braganza, J; Tatlock, J; Jewell, T; Zhou, JZ; Burke, B; Wang, J; Maegley, K; Mehta, PP; Yin, MJ; Gajiwala, KS; Hickey, MJ; Yamazaki, S; Smith, E; Kang, P; Sistla, A; Dovalsantos, E; Gehring, MR; Kania, R; Wythes, M; Kung, PP J Med Chem 54: 3368-85 (2011)
- Maccari, G; Sanfilippo, S; De Luca, F; Deodato, D; Casian, A; Dasso Lang, MC; Zamperini, C; Dreassi, E; Rossolini, GM; Docquier, JD; Botta, M Bioorg Med Chem Lett 24: 5525-9 (2014)
- Tahtouh, T; Elkins, JM; Filippakopoulos, P; Soundararajan, M; Burgy, G; Durieu, E; Cochet, C; Schmid, RS; Lo, DC; Delhommel, F; Oberholzer, AE; Pearl, LH; Carreaux, F; Bazureau, JP; Knapp, S; Meijer, L J Med Chem 55: 9312-30 (2012)
- Campbell, RM; Cartwright, C; Chen, W; Chen, Y; Duzic, E; Fu, JM; Loveland, M; Manning, R; McKibben, B; Pleiman, CM; Silverman, L; Trueheart, J; Webb, DR; Wilkinson, V; Witter, DJ; Xie, X; Castelhano, AL Bioorg Med Chem Lett 9: 2413-8 (1999)
- J., BM; E., FM; Marie, LH; J., MJ; J., RA; M., SK; J., SS WIPO WO2022115301 (2022)
- Giraud, F; Bourhis, M; Ebrahimi, E; Herfindal, L; Choudhury, RR; Bjørnstad, R; Døskeland, SO; Anizon, F; Moreau, P Bioorg Med Chem 23: 7313-23 (2015)
- Mahboobi, S; Uecker, A; Sellmer, A; Cénac, C; Höcher, H; Pongratz, H; Eichhorn, E; Hufsky, H; Trümpler, A; Sicker, M; Heidel, F; Fischer, T; Stocking, C; Elz, S; Böhmer, FD; Dove, S J Med Chem 49: 3101-15 (2006)
- Elhalem, E; Bellomo, A; Cooke, M; Scravaglieri, A; Pearce, LV; Peach, ML; Gandolfi Donadío, L; Kazanietz, MG; Comin, MJ J Med Chem 64: 11418-11431 (2021)
- Elzein, E; Kalla, RV; Koltun, D; Li, X; Parkhill, EQ; Perry, T; Simonovich, SP; Zablocki, J; Ziebenhaus, CA US Patent US10100058 (2018)
- Ayoup, MS; Barakat, MR; Abdel-Hamid, H; Emam, E; Al-Faiyz, YS; Masoud, AA; Ghareeb, DA; Sonousi, A; Kassab, AE RSC Med Chem 15: 2080-2097
- Lavogina, D; Enkvist, E; Viht, K; Uri, A Chembiochem 15: 443-50 (2014)
- Lefrançois, M; Lefebvre, MR; Saint-Onge, G; Boulais, PE; Lamothe, S; Leduc, R; Lavigne, P; Heveker, N; Escher, E ACS Med Chem Lett 2: 597-602 (2011)
- Ni, M; Esposito, E; Raj, VP; Muzi, L; Zunino, F; Zuco, V; Cominetti, D; Penco, S; Dal Pozzo, A Bioorg Med Chem 23: 6785-93 (2015)
- Sauerberg, P; Larsen, JJ; Falch, E; Krogsgaard-Larsen, P J Med Chem 29: 1004-9 (1986)
- Vidadala, RS; Rivas, KL; Ojo, KK; Hulverson, MA; Zambriski, JA; Bruzual, I; Schultz, TL; Huang, W; Zhang, Z; Scheele, S; DeRocher, AE; Choi, R; Barrett, LK; Siddaramaiah, LK; Hol, WG; Fan, E; Merritt, EA; Parsons, M; Freiberg, G; Marsh, K; Kempf, DJ; Carruthers, VB; Isoherranen, N; Doggett, JS; Van Voorhis, WC; Maly, DJ J Med Chem 59: 6531-46 (2016)
- Burns, CJ; Harte, MF; Bu, X; Fantino, E; Giarrusso, M; Joffe, M; Kurek, M; Legge, FS; Razzino, P; Su, S; Treutlein, H; Wan, SS; Zeng, J; Wilks, AF Bioorg Med Chem Lett 19: 1206-9 (2009)
- Li, K; McGee, LR; Fisher, B; Sudom, A; Liu, J; Rubenstein, SM; Anwer, MK; Cushing, TD; Shin, Y; Ayres, M; Lee, F; Eksterowicz, J; Faulder, P; Waszkowycz, B; Plotnikova, O; Farrelly, E; Xiao, SH; Chen, G; Wang, Z Bioorg Med Chem Lett 23: 1238-44 (2013)
- Di Fabio, R; St-Denis, Y; Sabbatini, FM; Andreotti, D; Arban, R; Bernasconi, G; Braggio, S; Blaney, FE; Capelli, AM; Castiglioni, E; Di Modugno, E; Donati, D; Fazzolari, E; Ratti, E; Feriani, A; Contini, S; Gentile, G; Ghirlanda, D; Provera, S; Marchioro, C; Roberts, KL; Mingardi, A; Mattioli, M; Nalin, A; Pavone, F; Spada, S; Trist, DG; Worby, A J Med Chem 51: 7370-9 (2009)
- McKinnell, RM; Fenster, E; Lam, TM; Palermo, AF US Patent US11339160 (2022)
- Leese, MP; Jourdan, FL; Gaukroger, K; Mahon, MF; Newman, SP; Foster, PA; Stengel, C; Regis-Lydi, S; Ferrandis, E; Di Fiore, A; De Simone, G; Supuran, CT; Purohit, A; Reed, MJ; Potter, BV J Med Chem 51: 1295-308 (2008)
- Gray, N; Zhang, T; Fischer, E; He, Z; Du, G; Donovan, K; Nowak, R; Yuan, JT US Patent US11530219 (2022)
- Lorthiois, E; Breitenstein, W; Cumin, F; Ehrhardt, C; Francotte, E; Jacoby, E; Ostermann, N; Sellner, H; Kosaka, T; Webb, RL; Rigel, DF; Hassiepen, U; Richert, P; Wagner, T; Maibaum, J J Med Chem 56: 2207-17 (2013)
- Kovács, D; Wölfling, J; Szabó, N; Szécsi, M; Kovács, I; Zupkó, I; Frank, E Eur J Med Chem 70: 649-60 (2013)
- Campbell, JC; Henning, P; Franz, E; Sankaran, B; Herberg, FW; Kim, C ACS Chem Biol 12: 2388-2398 (2017)
- Lalonde, JM; Elban, MA; Courter, JR; Sugawara, A; Soeta, T; Madani, N; Princiotto, AM; Kwon, YD; Kwong, PD; Schön, A; Freire, E; Sodroski, J; Smith, AB Bioorg Med Chem 19: 91-101 (2011)
- Toure, M; Johnson, T; Li, B; Schmidt, R; Ma, H; Neagu, C; Lopez, AU; Wang, Y; Guler, S; Xiao, Y; Henkes, R; Ho, K; Zhang, S; Chu, CL; Gundra, UM; Porichis, F; Li, L; Maurer, CK; Fang, Z; Musil, D; DiPoto, M; Friis, E; Jones, R; Jones, C; Cummings, J; Chekler, E; Tanzer, EM; Huck, B; Sherer, B Bioorg Med Chem 92: (2023)
- Berger, DM; Torres, N; Dutia, M; Powell, D; Ciszewski, G; Gopalsamy, A; Levin, JI; Kim, KH; Xu, W; Wilhelm, J; Hu, Y; Collins, K; Feldberg, L; Kim, S; Frommer, E; Wojciechowicz, D; Mallon, R Bioorg Med Chem Lett 19: 6519-23 (2009)
- Chua, K; Fung, E; Micewicz, ED; Ganz, T; Nemeth, E; Ruchala, P Bioorg Med Chem Lett 25: 4961-9 (2015)
- Casiraghi, G; Rassu, G; Auzzas, L; Burreddu, P; Gaetani, E; Battistini, L; Zanardi, F; Curti, C; Nicastro, G; Belvisi, L; Motto, I; Castorina, M; Giannini, G; Pisano, C J Med Chem 48: 7675-87 (2005)
- Malhotra, S; Siu, M; Wang, W; Wei, B; Zhou, A; Chan, BK; Gazzard, LJ; Heffron, T; Lainchbury, M; Madin, A; Seward, EM; Cartwright, MW; Gancia, E; Favor, D; Fong, KC; Good, A; Hu, Y US Patent US20240368170 (2024)
- Scott, JS; Bailey, A; Buttar, D; Carbajo, RJ; Curwen, J; Davey, PRJ; Davies, RDM; Degorce, SL; Donald, C; Gangl, E; Greenwood, R; Groombridge, SD; Johnson, T; Lamont, S; Lawson, M; Lister, A; Morrow, CJ; Moss, TA; Pink, JH; Polanski, R J Med Chem 62: 1593-1608 (2019)
- Carr&aagrovr;, G; Rizzi, A; Guerrini, R; Barnes, TA; McDonald, J; Hebbes, CP; Mela, F; Kenigs, VA; Marzola, G; Rizzi, D; Gavioli, E; Zucchini, S; Regoli, D; Morari, M; Salvadori, S; Rowbotham, DJ; Lambert, DG; Kapusta, DR; Calo', G J Pharmacol Exp Ther 312: 1114-23 (2005)
- Wijtmans, M; Celanire, S; Snip, E; Gillard, MR; Gelens, E; Collart, PP; Venhuis, BJ; Christophe, B; Hulscher, S; van der Goot, H; Lebon, F; Timmerman, H; Bakker, RA; Lallemand, BI; Leurs, R; Talaga, PE; de Esch, IJ J Med Chem 51: 2944-53 (2008)
- Heimburg, T; Kolbinger, FR; Zeyen, P; Ghazy, E; Herp, D; Schmidtkunz, K; Melesina, J; Shaik, TB; Erdmann, F; Schmidt, M; Romier, C; Robaa, D; Witt, O; Oehme, I; Jung, M; Sippl, W J Med Chem 60: 10188-10204 (2017)
- Carzaniga, L; Amari, G; Rizzi, A; Capaldi, C; De Fanti, R; Ghidini, E; Villetti, G; Carnini, C; Moretto, N; Facchinetti, F; Caruso, P; Marchini, G; Battipaglia, L; Patacchini, R; Cenacchi, V; Volta, R; Amadei, F; Pappani, A; Capacchi, S; Bagnacani, V; Delcanale, M; Puccini, P; Catinella, S; Civelli, M; Armani, E J Med Chem 60: 10026-10046 (2017)
- Moss, N; Beaulieu, P; Duceppe, JS; Ferland, JM; Garneau, M; Gauthier, J; Ghiro, E; Goulet, S; Guse, I; Jaramillo, J; Llinas-Brunet, M; Malenfant, E; Plante, R; Poirier, M; Soucy, F; Wernic, D; Yoakim, C; Déziel, R J Med Chem 39: 4173-80 (1996)
- Mohy El Dine, T; Jimmidi, R; Diaconu, A; Fransolet, M; Michiels, C; De Winter, J; Gillon, E; Imberty, A; Coenye, T; Vincent, SP J Med Chem 64: 14728-14744 (2021)
- Pellicciari, R; Costantino, G; Giovagnoni, E; Mattoli, L; Brabet, I; Pin, JP Bioorg Med Chem Lett 8: 1569-74 (1999)
- Tarragó, T; Kichik, N; Claasen, B; Prades, R; Teixidó, M; Giralt, E Bioorg Med Chem 16: 7516-24 (2008)
- Woltering, TJ; Adam, G; Wichmann, J; Goetschi, E; Kew, JN; Knoflach, F; Mutel, V; Gatti, S Bioorg Med Chem Lett 18: 1091-5 (2008)
- Nørholm, AB; Francotte, P; Olsen, L; Krintel, C; Frydenvang, K; Goffin, E; Challal, S; Danober, L; Botez-Pop, I; Lestage, P; Pirotte, B; Kastrup, JS J Med Chem 56: 8736-45 (2013)
- Castanedo, GM; Blaquiere, N; Beresini, M; Bravo, B; Brightbill, H; Chen, J; Cui, HF; Eigenbrot, C; Everett, C; Feng, J; Godemann, R; Gogol, E; Hymowitz, S; Johnson, A; Kayagaki, N; Kohli, PB; Knüppel, K; Kraemer, J; Krüger, S; Loke, P; McEwan, P; Montalbetti, C; Roberts, DA; Smith, M; Steinbacher, S; Sujatha-Bhaskar, S; Takahashi, R; Wang, X; Wu, LC; Zhang, Y; Staben, ST J Med Chem 60: 627-640 (2017)
- Hunt, HJ; Belanoff, JK; Golding, E; Gourdet, B; Phillips, T; Swift, D; Thomas, J; Unitt, JF; Walters, I Bioorg Med Chem Lett 25: 5720-5 (2015)
- Beebe, X; Darczak, D; Henry, RF; Vortherms, T; Janis, R; Namovic, M; Donnelly-Roberts, D; Kage, KL; Surowy, C; Milicic, I; Niforatos, W; Swensen, A; Marsh, KC; Wetter, JM; Franklin, P; Baker, S; Zhong, C; Simler, G; Gomez, E; Boyce-Rustay, JM; Zhu, CZ; Stewart, AO; Jarvis, MF; Scott, VE Bioorg Med Chem 20: 4128-39 (2012)
- Hoyt, SB; London, C; Ok, H; Gonzalez, E; Duffy, JL; Abbadie, C; Dean, B; Felix, JP; Garcia, ML; Jochnowitz, N; Karanam, BV; Li, X; Lyons, KA; McGowan, E; Macintyre, DE; Martin, WJ; Priest, BT; Smith, MM; Tschirret-Guth, R; Warren, VA; Williams, BS; Kaczorowski, GJ; Parsons, WH Bioorg Med Chem Lett 17: 6172-7 (2007)
- Barrish, JC; Gordon, E; Alam, M; Lin, PF; Bisacchi, GS; Chen, P; Cheng, PT; Fritz, AW; Greytok, JA; Hermsmeier, MA J Med Chem 37: 1758-68 (1994)
- Eddie, SL; Gregson, A; Graham, E; Burton, S; Harrison, T; Burden, R; Scott, CJ; Mullan, PB; Williams, R Bioorg Med Chem Lett 29: 1546-1548 (2019)
- Mukhopadhyaya, JK; Kozikowski, AP; Grajkowska, E; Pshenichkin, S; Wroblewski, JT Bioorg Med Chem Lett 11: 1919-24 (2001)
- Laufer, R; Forrest, B; Li, SW; Liu, Y; Sampson, P; Edwards, L; Lang, Y; Awrey, DE; Mao, G; Plotnikova, O; Leung, G; Hodgson, R; Beletskaya, I; Mason, JM; Luo, X; Wei, X; Yao, Y; Feher, M; Ban, F; Kiarash, R; Green, E; Mak, TW; Pan, G; Pauls, HW J Med Chem 56: 6069-87 (2013)
- Estiu, G; Greenberg, E; Harrison, CB; Kwiatkowski, NP; Mazitschek, R; Bradner, JE; Wiest, O J Med Chem 51: 2898-906 (2008)
- Spetea, M; Greiner, E; Aceto, MD; Harris, LS; Coop, A; Schmidhammer, H J Med Chem 48: 5052-5 (2005)
- Feng, Y; Yin, Y; Weiser, A; Griffin, E; Cameron, MD; Lin, L; Ruiz, C; Schürer, SC; Inoue, T; Rao, PV; Schröter, T; Lograsso, P J Med Chem 51: 6642-5 (2008)
- Li, CS; Black, WC; Brideau, C; Chan, CC; Charleson, S; Cromlish, WA; Claveau, D; Gauthier, JY; Gordon, R; Greig, G; Grimm, E; Guay, J; Lau, CK; Riendeau, D; Thérien, M; Visco, DM; Wong, E; Xu, L; Prasit, P Bioorg Med Chem Lett 9: 3181-6 (1999)
- Sergeev, A; Vorobyov, A; Yakubovskaya, M; Kirsanova, O; Gromova, E Bioorg Med Chem Lett 30: (2020)
- Doe, C; Bentley, R; Behm, DJ; Lafferty, R; Stavenger, R; Jung, D; Bamford, M; Panchal, T; Grygielko, E; Wright, LL; Smith, GK; Chen, Z; Webb, C; Khandekar, S; Yi, T; Kirkpatrick, R; Dul, E; Jolivette, L; Marino, JP; Willette, R; Lee, D; Hu, E J Pharmacol Exp Ther 320: 89-98 (2006)
- Stockwell, SR; Scott, DE; Fischer, G; Guarino, E; Rooney, TPC; Feng, TS; Moschetti, T; Srinivasan, R; Alza, E; Asteian, A; Dagostin, C; Alcaide, A; Rocaboy, M; Blaszczyk, B; Higueruelo, A; Wang, X; Rossmann, M; Perrior, TR; Blundell, TL; Spring, DR; McKenzie, G; Abell, C; Skidmore, J; Venkitaraman, AR; Hyvönen, M J Med Chem 67: 15521-15536
- Mougenot, P; Namane, C; Fett, E; Goumy, F; Dadji-Faïhun, R; Langot, G; Monseau, C; Onofri, B; Pacquet, F; Pascal, C; Crespin, O; Ben-Hassine, M; Ragot, JL; Van-Pham, T; Philippo, C; Chatelain-Egger, F; Péron, P; Le Bail, JC; Guillot, E; Chamiot-Clerc, P; Chabanaud, MA; Pruniaux, MP; Ménegotto, J; Schmidt, F; Venier, O; Viviani, F; Nicolai, E Bioorg Med Chem Lett 26: 25-32 (2016)
- Chappie, TA; Abdelmessih, M; Ambroise, CW; Boehm, M; Cai, M; Green, M; Guilmette, E; Steppan, CM; Stevens, LM; Wei, L; Xi, S; Hasson, SA ACS Med Chem Lett 13: 55-62 (2022)
- Sandham, DA; Arnold, N; Aschauer, H; Bala, K; Barker, L; Brown, L; Brown, Z; Budd, D; Cox, B; Docx, C; Dubois, G; Duggan, N; England, K; Everatt, B; Furegati, M; Hall, E; Kalthoff, F; King, A; Leblanc, CJ; Manini, J; Meingassner, J; Profit, R; Schmidt, A; Simmons, J; Sohal, B; Stringer, R; Thomas, M; Turner, KL; Walker, C; Watson, SJ; Westwick, J; Willis, J; Williams, G; Wilson, C Bioorg Med Chem 21: 6582-91 (2013)
- Kong, Y; Grembecka, J; Edler, MC; Hamel, E; Mooberry, SL; Sabat, M; Rieger, J; Brown, ML Chem Biol 12: 1007-14 (2005)
- de Gaetano, M; Butler, E; Gahan, K; Zanetti, A; Marai, M; Chen, J; Cacace, A; Hams, E; Maingot, C; McLoughlin, A; Brennan, E; Leroy, X; Loscher, CE; Fallon, P; Perretti, M; Godson, C; Guiry, PJ Eur J Med Chem 162: 80-108 (2019)
- Greenbaum, DC; Mackey, Z; Hansell, E; Doyle, P; Gut, J; Caffrey, CR; Lehrman, J; Rosenthal, PJ; McKerrow, JH; Chibale, K J Med Chem 47: 3212-9 (2004)
- Schühly, W; Hüfner, A; Pferschy-Wenzig, EM; Prettner, E; Adams, M; Bodensieck, A; Kunert, O; Oluwemimo, A; Haslinger, E; Bauer, R Bioorg Med Chem 17: 4459-65 (2009)
- Kapková, P; Heller, E; Unger, M; Folkers, G; Holzgrabe, U J Med Chem 48: 7496-9 (2005)
- Beard, RL; Chandraratna, RA; Colon, DF; Gillett, SJ; Henry, E; Marler, DK; Song, T; Denys, L; Garst, ME; Arefieg, T J Med Chem 38: 2820-9 (1995)
- Neochoritis, CG; Wang, K; Estrada-Ortiz, N; Herdtweck, E; Kubica, K; Twarda, A; Zak, KM; Holak, TA; Dömling, A Bioorg Med Chem Lett 25: 5661-6 (2015)
- Thoma, G; Nuninger, F; Falchetto, R; Hermes, E; Tavares, GA; Vangrevelinghe, E; Zerwes, HG J Med Chem 54: 284-8 (2011)
- Vlaar, CP; Castillo-Pichardo, L; Medina, JI; Marrero-Serra, CM; Vélez, E; Ramos, Z; Hernández, E Bioorg Med Chem 26: 884-890 (2018)
- Regan, J; Capolino, A; Cirillo, PF; Gilmore, T; Graham, AG; Hickey, E; Kroe, RR; Madwed, J; Moriak, M; Nelson, R; Pargellis, CA; Swinamer, A; Torcellini, C; Tsang, M; Moss, N J Med Chem 46: 4676-86 (2003)
- Uenohara, Y; Tsumura, S; Hirayama, S; Higashi, E; Watanabe, Y; Gouda, H; Nagase, H; Fujii, H Bioorg Med Chem 53: (2022)
- Kochanny, MJ; Adler, M; Ewing, J; Griedel, BD; Ho, E; Karanjawala, R; Lee, W; Lentz, D; Liang, AM; Morrissey, MM; Phillips, GB; Post, J; Sacchi, KL; Sakata, ST; Subramanyam, B; Vergona, R; Walters, J; White, KA; Whitlow, M; Ye, B; Zhao, Z; Shaw, KJ Bioorg Med Chem 15: 2127-46 (2007)
- Martinez Botella, G; Salituro, FG; Harrison, BL; Beresis, RT; Bai, Z; Blanco, MJ; Belfort, GM; Dai, J; Loya, CM; Ackley, MA; Althaus, AL; Grossman, SJ; Hoffmann, E; Doherty, JJ; Robichaud, AJ J Med Chem 60: 7810-7819 (2017)
- Geitmann, M; Retra, K; de Kloe, GE; Homan, E; Smit, AB; de Esch, IJ; Danielson, UH Biochemistry 49: 8143-54 (2010)
- Young, RJ; Adams, C; Blows, M; Brown, D; Burns-Kurtis, CL; Chan, C; Chaudry, L; Convery, MA; Davies, DE; Exall, AM; Foster, G; Harling, JD; Hortense, E; Irvine, S; Irving, WR; Jackson, S; Kleanthous, S; Pateman, AJ; Patikis, AN; Roethka, TJ; Senger, S; Stelman, GJ; Toomey, JR; West, RI; Whittaker, C; Zhou, P; Watson, NS Bioorg Med Chem Lett 21: 1582-7 (2011)
- Tang, H; Jensen, K; Houang, E; McRobb, FM; Bhat, S; Svensson, M; Bochevarov, A; Day, T; Dahlgren, MK; Bell, JA; Frye, L; Skene, RJ; Lewis, JH; Osborne, JD; Tierney, JP; Gordon, JA; Palomero, MA; Gallati, C; Chapman, RSL; Jones, DR; Hirst, KL; Sephton, M; Chauhan, A; Sharpe, A; Tardia, P; Dechaux, EA; Taylor, A; Waddell, RD; Valentine, A; Janssens, HB; Aziz, O; Bloomfield, DE; Ladha, S; Fraser, IJ; Ellard, JM J Med Chem 65: 6775-6802 (2022)
- Rzasa, RM; Hu, E; Rumfelt, S; Chen, N; Andrews, KL; Chmait, S; Falsey, JR; Zhong, W; Jones, AD; Porter, A; Louie, SW; Zhao, X; Treanor, JJ; Allen, JR Bioorg Med Chem Lett 22: 7371-5 (2012)
- Lopez-Tapia, F; Brotherton-Pleiss, C; Yue, P; Murakami, H; Costa Araujo, AC; Reis Dos Santos, B; Ichinotsubo, E; Rabkin, A; Shah, R; Lantz, M; Chen, S; Tius, MA; Turkson, J ACS Med Chem Lett 9: 250-255 (2018)
- Zakharova, O; Luzina, O; Zakharenko, A; Sokolov, D; Filimonov, A; Dyrkheeva, N; Chepanova, A; Ilina, E; Ilyina, A; Klabenkova, K; Chelobanov, B; Stetsenko, D; Zafar, A; Eurtivong, C; Reynisson, J; Volcho, K; Salakhutdinov, N; Lavrik, O Bioorg Med Chem 26: 4470-4480 (2018)
- Czudor, Z; Balogh, M; Bánhegyi, P; Boros, S; Breza, N; Dobos, J; Fábián, M; Horváth, Z; Illyés, E; Markó, P; Sipos, A; Szántai-Kis, C; Szokol, B; Őrfi, L Bioorg Med Chem Lett 28: 769-773 (2018)
- Imanishi, M; Tomishima, Y; Itou, S; Hamashima, H; Nakajima, Y; Washizuka, K; Sakurai, M; Matsui, S; Imamura, E; Ueshima, K; Yamamoto, T; Yamamoto, N; Ishikawa, H; Nakano, K; Unami, N; Hamada, K; Matsumura, Y; Takamura, F; Hattori, K J Med Chem 51: 1925-44 (2008)
- Isabel, E; Bateman, KP; Chauret, N; Cromlish, W; Desmarais, S; Duong, le T; Falgueyret, JP; Gauthier, JY; Lamontagne, S; Lau, CK; Léger, S; LeRiche, T; Lévesque, JF; Li, CS; Massé, F; McKay, DJ; Mellon, C; Nicoll-Griffith, DA; Oballa, RM; Percival, MD; Riendeau, D; Robichaud, J; Rodan, GA; Rodan, SB; Seto, C; Thérien, M; Truong, VL; Wesolowski, G; Young, RN; Zamboni, R; Black, WC Bioorg Med Chem Lett 20: 887-92 (2010)
- Bengtsson, C; Blaho, S; Saitton, DB; Brickmann, K; Broddefalk, J; Davidsson, O; Drmota, T; Folmer, R; Hallberg, K; Hallén, S; Hovland, R; Isin, E; Johannesson, P; Kull, B; Larsson, LO; Löfgren, L; Nilsson, KE; Noeske, T; Oakes, N; Plowright, AT; Schnecke, V; Ståhlberg, P; Sörme, P; Wan, H; Wellner, E; Oster, L Bioorg Med Chem 19: 3039-53 (2011)
- Lorthiois, E; Breitenstein, W; Cumin, F; Ehrhardt, C; Francotte, E; Jacoby, E; Ostermann, N; Sellner, H; Kosaka, T; Webb, RL; Rigel, DF; Hassiepen, U; Richert, P; Wagner, T; Maibaum, J J Med Chem 56: 2207-17 (2013)
- Madhav, H; Jameel, E; Rehan, M; Hoda, N RSC Med Chem 13: 258-279 (2022)
- Jecs, E; Tahirovic, YA; Wilson, RJ; Miller, EJ; Kim, M; Truax, V; Nguyen, HH; Akins, NS; Saindane, M; Wang, T; Sum, CS; Cvijic, ME; Schroeder, GM; Burton, SL; Derdeyn, CA; Xu, L; Jiang, Y; Wilson, LJ; Liotta, DC J Med Chem 65: 4058-4084 (2022)
- Guibbal, F; Bénard, S; Patché, J; Meneyrol, V; Couprie, J; Yong-Sang, J; Meilhac, O; Jestin, E Bioorg Med Chem Lett 28: 787-792 (2018)
- Harris, PA; Faucher, N; George, N; Eidam, PM; King, BW; White, GV; Anderson, NA; Bandyopadhyay, D; Beal, AM; Beneton, V; Berger, SB; Campobasso, N; Campos, S; Capriotti, CA; Cox, JA; Daugan, A; Donche, F; Fouchet, MH; Finger, JN; Geddes, B; Gough, PJ; Grondin, P; Hoffman, BL; Hoffman, SJ; Hutchinson, SE; Jeong, JU; Jigorel, E; Lamoureux, P; Leister, LK; Lich, JD; Mahajan, MK; Meslamani, J; Mosley, JE; Nagilla, R; Nassau, PM; Ng, SL; Ouellette, MT; Pasikanti, KK; Potvain, F; Reilly, MA; Rivera, EJ; Sautet, S; Schaeffer, MC; Sehon, CA; Sun, H; Thorpe, JH; Totoritis, RD; Ward, P; Wellaway, N; Wisnoski, DD; Woolven, JM; Bertin, J; Marquis, RW J Med Chem 62: 5096-5110 (2019)
- Pettersson, I; Ebdrup, S; Havranek, M; Pihera, P; Korínek, M; Mogensen, JP; Jeppesen, CB; Johansson, E; Sauerberg, P Bioorg Med Chem Lett 17: 4625-9 (2007)
- Tao, ZF; Wang, L; Stewart, KD; Chen, Z; Gu, W; Bui, MH; Merta, P; Zhang, H; Kovar, P; Johnson, E; Park, C; Judge, R; Rosenberg, S; Sowin, T; Lin, NH J Med Chem 50: 1514-27 (2007)
- Garton, NS; Barker, MD; Davis, RP; Douault, C; Hooper-Greenhill, E; Jones, E; Lewis, HD; Liddle, J; Lugo, D; McCleary, S; Preston, AGS; Ramirez-Molina, C; Neu, M; Shipley, TJ; Somers, DO; Watson, RJ; Wilson, DM Bioorg Med Chem Lett 26: 4606-4612 (2016)
- Preuss, J; Maloney, P; Peddibhotla, S; Hedrick, MP; Hershberger, P; Gosalia, P; Milewski, M; Li, YL; Sugarman, E; Hood, B; Suyama, E; Nguyen, K; Vasile, S; Sergienko, E; Mangravita-Novo, A; Vicchiarelli, M; McAnally, D; Smith, LH; Roth, GP; Diwan, J; Chung, TD; Jortzik, E; Rahlfs, S; Becker, K; Pinkerton, AB; Bode, L J Med Chem 55: 7262-72 (2012)
- Vázquez-Villa, H; González-Vera, JA; Benhamú, B; Viso, A; Fernández de la Pradilla, R; Junquera, E; Aicart, E; López-Rodríguez, ML; Ortega-Gutiérrez, S J Med Chem 53: 7095-106 (2010)
- Swahn, BM; Xue, Y; Arzel, E; Kallin, E; Magnus, A; Plobeck, N; Viklund, J Bioorg Med Chem Lett 16: 1397-401 (2006)
- Joubert, J; Kapp, E Bioorg Med Chem Lett 30: (2020)
- Hamilton, G; Bednar, D; Borosky, S; Huang, Z; Zubrowski, R; Ferkany, J; Karbon, E Bioorg Med Chem Lett 4: 2035-2040 (1994)
- Nomura, S; Sakamaki, S; Hongu, M; Kawanishi, E; Koga, Y; Sakamoto, T; Yamamoto, Y; Ueta, K; Kimata, H; Nakayama, K; Tsuda-Tsukimoto, M J Med Chem 53: 6355-60 (2010)
- Lane, T; Makarov, V; Nelson, JAE; Meeker, RB; Sanna, G; Riabova, O; Kazakova, E; Monakhova, N; Tsedilin, A; Urbina, F; Jones, T; Suchy, A; Ekins, S J Med Chem 66: 6193-6217 (2023)
- Borsari, C; Rageot, D; Beaufils, F; Bohnacker, T; Keles, E; Buslov, I; Melone, A; Sele, AM; Hebeisen, P; Fabbro, D; Hillmann, P; Wymann, MP ACS Med Chem Lett 10: 1473-1479 (2019)
- Ali, SM; Ashwell, MA; Kelleher, E; Koerner, S; Lapierre, J; Link, JS; Liu, Y; Moussa, M; Palma, R; Tandon, M; Vensel, D; Westlund, N; Wu, H; Yang, R US Patent US8541407 (2013)
- Muller-Steffner, H; Jacques, SA; Kuhn, I; Schultz, MD; Botta, D; Osswald, P; Maechling, C; Lund, FE; Kellenberger, E ACS Chem Biol 12: 1787-1795 (2017)
- Lowe, JD; Sanderson, HS; Cooke, AE; Ostovar, M; Tsisanova, E; Withey, SL; Chavkin, C; Husbands, SM; Kelly, E; Henderson, G; Bailey, CP Mol Pharmacol 88: 347-56
- Kim, C; Ann, J; Lee, S; Kim, E; Choi, S; Blumberg, PM; Frank-Foltyn, R; Bahrenberg, G; Stockhausen, H; Christoph, T; Lee, J Bioorg Med Chem 26: 4509-4517 (2018)
- Furber, M; Alcaraz, L; Luckhurst, C; Bahl, A; Beaton, H; Bowers, K; Collington, J; Denton, R; Donald, D; Kinchin, E; MacDonald, C; Rigby, A; Riley, R; Soars, M; Springthorpe, B; Webborn, P Bioorg Med Chem Lett 22: 7707-10 (2012)
- Kankanala, J; Ribeiro, CJA; Kiselev, E; Ravji, A; Williams, J; Xie, J; Aihara, H; Pommier, Y; Wang, Z J Med Chem 62: 4669-4682 (2019)
- Hebeisen, P; Kuhn, B; Kohler, P; Gubler, M; Huber, W; Kitas, E; Schott, B; Benz, J; Joseph, C; Ruf, A Bioorg Med Chem Lett 18: 4708-12 (2008)
- Carvalho, JF; Louvel, J; Doornbos, ML; Klaasse, E; Yu, Z; Brussee, J; IJzerman, AP J Med Chem 56: 2828-40 (2013)
- Tamamura, H; Omagari, A; Hiramatsu, K; Gotoh, K; Kanamoto, T; Xu, Y; Kodama, E; Matsuoka, M; Hattori, T; Yamamoto, N; Nakashima, H; Otaka, A; Fujii, N Bioorg Med Chem Lett 11: 1897-902 (2001)
- Blöcher, R; Lamers, C; Wittmann, SK; Merk, D; Hartmann, M; Weizel, L; Diehl, O; Brüggerhoff, A; Boß, M; Kaiser, A; Schader, T; Göbel, T; Grundmann, M; Angioni, C; Heering, J; Geisslinger, G; Wurglics, M; Kostenis, E; Brüne, B; Steinhilber, D; Schubert-Zsilavecz, M; Kahnt, AS; Proschak, E J Med Chem 59: 61-81 (2016)
- Kotsampasakou, E; Demopoulos, VJ Bioorg Med Chem 21: 869-73 (2013)
- Meza-Aviña, ME; Lingerfelt, MA; Console-Bram, LM; Gamage, TF; Sharir, H; Gettys, KE; Hurst, DP; Kotsikorou, E; Shore, DM; Caron, MG; Rao, N; Barak, LS; Abood, ME; Reggio, PH; Croatt, MP Bioorg Med Chem Lett 26: 1827-30 (2016)
- Zhang, P; Terefenko, EA; McComas, CC; Mahaney, PE; Vu, A; Trybulski, E; Koury, E; Johnston, G; Bray, J; Deecher, D Bioorg Med Chem Lett 18: 6067-70 (2008)
- Ahmad, W; Kumolosasi, E; Jantan, I; Bukhari, SN; Jasamai, M Chem Biol Drug Des 83: 670-81 (2014)
- Grebien, F; Vedadi, M; Getlik, M; Giambruno, R; Grover, A; Avellino, R; Skucha, A; Vittori, S; Kuznetsova, E; Smil, D; Barsyte-Lovejoy, D; Li, F; Poda, G; Schapira, M; Wu, H; Dong, A; Senisterra, G; Stukalov, A; Huber, KVM; Schönegger, A; Marcellus, R; Bilban, M; Bock, C; Brown, PJ; Zuber, J; Bennett, KL; Al-Awar, R; Delwel, R; Nerlov, C; Arrowsmith, CH; Superti-Furga, G Nat Chem Biol 11: 571-578
- Hsu, N; Cai, D; Damodaran, K; Gomez, RF; Keck, JG; Laborde, E; Lum, RT; Macke, TJ; Martin, G; Schow, SR; Simon, RJ; Villar, HO; Wick, MM; Beroza, P J Med Chem 47: 4875-80 (2004)
- Abate, C; Niso, M; Lacivita, E; Mosier, PD; Toscano, A; Perrone, R J Med Chem 54: 1022-32 (2011)
- Landagaray, E; Ettaoussi, M; Duroux, R; Boutin, JA; Caignard, DH; Delagrange, P; Melnyk, P; Berthelot, P; Yous, S Eur J Med Chem 109: 360-70 (2016)
- Eckhardt, M; Frattini, S; Langkopf, E; Wagner, H US Patent US9597310 (2017)
- Steffan, RJ; Ashwell, MA; Solvibile, WR; Matelan, E; Largis, E; Han, S; Tillet, J; Mulvey, R Bioorg Med Chem Lett 12: 2957-61 (2002)
- el Ahmad, Y; Laurent, E; Maillet, P; Talab, A; Teste, JF; Dokhan, R; Tran, G; Ollivier, R J Med Chem 40: 952-60 (1997)
- Zampieri, D; Laurini, E; Vio, L; Fermeglia, M; Pricl, S; Wünsch, B; Schepmann, D; Mamolo, MG Eur J Med Chem 90: 797-808 (2015)
- Carabet, LA; Lallous, N; Leblanc, E; Ban, F; Morin, H; Lawn, S; Ghaidi, F; Lee, J; Mills, IG; Gleave, ME; Rennie, PS; Cherkasov, A Eur J Med Chem 160: 108-119 (2018)
- Zhang, Y; Fu-Yang, Lin; Li, K; Zhu, W; Liu, YL; Cao, R; Pang, R; Lee, E; Axelson, J; Hensler, M; Wang, K; Molohon, KJ; Wang, Y; Mitchell, DA; Nizet, V; Oldfield, E ACS Med Chem Lett 3: 402-406 (2012)
- Paruch, K; Dwyer, MP; Alvarez, C; Brown, C; Chan, TY; Doll, RJ; Keertikar, K; Knutson, C; McKittrick, B; Rivera, J; Rossman, R; Tucker, G; Fischmann, TO; Hruza, A; Madison, V; Nomeir, AA; Wang, Y; Lees, E; Parry, D; Sgambellone, N; Seghezzi, W; Schultz, L; Shanahan, F; Wiswell, D; Xu, X; Zhou, Q; James, RA; Paradkar, VM; Park, H; Rokosz, LR; Stauffer, TM; Guzi, TJ Bioorg Med Chem Lett 17: 6220-3 (2007)
- Decaris, M; Turner, S; Lefebvre, E US Patent US11419869 (2022)
- Bitha, P; Li, Z; Francisco, GD; Yang, Y; Petersen, PJ; Lenoy, E; Lin, YI Bioorg Med Chem Lett 9: 997-1002 (1999)
- Petrocchi, A; Leo, E; Reyna, NJ; Hamilton, MM; Shi, X; Parker, CA; Mseeh, F; Bardenhagen, JP; Leonard, P; Cross, JB; Huang, S; Jiang, Y; Cardozo, M; Draetta, G; Marszalek, JR; Toniatti, C; Jones, P; Lewis, RT Bioorg Med Chem Lett 26: 1503-7 (2016)
- Kögler, M; Vanderhoydonck, B; De Jonghe, S; Rozenski, J; Van Belle, K; Herman, J; Louat, T; Parchina, A; Sibley, C; Lescrinier, E; Herdewijn, P J Med Chem 54: 4847-62 (2011)
- Moorjani, M; Zhang, X; Chen, Y; Lin, E; Rueter, JK; Gross, RS; Lanier, MC; Tellew, JE; Williams, JP; Lechner, SM; Malany, S; Santos, M; Ekhlassi, P; Castro-Palomino, JC; Crespo, MI; Prat, M; Gual, S; Díaz, JL; Saunders, J; Slee, DH Bioorg Med Chem Lett 18: 1269-73 (2008)
- Olsson, RI; Jacobson, I; Boström, J; Fex, T; Björe, A; Olsson, C; Sundell, J; Gran, U; Öhrn, A; Nordin, A; Gyll, J; Thorstensson, M; Hayen, A; Aplander, K; Hidestål, O; Jiang, F; Linhardt, G; Forsström, E; Collins, T; Sundqvist, M; Lindhardt, E; Åstrand, A; Löfberg, B Bioorg Med Chem Lett 23: 706-10 (2013)
- Lorthiois, E; Breitenstein, W; Cumin, F; Ehrhardt, C; Francotte, E; Jacoby, E; Ostermann, N; Sellner, H; Kosaka, T; Webb, RL; Rigel, DF; Hassiepen, U; Richert, P; Wagner, T; Maibaum, J J Med Chem 56: 2207-17 (2013)
- Papillon, JPN; Nakajima, K; Adair, CD; Hempel, J; Jouk, AO; Karki, RG; Mathieu, S; Möbitz, H; Ntaganda, R; Smith, T; Visser, M; Hill, SE; Hurtado, FK; Chenail, G; Bhang, HC; Bric, A; Xiang, K; Bushold, G; Gilbert, T; Vattay, A; Dooley, J; Costa, EA; Park, I; Li, A; Farley, D; Lounkine, E; Yue, QK; Xie, X; Zhu, X; Kulathila, R; King, D; Hu, T; Vulic, K; Cantwell, J; Luu, C; Jagani, Z J Med Chem 61: 10155-10172 (2018)
- Akgül, Ö; Lucarini, E; Mannelli, LDC; Ghelardini, C; D'Ambrosio, K; Buonanno, M; Monti, SM; De Simone, G; Angeli, A; Supuran, CT; Carta, F Eur J Med Chem 227: (2022)
- Wiles, JA; Song, Y; Wang, Q; Lucien, E; Hashimoto, A; Cheng, J; Marlor, CW; Ou, Y; Podos, SD; Thanassi, JA; Thoma, CL; Deshpande, M; Pucci, MJ; Bradbury, BJ Bioorg Med Chem Lett 16: 1277-81 (2006)
- Bianco, G; Meleddu, R; Distinto, S; Cottiglia, F; Gaspari, M; Melis, C; Corona, A; Angius, R; Angeli, A; Taverna, D; Alcaro, S; Leitans, J; Kazaks, A; Tars, K; Supuran, CT; Maccioni, E ACS Med Chem Lett 8: 792-796 (2017)
- Pelish, HE; Peterson, JR; Salvarezza, SB; Rodriguez-Boulan, E; Chen, JL; Stamnes, M; Macia, E; Feng, Y; Shair, MD; Kirchhausen, T Nat Chem Biol 2: 39-46 (2006)
- Valant, C; Maillet, E; Bourguignon, JJ; Bucher, B; Utard, V; Galzi, JL; Hibert, M J Med Chem 52: 5999-6011 (2009)
- Fader, LD; Malenfant, E; Parisien, M; Carson, R; Bilodeau, F; Landry, S; Pesant, M; Brochu, C; Morin, S; Chabot, C; Halmos, T; Bousquet, Y; Bailey, MD; Kawai, SH; Coulombe, R; LaPlante, S; Jakalian, A; Bhardwaj, PK; Wernic, D; Schroeder, P; Amad, M; Edwards, P; Garneau, M; Duan, J; Cordingley, M; Bethell, R; Mason, SW; Bös, M; Bonneau, P; Poupart, MA; Faucher, AM; Simoneau, B; Fenwick, C; Yoakim, C; Tsantrizos, Y ACS Med Chem Lett 5: 422-7 (2014)
- Lesuisse, D; Deprez, P; Albert, E; Duc, TT; Sortais, B; Gofflo, D; Jean-Baptiste, V; Marquette, J; Schoot, B; Sarubbi, E; Lange, G; Broto, P; Mandine, E Bioorg Med Chem Lett 11: 2127-31 (2001)
- Palani, A; Nawrocki, AR; Orvieto, F; Bianchi, E; Mandić, E; Pessi, A; Huang, C; Deng, Q; Toussaint, N; Walsh, E; Reddy, V; Ashley, E; He, H; Mumick, S; Hawes, B; Marsh, D; Erion, M; Nargund, R; Carrington, PE ACS Med Chem Lett 13: 1248-1254 (2022)
- Li, M; Konteatis, Z; Nagaraja, N; Chen, Y; Zhou, S; Ma, G; Gross, S; Marjon, K; Hyer, ML; Mandley, E; Lein, M; Padyana, AK; Jin, L; Tong, S; Peters, R; Murtie, J; Travins, J; Medeiros, M; Liu, P; Frank, V; Judd, ET; Biller, SA; Marks, KM; Sui, Z; Reznik, SK J Med Chem 65: 4600-4615 (2022)
- Bigioni, M; Ettorre, A; Felicetti, P; Mauro, S; Rossi, C; Maggi, CA; Marastoni, E; Binaschi, M; Parlani, M; Fattori, D Bioorg Med Chem Lett 22: 5360-2 (2012)
- Serrán-Aguilera, L; Mariotto, E; Rubbini, G; Castro Navas, FF; Marco, C; Carrasco-Jiménez, MP; Ballarotto, M; Macchiarulo, A; Hurtado-Guerrero, R; Viola, G; Lopez-Cara, LC Eur J Med Chem 207: (2020)
- Verhoest, PR; Proulx-Lafrance, C; Corman, M; Chenard, L; Helal, CJ; Hou, X; Kleiman, R; Liu, S; Marr, E; Menniti, FS; Schmidt, CJ; Vanase-Frawley, M; Schmidt, AW; Williams, RD; Nelson, FR; Fonseca, KR; Liras, S J Med Chem 52: 7946-9 (2009)
- Marsault, E; Peterson, ML J Med Chem 54: 1961-2004 (2011)
- Côté, B; Boulet, L; Brideau, C; Claveau, D; Ethier, D; Frenette, R; Gagnon, M; Giroux, A; Guay, J; Guiral, S; Mancini, J; Martins, E; Massé, F; Méthot, N; Riendeau, D; Rubin, J; Xu, D; Yu, H; Ducharme, Y; Friesen, RW Bioorg Med Chem Lett 17: 6816-20 (2008)
- Albanese, V; Ruzza, C; Marzola, E; Bernardi, T; Fabbri, M; Fantinati, A; Trapella, C; Reinscheid, RK; Ferrari, F; Sturaro, C; Calò, G; Amendola, G; Cosconati, S; Pacifico, S; Guerrini, R; Preti, D J Med Chem 64: 4089-4108 (2021)
- Nocentini, A; Ferraroni, M; Carta, F; Ceruso, M; Gratteri, P; Lanzi, C; Masini, E; Supuran, CT J Med Chem 59: 10692-10704 (2016)
- Schroeder, B; Demirel, P; Fischer, C; Masri, E; Kallis, S; Redl, L; Rudolf, T; Bergemann, S; Arkona, C; Nitsche, C; Bartenschlager, R; Rademann, J ACS Med Chem Lett 12: 1955-1961 (2021)
- Bhamidipati, S; Shaw, S; Darwish, I; Yu, J; Kolluri, R; Taylor, V; Masuda, E; Irving, M US Patent US11667643 (2023)
- Steffan, RJ; Ashwell, MA; Solvibile, WR; Matelan, E; Largis, E; Han, S; Tillet, J; Mulvey, R Bioorg Med Chem Lett 12: 2963-7 (2002)
- Andrés, JI; Alonso, JM; Díaz, A; Fernández, J; Iturrino, L; Martínez, P; Matesanz, E; Freyne, EJ; Deroose, F; Boeckx, G; Petit, D; Diels, G; Megens, A; Somers, M; Van Wauwe, J; Stoppie, P; Cools, M; De Clerck, F; Peeters, D; de Chaffoy, D Bioorg Med Chem Lett 12: 653-8 (2002)
- Ueno, T; Matsuoka, E; Asada, N; Yamamoto, S; Kanegawa, N; Ito, M; Ito, H; Moechars, D; Rombouts, FJR; Gijsen, HJM; Kusakabe, KI J Med Chem 64: 14165-14174 (2021)
- Romagnoli, R; Prencipe, F; Oliva, P; Baraldi, S; Baraldi, PG; Schiaffino Ortega, S; Chayah, M; Kimatrai Salvador, M; Lopez-Cara, LC; Brancale, A; Ferla, S; Hamel, E; Ronca, R; Bortolozzi, R; Mariotto, E; Mattiuzzo, E; Viola, G J Med Chem 62: 1274-1290 (2019)
- Sisay, MT; Steinmetzer, T; Stirnberg, M; Maurer, E; Hammami, M; Bajorath, J; Gütschow, M J Med Chem 53: 5523-35 (2010)
- Mazur, M; Koralewski, R; Borek, B; Olejniczak, S; Czestkowski, WJ; Piotrowicz, MC; Olczak, JP; Golebiowski, AA; Bartoszewicz, A; Maziarz, E; Kowalski, M US Patent US9944624 (2018)
- Pass, M; Abu-Rabie, S; Baxter, A; Conroy, R; Coote, SJ; Craven, AP; Finch, H; Hindley, S; Kelly, HA; Lowdon, AW; McDonald, E; Mitchell, WL; Pegg, NA; Procopiou, PA; Ramsden, NG; Thomas, R; Walker, DA; Watson, NS; Jhoti, H; Mooney, CJ; Tang, CM; Thomas, PJ; Parry, S; Patel, C Bioorg Med Chem Lett 9: 1657-62 (1999)
- Starr, J; Brown, MF; Aschenbrenner, L; Caspers, N; Che, Y; Gerstenberger, BS; Huband, M; Knafels, JD; Lemmon, MM; Li, C; McCurdy, SP; McElroy, E; Rauckhorst, MR; Tomaras, AP; Young, JA; Zaniewski, RP; Shanmugasundaram, V; Han, S J Med Chem 57: 3845-55 (2014)
- Shao, PP; Ye, F; Chakravarty, PK; Varughese, DJ; Herrington, JB; Dai, G; Bugianesi, RM; Haedo, RJ; Swensen, AM; Warren, VA; Smith, MM; Garcia, ML; McManus, OB; Lyons, KA; Li, X; Green, M; Jochnowitz, N; McGowan, E; Mistry, S; Sun, SY; Abbadie, C; Kaczorowski, GJ; Duffy, JL J Med Chem 55: 9847-55 (2012)
- Flick, AC; Leverett, CA; Ding, HX; McInturff, E; Fink, SJ; Mahapatra, S; Carney, DW; Lindsey, EA; DeForest, JC; France, SP; Berritt, S; Bigi-Botterill, SV; Gibson, TS; Liu, Y; O'Donnell, CJ J Med Chem 64: 3604-3657 (2021)
- Combs, AP; Zhu, W; Crawley, ML; Glass, B; Polam, P; Sparks, RB; Modi, D; Takvorian, A; McLaughlin, E; Yue, EW; Wasserman, Z; Bower, M; Wei, M; Rupar, M; Ala, PJ; Reid, BM; Ellis, D; Gonneville, L; Emm, T; Taylor, N; Yeleswaram, S; Li, Y; Wynn, R; Burn, TC; Hollis, G; Liu, PC; Metcalf, B J Med Chem 49: 3774-89 (2006)
- Ndubaku, CO; Crawford, TD; Chen, H; Boggs, JW; Drobnick, J; Harris, SF; Jesudason, R; McNamara, E; Nonomiya, J; Sambrone, A; Schmidt, S; Smyczek, T; Vitorino, P; Wang, L; Wu, P; Yeung, S; Chen, J; Chen, K; Ding, CZ; Wang, T; Xu, Z; Gould, SE; Murray, LJ; Ye, W ACS Med Chem Lett 6: 913-8 (2015)
- Frecer, V; Megnassan, E; Miertus, S Eur J Med Chem 44: 3009-19 (2009)
- Perregaard, J; Moltzen, EK; Meier, E; Sánchez, C J Med Chem 38: 1998-2008 (1995)
- Adams, CM; Hu, CW; Jeng, AY; Karki, R; Ksander, G; Lasala, D; Leung-Chu, J; Liang, G; Liu, Q; Meredith, E; Rao, C; Rigel, DF; Shi, J; Smith, S; Springer, C; Zhang, C Bioorg Med Chem Lett 20: 4324-7 (2010)
- Vandeveer, GH; Arduini, RM; Baker, DP; Barry, K; Bohnert, T; Bowden-Verhoek, JK; Conlon, P; Cullen, PF; Guan, B; Jenkins, TJ; Liao, SY; Lin, L; Liu, YT; Marcotte, D; Mertsching, E; Metrick, CM; Negrou, E; Powell, N; Scott, D; Silvian, LF; Hopkins, BT Bioorg Med Chem Lett 80: (2023)
- Hepnarova, V; Korabecny, J; Matouskova, L; Jost, P; Muckova, L; Hrabinova, M; Vykoukalova, N; Kerhartova, M; Kucera, T; Dolezal, R; Nepovimova, E; Spilovska, K; Mezeiova, E; Pham, NL; Jun, D; Staud, F; Kaping, D; Kuca, K; Soukup, O Eur J Med Chem 150: 292-306 (2018)
- Myrianthopoulos, V; Kritsanida, M; Gaboriaud-Kolar, N; Magiatis, P; Ferandin, Y; Durieu, E; Lozach, O; Cappel, D; Soundararajan, M; Filippakopoulos, P; Sherman, W; Knapp, S; Meijer, L; Mikros, E; Skaltsounis, AL ACS Med Chem Lett 4: 22-26 (2013)
- Hu, LY; Ryder, TR; Nikam, SS; Millerman, E; Szoke, BG; Rafferty, MF Bioorg Med Chem Lett 9: 1121-6 (1999)
- Dei, S; Coronnello, M; Floriddia, E; Bartolucci, G; Bellucci, C; Guandalini, L; Manetti, D; Romanelli, MN; Salerno, M; Bello, I; Mini, E; Teodori, E Eur J Med Chem 87: 398-412 (2014)
- Ortega, JA; Riccardi, L; Minniti, E; Borgogno, M; Arencibia, JM; Greco, ML; Minarini, A; Sissi, C; De Vivo, M J Med Chem 61: 1375-1379 (2018)
- Ben-Daniel, R; Deuther-Conrad, W; Scheunemann, M; Steinbach, J; Brust, P; Mishani, E Bioorg Med Chem 16: 6364-70 (2008)
- Masubuchi, K; Okada, T; Kohchi, M; Sakaitani, M; Mizuguchi, E; Shirai, H; Aoki, M; Watanabe, T; Kondoh, O; Yamazaki, T; Satoh, Y; Kobayashi, K; Inoue, T; Horii, I; Shimma, N Bioorg Med Chem Lett 11: 395-8 (2001)
- Dallavalle, S; Musso, L; Cincinelli, R; Darwiche, N; Gervasoni, S; Vistoli, G; Guglielmi, MB; La Porta, I; Pizzulo, M; Modica, E; Prosperi, F; Signorino, G; Colelli, F; Cardile, F; Fucci, A; D'Andrea, EL; Riccio, A; Pisano, C Eur J Med Chem 228: (2022)
- Alagha, A; Moman, E; Adamo, MF; Nolan, KB; Chubb, AJ Bioorg Med Chem Lett 19: 4213-6 (2009)
- Campiani, G; Morelli, E; Gemma, S; Nacci, V; Butini, S; Hamon, M; Novellino, E; Greco, G; Cagnotto, A; Goegan, M; Cervo, L; Dalla Valle, F; Fracasso, C; Caccia, S; Mennini, T J Med Chem 42: 4362-79 (1999)
- Morera, E; Di Marzo, V; Monti, L; Allarà, M; Schiano Moriello, A; Nalli, M; Ortar, G; De Petrocellis, L Bioorg Med Chem Lett 26: 1401-5 (2016)
- Zabludoff, SD; Deng, C; Grondine, MR; Sheehy, AM; Ashwell, S; Caleb, BL; Green, S; Haye, HR; Horn, CL; Janetka, JW; Liu, D; Mouchet, E; Ready, S; Rosenthal, JL; Queva, C; Schwartz, GK; Taylor, KJ; Tse, AN; Walker, GE; White, AM Mol Cancer Ther 7: 2955-66
- Ryckebusch, A; Deprez-Poulain, R; Maes, L; Debreu-Fontaine, MA; Mouray, E; Grellier, P; Sergheraert, C J Med Chem 46: 542-57 (2003)
- Mascitti, V; Maurer, TS; Robinson, RP; Bian, J; Boustany-Kari, CM; Brandt, T; Collman, BM; Kalgutkar, AS; Klenotic, MK; Leininger, MT; Lowe, A; Maguire, RJ; Masterson, VM; Miao, Z; Mukaiyama, E; Patel, JD; Pettersen, JC; Préville, C; Samas, B; She, L; Sobol, Z; Steppan, CM; Stevens, BD; Thuma, BA; Tugnait, M; Zeng, D; Zhu, T J Med Chem 54: 2952-60 (2011)
- Gauthier, JY; Belley, M; Deschênes, D; Fournier, JF; Gagné, S; Gareau, Y; Hamel, M; Hénault, M; Hyjazie, H; Kargman, S; Lavallée, G; Levesque, JF; Li, L; Mamane, Y; Mancini, J; Morin, N; Mulrooney, E; Robichaud, J; Thérien, M; Tranmer, G; Wang, Z; Wu, J; Black, WC Bioorg Med Chem Lett 21: 2836-9 (2011)
- Caprioglio, D; Mattoteia, D; Pollastro, F; Negri, R; Lopatriello, A; Chianese, G; Minassi, A; Collado, JA; Munoz, E; Taglialatela-Scafati, O; Appendino, G J Nat Prod 83: 1711-1715 (2020)
- Maj, R; Pattarino, F; Mura, E; Barberis, A US Patent US9173935 (2015)
- Orvieto, F; Koch, U; Matassa, VG; Muraglia, E Bioorg Med Chem Lett 13: 2745-8 (2003)
- Du, J; Chun, BK; Mosley, RT; Bansal, S; Bao, H; Espiritu, C; Lam, AM; Murakami, E; Niu, C; Micolochick Steuer, HM; Furman, PA; Sofia, MJ J Med Chem 57: 1826-35 (2014)
- Kaldor, SW; Kanouni, T; Tyhonas, J; Murphy, E; Cox, J; Kania, R US Patent US11407737 (2022)
- Deiana, V; Gómez-Cañas, M; Pazos, MR; Fernández-Ruiz, J; Asproni, B; Cichero, E; Fossa, P; Muñoz, E; Deligia, F; Murineddu, G; García-Arencibia, M; Pinna, GA Eur J Med Chem 112: 66-80 (2016)
- Tang, J; Liu, F; Nagy, E; Miller, L; Kirby, KA; Wilson, DJ; Wu, B; Sarafianos, SG; Parniak, MA; Wang, Z J Med Chem 59: 2648-59 (2016)
- Takayama, W; Shirasaki, Y; Sakai, Y; Nakajima, E; Fujita, S; Sakamoto-Mizutani, K; Inoue, J Bioorg Med Chem Lett 13: 3273-6 (2003)
- Radhakrishnan, S; Syed, R; Takei, H; Kobayashi, IS; Nakamura, E; Sultana, F; Kamal, A; Tenen, DG; Kobayashi, SS Bioorg Med Chem Lett 29: 2286-2289 (2019)
- Nakashima, H; Uto, Y; Nakata, E; Nagasawa, H; Ikkyu, K; Hiraoka, N; Nakashima, K; Sasaki, Y; Sugimoto, H; Shiro, Y; Hashimoto, T; Okamoto, Y; Asakawa, Y; Hori, H Bioorg Med Chem 16: 8661-9 (2008)
- Mena-Barragán, T; García-Moreno, MI; Nanba, E; Higaki, K; Concia, AL; Clapés, P; García Fernández, JM; Ortiz Mellet, C Eur J Med Chem 121: 880-891 (2016)
- Vandeveer, GH; Arduini, RM; Baker, DP; Barry, K; Bohnert, T; Bowden-Verhoek, JK; Conlon, P; Cullen, PF; Guan, B; Jenkins, TJ; Liao, SY; Lin, L; Liu, YT; Marcotte, D; Mertsching, E; Metrick, CM; Negrou, E; Powell, N; Scott, D; Silvian, LF; Hopkins, BT Bioorg Med Chem Lett 80: (2023)
- Chua, K; Fung, E; Micewicz, ED; Ganz, T; Nemeth, E; Ruchala, P Bioorg Med Chem Lett 25: 4961-9 (2015)
- Oleksak, P; Nepovimova, E; Chrienova, Z; Musilek, K; Patocka, J; Kuca, K Eur J Med Chem 238: (2022)
- Crosignani, S; Campos, S; Bouix-Peter, C; Harris, C; Talbot, E; Hu, H; Wang, S; Maclean, J; Zanelli, U; Taylor, S; Foote, K; Hacini-Rachinel, F; Nicodeme, E; Julia, V Bioorg Med Chem Lett 100:
- Mougenot, P; Namane, C; Fett, E; Goumy, F; Dadji-Faïhun, R; Langot, G; Monseau, C; Onofri, B; Pacquet, F; Pascal, C; Crespin, O; Ben-Hassine, M; Ragot, JL; Van-Pham, T; Philippo, C; Chatelain-Egger, F; Péron, P; Le Bail, JC; Guillot, E; Chamiot-Clerc, P; Chabanaud, MA; Pruniaux, MP; Ménegotto, J; Schmidt, F; Venier, O; Viviani, F; Nicolai, E Bioorg Med Chem Lett 26: 25-32 (2016)
- Varming, T; Christophersen, P; Møller, A; Peters, D; Axelsson, O; Nielsen, E& Bioorg Med Chem Lett 6: 245-248 (1996)
- Kodra, JT; Jørgensen, AS; Andersen, B; Behrens, C; Brand, CL; Christensen, IT; Guldbrandt, M; Jeppesen, CB; Knudsen, LB; Madsen, P; Nishimura, E; Sams, C; Sidelmann, UG; Pedersen, RA; Lynn, FC; Lau, J J Med Chem 51: 5387-96 (2008)
- Pace, P; Di Francesco, ME; Gardelli, C; Harper, S; Muraglia, E; Nizi, E; Orvieto, F; Petrocchi, A; Poma, M; Rowley, M; Scarpelli, R; Laufer, R; Gonzalez Paz, O; Monteagudo, E; Bonelli, F; Hazuda, D; Stillmock, KA; Summa, V J Med Chem 50: 2225-39 (2007)
- Jones, CL; Njomen, E; Sjögren, B; Dexheimer, TS; Tepe, JJ ACS Chem Biol 12: 2240-2247 (2017)
- Gehling, VS; Vaswani, RG; Nasveschuk, CG; Duplessis, M; Iyer, P; Balasubramanian, S; Zhao, F; Good, AC; Campbell, R; Lee, C; Dakin, LA; Cook, AS; Gagnon, A; Harmange, JC; Audia, JE; Cummings, RT; Normant, E; Trojer, P; Albrecht, BK Bioorg Med Chem Lett 25: 3644-9 (2015)
- Cosconati, S; Hong, JA; Novellino, E; Carroll, KS; Goodsell, DS; Olson, AJ J Med Chem 51: 6627-30 (2008)
- Gilbert, AM; Kirisits, M; Toy, P; Nunn, DS; Failli, A; Dushin, EG; Novikova, E; Petersen, PJ; Joseph-McCarthy, D; McFadyen, I; Fritz, CC Bioorg Med Chem Lett 14: 37-41 (2003)
- Cuffaro, D; Burkhard, T; Bernardoni, BL; Di Leo, R; Zhang, X; Galati, S; Tuccinardi, T; Macchia, M; Rossello, A; Santamaria, S; de Groot, R; Nuti, E RSC Med Chem 15: 2806-2825
- Vallin, KS; Sterky, KJ; Nyman, E; Bernström, J; From, R; Linde, C; Minidis, AB; Nolting, A; Närhi, K; Santangelo, EM; Sehgelmeble, FW; Sohn, D; Strindlund, J; Weigelt, D Bioorg Med Chem Lett 22: 5485-92 (2012)
- Anumala, UR; Waaler, J; Nkizinkiko, Y; Ignatev, A; Lazarow, K; Lindemann, P; Olsen, PA; Murthy, S; Obaji, E; Majouga, AG; Leonov, S; von Kries, JP; Lehtiö, L; Krauss, S; Nazaré, M J Med Chem 60: 10013-10025 (2017)
- Shultz, MD; Cheung, AK; Kirby, CA; Firestone, B; Fan, J; Chen, CH; Chen, Z; Chin, DN; Dipietro, L; Fazal, A; Feng, Y; Fortin, PD; Gould, T; Lagu, B; Lei, H; Lenoir, F; Majumdar, D; Ochala, E; Palermo, MG; Pham, L; Pu, M; Smith, T; Stams, T; Tomlinson, RC; Touré, BB; Visser, M; Wang, RM; Waters, NJ; Shao, W J Med Chem 56: 6495-511 (2013)
- Misawa, T; Tsuji, G; Takahashi, T; Ochiai, E; Takagi, KI; Horie, K; Kakuda, S; Takimoto-Kamimura, M; Kurihara, M; Demizu, Y Bioorg Med Chem 26: 6146-6152 (2018)
- Onyameh, EK; Bricker, BA; Eyunni, SVK; Voshavar, C; Gonela, UM; Ofori, E; Jenkins, A; Ablordeppey, SY Bioorg Med Chem 30: (2021)
- Nishimura, S; Hitora, Y; Kawahara, T; Tanabe, M; Ogata, E; Kato, H; Srikoon, P; Watanabe, T; Tsukamoto, S Bioorg Med Chem Lett 59: (2022)
- Ohshima, E; Takami, H; Harakawa, H; Sato, H; Obase, H; Miki, I; Ishii, A; Ishii, H; Sasaki, Y; Ohmori, K J Med Chem 36: 417-20 (1993)
- Hagihara, M; Yoneda, K; Okanari, E; Shigetomi, M US Patent US8685986 (2014)
- Shreder, KR; Lin, EC; Wu, J; Cajica, J; Amantea, CM; Hu, Y; Okerberg, E; Brown, HE; Pham, LM; Chung, de M; Fraser, AS; McGee, E; Rosenblum, JS; Kozarich, JW Bioorg Med Chem Lett 22: 5748-51 (2012)
- Malwal, SR; Mazurek, B; Ko, J; Xie, P; Barnes, C; Varvitsiotis, C; Zimmerman, MD; Olatunji, S; Lee, J; Xie, M; Sarathy, J; Caffrey, M; Strynadka, NCJ; Dartois, V; Dick, T; Lee, BNR; Russell, DG; Oldfield, E J Med Chem 66: 7553-7569 (2023)
- Baraldi, PG; Cacciari, B; Spalluto, G; Bergonzoni, M; Dionisotti, S; Ongini, E; Varani, K; Borea, PA J Med Chem 41: 2126-33 (1998)
- Zhang, X; Hou, C; Hufnagel, H; Singer, M; Opas, E; McKenney, S; Johnson, D; Sui, Z ACS Med Chem Lett 3: 1039-1044 (2012)
- Macchia, B; Cervetto, L; Demontis, GC; Domiano, P; Longoni, B; Macchia, M; Minutolo, F; Orlandini, E; Ortore, G; Papi, C Bioorg Med Chem Lett 11: 223-6 (2001)
- Bochen, A; Marelli, UK; Otto, E; Pallarola, D; Mas-Moruno, C; Di Leva, FS; Boehm, H; Spatz, JP; Novellino, E; Kessler, H; Marinelli, L J Med Chem 56: 1509-19 (2013)
- Rabindran, SK; Discafani, CM; Rosfjord, EC; Baxter, M; Floyd, MB; Golas, J; Hallett, WA; Johnson, BD; Nilakantan, R; Overbeek, E; Reich, MF; Shen, R; Shi, X; Tsou, HR; Wang, YF; Wissner, A Cancer Res 64: 3958-65
- Jain, N; Kanojia, RM; Xu, J; Jian-Zhong, G; Pacia, E; Lai, MT; Du, F; Musto, A; Allan, G; Hahn, D; Lundeen, S; Sui, Z J Med Chem 49: 3056-9 (2006)
- Xiao, Y; Araldi, GL; Zhao, Z; Brugger, N; Karra, S; Fischer, D; Palmer, E Bioorg Med Chem Lett 17: 4323-7 (2007)
- Battistutta, R; Cozza, G; Pierre, F; Papinutto, E; Lolli, G; Sarno, S; O'Brien, SE; Siddiqui-Jain, A; Haddach, M; Anderes, K; Ryckman, DM; Meggio, F; Pinna, LA Biochemistry 50: 8478-88 (2011)
- Crawford, TD; Vartanian, S; Côté, A; Bellon, S; Duplessis, M; Flynn, EM; Hewitt, M; Huang, HR; Kiefer, JR; Murray, J; Nasveschuk, CG; Pardo, E; Romero, FA; Sandy, P; Tang, Y; Taylor, AM; Tsui, V; Wang, J; Wang, S; Zawadzke, L; Albrecht, BK; Magnuson, SR; Cochran, AG; Stokoe, D Bioorg Med Chem Lett 27: 3534-3541 (2017)
- Chevillard, F; Rimmer, H; Betti, C; Pardon, E; Ballet, S; van Hilten, N; Steyaert, J; Diederich, WE; Kolb, P J Med Chem 61: 1118-1129 (2018)
- Lee, JY; Ryu, K; Kim, J; Kim, Y; Shin, D; Lee, B; Kang, S; Lee, H; Jung, H; Shin, YA; Park, E; Ahn, J; Kim, H; Ryu, JH US Patent US10155763 (2018)
- Thonhofer, M; Weber, P; Santana, AG; Fischer, R; Pabst, BM; Paschke, E; Schalli, M; Stütz, AE; Tschernutter, M; Windischhofer, W; Withers, SG Bioorg Med Chem Lett 26: 1438-42 (2016)
- Zhong, M; Peng, E; Huang, N; Huang, Q; Huq, A; Lau, M; Colonno, R; Li, L Bioorg Med Chem Lett 26: 4508-4512 (2016)
- Fiorino, F; Perissutti, E; Severino, B; Santagada, V; Cirillo, D; Terracciano, S; Massarelli, P; Bruni, G; Collavoli, E; Renner, C; Caliendo, G J Med Chem 48: 5495-503 (2005)
- Shaw, S; Bian, Z; Zhao, B; Tarr, JC; Veerasamy, N; Jeon, KO; Belmar, J; Arnold, AL; Fogarty, SA; Perry, E; Sensintaffar, JL; Camper, DV; Rossanese, OW; Lee, T; Olejniczak, ET; Fesik, SW J Med Chem 61: 2410-2421 (2018)
- Parodi, A; Righetti, G; Pesce, E; Salis, A; Tasso, B; Urbinati, C; Tomati, V; Damonte, G; Rusnati, M; Pedemonte, N; Cichero, E; Millo, E Eur J Med Chem 208: (2020)
- Menichincheri, M; Albanese, C; Alli, C; Ballinari, D; Bargiotti, A; Caldarelli, M; Ciavolella, A; Cirla, A; Colombo, M; Colotta, F; Croci, V; D'Alessio, R; D'Anello, M; Ermoli, A; Fiorentini, F; Forte, B; Galvani, A; Giordano, P; Isacchi, A; Martina, K; Molinari, A; Moll, JK; Montagnoli, A; Orsini, P; Orzi, F; Pesenti, E; Pillan, A; Roletto, F; Scolaro, A; Tatò, M; Tibolla, M; Valsasina, B; Varasi, M; Vianello, P; Volpi, D; Santocanale, C; Vanotti, E J Med Chem 53: 7296-315 (2010)
- Xu, YZ; Smith, JL; Semko, CM; Rossiter, KI; Fukuda, JY; Dappen, MS; Quincy, DA; Konradi, AW; Mao, W; Welch, B; Dreyer, ML; Samant, B; Zhang, H; Lugar, J; Liao, Z; Henschel, C; Petersen, E; Vandevert, C; Shoemaker, M; Wehner, N; Mutter, L; Shopp, G; Krimm, M; Chen, L; Wipke, B; Dofiles, L; Gallager, I; Sauer, JM; Messersmith, EK; Pleiss, MA; Bard, F; Yednock, TA Bioorg Med Chem Lett 23: 4370-3 (2013)
- Rej, RK; Wang, C; Lu, J; Wang, M; Petrunak, E; Zawacki, KP; McEachern, D; Yang, CY; Wang, L; Li, R; Chinnaswamy, K; Wen, B; Sun, D; Stuckey, JA; Zhou, Y; Chen, J; Tang, G; Wang, S J Med Chem 64: 14540-14556 (2021)
- Schwarz, S; Loesche, A; Lucas, SD; Sommerwerk, S; Serbian, I; Siewert, B; Pianowski, E; Csuk, R Eur J Med Chem 103: 438-45 (2015)
- Jolidon, S; Alberati, D; Dowle, A; Fischer, H; Hainzl, D; Narquizian, R; Norcross, R; Pinard, E Bioorg Med Chem Lett 18: 5533-6 (2008)
- Chatterjee, J; Laufer, B; Beck, JG; Helyes, Z; Pintér, E; Szolcsányi, J; Horvath, A; Mandl, J; Reubi, JC; Kéri, G; Kessler, H ACS Med Chem Lett 2: 509-514 (2011)
- Gornati, D; Ciccone, R; Vinciguerra, A; Ippati, S; Pannaccione, A; Petrozziello, T; Pizzi, E; Hassan, A; Colombo, E; Barbini, S; Milani, M; Caccavone, C; Randazzo, P; Muzio, L; Annunziato, L; Menegon, A; Secondo, A; Mastrangelo, E; Pignataro, G; Seneci, P J Med Chem 64: 8333-8353 (2021)
- Plut, E; Calderón, JC; Stanojlović, V; Gattor, AO; Höring, C; Humphrys, LJ; Konieczny, A; Kerres, S; Schubert, M; Keller, M; Cabrele, C; Clark, T; Reiser, O J Med Chem 66: 9642-9657 (2023)
- Koralewski, R; Dymek, B; Mazur, M; Sklepkiewicz, P; Olejniczak, S; Czestkowski, W; Matyszewski, K; Andryianau, G; Niedziejko, P; Kowalski, M; Gruza, M; Borek, B; Jedrzejczak, K; Bartoszewicz, A; Pluta, E; Rymaszewska, A; Kania, M; Rejczak, T; Piasecka, S; Mlacki, M; Mazurkiewicz, M; Piotrowicz, M; Salamon, M; Zagozdzon, A; Napiorkowska-Gromadzka, A; Bartlomiejczak, A; Mozga, W; Dobrzański, P; Dzwonek, K; Golab, J; Nowotny, M; Olczak, J; Golebiowski, A J Med Chem 63: 15527-15540 (2020)
- Purohit, MK; Poduch, E; Wei, LW; Crandall, IE; To, T; Kain, KC; Pai, EF; Kotra, LP J Med Chem 55: 9988-97 (2012)
- Guardigni, M; Greco, G; Poeta, E; Santini, A; Tassinari, E; Bergamini, C; Zalambani, C; De Simone, A; Andrisano, V; Uliassi, E; Monti, B; Bolognesi, ML; Fimognari, C; Milelli, A RSC Med Chem 15: 2045-2062
- Prchalová, E; Hin, N; Thomas, AG; Veeravalli, V; Ng, J; Alt, J; Rais, R; Rojas, C; Li, Z; Hihara, H; Aoki, M; Yoshizawa, K; Nishioka, T; Suzuki, S; Kopajtic, T; Chatrath, S; Liu, Q; Dong, X; Slusher, BS; Tsukamoto, T J Med Chem 62: 8631-8641 (2019)
- Cole, DC; Olland, AM; Jacob, J; Brooks, J; Bursavich, MG; Czerwinski, R; DeClercq, C; Johnson, M; Joseph-McCarthy, D; Ellingboe, JW; Lin, L; Nowak, P; Presman, E; Strand, J; Tam, A; Williams, CM; Yao, S; Tsao, DH; Fitz, LJ J Med Chem 53: 6122-8 (2010)
- Schühly, W; Hüfner, A; Pferschy-Wenzig, EM; Prettner, E; Adams, M; Bodensieck, A; Kunert, O; Oluwemimo, A; Haslinger, E; Bauer, R Bioorg Med Chem 17: 4459-65 (2009)
- Hernandez-Olmos, V; Knape, T; Heering, J; von Knethen, A; Kilu, W; Kaiser, A; Wurglics, M; Helmstädter, M; Merk, D; Schubert-Zsilavecz, M; Parnham, MJ; Steinhilber, D; Proschak, E Bioorg Med Chem 27: (2019)
- Vanda, D; Soural, M; Canale, V; Chaumont-Dubel, S; Satała, G; Kos, T; Funk, P; Fülöpová, V; Lemrová, B; Koczurkiewicz, P; Pękala, E; Bojarski, AJ; Popik, P; Marin, P; Zajdel, P Eur J Med Chem 144: 716-729 (2018)
- Santana, L; González-Díaz, H; Quezada, E; Uriarte, E; Yáñez, M; Viña, D; Orallo, F J Med Chem 51: 6740-51 (2008)
- Ullrich, JW; Morris, R; Bernotas, RC; Travins, JM; Jetter, J; Unwalla, R; Quinet, E; Nambi, P; Feingold, I; Huselton, C; Enroth, C; Wilhelmsson, A; Goos-Nilsson, A; Wrobel, J Bioorg Med Chem Lett 20: 2903-7 (2010)
- Van der Plas, SE; Kelgtermans, H; De Munck, T; Martina, SLX; Dropsit, S; Quinton, E; De Blieck, A; Joannesse, C; Tomaskovic, L; Jans, M; Christophe, T; van der Aar, E; Borgonovi, M; Nelles, L; Gees, M; Stouten, P; Van Der Schueren, J; Mammoliti, O; Conrath, K; Andrews, M J Med Chem 61: 1425-1435 (2018)
- Garsi, JB; Komjáti, B; Cullia, G; Fejes, I; Sipos, M; Sipos, Z; Fördős, E; Markacz, P; Balázs, B; Lancelot, N; Berger, S; Raimbaud, E; Brown, D; Vuillard, LM; Haberkorn, L; Cukier, C; Szlávik, Z; Hanessian, S ACS Med Chem Lett 13: 949-954 (2022)
- Pompliano, DL; Rands, E; Schaber, MD; Mosser, SD; Anthony, NJ; Gibbs, JB Biochemistry 31: 3800-7 (1992)
- Lazo, JS; Sharlow, E; Wipf, P; Tasker, N; Rastelli, E US Patent US12202839 (2025)
- Di Fabio, R; Pellacani, A; Faedo, S; Roth, A; Piccoli, L; Gerrard, P; Porter, RA; Johnson, CN; Thewlis, K; Donati, D; Stasi, L; Spada, S; Stemp, G; Nash, D; Branch, C; Kindon, L; Massagrande, M; Poffe, A; Braggio, S; Chiarparin, E; Marchioro, C; Ratti, E; Corsi, M Bioorg Med Chem Lett 21: 5562-7 (2011)
- Amssoms, K; Oza, SL; Ravaschino, E; Yamani, A; Lambeir, A; Rajan, P; Bal, G; Rodriguez, J; Fairlamb, AH; Augustyns, K; Haemers, A Bioorg Med Chem Lett 12: 2553-6 (2002)
- Salomé, C; Narbonne, V; Ribeiro, N; Thuaud, F; Serova, M; de Gramont, A; Faivre, S; Raymond, E; Désaubry, L Eur J Med Chem 74: 41-9 (2014)
- Raux, B; Voitovich, Y; Derviaux, C; Lugari, A; Rebuffet, E; Milhas, S; Priet, S; Roux, T; Trinquet, E; Guillemot, JC; Knapp, S; Brunel, JM; Fedorov, AY; Collette, Y; Roche, P; Betzi, S; Combes, S; Morelli, X J Med Chem 59: 1634-41 (2016)
- Liu, J; Steigel, A; Reininger, E; Bauer, R J Nat Prod 63: 403-5 (2000)
- Kurz, JL; Pedroso, MM; Richard, E; McGeary, RP; Schenk, G Bioorg Med Chem Lett 92: (2023)
- Hopkins, CR; O'neil, SV; Laufersweiler, MC; Wang, Y; Pokross, M; Mekel, M; Evdokimov, A; Walter, R; Kontoyianni, M; Petrey, ME; Sabatakos, G; Roesgen, JT; Richardson, E; Demuth, TP Bioorg Med Chem Lett 16: 5659-63 (2006)
- Richelson, E; Fauq, AH; Carlier, P; Monceaux, CJ US Patent US9944618 (2018)
- Castellano, S; Taliani, S; Milite, C; Pugliesi, I; Da Pozzo, E; Rizzetto, E; Bendinelli, S; Costa, B; Cosconati, S; Greco, G; Novellino, E; Sbardella, G; Stefancich, G; Martini, C; Da Settimo, F J Med Chem 55: 4506-10 (2012)
- Plobeck, N; Delorme, D; Wei, ZY; Yang, H; Zhou, F; Schwarz, P; Gawell, L; Gagnon, H; Pelcman, B; Schmidt, R; Yue, SY; Walpole, C; Brown, W; Zhou, E; Labarre, M; Payza, K; St-Onge, S; Kamassah, A; Morin, PE; Projean, D; Ducharme, J; Roberts, E J Med Chem 43: 3878-94 (2000)
- Greiner, D; Bonaldi, T; Eskeland, R; Roemer, E; Imhof, A Nat Chem Biol 1: 143-5 (2005)
- Lambruschini, C; Veronesi, M; Romeo, E; Garau, G; Bandiera, T; Piomelli, D; Scarpelli, R; Dalvit, C Chembiochem 14: 1611-9 (2013)
- Romero, E; Oueslati, S; Benchekroun, M; D'Hollander, ACA; Ventre, S; Vijayakumar, K; Minard, C; Exilie, C; Tlili, L; Retailleau, P; Zavala, A; Elisée, E; Selwa, E; Nguyen, LA; Pruvost, A; Naas, T; Iorga, BI; Dodd, RH; Cariou, K Eur J Med Chem 219: (2021)
- Lange, JH; Coolen, HK; van Stuivenberg, HH; Dijksman, JA; Herremans, AH; Ronken, E; Keizer, HG; Tipker, K; McCreary, AC; Veerman, W; Wals, HC; Stork, B; Verveer, PC; den Hartog, AP; de Jong, NM; Adolfs, TJ; Hoogendoorn, J; Kruse, CG J Med Chem 47: 627-43 (2004)
- Vogensen, SB; Jørgensen, L; Madsen, KK; Jurik, A; Borkar, N; Rosatelli, E; Nielsen, B; Ecker, GF; Schousboe, A; Clausen, RP Bioorg Med Chem 23: 2480-8 (2015)
- Goracci, L; Nurisso, A; Roussel, E; Pérès, B; Chaptal, V; Falson, P; Marminon, C; Jose, J; Le Borgne, M; Boumendjel, A Eur J Med Chem 248: (2023)
- Aghazadeh Tabrizi, M; Baraldi, PG; Ruggiero, E; Saponaro, G; Baraldi, S; Poli, G; Tuccinardi, T; Ravani, A; Vincenzi, F; Borea, PA; Varani, K Eur J Med Chem 113: 11-27 (2016)
- Gitto, R; Ferro, S; Agnello, S; De Luca, L; De Sarro, G; Russo, E; Vullo, D; Supuran, CT; Chimirri, A Bioorg Med Chem 17: 3659-64 (2009)
- Plazinska, A; Pajak, K; Rutkowska, E; Jimenez, L; Kozocas, J; Koolpe, G; Tanga, M; Toll, L; Wainer, IW; Jozwiak, K Bioorg Med Chem 22: 234-46 (2014)
- Sit, SY; Xie, K; Jacutin-Porte, S; Taber, MT; Gulwadi, AG; Korpinen, CD; Burris, KD; Molski, TF; Ryan, E; Xu, C; Wong, H; Zhu, J; Krishnananthan, S; Gao, Q; Verdoorn, T; Johnson, G J Med Chem 45: 3660-8 (2002)
- Epple, R; Azimioara, M; Russo, R; Xie, Y; Wang, X; Cow, C; Wityak, J; Karanewsky, D; Bursulaya, B; Kreusch, A; Tuntland, T; Gerken, A; Iskandar, M; Saez, E; Martin Seidel, H; Tian, SS Bioorg Med Chem Lett 16: 5488-92 (2006)
- Fensome, A; Gopalsamy, A; Gerstenberger, BS; Efremov, IV; Wan, Z; Pierce, B; Telliez, J; Trujillo, JI; Zhang, L; Xing, L; Saiah, E US Patent US10463675 (2019)
- Davies, HM; Saikali, E; Huby, NJ; Gilliatt, VJ; Matasi, JJ; Sexton, T; Childers, SR J Med Chem 37: 1262-8 (1994)
- El-Awady, R; Saleh, E; Hamoudi, R; Ramadan, WS; Mazitschek, R; Nael, MA; Elokely, KM; Abou-Gharbia, M; Childers, WE; Srinivasulu, V; Aloum, L; Menon, V; Al-Tel, TH Bioorg Med Chem 42: (2021)
- McClure, KF; Darout, E; Guimarães, CR; DeNinno, MP; Mascitti, V; Munchhof, MJ; Robinson, RP; Kohrt, J; Harris, AR; Moore, DE; Li, B; Samp, L; Lefker, BA; Futatsugi, K; Kung, D; Bonin, PD; Cornelius, P; Wang, R; Salter, E; Hornby, S; Kalgutkar, AS; Chen, Y J Med Chem 54: 1948-52 (2011)
- Musella, S; Carotenuto, L; Iraci, N; Baroli, G; Ciaglia, T; Nappi, P; Basilicata, MG; Salviati, E; Barrese, V; Vestuto, V; Pignataro, G; Pepe, G; Sommella, E; Di Sarno, V; Manfra, M; Campiglia, P; Gomez-Monterrey, I; Bertamino, A; Taglialatela, M; Ostacolo, C; Miceli, F J Med Chem 65: 11340-11364 (2022)
- Shrader, WD; Kolesnikov, A; Burgess-Henry, J; Rai, R; Hendrix, J; Hu, H; Torkelson, S; Ton, T; Young, WB; Katz, BA; Yu, C; Tang, J; Cabuslay, R; Sanford, E; Janc, JW; Sprengeler, PA Bioorg Med Chem Lett 16: 1596-600 (2006)
- Vaiana, N; Marzahn, M; Parapini, S; Liu, P; Dell'Agli, M; Pancotti, A; Sangiovanni, E; Basilico, N; Bosisio, E; Dunn, BM; Taramelli, D; Romeo, S Bioorg Med Chem Lett 22: 5915-8 (2012)
- Alnabulsi, S; Santina, E; Russo, I; Hussein, B; Kadirvel, M; Chadwick, A; Bichenkova, EV; Bryce, RA; Nolan, K; Demonacos, C; Stratford, IJ; Freeman, S Eur J Med Chem 111: 33-45 (2016)
- Lesuisse, D; Deprez, P; Albert, E; Duc, TT; Sortais, B; Gofflo, D; Jean-Baptiste, V; Marquette, J; Schoot, B; Sarubbi, E; Lange, G; Broto, P; Mandine, E Bioorg Med Chem Lett 11: 2127-31 (2001)
- Travelli, C; Aprile, S; Mattoteia, D; Colombo, G; Clemente, N; Scanziani, E; Terrazzino, S; Alisi, MA; Polenzani, L; Grosa, G; Genazzani, AA; Tron, GC; Galli, U Eur J Med Chem 181: (2019)
- Schirrmacher, E; Schirrmacher, R; Thews, O; Dillenburg, W; Helisch, A; Wessler, I; Buhl, R; Höhnemann, S; Buchholz, HG; Bartenstein, P; Machulla, HJ; Rösch, F Bioorg Med Chem Lett 13: 2687-92 (2003)
- Hodge, CN; Aldrich, PE; Wasserman, ZR; Fernandez, CH; Nemeth, GA; Arvanitis, A; Cheeseman, RS; Chorvat, RJ; Ciganek, E; Christos, TE; Gilligan, PJ; Krenitsky, P; Scholfield, E; Strucely, P J Med Chem 42: 819-32 (1999)
- Scholz, D; Billich, A; Charpiot, B; Ettmayer, P; Lehr, P; Rosenwirth, B; Schreiner, E; Gstach, H J Med Chem 37: 3079-89 (1994)
- Muthengi, A; Wimalasena, VK; Yosief, HO; Bikowitz, MJ; Sigua, LH; Wang, T; Li, D; Gaieb, Z; Dhawan, G; Liu, S; Erickson, J; Amaro, RE; Schönbrunn, E; Qi, J; Zhang, W J Med Chem 64: 5787-5801 (2021)
- Jorda, R; Schütznerová, E; Cankař, P; Brychtová, V; Navrátilová, J; Kryštof, V Bioorg Med Chem 23: 1975-81 (2015)
- Morwick, T; Berry, A; Brickwood, J; Cardozo, M; Catron, K; DeTuri, M; Emeigh, J; Homon, C; Hrapchak, M; Jacober, S; Jakes, S; Kaplita, P; Kelly, TA; Ksiazek, J; Liuzzi, M; Magolda, R; Mao, C; Marshall, D; McNeil, D; Prokopowicz, A; Sarko, C; Scouten, E; Sledziona, C; Sun, S; Watrous, J; Wu, JP; Cywin, CL J Med Chem 49: 2898-908 (2006)
- Braun, MG; Ashkenazi, A; Beveridge, RE; Castanedo, G; Wallweber, HA; Beresini, MH; Clark, KR; De Bruyn, T; Fu, L; Gibbons, P; Jiang, F; Kaufman, S; Kan, D; Kiefer, JR; Leclerc, JP; Lemire, A; Ly, C; Segal, E; Sims, J; Wang, W; Wei, W; Zhao, L; Schwarz, JB; Rudolph, J J Med Chem 67: 8708-8729
- Fidan, I; Salmas, RE; Arslan, M; Sentürk, M; Durdagi, S; Ekinci, D; Sentürk, E; Cosgun, S; Supuran, CT Bioorg Med Chem 23: 7353-8 (2015)
- Preuss, J; Maloney, P; Peddibhotla, S; Hedrick, MP; Hershberger, P; Gosalia, P; Milewski, M; Li, YL; Sugarman, E; Hood, B; Suyama, E; Nguyen, K; Vasile, S; Sergienko, E; Mangravita-Novo, A; Vicchiarelli, M; McAnally, D; Smith, LH; Roth, GP; Diwan, J; Chung, TD; Jortzik, E; Rahlfs, S; Becker, K; Pinkerton, AB; Bode, L J Med Chem 55: 7262-72 (2012)
- Crane, SN; Black, WC; Palmer, JT; Davis, DE; Setti, E; Robichaud, J; Paquet, J; Oballa, RM; Bayly, CI; McKay, DJ; Somoza, JR; Chauret, N; Seto, C; Scheigetz, J; Wesolowski, G; Massé, F; Desmarais, S; Ouellet, M J Med Chem 49: 1066-79 (2006)
- Cosimelli, B; Simorini, F; Taliani, S; La Motta, C; Da Settimo, F; Severi, E; Greco, G; Novellino, E; Costa, B; Da Pozzo, E; Bendinelli, S; Martini, C Eur J Med Chem 46: 4506-20 (2011)
- Mostinski, Y; Heynen, GJJE; López-Alberca, MP; Paul, J; Miksche, S; Radetzki, S; Schaller, D; Shanina, E; Seyffarth, C; Kolomeets, Y; Ziebart, N; de Schryver, J; Oestreich, S; Neuenschwander, M; Roske, Y; Heinemann, U; Rademacher, C; Volkamer, A; von Kries, JP; Birchmeier, W; Nazaré, M J Med Chem 63: 14780-14804 (2020)
- Lazo, JS; Sharlow, E; Wipf, P; Tasker, N; Rastelli, E US Patent US12202839 (2025)
- Conway, JG; McDonald, B; Parham, J; Keith, B; Rusnak, DW; Shaw, E; Jansen, M; Lin, P; Payne, A; Crosby, RM; Johnson, JH; Frick, L; Lin, MH; Depee, S; Tadepalli, S; Votta, B; James, I; Fuller, K; Chambers, TJ; Kull, FC; Chamberlain, SD; Hutchins, JT Proc Natl Acad Sci U S A 102: 16078-83 (2005)
- Cumming, JG; Brown, SJ; Cooper, AE; Faull, AW; Flynn, AP; Grime, K; Oldfield, J; Shaw, JS; Shepherd, E; Tucker, H; Whittaker, D Bioorg Med Chem Lett 16: 3533-6 (2006)
- Zhang, C; Xu, M; He, C; Zhuo, J; Burns, DM; Qian, DQ; Lin, Q; Li, YL; Chen, L; Shi, E; Agrios, C; Weng, L; Sharief, V; Jalluri, R; Li, Y; Scherle, P; Diamond, S; Hunter, D; Covington, M; Marando, C; Wynn, R; Katiyar, K; Contel, N; Vaddi, K; Yeleswaram, S; Hollis, G; Huber, R; Friedman, S; Metcalf, B; Yao, W Bioorg Med Chem Lett 69: (2022)
- Uchida, T; Koshino, H; Takahashi, S; Shimizu, E; Takahashi, H; Yoshida, J; Shinden, H; Tsujimura, M; Kofujita, H; Uesugi, S; Kimura, KI J Nat Prod 81: 1070-1074 (2018)
- Russell, AJ; Westwood, IM; Crawford, MH; Robinson, J; Kawamura, A; Redfield, C; Laurieri, N; Lowe, ED; Davies, SG; Sim, E Bioorg Med Chem 17: 905-18 (2009)
- Su, S; Clarke, A; Han, Y; Chao, HJ; Bostwick, J; Schumacher, W; Wang, T; Yan, M; Hsu, MY; Simmons, E; Luk, C; Xu, C; Dabros, M; Galella, M; Onorato, J; Gordon, D; Wexler, R; Gargalovic, PS; Lawrence, RM J Med Chem 62: 10456-10465 (2019)
- Simoni, E; Daniele, S; Bottegoni, G; Pizzirani, D; Trincavelli, ML; Goldoni, L; Tarozzo, G; Reggiani, A; Martini, C; Piomelli, D; Melchiorre, C; Rosini, M; Cavalli, A J Med Chem 55: 9708-21 (2012)
- Gentry, PR; Kokubo, M; Bridges, TM; Kett, NR; Harp, JM; Cho, HP; Smith, E; Chase, P; Hodder, PS; Niswender, CM; Daniels, JS; Conn, PJ; Wood, MR; Lindsley, CW J Med Chem 56: 9351-5 (2013)
- Wijtmans, M; Celanire, S; Snip, E; Gillard, MR; Gelens, E; Collart, PP; Venhuis, BJ; Christophe, B; Hulscher, S; van der Goot, H; Lebon, F; Timmerman, H; Bakker, RA; Lallemand, BI; Leurs, R; Talaga, PE; de Esch, IJ J Med Chem 51: 2944-53 (2008)
- Bago, R; Malik, N; Munson, MJ; Prescott, AR; Davies, P; Sommer, E; Shpiro, N; Ward, R; Cross, D; Ganley, IG; Alessi, DR Biochem J 463: 413-27
- Martínez, A; Gutiérrez-de-Terán, H; Brea, J; Raviña, E; Loza, MI; Cadavid, MI; Sanz, F; Vidal, B; Segarra, V; Sotelo, E Bioorg Med Chem 16: 2103-13 (2008)
- Specker, E; Böttcher, J; Böttcher, S; Heine, A; Lilie, H; Schoop, A; Müller, G; Müller, N; Klebe, G ChemMedChem 1: 106-17 (2006)
- Meibom, D; Wasnaire, P; Beyer, K; Broehl, A; Cancho-Grande, Y; Elowe, N; Henninger, K; Johannes, S; Jungmann, N; Krainz, T; Lindner, N; Maassen, S; MacDonald, B; Menshykau, D; Mittendorf, J; Sanchez, G; Schaefer, M; Stefan, E; Torge, A; Xing, Y; Zubov, D J Med Chem 67: 2907-2940
- Carson, KG; Goodwin, NC; Harrison, BA; Rawlins, DB; Strobel, E; Zambrowicz, B US Patent US9688710 (2017)
- Kovada, V; Withers-Martinez, C; Bobrovs, R; Ce Rule, HN; Liepins, E; Grinberga, S; Hackett, F; Collins, CR; Kreicberga, A; Jiménez-Díaz, MB; Angulo-Barturen, I; Rasina, D; Suna, E; Jaudzems, K; Blackman, MJ; Jirgensons, A J Med Chem 66: 10658-10680 (2023)
- Kozikowski, AP; Araldi, GL; Tückmantel, W; Pshenichkin, S; Surina, E; Wroblewski, JT Bioorg Med Chem Lett 9: 1721-6 (1999)
- Neochoritis, CG; Atmaj, J; Twarda-Clapa, A; Surmiak, E; Skalniak, L; Köhler, LM; Muszak, D; Kurpiewska, K; Kalinowska-Tłuścik, J; Beck, B; Holak, TA; Dömling, A Eur J Med Chem 182: (2019)
- Blaquiere, N; Castanedo, GM; Burch, JD; Berezhkovskiy, LM; Brightbill, H; Brown, S; Chan, C; Chiang, PC; Crawford, JJ; Dong, T; Fan, P; Feng, J; Ghilardi, N; Godemann, R; Gogol, E; Grabbe, A; Hole, AJ; Hu, B; Hymowitz, SG; Alaoui Ismaili, MH; Le, H; Lee, P; Lee, W; Lin, X; Liu, N; McEwan, PA; McKenzie, B; Silvestre, HL; Suto, E; Sujatha-Bhaskar, S; Wu, G; Wu, LC; Zhang, Y; Zhong, Z; Staben, ST J Med Chem 61: 6801-6813 (2018)
- Preuss, J; Maloney, P; Peddibhotla, S; Hedrick, MP; Hershberger, P; Gosalia, P; Milewski, M; Li, YL; Sugarman, E; Hood, B; Suyama, E; Nguyen, K; Vasile, S; Sergienko, E; Mangravita-Novo, A; Vicchiarelli, M; McAnally, D; Smith, LH; Roth, GP; Diwan, J; Chung, TD; Jortzik, E; Rahlfs, S; Becker, K; Pinkerton, AB; Bode, L J Med Chem 55: 7262-72 (2012)
- Baska, F; Sipos, A; Őrfi, Z; Nemes, Z; Dobos, J; Szántai-Kis, C; Szabó, E; Szénási, G; Dézsi, L; Hamar, P; Cserepes, MT; Tóvári, J; Garamvölgyi, R; Krekó, M; Őrfi, L Eur J Med Chem 184: (2019)
- Handzlik, J; Szymańska, E; Wójcik, R; Dela, A; Jastrzębska-Więsek, M; Karolak-Wojciechowska, J; Fruziński, A; Siwek, A; Filipek, B; Kieć-Kononowicz, K Bioorg Med Chem 20: 4245-57 (2012)
- Yamasaki, K; Tani, O; Tateishi, Y; Tanabe, E; Namatame, I; Niimi, T; Furukawa, K; Sakashita, H J Med Chem 59: 2261-6 (2016)
- Tobinaga, H; Kameyama, T; Asahi, K; Horiguchi, T; Oohara, M; Tada, Y; Fuchino, K; Jikihara, S; Endoh, T; Kurihara, N; Kanda, Y; Ogawa, M; Tamura, N; Yagi, S; Taniguchi, E; Takahara, Y; Shimada, S; Takeyama, C; Yamamoto, S; Shinohara, S; Kai, H Bioorg Med Chem Lett 29: 688-693 (2019)
- Guardigni, M; Greco, G; Poeta, E; Santini, A; Tassinari, E; Bergamini, C; Zalambani, C; De Simone, A; Andrisano, V; Uliassi, E; Monti, B; Bolognesi, ML; Fimognari, C; Milelli, A RSC Med Chem 15: 2045-2062
- Abdul-Hay, S; Schiefer, IT; Chandrasena, RE; Li, M; Abdelhamid, R; Wang, YT; Tavassoli, E; Michalsen, B; Asghodom, RT; Luo, J; Thatcher, GR ACS Med Chem Lett 2: 656-661 (2011)
- Dei, S; Coronnello, M; Floriddia, E; Bartolucci, G; Bellucci, C; Guandalini, L; Manetti, D; Romanelli, MN; Salerno, M; Bello, I; Mini, E; Teodori, E Eur J Med Chem 87: 398-412 (2014)
- Hanessian, S; Therrien, E; van Otterlo, WA; Bayrakdarian, M; Nilsson, I; Fjellström, O; Xue, Y Bioorg Med Chem Lett 16: 1032-6 (2006)
- Nencka, R; Votruba, I; Hrebabecký, H; Jansa, P; Tloustamppound39ova, E; Horska, K; Masojídkova, M; Holý, A J Med Chem 50: 6016-23 (2007)
- Skácel, J; Djukic, S; Baszczyňski, O; Kalčic, F; Bílek, T; Chalupský, K; Kozák, J; Dvořáková, A; Tloušt'ová, E; Král'ová, Z; Šmídková, M; Voldřich, J; Rumlová, M; Pachl, P; Brynda, J; Vučková, T; Fábry, M; Snášel, J; Pichová, I; Řezáčová, P; Mertlíková-Kaiserová, H; Janeba, Z J Med Chem 66: 6652-6681 (2023)
- Li, H; Anderes, KL; Kraynov, EA; Luthin, DR; Do, QQ; Hong, Y; Tompkins, E; Sun, ET; Rajapakse, R; Pathak, VP; Christie, LC; Feng, J; Vazir, H; Castillo, R; Gregory, ML; Castro, M; Nared-Hood, K; Paderes, G; Anderson, MB J Med Chem 49: 3362-7 (2006)
- Griglio, A; Torre, E; Serafini, M; Bianchi, A; Schmid, R; Coda Zabetta, G; Massarotti, A; Sorba, G; Pirali, T; Fallarini, S Bioorg Med Chem Lett 28: 651-657 (2018)
- Ontoria, JM; Biancofiore, I; Fezzardi, P; Ferrigno, F; Torrente, E; Colarusso, S; Bianchi, E; Andreini, M; Patsilinakos, A; Kempf, G; Augustin, M; Steinbacher, S; Summa, V; Pacifici, R; Muñoz-Sanjuan, I; Park, L; Bresciani, A; Dominguez, C; Sherman, LT; Harper, S ACS Med Chem Lett 11: 740-746 (2020)
- Kuzikov, M; Costanzi, E; Reinshagen, J; Esposito, F; Vangeel, L; Wolf, M; Ellinger, B; Claussen, C; Geisslinger, G; Corona, A; Iaconis, D; Talarico, C; Manelfi, C; Cannalire, R; Rossetti, G; Gossen, J; Albani, S; Musiani, F; Herzog, K; Ye, Y; Giabbai, B; Demitri, N; Jochmans, D; De Jonghe, S; Rymenants, J; Summa, V; Tramontano, E; Beccari, AR; Leyssen, P; Storici, P; Neyts, J; Gribbon, P; Zaliani, A bioRxiv 2020: (2020)
- Raux, B; Voitovich, Y; Derviaux, C; Lugari, A; Rebuffet, E; Milhas, S; Priet, S; Roux, T; Trinquet, E; Guillemot, JC; Knapp, S; Brunel, JM; Fedorov, AY; Collette, Y; Roche, P; Betzi, S; Combes, S; Morelli, X J Med Chem 59: 1634-41 (2016)
- Fernandez, MC; Castaño, A; Dominguez, E; Escribano, A; Jiang, D; Jimenez, A; Hong, E; Hornback, WJ; Nisenbaum, ES; Rankl, N; Tromiczak, E; Vaught, G; Zarrinmayeh, H; Zimmerman, DM Bioorg Med Chem Lett 16: 5057-61 (2006)
- Zhang, P; Terefenko, EA; McComas, CC; Mahaney, PE; Vu, A; Trybulski, E; Koury, E; Johnston, G; Bray, J; Deecher, D Bioorg Med Chem Lett 18: 6067-70 (2008)
- Lowe, JD; Sanderson, HS; Cooke, AE; Ostovar, M; Tsisanova, E; Withey, SL; Chavkin, C; Husbands, SM; Kelly, E; Henderson, G; Bailey, CP Mol Pharmacol 88: 347-56
- Hoyt, SB; Taylor, J; London, C; Ali, A; Ujjainwalla, F; Tata, J; Struthers, M; Cully, D; Wisniewski, T; Ren, N; Bopp, C; Sok, A; Verras, A; McMasters, D; Chen, Q; Tung, E; Tang, W; Salituro, G; Clemas, J; Zhou, G; MacNeil, D; Duffy, R; Xiong, Y Bioorg Med Chem Lett 27: 2384-2388 (2017)
- Chong, PY; Shotwell, JB; Miller, J; Price, DJ; Maynard, A; Voitenleitner, C; Mathis, A; Williams, S; Pouliot, JJ; Creech, K; Wang, F; Fang, J; Zhang, H; Tai, VW; Turner, E; Kahler, KM; Crosby, R; Peat, AJ J Med Chem 62: 3254-3267 (2019)
- Smith, JM; Barlaam, B; Beattie, D; Bradshaw, L; Chan, HM; Chiarparin, E; Collingwood, O; Cooke, SL; Cronin, A; Cumming, I; Dean, E; Debreczeni, JÉ; Del Barco Barrantes, I; Diene, C; Gianni, D; Guerot, C; Guo, X; Guven, S; Hayhow, TG; Hong, T; Kemmitt, PD; Lamont, GM; Lamont, S; Lynch, JT; McWilliams, L; Moore, S; Raubo, P; Robb, GR; Robinson, J; Scott, JS; Srinivasan, B; Steward, O; Stubbs, CJ; Syson, K; Tan, L; Turner, O; Underwood, E; Urosevic, J; Vazquez-Chantada, M; Whittaker, AL; Wilson, DM; Winter-Holt, JJ J Med Chem 67: 13604-13638
- Kalaba, P; Aher, NY; Ilić, M; Dragačević, V; Wieder, M; Miklosi, AG; Zehl, M; Wackerlig, J; Roller, A; Beryozkina, T; Radoman, B; Saroja, SR; Lindner, W; Gonzalez, EP; Bakulev, V; Leban, JJ; Sitte, HH; Urban, E; Langer, T; Lubec, G J Med Chem 60: 9330-9348 (2017)
- Matos, MJ; Vilar, S; Kachler, S; Celeiro, M; Vazquez-Rodriguez, S; Santana, L; Uriarte, E; Hripcsak, G; Borges, F; Klotz, KN Bioorg Chem 61: 1-6 (2015)
- Golding, BT; Riedinger, C; Griffin, RJ; Hardcastle, IR; Valeur, E; Watson, AF; Noble, M US Patent US8618158 (2013)
- Arena, C; Gado, F; Di Cesare Mannelli, L; Cervetto, C; Carpi, S; Reynoso-Moreno, I; Polini, B; Vallini, E; Chicca, S; Lucarini, E; Bertini, S; D'Andrea, F; Digiacomo, M; Poli, G; Tuccinardi, T; Macchia, M; Gertsch, J; Marcoli, M; Nieri, P; Ghelardini, C; Chicca, A; Manera, C Eur J Med Chem 208: (2020)
- Pallavicini, M; Bolchi, C; Binda, M; Cilia, A; Clementi, F; Ferrara, R; Fumagalli, L; Gotti, C; Moretti, M; Pedretti, A; Vistoli, G; Valoti, E Bioorg Med Chem Lett 19: 854-9 (2009)
- Gehling, VS; Bellon, SF; Harmange, JC; LeBlanc, Y; Poy, F; Odate, S; Buker, S; Lan, F; Arora, S; Williamson, KE; Sandy, P; Cummings, RT; Bailey, CM; Bergeron, L; Mao, W; Gustafson, A; Liu, Y; VanderPorten, E; Audia, JE; Trojer, P; Albrecht, BK Bioorg Med Chem Lett 26: 4350-4 (2016)
- van Eis, MJ; Evenou, JP; Floersheim, P; Gaul, C; Cowan-Jacob, SW; Monovich, L; Rummel, G; Schuler, W; Stark, W; Strauss, A; von Matt, A; Vangrevelinghe, E; Wagner, J; Soldermann, N Bioorg Med Chem Lett 21: 7367-72 (2011)
- Vanotti, E; Amici, R; Bargiotti, A; Berthelsen, J; Bosotti, R; Ciavolella, A; Cirla, A; Cristiani, C; Damppound39Alessio, R; Forte, B; Isacchi, A; Martina, K; Menichincheri, M; Molinari, A; Montagnoli, A; Orsini, P; Pillan, A; Roletto, F; Scolaro, A; Tibolla, M; Valsasina, B; Varasi, M; Volpi, D; Santocanale, C J Med Chem 51: 487-501 (2008)
- Zobel, K; Wang, L; Varfolomeev, E; Franklin, MC; Elliott, LO; Wallweber, HJ; Okawa, DC; Flygare, JA; Vucic, D; Fairbrother, WJ; Deshayes, K ACS Chem Biol 1: 525-33 (2006)
- Martin, BP; Vasilieva, E; Dupureur, CM; Spilling, CD Bioorg Med Chem 23: 7529-34 (2015)
- Szeleczky, Z; Szakács, Z; Bozó, É; Baska, F; Vukics, K; Lévai, S; Temesvári, K; Vass, E; Béni, Z; Krámos, B; Magdó, I; Szántay, C; Kóti, J; Domány-Kovács, K; Greiner, I; Bata, I J Med Chem 64: 10445-10468 (2021)
- Venkateswararao, E; Manickam, M; Boggu, P; Kim, Y; Jung, SH Bioorg Med Chem 23: 2498-504 (2015)
- Maurer, B; Rumpf, T; Scharfe, M; Stolfa, DA; Schmitt, ML; He, W; Verdin, E; Sippl, W; Jung, M ACS Med Chem Lett 3: 1050-1053 (2012)
- Owens, T; Verner, E US Patent US9994576 (2018)
- Di Pietro, O; Vicente-García, E; Taylor, MC; Berenguer, D; Viayna, E; Lanzoni, A; Sola, I; Sayago, H; Riera, C; Fisa, R; Clos, MV; Pérez, B; Kelly, JM; Lavilla, R; Muñoz-Torrero, D Eur J Med Chem 105: 120-37 (2015)
- Biemans, B; Guba, W; Jaeschke, G; Ricci, A; Rueher, D; Vieira, E US Patent US9695128 (2017)
- Terrett, JA; Chen, H; Shore, DG; Villemure, E; Larouche-Gauthier, R; Déry, M; Beaumier, F; Constantineau-Forget, L; Grand-Maître, C; Lépissier, L; Ciblat, S; Sturino, C; Chen, Y; Hu, B; Lu, A; Wang, Y; Cridland, AP; Ward, SI; Hackos, DH; Reese, RM; Shields, SD; Chen, J; Balestrini, A; Riol-Blanco, L; Lee, WP; Liu, J; Suto, E; Wu, X; Zhang, J; Ly, JQ; La, H; Johnson, K; Baumgardner, M; Chou, KJ; Rohou, A; Rougé, L; Safina, BS; Magnuson, S; Volgraf, M J Med Chem 64: 3843-3869 (2021)
- Zapf, CW; Bloom, JD; McBean, JL; Dushin, RG; Golas, JM; Liu, H; Lucas, J; Boschelli, F; Vogan, E; Levin, JI Bioorg Med Chem Lett 21: 3627-31 (2011)
- Vlaar, CP; Castillo-Pichardo, L; Medina, JI; Marrero-Serra, CM; Vélez, E; Ramos, Z; Hernández, E Bioorg Med Chem 26: 884-890 (2018)
- Varnes, JG; Gardner, DS; Santella, JB; Duncia, JV; Estrella, M; Watson, PS; Clark, CM; Ko, SS; Welch, P; Covington, M; Stowell, N; Wadman, E; Davies, P; Solomon, K; Newton, RC; Trainor, GL; Decicco, CP; Wacker, DA Bioorg Med Chem Lett 14: 1645-9 (2004)
- Cole, DC; Stock, JR; Chopra, R; Cowling, R; Ellingboe, JW; Fan, KY; Harrison, BL; Hu, Y; Jacobsen, S; Jennings, LD; Jin, G; Lohse, PA; Malamas, MS; Manas, ES; Moore, WJ; O'Donnell, MM; Olland, AM; Robichaud, AJ; Svenson, K; Wu, J; Wagner, E; Bard, J Bioorg Med Chem Lett 18: 1063-6 (2008)
- Wikström, P; Walum, E US Patent US12202790 (2025)
- Wang, E; Kolb, HC; Szardenings, AK; Liu, C; Walsh, JC; Chen, G; Sinha, A; Kasi, D; Yu, C; Gangadharmath, UB; Zhang, W; Zhao, T; Mocharla, VP US Patent US10894807 (2021)
- Reuberson, J; Horsley, H; Franklin, RJ; Ford, D; Neuss, J; Brookings, D; Huang, Q; Vanderhoydonck, B; Gao, LJ; Jang, MY; Herdewijn, P; Ghawalkar, A; Fallah-Arani, F; Khan, AR; Henshall, J; Jairaj, M; Malcolm, S; Ward, E; Shuttleworth, L; Lin, Y; Li, S; Louat, T; Waer, M; Herman, J; Payne, A; Ceska, T; Doyle, C; Pitt, W; Calmiano, M; Augustin, M; Steinbacher, S; Lammens, A; Allen, R J Med Chem 61: 6705-6723 (2018)
- Tejeda, EJC; Bello, AM; Wasilewski, E; Koebel, A; Dunn, S; Kotra, LP J Med Chem 60: 8876-8887 (2017)
- Yoshikawa, M; Saitoh, M; Katoh, T; Seki, T; Bigi, SV; Shimizu, Y; Ishii, T; Okai, T; Kuno, M; Hattori, H; Watanabe, E; Saikatendu, KS; Zou, H; Nakakariya, M; Tatamiya, T; Nakada, Y; Yogo, T J Med Chem 61: 2384-2409 (2018)
- Reddy, NL; Fischer, JB; Burke-Howie, KJ; Barmettler, P; Rhodes, MR; Weber, E; Keana, JF Bioorg Med Chem Lett 3: 2113-2116 (1993)
- Bachovchin, DA; Zuhl, AM; Speers, AE; Wolfe, MR; Weerapana, E; Brown, SJ; Rosen, H; Cravatt, BF J Med Chem 54: 5229-36 (2011)
- Allegretta, G; Weidel, E; Empting, M; Hartmann, RW Eur J Med Chem 90: 351-9 (2015)
- Liu, F; Zhang, X; Weisberg, E; Chen, S; Hur, W; Wu, H; Zhao, Z; Wang, W; Mao, M; Cai, C; Simon, NI; Sanda, T; Wang, J; Look, AT; Griffin, JD; Balk, SP; Liu, Q; Gray, NS ACS Chem Biol 8: 1423-8 (2013)
- Bengtsson, C; Blaho, S; Saitton, DB; Brickmann, K; Broddefalk, J; Davidsson, O; Drmota, T; Folmer, R; Hallberg, K; Hallén, S; Hovland, R; Isin, E; Johannesson, P; Kull, B; Larsson, LO; Löfgren, L; Nilsson, KE; Noeske, T; Oakes, N; Plowright, AT; Schnecke, V; Ståhlberg, P; Sörme, P; Wan, H; Wellner, E; Oster, L Bioorg Med Chem 19: 3039-53 (2011)
- Lanning, ME; Yu, W; Yap, JL; Chauhan, J; Chen, L; Whiting, E; Pidugu, LS; Atkinson, T; Bailey, H; Li, W; Roth, BM; Hynicka, L; Chesko, K; Toth, EA; Shapiro, P; MacKerell, AD; Wilder, PT; Fletcher, S Eur J Med Chem 113: 273-92 (2016)
- Llona-Minguez, S; Höglund, A; Jacques, SA; Johansson, L; Calderón-Montaño, JM; Claesson, M; Loseva, O; Valerie, NC; Lundbäck, T; Piedrafita, J; Maga, G; Crespan, E; Meijer, L; Burgos Morón, E; Baranczewski, P; Hagbjörk, AL; Svensson, R; Wiita, E; Almlöf, I; Visnes, T; Jeppsson, F; Sigmundsson, K; Jensen, AJ; Artursson, P; Jemth, AS; Stenmark, P; Warpman Berglund, U; Scobie, M; Helleday, T J Med Chem 59: 1140-8 (2016)
- Hudson, L; Mui, J; Vázquez, S; Carvalho, DM; Williams, E; Jones, C; Bullock, AN; Hoelder, S J Med Chem 61: 7261-7272 (2018)
- Wu, T; Nagle, A; Kuhen, K; Gagaring, K; Borboa, R; Francek, C; Chen, Z; Plouffe, D; Goh, A; Lakshminarayana, SB; Wu, J; Ang, HQ; Zeng, P; Kang, ML; Tan, W; Tan, M; Ye, N; Lin, X; Caldwell, C; Ek, J; Skolnik, S; Liu, F; Wang, J; Chang, J; Li, C; Hollenbeck, T; Tuntland, T; Isbell, J; Fischli, C; Brun, R; Rottmann, M; Dartois, V; Keller, T; Diagana, T; Winzeler, E; Glynne, R; Tully, DC; Chatterjee, AK J Med Chem 54: 5116-30 (2011)
- Beattie, D; Beer, D; Bradley, ME; Bruce, I; Charlton, SJ; Cuenoud, BM; Fairhurst, RA; Farr, D; Fozard, JR; Janus, D; Rosethorne, EM; Sandham, DA; Sykes, DA; Trifilieff, A; Turner, KL; Wissler, E Bioorg Med Chem Lett 22: 6280-5 (2012)
- Li, CS; Black, WC; Brideau, C; Chan, CC; Charleson, S; Cromlish, WA; Claveau, D; Gauthier, JY; Gordon, R; Greig, G; Grimm, E; Guay, J; Lau, CK; Riendeau, D; Thérien, M; Visco, DM; Wong, E; Xu, L; Prasit, P Bioorg Med Chem Lett 9: 3181-6 (1999)
- Boja, JW; Kuhar, MJ; Kopajtic, T; Yang, E; Abraham, P; Lewin, AH; Carroll, FI J Med Chem 37: 1220-3 (1994)
- Craig, RA; Fox, BM; Hu, C; Lexa, KW; Osipov, M; Thottumkara, AP; Larhammar, M; Miyamoto, T; Rana, A; Kane, LA; Yulyaningsih, E; Solanoy, H; Nguyen, H; Chau, R; Earr, T; Kajiwara, Y; Fleck, D; Lucas, A; Haddick, PCG; Takahashi, RH; Tong, V; Wang, J; Canet, MJ; Poda, SB; Scearce-Levie, K; Srivastava, A; Sweeney, ZK; Xu, M; Zhang, R; He, J; Lei, Y; Zhuo, Z; de Vicente, J J Med Chem 65: 16290-16312 (2022)
- Pannek, M; Alhalabi, Z; Tomaselli, D; Menna, M; Fiorentino, F; Robaa, D; Weyand, M; Puhlmann, M; Tomassi, S; Barreca, F; Tafani, M; Zaganjor, E; Haigis, MC; Sippl, W; Rotili, D; Mai, A; Steegborn, C J Med Chem 67: 1843-1860
- Hagen, SE; Domagala, J; Gajda, C; Lovdahl, M; Tait, BD; Wise, E; Holler, T; Hupe, D; Nouhan, C; Urumov, A; Zeikus, G; Zeikus, E; Lunney, EA; Pavlovsky, A; Gracheck, SJ; Saunders, J; VanderRoest, S; Brodfuehrer, J J Med Chem 44: 2319-32 (2001)
- Plobeck, N; Delorme, D; Wei, ZY; Yang, H; Zhou, F; Schwarz, P; Gawell, L; Gagnon, H; Pelcman, B; Schmidt, R; Yue, SY; Walpole, C; Brown, W; Zhou, E; Labarre, M; Payza, K; St-Onge, S; Kamassah, A; Morin, PE; Projean, D; Ducharme, J; Roberts, E J Med Chem 43: 3878-94 (2000)
- Hartmann, R; Frotscher, M; Oberwinkler, S; Ziegler, E; Messinger, J; Thole, H US Patent US8546392 (2013)
- Zigmond, E; Ben Ya'acov, A; Lee, H; Lichtenstein, Y; Shalev, Z; Smith, Y; Zolotarov, L; Ziv, E; Kalman, R; Le, HV; Lu, H; Silverman, RB; Ilan, Y ACS Med Chem Lett 6: 840-4 (2015)
- Zigmond, E; Ben Ya'acov, A; Lee, H; Lichtenstein, Y; Shalev, Z; Smith, Y; Zolotarov, L; Ziv, E; Kalman, R; Le, HV; Lu, H; Silverman, RB; Ilan, Y ACS Med Chem Lett 6: 840-4 (2015)
- Zuccarello, E; Zhang, H; Acquarone, E; Pham, D; Staniszewski, A; Deng, SX; Landry, DW; Arancio, O; Fiorito, J Bioorg Med Chem Lett 92: (2023)
- Martin, SF; Austin, RE; Oalmann, CJ; Baker, WR; Condon, SL; deLara, E; Rosenberg, SH; Spina, KP; Stein, HH; Cohen, J J Med Chem 35: 1710-21 (1992)
- Joshi, P; Anderson, C; Binch, H; Hadida, S; Yoo, S; Bergeron, D; Decker, C; terHaar, E; Moore, J; Garcia-Guzman, M; Termin, A Bioorg Med Chem Lett 24: 845-9 (2014)
- Banoglu, E; Çelikoglu, E; Völker, S; Olgaç, A; Gerstmeier, J; Garscha, U; Çaliskan, B; Schubert, US; Carotti, A; Macchiarulo, A; Werz, O Eur J Med Chem 113: 1-10 (2016)
- Čapkauskaitė, E; Zakšauskas, A; Ruibys, V; Linkuvienė, V; Paketurytė, V; Gedgaudas, M; Kairys, V; Matulis, D Bioorg Med Chem 26: 675-687 (2018)
- Řezníčková, E; Tenora, L; Pospíšilová, P; Galeta, J; Jorda, R; Berka, K; Majer, P; Potáček, M; Kryštof, V Eur J Med Chem 127: 632-642 (2017)